BindingDB Reactant_set_id	Ligand SMILES	Ligand InChI	Ligand InChI Key	BindingDB MonomerID	BindingDB Ligand Name	Target Name	Target Source Organism According to Curator or DataSource	Ki (nM)	IC50 (nM)	Kd (nM)	EC50 (nM)	kon (M-1-s-1)	koff (s-1)	pH	Temp (C)	Curation/DataSource	Article DOI	BindingDB Entry DOI	PMID	PubChem AID	Patent Number	Authors	Date of publication	Date in BindingDB	Institution	Link to Ligand in BindingDB	Link to Target in BindingDB	Link to Ligand-Target Pair in BindingDB	Ligand HET ID in PDB	PDB ID(s) for Ligand-Target Complex	PubChem CID	PubChem SID	ChEBI ID of Ligand	ChEMBL ID of Ligand	DrugBank ID of Ligand	IUPHAR_GRAC ID of Ligand	KEGG ID of Ligand	ZINC ID of Ligand	Number of Protein Chains in Target (>1 implies a multichain complex)	BindingDB Target Chain Sequence 1	PDB ID(s) of Target Chain 1	UniProt (SwissProt) Recommended Name of Target Chain 1	UniProt (SwissProt) Entry Name of Target Chain 1	UniProt (SwissProt) Primary ID of Target Chain 1	UniProt (SwissProt) Secondary ID(s) of Target Chain 1	UniProt (SwissProt) Alternative ID(s) of Target Chain 1	UniProt (TrEMBL) Submitted Name of Target Chain 1	UniProt (TrEMBL) Entry Name of Target Chain 1	UniProt (TrEMBL) Primary ID of Target Chain 1	UniProt (TrEMBL) Secondary ID(s) of Target Chain 1	UniProt (TrEMBL) Alternative ID(s) of Target Chain 1	BindingDB Target Chain Sequence 2	PDB ID(s) of Target Chain 2	UniProt (SwissProt) Recommended Name of Target Chain 2	UniProt (SwissProt) Entry Name of Target Chain 2	UniProt (SwissProt) Primary ID of Target Chain 2	UniProt (SwissProt) Secondary ID(s) of Target Chain 2	UniProt (SwissProt) Alternative ID(s) of Target Chain 2	UniProt (TrEMBL) Submitted Name of Target Chain 2	UniProt (TrEMBL) Entry Name of Target Chain 2	UniProt (TrEMBL) Primary ID of Target Chain 2	UniProt (TrEMBL) Secondary ID(s) of Target Chain 2	UniProt (TrEMBL) Alternative ID(s) of Target Chain 2	BindingDB Target Chain Sequence 3	PDB ID(s) of Target Chain 3	UniProt (SwissProt) Recommended Name of Target Chain 3	UniProt (SwissProt) Entry Name of Target Chain 3	UniProt (SwissProt) Primary ID of Target Chain 3	UniProt (SwissProt) Secondary ID(s) of Target Chain 3	UniProt (SwissProt) Alternative ID(s) of Target Chain 3	UniProt (TrEMBL) Submitted Name of Target Chain 3	UniProt (TrEMBL) Entry Name of Target Chain 3	UniProt (TrEMBL) Primary ID of Target Chain 3	UniProt (TrEMBL) Secondary ID(s) of Target Chain 3	UniProt (TrEMBL) Alternative ID(s) of Target Chain 3	BindingDB Target Chain Sequence 4	PDB ID(s) of Target Chain 4	UniProt (SwissProt) Recommended Name of Target Chain 4	UniProt (SwissProt) Entry Name of Target Chain 4	UniProt (SwissProt) Primary ID of Target Chain 4	UniProt (SwissProt) Secondary ID(s) of Target Chain 4	UniProt (SwissProt) Alternative ID(s) of Target Chain 4	UniProt (TrEMBL) Submitted Name of Target Chain 4	UniProt (TrEMBL) Entry Name of Target Chain 4	UniProt (TrEMBL) Primary ID of Target Chain 4	UniProt (TrEMBL) Secondary ID(s) of Target Chain 4	UniProt (TrEMBL) Alternative ID(s) of Target Chain 4	BindingDB Target Chain Sequence 5	PDB ID(s) of Target Chain 5	UniProt (SwissProt) Recommended Name of Target Chain 5	UniProt (SwissProt) Entry Name of Target Chain 5	UniProt (SwissProt) Primary ID of Target Chain 5	UniProt (SwissProt) Secondary ID(s) of Target Chain 5	UniProt (SwissProt) Alternative ID(s) of Target Chain 5	UniProt (TrEMBL) Submitted Name of Target Chain 5	UniProt (TrEMBL) Entry Name of Target Chain 5	UniProt (TrEMBL) Primary ID of Target Chain 5	UniProt (TrEMBL) Secondary ID(s) of Target Chain 5	UniProt (TrEMBL) Alternative ID(s) of Target Chain 5	BindingDB Target Chain Sequence 6	PDB ID(s) of Target Chain 6	UniProt (SwissProt) Recommended Name of Target Chain 6	UniProt (SwissProt) Entry Name of Target Chain 6	UniProt (SwissProt) Primary ID of Target Chain 6	UniProt (SwissProt) Secondary ID(s) of Target Chain 6	UniProt (SwissProt) Alternative ID(s) of Target Chain 6	UniProt (TrEMBL) Submitted Name of Target Chain 6	UniProt (TrEMBL) Entry Name of Target Chain 6	UniProt (TrEMBL) Primary ID of Target Chain 6	UniProt (TrEMBL) Secondary ID(s) of Target Chain 6	UniProt (TrEMBL) Alternative ID(s) of Target Chain 6	BindingDB Target Chain Sequence 7	PDB ID(s) of Target Chain 7	UniProt (SwissProt) Recommended Name of Target Chain 7	UniProt (SwissProt) Entry Name of Target Chain 7	UniProt (SwissProt) Primary ID of Target Chain 7	UniProt (SwissProt) Secondary ID(s) of Target Chain 7	UniProt (SwissProt) Alternative ID(s) of Target Chain 7	UniProt (TrEMBL) Submitted Name of Target Chain 7	UniProt (TrEMBL) Entry Name of Target Chain 7	UniProt (TrEMBL) Primary ID of Target Chain 7	UniProt (TrEMBL) Secondary ID(s) of Target Chain 7	UniProt (TrEMBL) Alternative ID(s) of Target Chain 7	BindingDB Target Chain Sequence 8	PDB ID(s) of Target Chain 8	UniProt (SwissProt) Recommended Name of Target Chain 8	UniProt (SwissProt) Entry Name of Target Chain 8	UniProt (SwissProt) Primary ID of Target Chain 8	UniProt (SwissProt) Secondary ID(s) of Target Chain 8	UniProt (SwissProt) Alternative ID(s) of Target Chain 8	UniProt (TrEMBL) Submitted Name of Target Chain 8	UniProt (TrEMBL) Entry Name of Target Chain 8	UniProt (TrEMBL) Primary ID of Target Chain 8	UniProt (TrEMBL) Secondary ID(s) of Target Chain 8	UniProt (TrEMBL) Alternative ID(s) of Target Chain 8	BindingDB Target Chain Sequence 9	PDB ID(s) of Target Chain 9	UniProt (SwissProt) Recommended Name of Target Chain 9	UniProt (SwissProt) Entry Name of Target Chain 9	UniProt (SwissProt) Primary ID of Target Chain 9	UniProt (SwissProt) Secondary ID(s) of Target Chain 9	UniProt (SwissProt) Alternative ID(s) of Target Chain 9	UniProt (TrEMBL) Submitted Name of Target Chain 9	UniProt (TrEMBL) Entry Name of Target Chain 9	UniProt (TrEMBL) Primary ID of Target Chain 9	UniProt (TrEMBL) Secondary ID(s) of Target Chain 9	UniProt (TrEMBL) Alternative ID(s) of Target Chain 9	BindingDB Target Chain Sequence 10	PDB ID(s) of Target Chain 10	UniProt (SwissProt) Recommended Name of Target Chain 10	UniProt (SwissProt) Entry Name of Target Chain 10	UniProt (SwissProt) Primary ID of Target Chain 10	UniProt (SwissProt) Secondary ID(s) of Target Chain 10	UniProt (SwissProt) Alternative ID(s) of Target Chain 10	UniProt (TrEMBL) Submitted Name of Target Chain 10	UniProt (TrEMBL) Entry Name of Target Chain 10	UniProt (TrEMBL) Primary ID of Target Chain 10	UniProt (TrEMBL) Secondary ID(s) of Target Chain 10	UniProt (TrEMBL) Alternative ID(s) of Target Chain 10	BindingDB Target Chain Sequence 11	PDB ID(s) of Target Chain 11	UniProt (SwissProt) Recommended Name of Target Chain 11	UniProt (SwissProt) Entry Name of Target Chain 11	UniProt (SwissProt) Primary ID of Target Chain 11	UniProt (SwissProt) Secondary ID(s) of Target Chain 11	UniProt (SwissProt) Alternative ID(s) of Target Chain 11	UniProt (TrEMBL) Submitted Name of Target Chain 11	UniProt (TrEMBL) Entry Name of Target Chain 11	UniProt (TrEMBL) Primary ID of Target Chain 11	UniProt (TrEMBL) Secondary ID(s) of Target Chain 11	UniProt (TrEMBL) Alternative ID(s) of Target Chain 11	BindingDB Target Chain Sequence 12	PDB ID(s) of Target Chain 12	UniProt (SwissProt) Recommended Name of Target Chain 12	UniProt (SwissProt) Entry Name of Target Chain 12	UniProt (SwissProt) Primary ID of Target Chain 12	UniProt (SwissProt) Secondary ID(s) of Target Chain 12	UniProt (SwissProt) Alternative ID(s) of Target Chain 12	UniProt (TrEMBL) Submitted Name of Target Chain 12	UniProt (TrEMBL) Entry Name of Target Chain 12	UniProt (TrEMBL) Primary ID of Target Chain 12	UniProt (TrEMBL) Secondary ID(s) of Target Chain 12	UniProt (TrEMBL) Alternative ID(s) of Target Chain 12	BindingDB Target Chain Sequence 13	PDB ID(s) of Target Chain 13	UniProt (SwissProt) Recommended Name of Target Chain 13	UniProt (SwissProt) Entry Name of Target Chain 13	UniProt (SwissProt) Primary ID of Target Chain 13	UniProt (SwissProt) Secondary ID(s) of Target Chain 13	UniProt (SwissProt) Alternative ID(s) of Target Chain 13	UniProt (TrEMBL) Submitted Name of Target Chain 13	UniProt (TrEMBL) Entry Name of Target Chain 13	UniProt (TrEMBL) Primary ID of Target Chain 13	UniProt (TrEMBL) Secondary ID(s) of Target Chain 13	UniProt (TrEMBL) Alternative ID(s) of Target Chain 13	BindingDB Target Chain Sequence 14	PDB ID(s) of Target Chain 14	UniProt (SwissProt) Recommended Name of Target Chain 14	UniProt (SwissProt) Entry Name of Target Chain 14	UniProt (SwissProt) Primary ID of Target Chain 14	UniProt (SwissProt) Secondary ID(s) of Target Chain 14	UniProt (SwissProt) Alternative ID(s) of Target Chain 14	UniProt (TrEMBL) Submitted Name of Target Chain 14	UniProt (TrEMBL) Entry Name of Target Chain 14	UniProt (TrEMBL) Primary ID of Target Chain 14	UniProt (TrEMBL) Secondary ID(s) of Target Chain 14	UniProt (TrEMBL) Alternative ID(s) of Target Chain 14	BindingDB Target Chain Sequence 15	PDB ID(s) of Target Chain 15	UniProt (SwissProt) Recommended Name of Target Chain 15	UniProt (SwissProt) Entry Name of Target Chain 15	UniProt (SwissProt) Primary ID of Target Chain 15	UniProt (SwissProt) Secondary ID(s) of Target Chain 15	UniProt (SwissProt) Alternative ID(s) of Target Chain 15	UniProt (TrEMBL) Submitted Name of Target Chain 15	UniProt (TrEMBL) Entry Name of Target Chain 15	UniProt (TrEMBL) Primary ID of Target Chain 15	UniProt (TrEMBL) Secondary ID(s) of Target Chain 15	UniProt (TrEMBL) Alternative ID(s) of Target Chain 15	BindingDB Target Chain Sequence 16	PDB ID(s) of Target Chain 16	UniProt (SwissProt) Recommended Name of Target Chain 16	UniProt (SwissProt) Entry Name of Target Chain 16	UniProt (SwissProt) Primary ID of Target Chain 16	UniProt (SwissProt) Secondary ID(s) of Target Chain 16	UniProt (SwissProt) Alternative ID(s) of Target Chain 16	UniProt (TrEMBL) Submitted Name of Target Chain 16	UniProt (TrEMBL) Entry Name of Target Chain 16	UniProt (TrEMBL) Primary ID of Target Chain 16	UniProt (TrEMBL) Secondary ID(s) of Target Chain 16	UniProt (TrEMBL) Alternative ID(s) of Target Chain 16	BindingDB Target Chain Sequence 17	PDB ID(s) of Target Chain 17	UniProt (SwissProt) Recommended Name of Target Chain 17	UniProt (SwissProt) Entry Name of Target Chain 17	UniProt (SwissProt) Primary ID of Target Chain 17	UniProt (SwissProt) Secondary ID(s) of Target Chain 17	UniProt (SwissProt) Alternative ID(s) of Target Chain 17	UniProt (TrEMBL) Submitted Name of Target Chain 17	UniProt (TrEMBL) Entry Name of Target Chain 17	UniProt (TrEMBL) Primary ID of Target Chain 17	UniProt (TrEMBL) Secondary ID(s) of Target Chain 17	UniProt (TrEMBL) Alternative ID(s) of Target Chain 17	BindingDB Target Chain Sequence 18	PDB ID(s) of Target Chain 18	UniProt (SwissProt) Recommended Name of Target Chain 18	UniProt (SwissProt) Entry Name of Target Chain 18	UniProt (SwissProt) Primary ID of Target Chain 18	UniProt (SwissProt) Secondary ID(s) of Target Chain 18	UniProt (SwissProt) Alternative ID(s) of Target Chain 18	UniProt (TrEMBL) Submitted Name of Target Chain 18	UniProt (TrEMBL) Entry Name of Target Chain 18	UniProt (TrEMBL) Primary ID of Target Chain 18	UniProt (TrEMBL) Secondary ID(s) of Target Chain 18	UniProt (TrEMBL) Alternative ID(s) of Target Chain 18	BindingDB Target Chain Sequence 19	PDB ID(s) of Target Chain 19	UniProt (SwissProt) Recommended Name of Target Chain 19	UniProt (SwissProt) Entry Name of Target Chain 19	UniProt (SwissProt) Primary ID of Target Chain 19	UniProt (SwissProt) Secondary ID(s) of Target Chain 19	UniProt (SwissProt) Alternative ID(s) of Target Chain 19	UniProt (TrEMBL) Submitted Name of Target Chain 19	UniProt (TrEMBL) Entry Name of Target Chain 19	UniProt (TrEMBL) Primary ID of Target Chain 19	UniProt (TrEMBL) Secondary ID(s) of Target Chain 19	UniProt (TrEMBL) Alternative ID(s) of Target Chain 19	BindingDB Target Chain Sequence 20	PDB ID(s) of Target Chain 20	UniProt (SwissProt) Recommended Name of Target Chain 20	UniProt (SwissProt) Entry Name of Target Chain 20	UniProt (SwissProt) Primary ID of Target Chain 20	UniProt (SwissProt) Secondary ID(s) of Target Chain 20	UniProt (SwissProt) Alternative ID(s) of Target Chain 20	UniProt (TrEMBL) Submitted Name of Target Chain 20	UniProt (TrEMBL) Entry Name of Target Chain 20	UniProt (TrEMBL) Primary ID of Target Chain 20	UniProt (TrEMBL) Secondary ID(s) of Target Chain 20	UniProt (TrEMBL) Alternative ID(s) of Target Chain 20	BindingDB Target Chain Sequence 21	PDB ID(s) of Target Chain 21	UniProt (SwissProt) Recommended Name of Target Chain 21	UniProt (SwissProt) Entry Name of Target Chain 21	UniProt (SwissProt) Primary ID of Target Chain 21	UniProt (SwissProt) Secondary ID(s) of Target Chain 21	UniProt (SwissProt) Alternative ID(s) of Target Chain 21	UniProt (TrEMBL) Submitted Name of Target Chain 21	UniProt (TrEMBL) Entry Name of Target Chain 21	UniProt (TrEMBL) Primary ID of Target Chain 21	UniProt (TrEMBL) Secondary ID(s) of Target Chain 21	UniProt (TrEMBL) Alternative ID(s) of Target Chain 21	BindingDB Target Chain Sequence 22	PDB ID(s) of Target Chain 22	UniProt (SwissProt) Recommended Name of Target Chain 22	UniProt (SwissProt) Entry Name of Target Chain 22	UniProt (SwissProt) Primary ID of Target Chain 22	UniProt (SwissProt) Secondary ID(s) of Target Chain 22	UniProt (SwissProt) Alternative ID(s) of Target Chain 22	UniProt (TrEMBL) Submitted Name of Target Chain 22	UniProt (TrEMBL) Entry Name of Target Chain 22	UniProt (TrEMBL) Primary ID of Target Chain 22	UniProt (TrEMBL) Secondary ID(s) of Target Chain 22	UniProt (TrEMBL) Alternative ID(s) of Target Chain 22	BindingDB Target Chain Sequence 23	PDB ID(s) of Target Chain 23	UniProt (SwissProt) Recommended Name of Target Chain 23	UniProt (SwissProt) Entry Name of Target Chain 23	UniProt (SwissProt) Primary ID of Target Chain 23	UniProt (SwissProt) Secondary ID(s) of Target Chain 23	UniProt (SwissProt) Alternative ID(s) of Target Chain 23	UniProt (TrEMBL) Submitted Name of Target Chain 23	UniProt (TrEMBL) Entry Name of Target Chain 23	UniProt (TrEMBL) Primary ID of Target Chain 23	UniProt (TrEMBL) Secondary ID(s) of Target Chain 23	UniProt (TrEMBL) Alternative ID(s) of Target Chain 23	BindingDB Target Chain Sequence 24	PDB ID(s) of Target Chain 24	UniProt (SwissProt) Recommended Name of Target Chain 24	UniProt (SwissProt) Entry Name of Target Chain 24	UniProt (SwissProt) Primary ID of Target Chain 24	UniProt (SwissProt) Secondary ID(s) of Target Chain 24	UniProt (SwissProt) Alternative ID(s) of Target Chain 24	UniProt (TrEMBL) Submitted Name of Target Chain 24	UniProt (TrEMBL) Entry Name of Target Chain 24	UniProt (TrEMBL) Primary ID of Target Chain 24	UniProt (TrEMBL) Secondary ID(s) of Target Chain 24	UniProt (TrEMBL) Alternative ID(s) of Target Chain 24	BindingDB Target Chain Sequence 25	PDB ID(s) of Target Chain 25	UniProt (SwissProt) Recommended Name of Target Chain 25	UniProt (SwissProt) Entry Name of Target Chain 25	UniProt (SwissProt) Primary ID of Target Chain 25	UniProt (SwissProt) Secondary ID(s) of Target Chain 25	UniProt (SwissProt) Alternative ID(s) of Target Chain 25	UniProt (TrEMBL) Submitted Name of Target Chain 25	UniProt (TrEMBL) Entry Name of Target Chain 25	UniProt (TrEMBL) Primary ID of Target Chain 25	UniProt (TrEMBL) Secondary ID(s) of Target Chain 25	UniProt (TrEMBL) Alternative ID(s) of Target Chain 25	BindingDB Target Chain Sequence 26	PDB ID(s) of Target Chain 26	UniProt (SwissProt) Recommended Name of Target Chain 26	UniProt (SwissProt) Entry Name of Target Chain 26	UniProt (SwissProt) Primary ID of Target Chain 26	UniProt (SwissProt) Secondary ID(s) of Target Chain 26	UniProt (SwissProt) Alternative ID(s) of Target Chain 26	UniProt (TrEMBL) Submitted Name of Target Chain 26	UniProt (TrEMBL) Entry Name of Target Chain 26	UniProt (TrEMBL) Primary ID of Target Chain 26	UniProt (TrEMBL) Secondary ID(s) of Target Chain 26	UniProt (TrEMBL) Alternative ID(s) of Target Chain 26	BindingDB Target Chain Sequence 27	PDB ID(s) of Target Chain 27	UniProt (SwissProt) Recommended Name of Target Chain 27	UniProt (SwissProt) Entry Name of Target Chain 27	UniProt (SwissProt) Primary ID of Target Chain 27	UniProt (SwissProt) Secondary ID(s) of Target Chain 27	UniProt (SwissProt) Alternative ID(s) of Target Chain 27	UniProt (TrEMBL) Submitted Name of Target Chain 27	UniProt (TrEMBL) Entry Name of Target Chain 27	UniProt (TrEMBL) Primary ID of Target Chain 27	UniProt (TrEMBL) Secondary ID(s) of Target Chain 27	UniProt (TrEMBL) Alternative ID(s) of Target Chain 27	BindingDB Target Chain Sequence 28	PDB ID(s) of Target Chain 28	UniProt (SwissProt) Recommended Name of Target Chain 28	UniProt (SwissProt) Entry Name of Target Chain 28	UniProt (SwissProt) Primary ID of Target Chain 28	UniProt (SwissProt) Secondary ID(s) of Target Chain 28	UniProt (SwissProt) Alternative ID(s) of Target Chain 28	UniProt (TrEMBL) Submitted Name of Target Chain 28	UniProt (TrEMBL) Entry Name of Target Chain 28	UniProt (TrEMBL) Primary ID of Target Chain 28	UniProt (TrEMBL) Secondary ID(s) of Target Chain 28	UniProt (TrEMBL) Alternative ID(s) of Target Chain 28	BindingDB Target Chain Sequence 29	PDB ID(s) of Target Chain 29	UniProt (SwissProt) Recommended Name of Target Chain 29	UniProt (SwissProt) Entry Name of Target Chain 29	UniProt (SwissProt) Primary ID of Target Chain 29	UniProt (SwissProt) Secondary ID(s) of Target Chain 29	UniProt (SwissProt) Alternative ID(s) of Target Chain 29	UniProt (TrEMBL) Submitted Name of Target Chain 29	UniProt (TrEMBL) Entry Name of Target Chain 29	UniProt (TrEMBL) Primary ID of Target Chain 29	UniProt (TrEMBL) Secondary ID(s) of Target Chain 29	UniProt (TrEMBL) Alternative ID(s) of Target Chain 29	BindingDB Target Chain Sequence 30	PDB ID(s) of Target Chain 30	UniProt (SwissProt) Recommended Name of Target Chain 30	UniProt (SwissProt) Entry Name of Target Chain 30	UniProt (SwissProt) Primary ID of Target Chain 30	UniProt (SwissProt) Secondary ID(s) of Target Chain 30	UniProt (SwissProt) Alternative ID(s) of Target Chain 30	UniProt (TrEMBL) Submitted Name of Target Chain 30	UniProt (TrEMBL) Entry Name of Target Chain 30	UniProt (TrEMBL) Primary ID of Target Chain 30	UniProt (TrEMBL) Secondary ID(s) of Target Chain 30	UniProt (TrEMBL) Alternative ID(s) of Target Chain 30	BindingDB Target Chain Sequence 31	PDB ID(s) of Target Chain 31	UniProt (SwissProt) Recommended Name of Target Chain 31	UniProt (SwissProt) Entry Name of Target Chain 31	UniProt (SwissProt) Primary ID of Target Chain 31	UniProt (SwissProt) Secondary ID(s) of Target Chain 31	UniProt (SwissProt) Alternative ID(s) of Target Chain 31	UniProt (TrEMBL) Submitted Name of Target Chain 31	UniProt (TrEMBL) Entry Name of Target Chain 31	UniProt (TrEMBL) Primary ID of Target Chain 31	UniProt (TrEMBL) Secondary ID(s) of Target Chain 31	UniProt (TrEMBL) Alternative ID(s) of Target Chain 31	BindingDB Target Chain Sequence 32	PDB ID(s) of Target Chain 32	UniProt (SwissProt) Recommended Name of Target Chain 32	UniProt (SwissProt) Entry Name of Target Chain 32	UniProt (SwissProt) Primary ID of Target Chain 32	UniProt (SwissProt) Secondary ID(s) of Target Chain 32	UniProt (SwissProt) Alternative ID(s) of Target Chain 32	UniProt (TrEMBL) Submitted Name of Target Chain 32	UniProt (TrEMBL) Entry Name of Target Chain 32	UniProt (TrEMBL) Primary ID of Target Chain 32	UniProt (TrEMBL) Secondary ID(s) of Target Chain 32	UniProt (TrEMBL) Alternative ID(s) of Target Chain 32	BindingDB Target Chain Sequence 33	PDB ID(s) of Target Chain 33	UniProt (SwissProt) Recommended Name of Target Chain 33	UniProt (SwissProt) Entry Name of Target Chain 33	UniProt (SwissProt) Primary ID of Target Chain 33	UniProt (SwissProt) Secondary ID(s) of Target Chain 33	UniProt (SwissProt) Alternative ID(s) of Target Chain 33	UniProt (TrEMBL) Submitted Name of Target Chain 33	UniProt (TrEMBL) Entry Name of Target Chain 33	UniProt (TrEMBL) Primary ID of Target Chain 33	UniProt (TrEMBL) Secondary ID(s) of Target Chain 33	UniProt (TrEMBL) Alternative ID(s) of Target Chain 33	BindingDB Target Chain Sequence 34	PDB ID(s) of Target Chain 34	UniProt (SwissProt) Recommended Name of Target Chain 34	UniProt (SwissProt) Entry Name of Target Chain 34	UniProt (SwissProt) Primary ID of Target Chain 34	UniProt (SwissProt) Secondary ID(s) of Target Chain 34	UniProt (SwissProt) Alternative ID(s) of Target Chain 34	UniProt (TrEMBL) Submitted Name of Target Chain 34	UniProt (TrEMBL) Entry Name of Target Chain 34	UniProt (TrEMBL) Primary ID of Target Chain 34	UniProt (TrEMBL) Secondary ID(s) of Target Chain 34	UniProt (TrEMBL) Alternative ID(s) of Target Chain 34	BindingDB Target Chain Sequence 35	PDB ID(s) of Target Chain 35	UniProt (SwissProt) Recommended Name of Target Chain 35	UniProt (SwissProt) Entry Name of Target Chain 35	UniProt (SwissProt) Primary ID of Target Chain 35	UniProt (SwissProt) Secondary ID(s) of Target Chain 35	UniProt (SwissProt) Alternative ID(s) of Target Chain 35	UniProt (TrEMBL) Submitted Name of Target Chain 35	UniProt (TrEMBL) Entry Name of Target Chain 35	UniProt (TrEMBL) Primary ID of Target Chain 35	UniProt (TrEMBL) Secondary ID(s) of Target Chain 35	UniProt (TrEMBL) Alternative ID(s) of Target Chain 35	BindingDB Target Chain Sequence 36	PDB ID(s) of Target Chain 36	UniProt (SwissProt) Recommended Name of Target Chain 36	UniProt (SwissProt) Entry Name of Target Chain 36	UniProt (SwissProt) Primary ID of Target Chain 36	UniProt (SwissProt) Secondary ID(s) of Target Chain 36	UniProt (SwissProt) Alternative ID(s) of Target Chain 36	UniProt (TrEMBL) Submitted Name of Target Chain 36	UniProt (TrEMBL) Entry Name of Target Chain 36	UniProt (TrEMBL) Primary ID of Target Chain 36	UniProt (TrEMBL) Secondary ID(s) of Target Chain 36	UniProt (TrEMBL) Alternative ID(s) of Target Chain 36	BindingDB Target Chain Sequence 37	PDB ID(s) of Target Chain 37	UniProt (SwissProt) Recommended Name of Target Chain 37	UniProt (SwissProt) Entry Name of Target Chain 37	UniProt (SwissProt) Primary ID of Target Chain 37	UniProt (SwissProt) Secondary ID(s) of Target Chain 37	UniProt (SwissProt) Alternative ID(s) of Target Chain 37	UniProt (TrEMBL) Submitted Name of Target Chain 37	UniProt (TrEMBL) Entry Name of Target Chain 37	UniProt (TrEMBL) Primary ID of Target Chain 37	UniProt (TrEMBL) Secondary ID(s) of Target Chain 37	UniProt (TrEMBL) Alternative ID(s) of Target Chain 37	BindingDB Target Chain Sequence 38	PDB ID(s) of Target Chain 38	UniProt (SwissProt) Recommended Name of Target Chain 38	UniProt (SwissProt) Entry Name of Target Chain 38	UniProt (SwissProt) Primary ID of Target Chain 38	UniProt (SwissProt) Secondary ID(s) of Target Chain 38	UniProt (SwissProt) Alternative ID(s) of Target Chain 38	UniProt (TrEMBL) Submitted Name of Target Chain 38	UniProt (TrEMBL) Entry Name of Target Chain 38	UniProt (TrEMBL) Primary ID of Target Chain 38	UniProt (TrEMBL) Secondary ID(s) of Target Chain 38	UniProt (TrEMBL) Alternative ID(s) of Target Chain 38	BindingDB Target Chain Sequence 39	PDB ID(s) of Target Chain 39	UniProt (SwissProt) Recommended Name of Target Chain 39	UniProt (SwissProt) Entry Name of Target Chain 39	UniProt (SwissProt) Primary ID of Target Chain 39	UniProt (SwissProt) Secondary ID(s) of Target Chain 39	UniProt (SwissProt) Alternative ID(s) of Target Chain 39	UniProt (TrEMBL) Submitted Name of Target Chain 39	UniProt (TrEMBL) Entry Name of Target Chain 39	UniProt (TrEMBL) Primary ID of Target Chain 39	UniProt (TrEMBL) Secondary ID(s) of Target Chain 39	UniProt (TrEMBL) Alternative ID(s) of Target Chain 39	BindingDB Target Chain Sequence 40	PDB ID(s) of Target Chain 40	UniProt (SwissProt) Recommended Name of Target Chain 40	UniProt (SwissProt) Entry Name of Target Chain 40	UniProt (SwissProt) Primary ID of Target Chain 40	UniProt (SwissProt) Secondary ID(s) of Target Chain 40	UniProt (SwissProt) Alternative ID(s) of Target Chain 40	UniProt (TrEMBL) Submitted Name of Target Chain 40	UniProt (TrEMBL) Entry Name of Target Chain 40	UniProt (TrEMBL) Primary ID of Target Chain 40	UniProt (TrEMBL) Secondary ID(s) of Target Chain 40	UniProt (TrEMBL) Alternative ID(s) of Target Chain 40	BindingDB Target Chain Sequence 41	PDB ID(s) of Target Chain 41	UniProt (SwissProt) Recommended Name of Target Chain 41	UniProt (SwissProt) Entry Name of Target Chain 41	UniProt (SwissProt) Primary ID of Target Chain 41	UniProt (SwissProt) Secondary ID(s) of Target Chain 41	UniProt (SwissProt) Alternative ID(s) of Target Chain 41	UniProt (TrEMBL) Submitted Name of Target Chain 41	UniProt (TrEMBL) Entry Name of Target Chain 41	UniProt (TrEMBL) Primary ID of Target Chain 41	UniProt (TrEMBL) Secondary ID(s) of Target Chain 41	UniProt (TrEMBL) Alternative ID(s) of Target Chain 41	BindingDB Target Chain Sequence 42	PDB ID(s) of Target Chain 42	UniProt (SwissProt) Recommended Name of Target Chain 42	UniProt (SwissProt) Entry Name of Target Chain 42	UniProt (SwissProt) Primary ID of Target Chain 42	UniProt (SwissProt) Secondary ID(s) of Target Chain 42	UniProt (SwissProt) Alternative ID(s) of Target Chain 42	UniProt (TrEMBL) Submitted Name of Target Chain 42	UniProt (TrEMBL) Entry Name of Target Chain 42	UniProt (TrEMBL) Primary ID of Target Chain 42	UniProt (TrEMBL) Secondary ID(s) of Target Chain 42	UniProt (TrEMBL) Alternative ID(s) of Target Chain 42	BindingDB Target Chain Sequence 43	PDB ID(s) of Target Chain 43	UniProt (SwissProt) Recommended Name of Target Chain 43	UniProt (SwissProt) Entry Name of Target Chain 43	UniProt (SwissProt) Primary ID of Target Chain 43	UniProt (SwissProt) Secondary ID(s) of Target Chain 43	UniProt (SwissProt) Alternative ID(s) of Target Chain 43	UniProt (TrEMBL) Submitted Name of Target Chain 43	UniProt (TrEMBL) Entry Name of Target Chain 43	UniProt (TrEMBL) Primary ID of Target Chain 43	UniProt (TrEMBL) Secondary ID(s) of Target Chain 43	UniProt (TrEMBL) Alternative ID(s) of Target Chain 43	BindingDB Target Chain Sequence 44	PDB ID(s) of Target Chain 44	UniProt (SwissProt) Recommended Name of Target Chain 44	UniProt (SwissProt) Entry Name of Target Chain 44	UniProt (SwissProt) Primary ID of Target Chain 44	UniProt (SwissProt) Secondary ID(s) of Target Chain 44	UniProt (SwissProt) Alternative ID(s) of Target Chain 44	UniProt (TrEMBL) Submitted Name of Target Chain 44	UniProt (TrEMBL) Entry Name of Target Chain 44	UniProt (TrEMBL) Primary ID of Target Chain 44	UniProt (TrEMBL) Secondary ID(s) of Target Chain 44	UniProt (TrEMBL) Alternative ID(s) of Target Chain 44	BindingDB Target Chain Sequence 45	PDB ID(s) of Target Chain 45	UniProt (SwissProt) Recommended Name of Target Chain 45	UniProt (SwissProt) Entry Name of Target Chain 45	UniProt (SwissProt) Primary ID of Target Chain 45	UniProt (SwissProt) Secondary ID(s) of Target Chain 45	UniProt (SwissProt) Alternative ID(s) of Target Chain 45	UniProt (TrEMBL) Submitted Name of Target Chain 45	UniProt (TrEMBL) Entry Name of Target Chain 45	UniProt (TrEMBL) Primary ID of Target Chain 45	UniProt (TrEMBL) Secondary ID(s) of Target Chain 45	UniProt (TrEMBL) Alternative ID(s) of Target Chain 45	BindingDB Target Chain Sequence 46	PDB ID(s) of Target Chain 46	UniProt (SwissProt) Recommended Name of Target Chain 46	UniProt (SwissProt) Entry Name of Target Chain 46	UniProt (SwissProt) Primary ID of Target Chain 46	UniProt (SwissProt) Secondary ID(s) of Target Chain 46	UniProt (SwissProt) Alternative ID(s) of Target Chain 46	UniProt (TrEMBL) Submitted Name of Target Chain 46	UniProt (TrEMBL) Entry Name of Target Chain 46	UniProt (TrEMBL) Primary ID of Target Chain 46	UniProt (TrEMBL) Secondary ID(s) of Target Chain 46	UniProt (TrEMBL) Alternative ID(s) of Target Chain 46	BindingDB Target Chain Sequence 47	PDB ID(s) of Target Chain 47	UniProt (SwissProt) Recommended Name of Target Chain 47	UniProt (SwissProt) Entry Name of Target Chain 47	UniProt (SwissProt) Primary ID of Target Chain 47	UniProt (SwissProt) Secondary ID(s) of Target Chain 47	UniProt (SwissProt) Alternative ID(s) of Target Chain 47	UniProt (TrEMBL) Submitted Name of Target Chain 47	UniProt (TrEMBL) Entry Name of Target Chain 47	UniProt (TrEMBL) Primary ID of Target Chain 47	UniProt (TrEMBL) Secondary ID(s) of Target Chain 47	UniProt (TrEMBL) Alternative ID(s) of Target Chain 47	BindingDB Target Chain Sequence 48	PDB ID(s) of Target Chain 48	UniProt (SwissProt) Recommended Name of Target Chain 48	UniProt (SwissProt) Entry Name of Target Chain 48	UniProt (SwissProt) Primary ID of Target Chain 48	UniProt (SwissProt) Secondary ID(s) of Target Chain 48	UniProt (SwissProt) Alternative ID(s) of Target Chain 48	UniProt (TrEMBL) Submitted Name of Target Chain 48	UniProt (TrEMBL) Entry Name of Target Chain 48	UniProt (TrEMBL) Primary ID of Target Chain 48	UniProt (TrEMBL) Secondary ID(s) of Target Chain 48	UniProt (TrEMBL) Alternative ID(s) of Target Chain 48	BindingDB Target Chain Sequence 49	PDB ID(s) of Target Chain 49	UniProt (SwissProt) Recommended Name of Target Chain 49	UniProt (SwissProt) Entry Name of Target Chain 49	UniProt (SwissProt) Primary ID of Target Chain 49	UniProt (SwissProt) Secondary ID(s) of Target Chain 49	UniProt (SwissProt) Alternative ID(s) of Target Chain 49	UniProt (TrEMBL) Submitted Name of Target Chain 49	UniProt (TrEMBL) Entry Name of Target Chain 49	UniProt (TrEMBL) Primary ID of Target Chain 49	UniProt (TrEMBL) Secondary ID(s) of Target Chain 49	UniProt (TrEMBL) Alternative ID(s) of Target Chain 49	BindingDB Target Chain Sequence 50	PDB ID(s) of Target Chain 50	UniProt (SwissProt) Recommended Name of Target Chain 50	UniProt (SwissProt) Entry Name of Target Chain 50	UniProt (SwissProt) Primary ID of Target Chain 50	UniProt (SwissProt) Secondary ID(s) of Target Chain 50	UniProt (SwissProt) Alternative ID(s) of Target Chain 50	UniProt (TrEMBL) Submitted Name of Target Chain 50	UniProt (TrEMBL) Entry Name of Target Chain 50	UniProt (TrEMBL) Primary ID of Target Chain 50	UniProt (TrEMBL) Secondary ID(s) of Target Chain 50	UniProt (TrEMBL) Alternative ID(s) of Target Chain 50
126274	CC(C)Oc1cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2cc1F	InChI=1S/C19H16ClFN4O2/c1-8(2)27-15-5-10-14(6-13(15)21)24-19(26)17(22)16(10)9-3-4-12(20)18-11(9)7-23-25-18/h3-8H,22H2,1-2H3,(H,23,25)(H,24,26)	QHEONYKAIWOVCG-UHFFFAOYSA-N	794652	3-Amino-4-(7-chloro-1H-indazol-4-yl)-7-fluoro-6-propan-2-yloxy-1H-quinolin-2-one::US20260062412, Compound A1	Myelin transcription factor 1	Homo sapiens		 29.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794652	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794652&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293806	528826115							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126275	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(OCCC(F)F)c(F)cc2[nH]c1=O	InChI=1S/C19H14ClF3N4O2/c20-11-2-1-8(10-7-25-27-18(10)11)16-9-5-14(29-4-3-15(22)23)12(21)6-13(9)26-19(28)17(16)24/h1-2,5-7,15H,3-4,24H2,(H,25,27)(H,26,28)	NEMCMVVKARKURO-UHFFFAOYSA-N	794655	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-(3,3-difluoropropoxy)-7-fluoro-1H-quinolin-2-one::US20260062412, Compound A2	Myelin transcription factor 1	Homo sapiens		 9.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794655	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794655&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293288	528826118							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126276	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(OCC3CC3)c(F)cc2[nH]c1=O	InChI=1S/C20H16ClFN4O2/c21-13-4-3-10(12-7-24-26-19(12)13)17-11-5-16(28-8-9-1-2-9)14(22)6-15(11)25-20(27)18(17)23/h3-7,9H,1-2,8,23H2,(H,24,26)(H,25,27)	VUVPZFHPDMZIII-UHFFFAOYSA-N	794660	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-(cyclopropylmethoxy)-7-fluoro-1H-quinolin-2-one::US20260062412, Compound A3	Myelin transcription factor 1	Homo sapiens		 8.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794660	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794660&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293222	528826123							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126277	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(O[C@H]3C[C@H](F)C3)c(F)cc2[nH]c1=O	InChI=1S/C20H15ClF2N4O2/c21-13-2-1-10(12-7-25-27-19(12)13)17-11-5-16(29-9-3-8(22)4-9)14(23)6-15(11)26-20(28)18(17)24/h1-2,5-9H,3-4,24H2,(H,25,27)(H,26,28)	FWYYSRXGENGHEW-UHFFFAOYSA-N	794661	3-Amino-4-(7-chloro-1H-indazol-4-yl)-7-fluoro-6-((1r,3r)-3-fluorocyclobutyl)oxy-1H-quinolin-2-one::US20260062412, Compound A4	Myelin transcription factor 1	Homo sapiens		 3.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794661	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794661&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293619	528826124							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126278	N#C[C@H]1C[C@H](Oc2cc3c(-c4ccc(Cl)c5[nH]ncc45)c(N)c(=O)[nH]c3cc2F)C1	InChI=1S/C21H15ClFN5O2/c22-14-2-1-11(13-8-26-28-20(13)14)18-12-5-17(30-10-3-9(4-10)7-24)15(23)6-16(12)27-21(29)19(18)25/h1-2,5-6,8-10H,3-4,25H2,(H,26,28)(H,27,29)	JWCPFHPHVOMTES-UHFFFAOYSA-N	794662	(1r,3r)-3-[[3-Amino-4-(7-chloro-1H-indazol-4-yl)-7-fluoro-2-oxo-1H-quinolin-6-yl]oxy]cyclobutane-1-carbonitrile::US20260062412, Compound A5	Myelin transcription factor 1	Homo sapiens		 1.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794662	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794662&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293525	528826125							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126279	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(OCCCF)c(F)cc2[nH]c1=O	InChI=1S/C19H15ClF2N4O2/c20-12-3-2-9(11-8-24-26-18(11)12)16-10-6-15(28-5-1-4-21)13(22)7-14(10)25-19(27)17(16)23/h2-3,6-8H,1,4-5,23H2,(H,24,26)(H,25,27)	SCGMAKRGVWBIOT-UHFFFAOYSA-N	794663	3-Amino-4-(7-chloro-1H-indazol-4-yl)-7-fluoro-6-(3-fluoropropoxy)-1H-quinolin-2-one::US20260062412, Compound A6	Myelin transcription factor 1	Homo sapiens		 3.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794663	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794663&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293754	528826126							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126280	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(OC3CCC3)c(F)cc2[nH]c1=O	InChI=1S/C20H16ClFN4O2/c21-13-5-4-10(12-8-24-26-19(12)13)17-11-6-16(28-9-2-1-3-9)14(22)7-15(11)25-20(27)18(17)23/h4-9H,1-3,23H2,(H,24,26)(H,25,27)	WMVFZVNBMIYCSU-UHFFFAOYSA-N	794664	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-cyclobutyloxy-7-fluoro-1H-quinolin-2-one::US20260062412, Compound A7	Myelin transcription factor 1	Homo sapiens		 4.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794664	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794664&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293210	528826127							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126281	CC(C)Oc1cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2cc1Cl	InChI=1S/C19H16Cl2N4O2/c1-8(2)27-15-5-10-14(6-13(15)21)24-19(26)17(22)16(10)9-3-4-12(20)18-11(9)7-23-25-18/h3-8H,22H2,1-2H3,(H,23,25)(H,24,26)	CJVFOLKYLDNLDS-UHFFFAOYSA-N	794665	3-Amino-7-chloro-4-(7-chloro-1H-indazol-4-yl)-6-propan-2-yloxy-1H-quinolin-2-one::US20260062412, Compound A8	Myelin transcription factor 1	Homo sapiens		 23.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794665	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794665&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293199	528826128							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126282	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(OCCC(F)F)c(Cl)cc2[nH]c1=O	InChI=1S/C19H14Cl2F2N4O2/c20-11-2-1-8(10-7-25-27-18(10)11)16-9-5-14(29-4-3-15(22)23)12(21)6-13(9)26-19(28)17(16)24/h1-2,5-7,15H,3-4,24H2,(H,25,27)(H,26,28)	HSOVQMBJRFIYOT-UHFFFAOYSA-N	794666	3-Amino-7-chloro-4-(7-chloro-1H-indazol-4-yl)-6-(3,3-difluoropropoxy)-1H-quinolin-2-one::US20260062412, Compound A9	Myelin transcription factor 1	Homo sapiens		 3.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794666	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794666&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293611	528826129							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126283	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(OC3CCC3)c(Cl)cc2[nH]c1=O	InChI=1S/C20H16Cl2N4O2/c21-13-5-4-10(12-8-24-26-19(12)13)17-11-6-16(28-9-2-1-3-9)14(22)7-15(11)25-20(27)18(17)23/h4-9H,1-3,23H2,(H,24,26)(H,25,27)	ARBCACCEBDYAMK-UHFFFAOYSA-N	794667	3-Amino-7-chloro-4-(7-chloro-1H-indazol-4-yl)-6-cyclobutyloxy-1H-quinolin-2-one::US20260062412, Compound A10	Myelin transcription factor 1	Homo sapiens		 4.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794667	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794667&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293879	528826130							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126284	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(O[C@H]3C[C@H](F)C3)c(Cl)cc2[nH]c1=O	InChI=1S/C20H15Cl2FN4O2/c21-13-2-1-10(12-7-25-27-19(12)13)17-11-5-16(29-9-3-8(23)4-9)14(22)6-15(11)26-20(28)18(17)24/h1-2,5-9H,3-4,24H2,(H,25,27)(H,26,28)	KYWCRTUUUQMSSJ-UHFFFAOYSA-N	794668	3-Amino-7-chloro-4-(7-chloro-1H-indazol-4-yl)-6-((1r,3r)-3-fluorocyclobutyl)oxy-1H-quinolin-2-one::US20260062412, Compound A11	Myelin transcription factor 1	Homo sapiens		 3.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794668	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794668&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293416	528826131							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126285	N#C[C@H]1C[C@H](Oc2cc3c(-c4ccc(Cl)c5[nH]ncc45)c(N)c(=O)[nH]c3cc2Cl)C1	InChI=1S/C21H15Cl2N5O2/c22-14-2-1-11(13-8-26-28-20(13)14)18-12-5-17(30-10-3-9(4-10)7-24)15(23)6-16(12)27-21(29)19(18)25/h1-2,5-6,8-10H,3-4,25H2,(H,26,28)(H,27,29)	NYQWVQMLTLBLNI-UHFFFAOYSA-N	794669	(1r,3r)-3-[[3-Amino-7-chloro-4-(7-chloro-1H-indazol-4-yl)-2-oxo-1H-quinolin-6-yl]oxy]cyclobutane-1-carbonitrile::US20260062412, Compound A12	Myelin transcription factor 1	Homo sapiens		 2.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794669	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794669&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293807	528826132							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126286	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(OCC3CC3)c(Cl)cc2[nH]c1=O	InChI=1S/C20H16Cl2N4O2/c21-13-4-3-10(12-7-24-26-19(12)13)17-11-5-16(28-8-9-1-2-9)14(22)6-15(11)25-20(27)18(17)23/h3-7,9H,1-2,8,23H2,(H,24,26)(H,25,27)	AXGUNYUZVITTMY-UHFFFAOYSA-N	794670	3-Amino-7-chloro-4-(7-chloro-1H-indazol-4-yl)-6-(cyclopropylmethoxy)-1H-quinolin-2-one::US20260062412, Compound A13	Myelin transcription factor 1	Homo sapiens		 18.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794670	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794670&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293494	528826133							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126287	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(OCCCF)c(Cl)cc2[nH]c1=O	InChI=1S/C19H15Cl2FN4O2/c20-12-3-2-9(11-8-24-26-18(11)12)16-10-6-15(28-5-1-4-22)13(21)7-14(10)25-19(27)17(16)23/h2-3,6-8H,1,4-5,23H2,(H,24,26)(H,25,27)	RQRLOHXFRVDNJO-UHFFFAOYSA-N	794671	3-Amino-7-chloro-4-(7-chloro-1H-indazol-4-yl)-6-(3-fluoropropoxy)-1H-quinolin-2-one::US20260062412, Compound A14	Myelin transcription factor 1	Homo sapiens		 2.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794671	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794671&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293916	528826134							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126288	Cc1nc2[nH]c(=O)c(N)c(-c3ccc(Cl)c4[nH]ncc34)c2cc1O[C@H]1C[C@H](F)C1	InChI=1S/C20H17ClFN5O2/c1-8-15(29-10-4-9(22)5-10)6-12-16(17(23)20(28)26-19(12)25-8)11-2-3-14(21)18-13(11)7-24-27-18/h2-3,6-7,9-10H,4-5,23H2,1H3,(H,24,27)(H,25,26,28)	WGKKYFQPPPRSKG-UHFFFAOYSA-N	794672	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-((1r,3r)-3-fluorocyclobutyl)oxy-7-methyl-1H-1,8-naphthyridin-2-one::US20260062412, Compound A15	Myelin transcription factor 1	Homo sapiens		 13.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794672	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794672&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293821	528826135							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126289	Cc1nc2[nH]c(=O)c(N)c(-c3ccc(Cl)c4[nH]ncc34)c2cc1O[C@H]1C[C@H](C#N)C1	InChI=1S/C21H17ClN6O2/c1-9-16(30-11-4-10(5-11)7-23)6-13-17(18(24)21(29)27-20(13)26-9)12-2-3-15(22)19-14(12)8-25-28-19/h2-3,6,8,10-11H,4-5,24H2,1H3,(H,25,28)(H,26,27,29)	GSBMMFXCVVFENB-UHFFFAOYSA-N	794673	(1r,3r)-3-[[6-Amino-5-(7-chloro-1H-indazol-4-yl)-2-methyl-7-oxo-8H-1,8-naphthyridine-3-yl]oxy]cyclobutane-1-carbonitrile::US20260062412, Compound A16	Myelin transcription factor 1	Homo sapiens		 5.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794673	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794673&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293390	528826136							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126290	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Cl)cc(Br)c2[nH]c1=O	InChI=1S/C16H9BrCl2N4O/c17-10-4-6(18)3-8-12(13(20)16(24)22-14(8)10)7-1-2-11(19)15-9(7)5-21-23-15/h1-5H,20H2,(H,21,23)(H,22,24)	RKWWUDHFXDADSJ-UHFFFAOYSA-N	794674	3-Amino-8-bromo-6-chloro-4-(7-chloro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A17	Myelin transcription factor 1	Homo sapiens		 27.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794674	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794674&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293856	528826137							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126291	C#Cc1cc(Cl)cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C18H10Cl2N4O/c1-2-8-5-9(19)6-11-14(15(21)18(25)23-16(8)11)10-3-4-13(20)17-12(10)7-22-24-17/h1,3-7H,21H2,(H,22,24)(H,23,25)	NWQGFQSQIXINNK-UHFFFAOYSA-N	794675	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-8-ethynyl-1H-quinolin-2-one::US20260062412, Compound A18	Myelin transcription factor 1	Homo sapiens		 87.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794675	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794675&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293796	528826138							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126292	CC(C)c1cc(Cl)cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C19H16Cl2N4O/c1-8(2)11-5-9(20)6-12-15(16(22)19(26)24-17(11)12)10-3-4-14(21)18-13(10)7-23-25-18/h3-8H,22H2,1-2H3,(H,23,25)(H,24,26)	PMFALPQGGKNLJK-UHFFFAOYSA-N	794676	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-8-propan-2-yl-1H-quinolin-2-one::US20260062412, Compound A19	Myelin transcription factor 1	Homo sapiens		 600							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794676	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794676&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293207	528826139							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126293	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Cl)cc(Cl)c2[nH]c1=O	InChI=1S/C16H9Cl3N4O/c17-6-3-8-12(13(20)16(24)22-14(8)11(19)4-6)7-1-2-10(18)15-9(7)5-21-23-15/h1-5H,20H2,(H,21,23)(H,22,24)	MQICUHHIBTVHTR-UHFFFAOYSA-N	794677	3-Amino-6,8-dichloro-4-(7-chloro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A20	Myelin transcription factor 1	Homo sapiens		 12.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794677	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794677&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293549	528826140							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126294	N#Cc1cc(Cl)cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C17H9Cl2N5O/c18-8-3-7(5-20)15-10(4-8)13(14(21)17(25)23-15)9-1-2-12(19)16-11(9)6-22-24-16/h1-4,6H,21H2,(H,22,24)(H,23,25)	FIMUPDPURKXAMK-UHFFFAOYSA-N	794678	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-2-oxo-1H-quinoline-8-carbonitrile::US20260062412, Compound A21	Myelin transcription factor 1	Homo sapiens		 20.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794678	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794678&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293623	528826141							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126295	CCCc1cc(Cl)cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C19H16Cl2N4O/c1-2-3-9-6-10(20)7-12-15(16(22)19(26)24-17(9)12)11-4-5-14(21)18-13(11)8-23-25-18/h4-8H,2-3,22H2,1H3,(H,23,25)(H,24,26)	XUWOEAARJAAZFI-UHFFFAOYSA-N	794679	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-8-propyl-1H-quinolin-2-one::US20260062412, Compound A22	Myelin transcription factor 1	Homo sapiens		 270							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794679	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794679&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293502	528826142							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126296	C=Cc1cc(Cl)cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C18H12Cl2N4O/c1-2-8-5-9(19)6-11-14(15(21)18(25)23-16(8)11)10-3-4-13(20)17-12(10)7-22-24-17/h2-7H,1,21H2,(H,22,24)(H,23,25)	OBOCTNPBEABGBT-UHFFFAOYSA-N	794680	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-8-ethenyl-1H-quinolin-2-one::US20260062412, Compound A23	Myelin transcription factor 1	Homo sapiens		 34.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794680	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794680&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293387	528826143							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126297	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Cl)cc(C3CC3)c2[nH]c1=O	InChI=1S/C19H14Cl2N4O/c20-9-5-11(8-1-2-8)17-12(6-9)15(16(22)19(26)24-17)10-3-4-14(21)18-13(10)7-23-25-18/h3-8H,1-2,22H2,(H,23,25)(H,24,26)	BBLSHLFKXWPZCS-UHFFFAOYSA-N	794681	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-8-cyclopropyl-1H-quinolin-2-one::US20260062412, Compound A24	Myelin transcription factor 1	Homo sapiens		 110							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794681	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794681&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293517	528826144							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126298	CCc1cc(Cl)cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C18H14Cl2N4O/c1-2-8-5-9(19)6-11-14(15(21)18(25)23-16(8)11)10-3-4-13(20)17-12(10)7-22-24-17/h3-7H,2,21H2,1H3,(H,22,24)(H,23,25)	XOKVETMICBJOKR-UHFFFAOYSA-N	794682	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-8-ethyl-1H-quinolin-2-one::US20260062412, Compound A25	Myelin transcription factor 1	Homo sapiens		 45.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794682	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794682&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293731	528826145							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126299	Cc1cc(Cl)cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C17H12Cl2N4O/c1-7-4-8(18)5-10-13(14(20)17(24)22-15(7)10)9-2-3-12(19)16-11(9)6-21-23-16/h2-6H,20H2,1H3,(H,21,23)(H,22,24)	KXOARNHKMWHQRX-UHFFFAOYSA-N	794683	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-8-methyl-1H-quinolin-2-one::US20260062412, Compound A26	Myelin transcription factor 1	Homo sapiens		 11.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794683	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794683&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293690	528826146							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126300	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Cl)c(Br)cc2[nH]c1=O	InChI=1S/C16H9BrCl2N4O/c17-9-4-12-7(3-11(9)19)13(14(20)16(24)22-12)6-1-2-10(18)15-8(6)5-21-23-15/h1-5H,20H2,(H,21,23)(H,22,24)	KTSKQHONYLQJGZ-UHFFFAOYSA-N	794684	3-Amino-7-bromo-6-chloro-4-(7-chloro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A27	Myelin transcription factor 1	Homo sapiens		 40.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794684	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794684&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293616	528826147							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126301	CCc1cc2[nH]c(=O)c(N)c(-c3ccc(Cl)c4[nH]ncc34)c2cc1Cl	InChI=1S/C18H14Cl2N4O/c1-2-8-5-14-10(6-13(8)20)15(16(21)18(25)23-14)9-3-4-12(19)17-11(9)7-22-24-17/h3-7H,2,21H2,1H3,(H,22,24)(H,23,25)	DRRLUOMJMCRUOJ-UHFFFAOYSA-N	794685	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-7-ethyl-1H-quinolin-2-one::US20260062412, Compound A28	Myelin transcription factor 1	Homo sapiens		 47.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794685	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794685&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293732	528826148							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126302	N#Cc1cc2[nH]c(=O)c(N)c(-c3ccc(Cl)c4[nH]ncc34)c2cc1Cl	InChI=1S/C17H9Cl2N5O/c18-11-2-1-8(10-6-22-24-16(10)11)14-9-4-12(19)7(5-20)3-13(9)23-17(25)15(14)21/h1-4,6H,21H2,(H,22,24)(H,23,25)	ONYARRBZMDMFDQ-UHFFFAOYSA-N	794686	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-2-oxo-1H-quinoline-7-carbonitrile::US20260062412, Compound A29	Myelin transcription factor 1	Homo sapiens		 29.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794686	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794686&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293464	528826149							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126303	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Cl)c(OC(F)F)cc2[nH]c1=O	InChI=1S/C17H10Cl2F2N4O2/c18-9-2-1-6(8-5-23-25-15(8)9)13-7-3-10(19)12(27-17(20)21)4-11(7)24-16(26)14(13)22/h1-5,17H,22H2,(H,23,25)(H,24,26)	YNIHNDYYBMUDRX-UHFFFAOYSA-N	794687	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-7-(difluoromethoxy)-1H-quinolin-2-one::US20260062412, Compound A30	Myelin transcription factor 1	Homo sapiens		 43.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794687	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794687&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293316	528826150							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126304	CC(=O)c1ccc2[nH]c(=O)c(N)c(-c3ccc(Cl)c4[nH]ncc34)c2c1	InChI=1S/C18H13ClN4O2/c1-8(24)9-2-5-14-11(6-9)15(16(20)18(25)22-14)10-3-4-13(19)17-12(10)7-21-23-17/h2-7H,20H2,1H3,(H,21,23)(H,22,25)	HLAGVFFVRHCMSM-UHFFFAOYSA-N	794688	6-Acetyl-3-amino-4-(7-chloro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A31	Myelin transcription factor 1	Homo sapiens		 7.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794688	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794688&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293346	528826151							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126305	CC(O)c1ccc2[nH]c(=O)c(N)c(-c3ccc(Cl)c4[nH]ncc34)c2c1	InChI=1S/C18H15ClN4O2/c1-8(24)9-2-5-14-11(6-9)15(16(20)18(25)22-14)10-3-4-13(19)17-12(10)7-21-23-17/h2-8,24H,20H2,1H3,(H,21,23)(H,22,25)	RNOWJBWJUNSCTJ-UHFFFAOYSA-N	794689	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-(1-hydroxyethyl)-1H-quinolin-2-one::US20260062412, Compound A32	Myelin transcription factor 1	Homo sapiens		 16.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794689	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794689&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293711	528826152							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126306	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C3CCNCC3)ccc2[nH]c1=O	InChI=1S/C21H20ClN5O/c22-16-3-2-13(15-10-25-27-20(15)16)18-14-9-12(11-5-7-24-8-6-11)1-4-17(14)26-21(28)19(18)23/h1-4,9-11,24H,5-8,23H2,(H,25,27)(H,26,28)	HIPHGESAVANUEL-UHFFFAOYSA-N	794690	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-piperidin-4-yl-1H-quinolin-2-one; 2,2,2-trifluoroacetate::US20260062412, Compound A33	Myelin transcription factor 1	Homo sapiens		 13.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794690	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794690&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293812	528826153							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126307	CC(C)N1CCC(c2ccc3[nH]c(=O)c(N)c(-c4ccc(F)c5[nH]ncc45)c3c2)CC1	InChI=1S/C24H26FN5O/c1-13(2)30-9-7-14(8-10-30)15-3-6-20-17(11-15)21(22(26)24(31)28-20)16-4-5-19(25)23-18(16)12-27-29-23/h3-6,11-14H,7-10,26H2,1-2H3,(H,27,29)(H,28,31)	AHIZPOOQGWJEGU-UHFFFAOYSA-N	794691	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-(1-propan-2-ylpiperidin-4-yl)-1H-quinolin-2-one::US20260062412, Compound A34	Myelin transcription factor 1	Homo sapiens		 26.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794691	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794691&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			178423163	528826154							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126308	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C3CCN(C4CCC4)CC3)ccc2[nH]c1=O	InChI=1S/C25H26ClN5O/c26-20-6-5-17(19-13-28-30-24(19)20)22-18-12-15(4-7-21(18)29-25(32)23(22)27)14-8-10-31(11-9-14)16-2-1-3-16/h4-7,12-14,16H,1-3,8-11,27H2,(H,28,30)(H,29,32)	IPLNEIDYDFNYHY-UHFFFAOYSA-N	794692	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-(1-cyclobutylpiperidin-4-yl)-1H-quinolin-2-one::US20260062412, Compound A35	Myelin transcription factor 1	Homo sapiens		 19.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794692	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794692&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293722	528826155							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126309	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C3CCN(C4COC4)CC3)ccc2[nH]c1=O	InChI=1S/C24H24ClN5O2/c25-19-3-2-16(18-10-27-29-23(18)19)21-17-9-14(1-4-20(17)28-24(31)22(21)26)13-5-7-30(8-6-13)15-11-32-12-15/h1-4,9-10,13,15H,5-8,11-12,26H2,(H,27,29)(H,28,31)	ABULMBQTBYAIEO-UHFFFAOYSA-N	794693	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-[1-(oxetane-3-yl) piperidin-4-yl]-1H-quinolin-2-one::US20260062412, Compound A36	Myelin transcription factor 1	Homo sapiens		 18.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794693	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794693&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293202	528826156							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126310	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C(=O)NC3CC3)ccc2[nH]c1=O	InChI=1S/C20H16ClN5O2/c21-14-5-4-11(13-8-23-26-18(13)14)16-12-7-9(19(27)24-10-2-3-10)1-6-15(12)25-20(28)17(16)22/h1,4-8,10H,2-3,22H2,(H,23,26)(H,24,27)(H,25,28)	WAAUGEQDOCTESA-UHFFFAOYSA-N	794694	3-Amino-4-(7-chloro-1H-indazol-4-yl)-N-cyclopropyl-2-oxo-1H-quinoline-6-carboxamide::US20260062412, Compound A37	Myelin transcription factor 1	Homo sapiens		 5.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794694	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794694&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293383	528826157							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126311	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C(=O)N3CCOCC3)ccc2[nH]c1=O	InChI=1S/C21H18ClN5O3/c22-15-3-2-12(14-10-24-26-19(14)15)17-13-9-11(21(29)27-5-7-30-8-6-27)1-4-16(13)25-20(28)18(17)23/h1-4,9-10H,5-8,23H2,(H,24,26)(H,25,28)	ANSWROWQBRFUJJ-UHFFFAOYSA-N	794695	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-(morpholine-4-carbonyl)-1H-quinolin-2-one::US20260062412, Compound A38	Myelin transcription factor 1	Homo sapiens		 20.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794695	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794695&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293857	528826158							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126312	CN1CC(c2ccc3[nH]c(=O)c(N)c(-c4ccc(Cl)c5[nH]ncc45)c3c2)C1	InChI=1S/C20H18ClN5O/c1-26-8-11(9-26)10-2-5-16-13(6-10)17(18(22)20(27)24-16)12-3-4-15(21)19-14(12)7-23-25-19/h2-7,11H,8-9,22H2,1H3,(H,23,25)(H,24,27)	JHNQKTXIFGGUEW-UHFFFAOYSA-N	794696	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-(1-methylazetidin-3-yl)-1H-quinolin-2-one::US20260062412, Compound A39	Myelin transcription factor 1	Homo sapiens		 23.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794696	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794696&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293179	528826159							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126313	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2ccc(Cl)cc2[nH]c1=O	InChI=1S/C16H10Cl2N4O/c17-7-1-2-9-12(5-7)21-16(23)14(19)13(9)8-3-4-11(18)15-10(8)6-20-22-15/h1-6H,19H2,(H,20,22)(H,21,23)	FKXWRVKBURLAJY-UHFFFAOYSA-N	794697	3-Amino-7-chloro-4-(7-chloro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A40	Myelin transcription factor 1	Homo sapiens		 8.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794697	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794697&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293239	528826160							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126314	Nc1c(-c2cccc(O)c2)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C15H11ClN2O2/c16-9-4-5-12-11(7-9)13(14(17)15(20)18-12)8-2-1-3-10(19)6-8/h1-7,19H,17H2,(H,18,20)	ZKBHGHWWUQGAFG-UHFFFAOYSA-N	50661014	CHEMBL6172134::US20260062412, Compound A41	Myelin transcription factor 1	Homo sapiens		 140							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=50661014	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=50661014&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293890	528507709							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126315	COc1cccc(-c2c(N)c(=O)[nH]c3ccc(Cl)cc23)c1	InChI=1S/C16H13ClN2O2/c1-21-11-4-2-3-9(7-11)14-12-8-10(17)5-6-13(12)19-16(20)15(14)18/h2-8H,18H2,1H3,(H,19,20)	DLBXWTNDJLLZKZ-UHFFFAOYSA-N	794699	3-Amino-6-chloro-4-(3-methoxyphenyl)-1H-quinolin-2-one::US20260062412, Compound A42	Myelin transcription factor 1	Homo sapiens		 450							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794699	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794699&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293628	528826162							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126316	Nc1c(-c2cccc3[nH]ncc23)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H11ClN4O/c17-8-4-5-12-10(6-8)14(15(18)16(22)20-12)9-2-1-3-13-11(9)7-19-21-13/h1-7H,18H2,(H,19,21)(H,20,22)	HYWIKRVIDIVJLY-UHFFFAOYSA-N	794700	3-Amino-6-chloro-4-(1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A43	Myelin transcription factor 1	Homo sapiens		 48.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794700	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794700&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293577	528826163							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126317	Nc1c(-c2ccncc2)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C14H10ClN3O/c15-9-1-2-11-10(7-9)12(13(16)14(19)18-11)8-3-5-17-6-4-8/h1-7H,16H2,(H,18,19)	ADDNTJDLYMXGHM-UHFFFAOYSA-N	794701	3-Amino-6-chloro-4-pyridin-4-yl-1H-quinolin-2-one::US20260062412, Compound A44	Myelin transcription factor 1	Homo sapiens		 5000							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794701	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794701&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293815	528826164							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126318	Nc1c(-c2cccnc2)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C14H10ClN3O/c15-9-3-4-11-10(6-9)12(13(16)14(19)18-11)8-2-1-5-17-7-8/h1-7H,16H2,(H,18,19)	OPTRZTVDXKFDKO-UHFFFAOYSA-N	794702	3-Amino-6-chloro-4-pyridin-3-yl-1H-quinolin-2-one::US20260062412, Compound A45	Myelin transcription factor 1	Homo sapiens		 5000							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794702	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794702&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293741	528826165							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126319	CS(=O)(=O)Nc1cccc(-c2c(N)c(=O)[nH]c3ccc(Cl)cc23)c1	InChI=1S/C16H14ClN3O3S/c1-24(22,23)20-11-4-2-3-9(7-11)14-12-8-10(17)5-6-13(12)19-16(21)15(14)18/h2-8,20H,18H2,1H3,(H,19,21)	VSKQJUXEEPZTEI-UHFFFAOYSA-N	794703	N-[3-(3-amino-6-chloro-2-oxo-1H-quinolin-4-yl)phenyl]methanesulfonamide::US20260062412, Compound A46	Myelin transcription factor 1	Homo sapiens		 5900							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794703	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794703&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293368	528826166							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126320	Nc1cc(-c2c(N)c(=O)[nH]c3ccc(Cl)cc23)ccn1	InChI=1S/C14H11ClN4O/c15-8-1-2-10-9(6-8)12(13(17)14(20)19-10)7-3-4-18-11(16)5-7/h1-6H,17H2,(H2,16,18)(H,19,20)	GKXJDUBCAUSSSK-UHFFFAOYSA-N	794704	3-Amino-4-(2-aminopyridin-4-yl)-6-chloro-1H-quinolin-2-one::US20260062412, Compound A47	Myelin transcription factor 1	Homo sapiens		 3300							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794704	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794704&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293804	528826167							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126321	Nc1c(-c2ccc3nc[nH]c3c2)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H11ClN4O/c17-9-2-4-11-10(6-9)14(15(18)16(22)21-11)8-1-3-12-13(5-8)20-7-19-12/h1-7H,18H2,(H,19,20)(H,21,22)	GKUIDTICVATVLA-UHFFFAOYSA-N	794705	3-Amino-4-(3H-benzimidazol-5-yl)-6-chloro-1H-quinolin-2-one::US20260062412, Compound A48	Myelin transcription factor 1	Homo sapiens		 5300							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794705	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794705&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293466	528826168							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126322	Nc1c(-c2ccc3cn[nH]c3c2)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H11ClN4O/c17-10-3-4-12-11(6-10)14(15(18)16(22)20-12)8-1-2-9-7-19-21-13(9)5-8/h1-7H,18H2,(H,19,21)(H,20,22)	XCGCFBKMXWDTCW-UHFFFAOYSA-N	794706	3-Amino-6-chloro-4-(1H-indazol-6-yl)-1H-quinolin-2-one::US20260062412, Compound A49	Myelin transcription factor 1	Homo sapiens		 790							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794706	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794706&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293925	528826169							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126323	Nc1c(-c2cccc(OC(F)F)c2)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H11ClF2N2O2/c17-9-4-5-12-11(7-9)13(14(20)15(22)21-12)8-2-1-3-10(6-8)23-16(18)19/h1-7,16H,20H2,(H,21,22)	QIDOCGFQUXUVQD-UHFFFAOYSA-N	794707	3-Amino-6-chloro-4-[3-(difluoromethoxy)phenyl]-1H-quinolin-2-one::US20260062412, Compound A50	Myelin transcription factor 1	Homo sapiens		 5800							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794707	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794707&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293624	528826170							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126324	Nc1c(-c2cccc(C(F)F)c2)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H11ClF2N2O/c17-10-4-5-12-11(7-10)13(14(20)16(22)21-12)8-2-1-3-9(6-8)15(18)19/h1-7,15H,20H2,(H,21,22)	QTUGGYSKPHSHSC-UHFFFAOYSA-N	794708	3-Amino-6-chloro-4-[3-(difluoromethyl)phenyl]-1H-quinolin-2-one::US20260062412, Compound A51	Myelin transcription factor 1	Homo sapiens		 2700							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794708	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794708&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293444	528826171							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126325	Cn1ccc(-c2c(N)c(=O)[nH]c3ccc(Cl)cc23)cc1=O	InChI=1S/C15H12ClN3O2/c1-19-5-4-8(6-12(19)20)13-10-7-9(16)2-3-11(10)18-15(21)14(13)17/h2-7H,17H2,1H3,(H,18,21)	RPYKHDHXAVGJGI-UHFFFAOYSA-N	794709	3-Amino-6-chloro-4-(1-methyl-2-oxopyridin-4-yl)-1H-quinolin-2-one::US20260062412, Compound A52	Myelin transcription factor 1	Homo sapiens		 4400							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794709	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794709&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293406	528826172							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126326	Nc1c(-c2cccc3[nH]ccc23)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C17H12ClN3O/c18-9-4-5-14-12(8-9)15(16(19)17(22)21-14)11-2-1-3-13-10(11)6-7-20-13/h1-8,20H,19H2,(H,21,22)	ACPWWFWJOXESPR-UHFFFAOYSA-N	794710	3-Amino-6-chloro-4-(1H-indol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A53	Myelin transcription factor 1	Homo sapiens		 980							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794710	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794710&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293314	528826173							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126327	Cc1cc(-c2c(N)c(=O)[nH]c3ccc(Cl)cc23)c2cn[nH]c2c1	InChI=1S/C17H13ClN4O/c1-8-4-10(12-7-20-22-14(12)5-8)15-11-6-9(18)2-3-13(11)21-17(23)16(15)19/h2-7H,19H2,1H3,(H,20,22)(H,21,23)	WWLBKTSDXVSZAY-UHFFFAOYSA-N	794711	3-Amino-6-chloro-4-(6-methyl-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A55	Myelin transcription factor 1	Homo sapiens		 480							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794711	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794711&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293358	528826174							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126328	Nc1c(-c2cc(F)cc3[nH]ncc23)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H10ClFN4O/c17-7-1-2-12-10(3-7)14(15(19)16(23)21-12)9-4-8(18)5-13-11(9)6-20-22-13/h1-6H,19H2,(H,20,22)(H,21,23)	CTYWKJSVQRBRSV-UHFFFAOYSA-N	794712	3-Amino-6-chloro-4-(6-fluoro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A56	Myelin transcription factor 1	Homo sapiens		 58.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794712	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794712&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293140	528826175							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126329	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H10ClFN4O/c17-7-1-4-12-9(5-7)13(14(19)16(23)21-12)8-2-3-11(18)15-10(8)6-20-22-15/h1-6H,19H2,(H,20,22)(H,21,23)	USGRRVXARARGEO-UHFFFAOYSA-N	794713	3-Amino-6-chloro-4-(7-fluoro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A57	Myelin transcription factor 1	Homo sapiens		 13.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794713	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794713&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293831	528826176							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126330	Nc1c(-c2cc(Cl)cc3[nH]ncc23)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H10Cl2N4O/c17-7-1-2-12-10(3-7)14(15(19)16(23)21-12)9-4-8(18)5-13-11(9)6-20-22-13/h1-6H,19H2,(H,20,22)(H,21,23)	IYYNPMMVJLJXPC-UHFFFAOYSA-N	794714	3-Amino-6-chloro-4-(6-chloro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A58	Myelin transcription factor 1	Homo sapiens		 360							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794714	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794714&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293791	528826177							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126331	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H10Cl2N4O/c17-7-1-4-12-9(5-7)13(14(19)16(23)21-12)8-2-3-11(18)15-10(8)6-20-22-15/h1-6H,19H2,(H,20,22)(H,21,23)	YXKVRHAAENFPKJ-UHFFFAOYSA-N	794715	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A59	Myelin transcription factor 1	Homo sapiens		 5.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794715	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794715&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293613	528826178							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126332	Cc1ccc(-c2c(N)c(=O)[nH]c3ccc(Cl)cc23)c2cn[nH]c12	InChI=1S/C17H13ClN4O/c1-8-2-4-10(12-7-20-22-16(8)12)14-11-6-9(18)3-5-13(11)21-17(23)15(14)19/h2-7H,19H2,1H3,(H,20,22)(H,21,23)	RQHRSWSSLBGBBW-UHFFFAOYSA-N	794716	3-Amino-6-chloro-4-(7-methyl-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A60	Myelin transcription factor 1	Homo sapiens		 7.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794716	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794716&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293475	528826179							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126333	Nc1c(-c2ccc(C(F)(F)F)c3[nH]ncc23)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C17H10ClF3N4O/c18-7-1-4-12-9(5-7)13(14(22)16(26)24-12)8-2-3-11(17(19,20)21)15-10(8)6-23-25-15/h1-6H,22H2,(H,23,25)(H,24,26)	NMVHRSCBOHNZMV-UHFFFAOYSA-N	794717	3-Amino-6-chloro-4-[7-(trifluoromethyl)-1H-indazol-4-yl]-1H-quinolin-2-one::US20260062412, Compound A61	Myelin transcription factor 1	Homo sapiens		 140							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794717	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794717&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293441	528826180							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126334	Cc1n[nH]c2cccc(-c3c(N)c(=O)[nH]c4ccc(Cl)cc34)c12	InChI=1S/C17H13ClN4O/c1-8-14-10(3-2-4-13(14)22-21-8)15-11-7-9(18)5-6-12(11)20-17(23)16(15)19/h2-7H,19H2,1H3,(H,20,23)(H,21,22)	SJYJIYWAVYWXIC-UHFFFAOYSA-N	794718	3-Amino-6-chloro-4-(3-methyl-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A62	Myelin transcription factor 1	Homo sapiens		 3900							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794718	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794718&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293289	528826181							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126335	Cc1ccc2[nH]ncc2c1-c1c(N)c(=O)[nH]c2ccc(Cl)cc12	InChI=1S/C17H13ClN4O/c1-8-2-4-13-11(7-20-22-13)14(8)15-10-6-9(18)3-5-12(10)21-17(23)16(15)19/h2-7H,19H2,1H3,(H,20,22)(H,21,23)	BJHKLGXLFGHAHN-UHFFFAOYSA-N	794719	3-Amino-6-chloro-4-(5-methyl-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A63	Myelin transcription factor 1	Homo sapiens		 710							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794719	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794719&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293761	528826182							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126336	Nc1c(-c2cccc(O)c2)c2cc(C3CC3)ccc2[nH]c1=O	InChI=1S/C18H16N2O2/c19-17-16(12-2-1-3-13(21)8-12)14-9-11(10-4-5-10)6-7-15(14)20-18(17)22/h1-3,6-10,21H,4-5,19H2,(H,20,22)	UNPIOEPLUVZGLL-UHFFFAOYSA-N	794720	3-Amino-6-cyclopropyl-4-(3-hydroxyphenyl)-1H-quinolin-2-one::US20260062412, Compound A65	Myelin transcription factor 1	Homo sapiens		 190							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794720	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794720&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293213	528826183							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126337	Nc1c(-c2cccc(O)c2)c2ccccc2[nH]c1=O	InChI=1S/C15H12N2O2/c16-14-13(9-4-3-5-10(18)8-9)11-6-1-2-7-12(11)17-15(14)19/h1-8,18H,16H2,(H,17,19)	BDJDIWNSWGMJJC-UHFFFAOYSA-N	794721	3-Amino-4-(3-hydroxyphenyl)-1H-quinolin-2-one::US20260062412, Compound A66	Myelin transcription factor 1	Homo sapiens		 380							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794721	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794721&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293892	528826184							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126338	Nc1c(-c2c(F)ccc3[nH]ncc23)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H10ClFN4O/c17-7-1-3-11-8(5-7)14(15(19)16(23)21-11)13-9-6-20-22-12(9)4-2-10(13)18/h1-6H,19H2,(H,20,22)(H,21,23)	ZCPMXVGZCWOWBD-UHFFFAOYSA-N	794722	3-Amino-6-chloro-4-(5-fluoro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A67	Myelin transcription factor 1	Homo sapiens		 130							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794722	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794722&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293381	528826185							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126339	Nc1c(-c2cc[nH]c(=O)c2)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C14H10ClN3O2/c15-8-1-2-10-9(6-8)12(13(16)14(20)18-10)7-3-4-17-11(19)5-7/h1-6H,16H2,(H,17,19)(H,18,20)	AMYLIWWYXWYHCF-UHFFFAOYSA-N	794723	3-Amino-6-chloro-4-(2-oxo-1H-pyridin-4-yl)-1H-quinolin-2-one::US20260062412, Compound A68	Myelin transcription factor 1	Homo sapiens		 8000							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794723	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794723&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293505	528826186							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126340	Nc1nccc(-c2c(N)c(=O)[nH]c3ccc(Cl)cc23)n1	InChI=1S/C13H10ClN5O/c14-6-1-2-8-7(5-6)10(11(15)12(20)18-8)9-3-4-17-13(16)19-9/h1-5H,15H2,(H,18,20)(H2,16,17,19)	MVKZLZYHXCWMOJ-UHFFFAOYSA-N	794724	3-Amino-4-(2-aminopyrimidin-4-yl)-6-chloro-1H-quinolin-2-one::US20260062412, Compound A69	Myelin transcription factor 1	Homo sapiens		 2500							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794724	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794724&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293200	528826187							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126341	Nc1c(-c2ccccc2)c2ccccc2[nH]c1=O	InChI=1S/C15H12N2O/c16-14-13(10-6-2-1-3-7-10)11-8-4-5-9-12(11)17-15(14)18/h1-9H,16H2,(H,17,18)	ZUYDHEBASIFXCJ-UHFFFAOYSA-N	794725	3-Amino-4-phenyl-1H-quinolin-2-one::US20260062412, Compound A70	Myelin transcription factor 1	Homo sapiens		 6200							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794725	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794725&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			12695718	528826188							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126342	Nc1c(N2CCCC(CO)C2)c2cc(Br)ccc2[nH]c1=O	InChI=1S/C15H18BrN3O2/c16-10-3-4-12-11(6-10)14(13(17)15(21)18-12)19-5-1-2-9(7-19)8-20/h3-4,6,9,20H,1-2,5,7-8,17H2,(H,18,21)	ROXSIWLDULTSLA-UHFFFAOYSA-N	794726	3-Amino-6-bromo-4-[3-(hydroxymethyl) piperidin-1-yl]-1H-quinolin-2-one 2,2,2-trifluoroacetate::US20260062412, Compound A71	Myelin transcription factor 1	Homo sapiens		 1400							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794726	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794726&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293377	528826189							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126343	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(OCC3(F)CC3)c(F)cc2[nH]c1=O	InChI=1S/C20H15ClF2N4O2/c21-12-2-1-9(11-7-25-27-18(11)12)16-10-5-15(29-8-20(23)3-4-20)13(22)6-14(10)26-19(28)17(16)24/h1-2,5-7H,3-4,8,24H2,(H,25,27)(H,26,28)	ATHGTEFXOWAQDG-UHFFFAOYSA-N	794727	3-Amino-4-(7-chloro-1H-indazol-4-yl)-7-fluoro-6-[(1-fluorocyclopropyl)methoxy]-1H-quinolin-2-one::US20260062412, Compound A72	Myelin transcription factor 1	Homo sapiens		 96.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794727	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794727&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293329	528826190							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126344	COc1cccc(-c2c(N)c(=O)[nH]c3c2ccc2ccccc23)c1	InChI=1S/C20H16N2O2/c1-24-14-7-4-6-13(11-14)17-16-10-9-12-5-2-3-8-15(12)19(16)22-20(23)18(17)21/h2-11H,21H2,1H3,(H,22,23)	DMXIVHDUUSCSDJ-UHFFFAOYSA-N	794728	3-Amino-4-(3-methoxyphenyl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B1	Myelin transcription factor 1	Homo sapiens		 5600							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794728	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794728&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293597	528826191							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126345	Nc1c(-c2cccc(O)c2)c2ccc3ccccc3c2[nH]c1=O	InChI=1S/C19H14N2O2/c20-17-16(12-5-3-6-13(22)10-12)15-9-8-11-4-1-2-7-14(11)18(15)21-19(17)23/h1-10,22H,20H2,(H,21,23)	MBPNONCSDWAHCA-UHFFFAOYSA-N	794729	3-Amino-4-(3-hydroxyphenyl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B2	Myelin transcription factor 1	Homo sapiens		 22.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794729	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794729&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293937	528826192							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126346	Nc1c(-c2cccc(O)c2)c2cc(C3CC3)c3ccccc3c2[nH]c1=O	InChI=1S/C22H18N2O2/c23-20-19(13-4-3-5-14(25)10-13)18-11-17(12-8-9-12)15-6-1-2-7-16(15)21(18)24-22(20)26/h1-7,10-12,25H,8-9,23H2,(H,24,26)	BPJSTDLWYAENHZ-UHFFFAOYSA-N	794730	3-Amino-6-cyclopropyl-4-(3-hydroxyphenyl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B3	Myelin transcription factor 1	Homo sapiens		 7.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794730	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794730&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293234	528826193							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126347	Nc1c(-c2cccc(O)c2)c2cc(Br)c3ccccc3c2[nH]c1=O	InChI=1S/C19H13BrN2O2/c20-15-9-14-16(10-4-3-5-11(23)8-10)17(21)19(24)22-18(14)13-7-2-1-6-12(13)15/h1-9,23H,21H2,(H,22,24)	HEFQXQLNGUCOIB-UHFFFAOYSA-N	794731	3-Amino-6-bromo-4-(3-hydroxyphenyl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B4	Myelin transcription factor 1	Homo sapiens		 27.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794731	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794731&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293834	528826194							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126348	Nc1c(-c2cccc(O)c2)c2cc(-c3ccccc3)c3ccccc3c2[nH]c1=O	InChI=1S/C25H18N2O2/c26-23-22(16-9-6-10-17(28)13-16)21-14-20(15-7-2-1-3-8-15)18-11-4-5-12-19(18)24(21)27-25(23)29/h1-14,28H,26H2,(H,27,29)	XRKGNVJYXCCGBH-UHFFFAOYSA-N	794732	3-Amino-4-(3-hydroxyphenyl)-6-phenyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B5	Myelin transcription factor 1	Homo sapiens		 420							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794732	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794732&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293227	528826195							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126349	Cc1cc2c(-c3cccc(O)c3)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C20H16N2O2/c1-11-9-16-17(12-5-4-6-13(23)10-12)18(21)20(24)22-19(16)15-8-3-2-7-14(11)15/h2-10,23H,21H2,1H3,(H,22,24)	IKNTVXJLTFMMOI-UHFFFAOYSA-N	794733	3-Amino-4-(3-hydroxyphenyl)-6-methyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B6	Myelin transcription factor 1	Homo sapiens		 7.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794733	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794733&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293637	528826196							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126350	N#Cc1cc2c(-c3cccc(O)c3)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C20H13N3O2/c21-10-12-9-16-17(11-4-3-5-13(24)8-11)18(22)20(25)23-19(16)15-7-2-1-6-14(12)15/h1-9,24H,22H2,(H,23,25)	YHYNXXIZLMHJKC-UHFFFAOYSA-N	794734	3-Amino-4-(3-hydroxyphenyl)-2-oxo-1H-benzo[h]quinoline-6-carbonitrile::US20260062412, Compound B7	Myelin transcription factor 1	Homo sapiens		 6.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794734	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794734&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293881	528826197							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126351	Nc1c(-c2cccc(O)c2)c2cc(Cl)c3ccccc3c2[nH]c1=O	InChI=1S/C19H13ClN2O2/c20-15-9-14-16(10-4-3-5-11(23)8-10)17(21)19(24)22-18(14)13-7-2-1-6-12(13)15/h1-9,23H,21H2,(H,22,24)	PZVOEQDOQOELME-UHFFFAOYSA-N	794735	3-Amino-6-chloro-4-(3-hydroxyphenyl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B8	Myelin transcription factor 1	Homo sapiens		 12.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794735	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794735&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293640	528826198							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126352	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(I)c3ccc(Cl)cc3c2[nH]c1=O	InChI=1S/C20H11ClFIN4O/c21-8-1-2-9-11(5-8)18-12(6-15(9)23)16(17(24)20(28)26-18)10-3-4-14(22)19-13(10)7-25-27-19/h1-7H,24H2,(H,25,27)(H,26,28)	GWRDNRPFHIYUFT-UHFFFAOYSA-N	794736	3-Amino-9-chloro-4-(7-fluoro-1H-indazol-4-yl)-6-iodo-1H-benzo[h]quinolin-2-one::US20260062412, Compound B9	Myelin transcription factor 1	Homo sapiens		 120							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794736	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794736&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293868	528826199							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126353	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3ccc(Cl)cc3c2[nH]c1=O	InChI=1S/C23H16ClFN4O/c24-11-3-4-12-14(10-1-2-10)8-16-19(20(26)23(30)28-21(16)15(12)7-11)13-5-6-18(25)22-17(13)9-27-29-22/h3-10H,1-2,26H2,(H,27,29)(H,28,30)	BLTYYROZTSQECN-UHFFFAOYSA-N	794737	3-Amino-9-chloro-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B10	Myelin transcription factor 1	Homo sapiens		 36.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794737	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794737&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293867	528826200							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126354	Nc1c(-c2ccc(F)c3[nH]ncc23)c2ccc3ccc(Cl)cc3c2[nH]c1=O	InChI=1S/C20H12ClFN4O/c21-10-3-1-9-2-4-12-16(17(23)20(27)25-18(12)13(9)7-10)11-5-6-15(22)19-14(11)8-24-26-19/h1-8H,23H2,(H,24,26)(H,25,27)	TUDBWPYFRLPOJG-UHFFFAOYSA-N	794738	3-Amino-9-chloro-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B11	Myelin transcription factor 1	Homo sapiens		 30.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794738	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794738&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293352	528826201							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126355	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cc(Cl)ccc12	InChI=1S/C21H14ClFN4O/c1-9-6-14-17(12-4-5-16(23)20-15(12)8-25-27-20)18(24)21(28)26-19(14)13-7-10(22)2-3-11(9)13/h2-8H,24H2,1H3,(H,25,27)(H,26,28)	RWSRKPTZPCZTHQ-UHFFFAOYSA-N	794739	3-Amino-9-chloro-4-(7-fluoro-1H-indazol-4-yl)-6-methyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B12	Myelin transcription factor 1	Homo sapiens		 20.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794739	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794739&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293437	528826202							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126356	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(I)c3cc(Cl)ccc3c2[nH]c1=O	InChI=1S/C20H11ClFIN4O/c21-8-1-2-10-11(5-8)15(23)6-12-16(17(24)20(28)26-18(10)12)9-3-4-14(22)19-13(9)7-25-27-19/h1-7H,24H2,(H,25,27)(H,26,28)	UPIBGDIVWFFWRV-UHFFFAOYSA-N	794740	3-Amino-8-chloro-4-(7-fluoro-1H-indazol-4-yl)-6-iodo-1H-benzo[h]quinolin-2-one::US20260062412, Compound B13	Myelin transcription factor 1	Homo sapiens		 85.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794740	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794740&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293742	528826203							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126357	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3cc(Cl)ccc3c2[nH]c1=O	InChI=1S/C23H16ClFN4O/c24-11-3-4-13-15(7-11)14(10-1-2-10)8-16-19(20(26)23(30)28-21(13)16)12-5-6-18(25)22-17(12)9-27-29-22/h3-10H,1-2,26H2,(H,27,29)(H,28,30)	NRQRQRIARKMWPA-UHFFFAOYSA-N	794741	3-Amino-8-chloro-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B14	Myelin transcription factor 1	Homo sapiens		 18.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794741	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794741&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293223	528826204							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126358	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccc(Cl)cc12	InChI=1S/C21H14ClFN4O/c1-9-6-14-17(11-4-5-16(23)20-15(11)8-25-27-20)18(24)21(28)26-19(14)12-3-2-10(22)7-13(9)12/h2-8H,24H2,1H3,(H,25,27)(H,26,28)	FVALLGOHMFNFNL-UHFFFAOYSA-N	794742	3-Amino-8-chloro-4-(7-fluoro-1H-indazol-4-yl)-6-methyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B15	Myelin transcription factor 1	Homo sapiens		 8.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794742	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794742&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293281	528826205							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126359	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3c(Cl)cccc3c2[nH]c1=O	InChI=1S/C20H11BrClFN4O/c21-12-6-10-15(8-4-5-14(23)19-11(8)7-25-27-19)17(24)20(28)26-18(10)9-2-1-3-13(22)16(9)12/h1-7H,24H2,(H,25,27)(H,26,28)	PSECXWFYFDGNKV-UHFFFAOYSA-N	794743	3-Amino-6-bromo-7-chloro-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B16	Myelin transcription factor 1	Homo sapiens		 46.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794743	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794743&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293843	528826206							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126360	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3c(Cl)cccc3c2[nH]c1=O	InChI=1S/C23H16ClFN4O/c24-16-3-1-2-12-18(16)13(10-4-5-10)8-14-19(20(26)23(30)28-21(12)14)11-6-7-17(25)22-15(11)9-27-29-22/h1-3,6-10H,4-5,26H2,(H,27,29)(H,28,30)	QAMPSUXFZGGTKI-UHFFFAOYSA-N	794744	3-Amino-7-chloro-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B17	Myelin transcription factor 1	Homo sapiens		 15.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794744	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794744&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293902	528826207							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126361	Nc1c(-c2ccc(F)c3[nH]ncc23)c2ccc3c(Cl)cccc3c2[nH]c1=O	InChI=1S/C20H12ClFN4O/c21-14-3-1-2-11-9(14)4-5-12-16(17(23)20(27)25-18(11)12)10-6-7-15(22)19-13(10)8-24-26-19/h1-8H,23H2,(H,24,26)(H,25,27)	MJBBJYILIVPZHU-UHFFFAOYSA-N	794745	3-Amino-7-chloro-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B18	Myelin transcription factor 1	Homo sapiens		 23.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794745	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794745&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293194	528826208							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126362	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccc(Cl)c12	InChI=1S/C21H14ClFN4O/c1-9-7-12-17(10-5-6-15(23)20-13(10)8-25-27-20)18(24)21(28)26-19(12)11-3-2-4-14(22)16(9)11/h2-8H,24H2,1H3,(H,25,27)(H,26,28)	PAYBMNLPDFPPKD-UHFFFAOYSA-N	794746	3-Amino-7-chloro-4-(7-fluoro-1H-indazol-4-yl)-6-methyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B19	Myelin transcription factor 1	Homo sapiens		 22.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794746	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794746&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293167	528826209							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126363	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3cccc(Cl)c3c2[nH]c1=O	InChI=1S/C23H16ClFN4O/c24-16-3-1-2-11-13(10-4-5-10)8-14-18(20(26)23(30)28-22(14)19(11)16)12-6-7-17(25)21-15(12)9-27-29-21/h1-3,6-10H,4-5,26H2,(H,27,29)(H,28,30)	BCYAWWNFOALVNN-UHFFFAOYSA-N	794747	3-Amino-10-chloro-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B20	Myelin transcription factor 1	Homo sapiens		 42.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794747	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794747&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293413	528826210							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126364	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3ccccc3c2[nH]c1=O	InChI=1S/C20H12BrFN4O/c21-14-7-12-16(10-5-6-15(22)19-13(10)8-24-26-19)17(23)20(27)25-18(12)11-4-2-1-3-9(11)14/h1-8H,23H2,(H,24,26)(H,25,27)	WRVOFHPLHSUTDF-UHFFFAOYSA-N	794748	3-Amino-6-bromo-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B21	Myelin transcription factor 1	Homo sapiens		 20.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794748	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794748&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293550	528826211							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126365	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3ccccc3c2[nH]c1=O	InChI=1S/C23H17FN4O/c24-18-8-7-13(17-10-26-28-22(17)18)19-16-9-15(11-5-6-11)12-3-1-2-4-14(12)21(16)27-23(29)20(19)25/h1-4,7-11H,5-6,25H2,(H,26,28)(H,27,29)	ZMVUHEXIDZMTQF-UHFFFAOYSA-N	794749	3-Amino-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B22	Myelin transcription factor 1	Homo sapiens		 11.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794749	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794749&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293622	528826212							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126366	CCc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C22H17FN4O/c1-2-11-9-15-18(13-7-8-17(23)21-16(13)10-25-27-21)19(24)22(28)26-20(15)14-6-4-3-5-12(11)14/h3-10H,2,24H2,1H3,(H,25,27)(H,26,28)	WXFGCKNRGPCFQC-UHFFFAOYSA-N	794750	3-Amino-6-ethyl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B23	Myelin transcription factor 1	Homo sapiens		 8.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794750	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794750&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293398	528826213							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126367	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCC3)c3ccccc3c2[nH]c1=O	InChI=1S/C24H19FN4O/c25-19-9-8-14(18-11-27-29-23(18)19)20-17-10-16(12-4-3-5-12)13-6-1-2-7-15(13)22(17)28-24(30)21(20)26/h1-2,6-12H,3-5,26H2,(H,27,29)(H,28,30)	WSIHCUQKGHWPIW-UHFFFAOYSA-N	794751	3-Amino-6-cyclobutyl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B24	Myelin transcription factor 1	Homo sapiens		 16.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794751	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794751&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293214	528826214							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126368	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCCC3)c3ccccc3c2[nH]c1=O	InChI=1S/C25H21FN4O/c26-20-10-9-15(19-12-28-30-24(19)20)21-18-11-17(13-5-1-2-6-13)14-7-3-4-8-16(14)23(18)29-25(31)22(21)27/h3-4,7-13H,1-2,5-6,27H2,(H,28,30)(H,29,31)	XYWFJMZNMSUPII-UHFFFAOYSA-N	794752	3-Amino-6-cyclopentyl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B25	Myelin transcription factor 1	Homo sapiens		 24.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794752	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794752&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293923	528826215							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126369	N#Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C21H12FN5O/c22-16-6-5-12(15-9-25-27-20(15)16)17-14-7-10(8-23)11-3-1-2-4-13(11)19(14)26-21(28)18(17)24/h1-7,9H,24H2,(H,25,27)(H,26,28)	YUBIURDSEFTDEV-UHFFFAOYSA-N	794753	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-benzo[h]quinoline-6-carbonitrile::US20260062412, Compound B26	Myelin transcription factor 1	Homo sapiens		 10.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794753	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794753&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293500	528826216							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126370	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C21H15FN4O/c1-10-8-14-17(12-6-7-16(22)20-15(12)9-24-26-20)18(23)21(27)25-19(14)13-5-3-2-4-11(10)13/h2-9H,23H2,1H3,(H,24,26)(H,25,27)	QMANJWPRNPRPCY-UHFFFAOYSA-N	794754	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-methyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B27	Myelin transcription factor 1	Homo sapiens		 7.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794754	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794754&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293854	528826217							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126371	CC#Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C23H15FN4O/c1-2-5-12-10-16-19(14-8-9-18(24)22-17(14)11-26-28-22)20(25)23(29)27-21(16)15-7-4-3-6-13(12)15/h3-4,6-11H,25H2,1H3,(H,26,28)(H,27,29)	PEUUKALECFUQKT-UHFFFAOYSA-N	794755	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-prop-1-inyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B28	Myelin transcription factor 1	Homo sapiens		 22.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794755	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794755&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293510	528826218							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126372	Cn1cc(-c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3ccccc23)cn1	InChI=1S/C24H17FN6O/c1-31-11-12(9-28-31)16-8-17-20(14-6-7-19(25)23-18(14)10-27-30-23)21(26)24(32)29-22(17)15-5-3-2-4-13(15)16/h2-11H,26H2,1H3,(H,27,30)(H,29,32)	FJUGQUHIYZLINF-UHFFFAOYSA-N	794756	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-methylpyrazole-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B29	Myelin transcription factor 1	Homo sapiens		 9.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794756	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794756&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293927	528826219							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126373	C=Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C22H15FN4O/c1-2-11-9-15-18(13-7-8-17(23)21-16(13)10-25-27-21)19(24)22(28)26-20(15)14-6-4-3-5-12(11)14/h2-10H,1,24H2,(H,25,27)(H,26,28)	ZIRNZJULOYMAPU-UHFFFAOYSA-N	794757	3-Amino-6-ethenyl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B30	Myelin transcription factor 1	Homo sapiens		 15.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794757	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794757&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293395	528826220							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126374	CP(C)(=O)c1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C22H18FN4O2P/c1-30(2,29)17-9-14-18(12-7-8-16(23)21-15(12)10-25-27-21)19(24)22(28)26-20(14)13-6-4-3-5-11(13)17/h3-10H,24H2,1-2H3,(H,25,27)(H,26,28)	KATJVJFDXQPFPI-UHFFFAOYSA-N	794758	3-Amino-6-dimethylphosphoryl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B31	Myelin transcription factor 1	Homo sapiens		 19.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794758	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794758&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293657	528826221							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126375	Nc1c(-c2ccc(F)c3[nH]ncc23)c2ccc3ccccc3c2[nH]c1=O	InChI=1S/C20H13FN4O/c21-15-8-7-12(14-9-23-25-19(14)15)16-13-6-5-10-3-1-2-4-11(10)18(13)24-20(26)17(16)22/h1-9H,22H2,(H,23,25)(H,24,26)	AFCDRYCMAJNTBS-UHFFFAOYSA-N	794759	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B32	Myelin transcription factor 1	Homo sapiens		 3.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794759	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794759&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293220	528826222							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126376	Cn1c(=O)c(N)c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3ccccc3c21	InChI=1S/C21H14BrFN4O/c1-27-20-12-5-3-2-4-10(12)15(22)8-13(20)17(18(24)21(27)28)11-6-7-16(23)19-14(11)9-25-26-19/h2-9H,24H2,1H3,(H,25,26)	AIAKHXPRMNRGQB-UHFFFAOYSA-N	794760	3-Amino-6-bromo-4-(7-fluoro-1H-indazol-4-yl)-1-methylbenzo[h]quinolin-2-one::US20260062412, Compound B33	Myelin transcription factor 1	Homo sapiens		 2600							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794760	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794760&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293284	528826223							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126377	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Cl)c3ccccc3c2[nH]c1=O	InChI=1S/C20H12ClFN4O/c21-14-7-12-16(10-5-6-15(22)19-13(10)8-24-26-19)17(23)20(27)25-18(12)11-4-2-1-3-9(11)14/h1-8H,23H2,(H,24,26)(H,25,27)	LZYBABQGXSNVHJ-UHFFFAOYSA-N	794761	3-Amino-6-chloro-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B34	Myelin transcription factor 1	Homo sapiens		 33.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794761	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794761&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293813	528826224							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126378	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(F)c3ccccc3c2[nH]c1=O	InChI=1S/C20H12F2N4O/c21-14-6-5-10(13-8-24-26-19(13)14)16-12-7-15(22)9-3-1-2-4-11(9)18(12)25-20(27)17(16)23/h1-8H,23H2,(H,24,26)(H,25,27)	JNZVVFYRJTWAJV-UHFFFAOYSA-N	794762	3-Amino-6-fluoro-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B35	Myelin transcription factor 1	Homo sapiens		 3.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794762	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794762&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293568	528826225							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126379	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Br)c3ccccc3c2[nH]c1=O	InChI=1S/C20H12BrClN4O/c21-14-7-12-16(10-5-6-15(22)19-13(10)8-24-26-19)17(23)20(27)25-18(12)11-4-2-1-3-9(11)14/h1-8H,23H2,(H,24,26)(H,25,27)	QECQFPQAPVMWGS-UHFFFAOYSA-N	794763	3-Amino-6-bromo-4-(7-chloro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B36	Myelin transcription factor 1	Homo sapiens		 14.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794763	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794763&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293309	528826226							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126380	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C3CC3)c3ccccc3c2[nH]c1=O	InChI=1S/C23H17ClN4O/c24-18-8-7-13(17-10-26-28-22(17)18)19-16-9-15(11-5-6-11)12-3-1-2-4-14(12)21(16)27-23(29)20(19)25/h1-4,7-11H,5-6,25H2,(H,26,28)(H,27,29)	NKEOCOBPKVNCLZ-UHFFFAOYSA-N	794764	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-cyclopropyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B37	Myelin transcription factor 1	Homo sapiens		 6.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794764	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794764&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293443	528826227							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126381	CCc1cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C22H17ClN4O/c1-2-11-9-15-18(13-7-8-17(23)21-16(13)10-25-27-21)19(24)22(28)26-20(15)14-6-4-3-5-12(11)14/h3-10H,2,24H2,1H3,(H,25,27)(H,26,28)	AFVUQUFXEMUZMX-UHFFFAOYSA-N	794765	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-ethyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B38	Myelin transcription factor 1	Homo sapiens		 4.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794765	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794765&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293196	528826228							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126382	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C3CCC3)c3ccccc3c2[nH]c1=O	InChI=1S/C24H19ClN4O/c25-19-9-8-14(18-11-27-29-23(18)19)20-17-10-16(12-4-3-5-12)13-6-1-2-7-15(13)22(17)28-24(30)21(20)26/h1-2,6-12H,3-5,26H2,(H,27,29)(H,28,30)	YSXPMKJIPMRUHE-UHFFFAOYSA-N	794766	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-cyclobutyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B39	Myelin transcription factor 1	Homo sapiens		 10.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794766	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794766&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293906	528826229							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126383	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C3CCCC3)c3ccccc3c2[nH]c1=O	InChI=1S/C25H21ClN4O/c26-20-10-9-15(19-12-28-30-24(19)20)21-18-11-17(13-5-1-2-6-13)14-7-3-4-8-16(14)23(18)29-25(31)22(21)27/h3-4,7-13H,1-2,5-6,27H2,(H,28,30)(H,29,31)	MCRVDXNEEYHGCF-UHFFFAOYSA-N	794767	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-cyclopentyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B40	Myelin transcription factor 1	Homo sapiens		 13.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794767	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794767&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293463	528826230							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126384	N#Cc1cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C21H12ClN5O/c22-16-6-5-12(15-9-25-27-20(15)16)17-14-7-10(8-23)11-3-1-2-4-13(11)19(14)26-21(28)18(17)24/h1-7,9H,24H2,(H,25,27)(H,26,28)	VYNUQDHLXJKRKY-UHFFFAOYSA-N	794768	3-Amino-4-(7-chloro-1H-indazol-4-yl)-2-oxo-1H-benzo[h]quinoline-6-carbonitrile::US20260062412, Compound B41	Myelin transcription factor 1	Homo sapiens		 14.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794768	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794768&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293758	528826231							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126385	N#Cc1cc2c(-c3ccc(C#N)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C22H12N6O/c23-8-11-5-6-14(17-10-26-28-20(11)17)18-16-7-12(9-24)13-3-1-2-4-15(13)21(16)27-22(29)19(18)25/h1-7,10H,25H2,(H,26,28)(H,27,29)	QGSQBJPWQLEMDO-UHFFFAOYSA-N	794769	3-Amino-4-(7-cyano-1H-indazol-4-yl)-2-oxo-1H-benzo[h]quinoline-6-carbonitrile::US20260062412, Compound B42	Myelin transcription factor 1	Homo sapiens		 250							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794769	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794769&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293634	528826232							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126386	Cc1cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C21H15ClN4O/c1-10-8-14-17(12-6-7-16(22)20-15(12)9-24-26-20)18(23)21(27)25-19(14)13-5-3-2-4-11(10)13/h2-9H,23H2,1H3,(H,24,26)(H,25,27)	SUBLJJQFHUTFTN-UHFFFAOYSA-N	794770	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-methyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B43	Myelin transcription factor 1	Homo sapiens		 15.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794770	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794770&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293553	528826233							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126387	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2ccc3ccccc3c2[nH]c1=O	InChI=1S/C20H13ClN4O/c21-15-8-7-12(14-9-23-25-19(14)15)16-13-6-5-10-3-1-2-4-11(10)18(13)24-20(26)17(16)22/h1-9H,22H2,(H,23,25)(H,24,26)	GMVHBDIILDFWNG-UHFFFAOYSA-N	794771	3-Amino-4-(7-chloro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B44	Myelin transcription factor 1	Homo sapiens		 14.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794771	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794771&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293859	528826234							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126388	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Cl)c3ccccc3c2[nH]c1=O	InChI=1S/C20H12Cl2N4O/c21-14-6-5-10(13-8-24-26-19(13)14)16-12-7-15(22)9-3-1-2-4-11(9)18(12)25-20(27)17(16)23/h1-8H,23H2,(H,24,26)(H,25,27)	RHZNNIQPOYXLNA-UHFFFAOYSA-N	794772	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B45	Myelin transcription factor 1	Homo sapiens		 33.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794772	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794772&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293567	528826235							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126389	Nc1c(-c2cccc3[nH]ncc23)c2ccc3ccccc3c2[nH]c1=O	InChI=1S/C20H14N4O/c21-18-17(13-6-3-7-16-15(13)10-22-24-16)14-9-8-11-4-1-2-5-12(11)19(14)23-20(18)25/h1-10H,21H2,(H,22,24)(H,23,25)	QMDOHABESUHWFL-UHFFFAOYSA-N	794773	3-Amino-4-(1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B46	Myelin transcription factor 1	Homo sapiens		 6.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794773	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794773&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293254	528826236							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126390	Nc1c(-c2cccc3[nH]ncc23)c2cc(C3CC3)c3ccc(F)cc3c2[nH]c1=O	InChI=1S/C23H17FN4O/c24-12-6-7-13-15(11-4-5-11)9-17-20(14-2-1-3-19-18(14)10-26-28-19)21(25)23(29)27-22(17)16(13)8-12/h1-3,6-11H,4-5,25H2,(H,26,28)(H,27,29)	MJDLGQBGEZVCMO-UHFFFAOYSA-N	794774	3-Amino-6-cyclopropyl-9-fluoro-4-(1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B47	Myelin transcription factor 1	Homo sapiens		 10.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794774	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794774&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293334	528826237							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126391	Nc1c(-c2cccc3[nH]ncc23)c2cc(C3CC3)c3cc(F)ccc3c2[nH]c1=O	InChI=1S/C23H17FN4O/c24-12-6-7-14-16(8-12)15(11-4-5-11)9-17-20(21(25)23(29)27-22(14)17)13-2-1-3-19-18(13)10-26-28-19/h1-3,6-11H,4-5,25H2,(H,26,28)(H,27,29)	MPSOQTIARBCFIO-UHFFFAOYSA-N	794775	3-Amino-6-cyclopropyl-8-fluoro-4-(1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one; hydrochloride::US20260062412, Compound B48	Myelin transcription factor 1	Homo sapiens		 18.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794775	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794775&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293249	528826238							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126392	Nc1c(-c2cccc3[nH]ncc23)c2cc(C3CC3)c3ccccc3c2[nH]c1=O	InChI=1S/C23H18N4O/c24-21-20(14-6-3-7-19-18(14)11-25-27-19)17-10-16(12-8-9-12)13-4-1-2-5-15(13)22(17)26-23(21)28/h1-7,10-12H,8-9,24H2,(H,25,27)(H,26,28)	QHZKNLUIVZGKCR-UHFFFAOYSA-N	794776	3-Amino-6-cyclopropyl-4-(1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one 2-propanol solvate::US20260062412, Compound B49	Myelin transcription factor 1	Homo sapiens		 6.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794776	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794776&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293863	528826239							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126393	Nc1c(-c2cccc(F)c2)c2ccc3ccccc3c2[nH]c1=O	InChI=1S/C19H13FN2O/c20-13-6-3-5-12(10-13)16-15-9-8-11-4-1-2-7-14(11)18(15)22-19(23)17(16)21/h1-10H,21H2,(H,22,23)	NSOFAMMWRKVIDV-UHFFFAOYSA-N	794777	3-Amino-4-(3-fluorophenyl)-1H-benzo[h]quinolin-2-one; hydrochloride::US20260062412, Compound B50	Myelin transcription factor 1	Homo sapiens		 750							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794777	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794777&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293371	528826240							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126394	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3ncccc3c2[nH]c1=O	InChI=1S/C19H11BrFN5O/c20-12-6-10-14(8-3-4-13(21)18-11(8)7-24-26-18)15(22)19(27)25-16(10)9-2-1-5-23-17(9)12/h1-7H,22H2,(H,24,26)(H,25,27)	DQRRECKYKYCQAW-UHFFFAOYSA-N	794778	3-Amino-6-bromo-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C1	Myelin transcription factor 1	Homo sapiens		 2.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794778	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794778&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293706	528826241							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126395	Cn1ncc2c(-c3c(N)c(=O)[nH]c4c3cc(Br)c3ncccc34)ccc(F)c21	InChI=1S/C20H13BrFN5O/c1-27-19-12(8-25-27)9(4-5-14(19)22)15-11-7-13(21)18-10(3-2-6-24-18)17(11)26-20(28)16(15)23/h2-8H,23H2,1H3,(H,26,28)	BIJUIAYCUIDRCX-UHFFFAOYSA-N	794779	3-Amino-6-bromo-4-(7-fluoro-1-methylindazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C2	Myelin transcription factor 1	Homo sapiens		 1100							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794779	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794779&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293400	528826242							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126396	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(O)c3ncccc3c2[nH]c1=O	InChI=1S/C19H12FN5O2/c20-12-4-3-8(11-7-23-25-17(11)12)14-10-6-13(26)18-9(2-1-5-22-18)16(10)24-19(27)15(14)21/h1-7,26H,21H2,(H,23,25)(H,24,27)	HORDDPWVIIPRCX-UHFFFAOYSA-N	794780	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-hydroxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C3	Myelin transcription factor 1	Homo sapiens		 3.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794780	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794780&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293245	528826243							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126397	COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H14FN5O2/c1-28-14-7-11-15(9-4-5-13(21)18-12(9)8-24-26-18)16(22)20(27)25-17(11)10-3-2-6-23-19(10)14/h2-8H,22H2,1H3,(H,24,26)(H,25,27)	UZGVOKWMDFZQCU-UHFFFAOYSA-N	794781	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-methoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C4	Myelin transcription factor 1	Homo sapiens		 1.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794781	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794781&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293492	528826244							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126398	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(O[C@@H]3CCOC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H18FN5O3/c24-16-4-3-12(15-9-27-29-21(15)16)18-14-8-17(32-11-5-7-31-10-11)22-13(2-1-6-26-22)20(14)28-23(30)19(18)25/h1-4,6,8-9,11H,5,7,10,25H2,(H,27,29)(H,28,30)	WDNFEZCOBPOONI-UHFFFAOYSA-N	794782	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[(3R)-oxolan-3-yl]oxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C5	Myelin transcription factor 1	Homo sapiens		 1.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794782	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794782&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293293	528826245							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126399	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC3CCCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20FN5O2/c25-17-8-7-13(16-11-28-30-22(16)17)19-15-10-18(32-12-4-1-2-5-12)23-14(6-3-9-27-23)21(15)29-24(31)20(19)26/h3,6-12H,1-2,4-5,26H2,(H,28,30)(H,29,31)	UUYKPVJMSHUABU-UHFFFAOYSA-N	794783	3-Amino-6-cyclopentyloxy-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C6	Myelin transcription factor 1	Homo sapiens		 1.000							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794783	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794783&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293659	528826246							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126400	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC3CCOCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20FN5O3/c25-17-4-3-13(16-11-28-30-22(16)17)19-15-10-18(33-12-5-8-32-9-6-12)23-14(2-1-7-27-23)21(15)29-24(31)20(19)26/h1-4,7,10-12H,5-6,8-9,26H2,(H,28,30)(H,29,31)	ZJOPXBQFRRZNQX-UHFFFAOYSA-N	794784	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(oxan-4-yloxy)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C7	Myelin transcription factor 1	Homo sapiens		 1.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794784	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794784&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293471	528826247							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126401	CCOc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H16FN5O2/c1-2-29-15-8-12-16(10-5-6-14(22)19-13(10)9-25-27-19)17(23)21(28)26-18(12)11-4-3-7-24-20(11)15/h3-9H,2,23H2,1H3,(H,25,27)(H,26,28)	MRTXNVJHKIGLQK-UHFFFAOYSA-N	794785	3-Amino-6-ethoxy-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C8	Myelin transcription factor 1	Homo sapiens		 1.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794785	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794785&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293442	528826248							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126402	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCC3CCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20FN5O2/c25-17-7-6-13(16-10-28-30-22(16)17)19-15-9-18(32-11-12-3-1-4-12)23-14(5-2-8-27-23)21(15)29-24(31)20(19)26/h2,5-10,12H,1,3-4,11,26H2,(H,28,30)(H,29,31)	XSRRCTJDUYDITE-UHFFFAOYSA-N	794786	3-Amino-6-(cyclobutylmethoxy)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C9	Myelin transcription factor 1	Homo sapiens		 3.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794786	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794786&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293736	528826249							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126403	CC(C)CCOc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C24H22FN5O2/c1-12(2)7-9-32-18-10-15-19(13-5-6-17(25)22-16(13)11-28-30-22)20(26)24(31)29-21(15)14-4-3-8-27-23(14)18/h3-6,8,10-12H,7,9,26H2,1-2H3,(H,28,30)(H,29,31)	SDRAWGGRFHFOCN-UHFFFAOYSA-N	794787	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(3-methylbutoxy)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C10	Myelin transcription factor 1	Homo sapiens		 2.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794787	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794787&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293158	528826250							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126404	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCC3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H18FN5O2/c24-16-6-5-12(15-9-27-29-21(15)16)18-14-8-17(31-10-11-3-4-11)22-13(2-1-7-26-22)20(14)28-23(30)19(18)25/h1-2,5-9,11H,3-4,10,25H2,(H,27,29)(H,28,30)	FQQZHYOVRFONNF-UHFFFAOYSA-N	794788	3-Amino-6-(cyclopropylmethoxy)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C11	Myelin transcription factor 1	Homo sapiens		 1.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794788	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794788&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293226	528826251							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126405	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC3CCOC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H18FN5O3/c24-16-4-3-12(15-9-27-29-21(15)16)18-14-8-17(32-11-5-7-31-10-11)22-13(2-1-6-26-22)20(14)28-23(30)19(18)25/h1-4,6,8-9,11H,5,7,10,25H2,(H,27,29)(H,28,30)	WDNFEZCOBPOONI-UHFFFAOYSA-N	794789	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[(3S)-oxolan-3-yl]oxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C12	Myelin transcription factor 1	Homo sapiens		 2.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794789	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794789&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			178423165	528826252							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126406	CC(C)Oc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H18FN5O2/c1-10(2)30-16-8-13-17(11-5-6-15(23)20-14(11)9-26-28-20)18(24)22(29)27-19(13)12-4-3-7-25-21(12)16/h3-10H,24H2,1-2H3,(H,26,28)(H,27,29)	JHGYBATVADJEKA-UHFFFAOYSA-N	794790	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-propan-2-yloxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C13	Myelin transcription factor 1	Homo sapiens		 1.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794790	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794790&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293767	528826253							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126407	COCCOc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H18FN5O3/c1-30-7-8-31-16-9-13-17(11-4-5-15(23)20-14(11)10-26-28-20)18(24)22(29)27-19(13)12-3-2-6-25-21(12)16/h2-6,9-10H,7-8,24H2,1H3,(H,26,28)(H,27,29)	DEOVWGVLKHEXJK-UHFFFAOYSA-N	794791	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(2-methoxyethoxy)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C14	Myelin transcription factor 1	Homo sapiens		 2.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794791	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794791&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293374	528826254							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126408	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCC(F)(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C21H13F4N5O2/c22-13-4-3-9(12-7-28-30-18(12)13)15-11-6-14(32-8-21(23,24)25)19-10(2-1-5-27-19)17(11)29-20(31)16(15)26/h1-7H,8,26H2,(H,28,30)(H,29,31)	UBFYPLLBSMYPGI-UHFFFAOYSA-N	794792	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(2,2,2-trifluoroethoxy)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C15	Myelin transcription factor 1	Homo sapiens		 2.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794792	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794792&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293262	528826255							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126409	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCC(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C21H14F3N5O2/c22-13-4-3-9(12-7-27-29-19(12)13)16-11-6-14(31-8-15(23)24)20-10(2-1-5-26-20)18(11)28-21(30)17(16)25/h1-7,15H,8,25H2,(H,27,29)(H,28,30)	AHOWGKCZHMCVBX-UHFFFAOYSA-N	794793	3-Amino-6-(2,2-difluoroethoxy)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C16	Myelin transcription factor 1	Homo sapiens		 1.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794793	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794793&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293626	528826256							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126410	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC3CCCCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C25H22FN5O2/c26-18-9-8-14(17-12-29-31-23(17)18)20-16-11-19(33-13-5-2-1-3-6-13)24-15(7-4-10-28-24)22(16)30-25(32)21(20)27/h4,7-13H,1-3,5-6,27H2,(H,29,31)(H,30,32)	BILRANUGPZKHLA-UHFFFAOYSA-N	794794	3-Amino-6-cyclohexyloxy-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C17	Myelin transcription factor 1	Homo sapiens		 4.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794794	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794794&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293134	528826257							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126411	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC3CCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H18FN5O2/c24-16-7-6-12(15-10-27-29-21(15)16)18-14-9-17(31-11-3-1-4-11)22-13(5-2-8-26-22)20(14)28-23(30)19(18)25/h2,5-11H,1,3-4,25H2,(H,27,29)(H,28,30)	ISDFJCWLLPEYQY-UHFFFAOYSA-N	794795	3-Amino-6-cyclobutyloxy-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C18	Myelin transcription factor 1	Homo sapiens		 2.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794795	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794795&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293528	528826258							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126412	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCCCF)c3ncccc3c2[nH]c1=O	InChI=1S/C22H17F2N5O2/c23-6-2-8-31-16-9-13-17(11-4-5-15(24)20-14(11)10-27-29-20)18(25)22(30)28-19(13)12-3-1-7-26-21(12)16/h1,3-5,7,9-10H,2,6,8,25H2,(H,27,29)(H,28,30)	ZGJLNVIPBMQUBK-UHFFFAOYSA-N	794796	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(3-fluoropropoxy)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C19	Myelin transcription factor 1	Homo sapiens		 2.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794796	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794796&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293578	528826259							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126413	CC(C)(O)CCOc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C24H22FN5O3/c1-24(2,32)7-9-33-17-10-14-18(12-5-6-16(25)21-15(12)11-28-30-21)19(26)23(31)29-20(14)13-4-3-8-27-22(13)17/h3-6,8,10-11,32H,7,9,26H2,1-2H3,(H,28,30)(H,29,31)	YMTXXWOTJZXZRO-UHFFFAOYSA-N	794797	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(3-hydroxy-3-methylbutoxy)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C20	Myelin transcription factor 1	Homo sapiens		 3.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794797	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794797&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293942	528826260							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126414	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C20H12F3N5O2/c21-12-4-3-8(11-7-26-28-17(11)12)14-10-6-13(30-20(22)23)18-9(2-1-5-25-18)16(10)27-19(29)15(14)24/h1-7,20H,24H2,(H,26,28)(H,27,29)	CKIDBTAZJFZURM-UHFFFAOYSA-N	794798	3-Amino-6-(difluoromethoxy)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C21	Myelin transcription factor 1	Homo sapiens		 2.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794798	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794798&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293479	528826261							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126415	C[C@H](Oc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12)C(F)(F)F	InChI=1S/C22H15F4N5O2/c1-9(22(24,25)26)33-15-7-12-16(10-4-5-14(23)19-13(10)8-29-31-19)17(27)21(32)30-18(12)11-3-2-6-28-20(11)15/h2-9H,27H2,1H3,(H,29,31)(H,30,32)	ILBQLXOSVYHDKI-UHFFFAOYSA-N	794799	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[(2S)-1,1,1-trifluoropropan-2-yl]oxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C22	Myelin transcription factor 1	Homo sapiens		 7.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794799	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794799&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293572	528826262							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126416	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC3CC(F)(F)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H16F3N5O2/c24-15-4-3-11(14-9-29-31-20(14)15)17-13-6-16(33-10-7-23(25,26)8-10)21-12(2-1-5-28-21)19(13)30-22(32)18(17)27/h1-6,9-10H,7-8,27H2,(H,29,31)(H,30,32)	BALAFJZMTPSJCC-UHFFFAOYSA-N	794800	3-Amino-6-(3,3-difluorocyclobutyl)oxy-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C23	Myelin transcription factor 1	Homo sapiens		 5.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794800	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794800&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293882	528826263							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126417	CC(C)(O)COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C23H20FN5O3/c1-23(2,31)10-32-16-8-13-17(11-5-6-15(24)20-14(11)9-27-29-20)18(25)22(30)28-19(13)12-4-3-7-26-21(12)16/h3-9,31H,10,25H2,1-2H3,(H,27,29)(H,28,30)	OSHNHYFMTQNWDD-UHFFFAOYSA-N	794801	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(2-hydroxy-2-methylpropoxy)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C24	Myelin transcription factor 1	Homo sapiens		 6.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794801	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794801&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293661	528826264							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126418	CC(F)(F)COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H16F3N5O2/c1-22(24,25)9-32-15-7-12-16(10-4-5-14(23)19-13(10)8-28-30-19)17(26)21(31)29-18(12)11-3-2-6-27-20(11)15/h2-8H,9,26H2,1H3,(H,28,30)(H,29,31)	VFQYWKDOOYTMNT-UHFFFAOYSA-N	794802	3-Amino-6-(2,2-difluoropropoxy)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C25	Myelin transcription factor 1	Homo sapiens		 2.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794802	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794802&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293527	528826265							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126419	COCC(F)(F)COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C23H18F3N5O3/c1-33-9-23(25,26)10-34-16-7-13-17(11-4-5-15(24)20-14(11)8-29-31-20)18(27)22(32)30-19(13)12-3-2-6-28-21(12)16/h2-8H,9-10,27H2,1H3,(H,29,31)(H,30,32)	PUDOACZSKDKFOO-UHFFFAOYSA-N	794803	3-Amino-6-(2,2-difluoro-3-methoxypropoxy)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C26	Myelin transcription factor 1	Homo sapiens		 2.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794803	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794803&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293889	528826266							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126420	C[C@@H](Oc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12)C(F)(F)F	InChI=1S/C22H15F4N5O2/c1-9(22(24,25)26)33-15-7-12-16(10-4-5-14(23)19-13(10)8-29-31-19)17(27)21(32)30-18(12)11-3-2-6-28-20(11)15/h2-9H,27H2,1H3,(H,29,31)(H,30,32)	ILBQLXOSVYHDKI-UHFFFAOYSA-N	794804	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[(2R)-1,1,1-trifluoropropan-2-yl]oxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C27	Myelin transcription factor 1	Homo sapiens		 4.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794804	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794804&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293605	528826267							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126421	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(O[C@H]3C[C@@H](F)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H17F2N5O2/c24-10-6-11(7-10)32-17-8-14-18(12-3-4-16(25)21-15(12)9-28-30-21)19(26)23(31)29-20(14)13-2-1-5-27-22(13)17/h1-5,8-11H,6-7,26H2,(H,28,30)(H,29,31)	SXVHVHDRZDKHET-UHFFFAOYSA-N	794805	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-((1s,3s)-3-fluorocyclobutoxy)-1,7-phenanthrolin-2(1H)-one::US20260062412, Compound C28	Myelin transcription factor 1	Homo sapiens		 1.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794805	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794805&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293666	528826268							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126422	CO[C@H]1C[C@@H](Oc2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)C1	InChI=1S/C24H20FN5O3/c1-32-11-7-12(8-11)33-18-9-15-19(13-4-5-17(25)22-16(13)10-28-30-22)20(26)24(31)29-21(15)14-3-2-6-27-23(14)18/h2-6,9-12H,7-8,26H2,1H3,(H,28,30)(H,29,31)	PYGUNNRIUPSDLO-UHFFFAOYSA-N	794806	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-((1s,3s)-3-methoxycyclobutoxy)-1,7-phenanthrolin-2(1H)-one::US20260062412, Compound C29	Myelin transcription factor 1	Homo sapiens		 3.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794806	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794806&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293797	528826269							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126423	CO[C@H]1C[C@H](Oc2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)C1	InChI=1S/C24H20FN5O3/c1-32-11-7-12(8-11)33-18-9-15-19(13-4-5-17(25)22-16(13)10-28-30-22)20(26)24(31)29-21(15)14-3-2-6-27-23(14)18/h2-6,9-12H,7-8,26H2,1H3,(H,28,30)(H,29,31)	PYGUNNRIUPSDLO-UHFFFAOYSA-N	794807	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-((1r,3r)-3-methoxycyclobutoxy)-1,7-phenanthrolin-2(1H)-one::US20260062412, Compound C30	Myelin transcription factor 1	Homo sapiens		 5.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794807	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794807&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293797	528826270							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126424	N#C[C@H]1C[C@H](Oc2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)C1	InChI=1S/C24H17FN6O2/c25-17-4-3-13(16-10-29-31-22(16)17)19-15-8-18(33-12-6-11(7-12)9-26)23-14(2-1-5-28-23)21(15)30-24(32)20(19)27/h1-5,8,10-12H,6-7,27H2,(H,29,31)(H,30,32)	OSRYMJQFONWWTK-UHFFFAOYSA-N	794808	(1r,3r)-3-[[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]oxy]cyclobutane-1-carbonitrile::US20260062412, Compound C31	Myelin transcription factor 1	Homo sapiens		 4.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794808	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794808&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293840	528826271							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126425	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCCC(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C22H16F3N5O2/c23-14-4-3-10(13-9-28-30-20(13)14)17-12-8-15(32-7-5-16(24)25)21-11(2-1-6-27-21)19(12)29-22(31)18(17)26/h1-4,6,8-9,16H,5,7,26H2,(H,28,30)(H,29,31)	ZRKHKKAYAYBRRD-UHFFFAOYSA-N	794809	3-Amino-6-(3,3-difluoropropoxy)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C32	Myelin transcription factor 1	Homo sapiens		 3.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794809	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794809&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293734	528826272							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126426	N#C[C@H]1C[C@@H](Oc2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)C1	InChI=1S/C24H17FN6O2/c25-17-4-3-13(16-10-29-31-22(16)17)19-15-8-18(33-12-6-11(7-12)9-26)23-14(2-1-5-28-23)21(15)30-24(32)20(19)27/h1-5,8,10-12H,6-7,27H2,(H,29,31)(H,30,32)	OSRYMJQFONWWTK-UHFFFAOYSA-N	794810	(1s,3s)-3-[[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]oxy]cyclobutane-1-carbonitrile::US20260062412, Compound C33	Myelin transcription factor 1	Homo sapiens		 3.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794810	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794810&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293840	528826273							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126427	CC[C@H](C)Oc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C23H20FN5O2/c1-3-11(2)31-17-9-14-18(12-6-7-16(24)21-15(12)10-27-29-21)19(25)23(30)28-20(14)13-5-4-8-26-22(13)17/h4-11H,3,25H2,1-2H3,(H,27,29)(H,28,30)	KWYHRXRCMSSWSV-UHFFFAOYSA-N	794811	3-Amino-6-[(2S)-butan-2-yl]oxy-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C34	Myelin transcription factor 1	Homo sapiens		 3.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794811	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794811&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293620	528826274							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126428	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC[C@H]3CCCO3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20FN5O3/c25-17-6-5-13(16-10-28-30-22(16)17)19-15-9-18(33-11-12-3-2-8-32-12)23-14(4-1-7-27-23)21(15)29-24(31)20(19)26/h1,4-7,9-10,12H,2-3,8,11,26H2,(H,28,30)(H,29,31)	HDYYBVOXXIVGQL-UHFFFAOYSA-N	794812	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[[(2R)-oxolan-2-yl]methoxy]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C35	Myelin transcription factor 1	Homo sapiens		 4.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794812	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794812&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293350	528826275							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126429	CC[C@@H](C)Oc1cc2c(c3cccnc13)NC(=O)C(N)C2c1ccc(F)c2[nH]ncc12	InChI=1S/C23H22FN5O2/c1-3-11(2)31-17-9-14-18(12-6-7-16(24)21-15(12)10-27-29-21)19(25)23(30)28-20(14)13-5-4-8-26-22(13)17/h4-11,18-19H,3,25H2,1-2H3,(H,27,29)(H,28,30)	IHEUWHASRPQHAQ-UHFFFAOYSA-N	794813	3-Amino-6-[(2R)-butan-2-yl]oxy-4-(7-fluoro-1H-indazol-4-yl)-3,4-dihydro-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C36	Myelin transcription factor 1	Homo sapiens		 4.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794813	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794813&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293569	528826276							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126430	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC[C@@H]3CCCO3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20FN5O3/c25-17-6-5-13(16-10-28-30-22(16)17)19-15-9-18(33-11-12-3-2-8-32-12)23-14(4-1-7-27-23)21(15)29-24(31)20(19)26/h1,4-7,9-10,12H,2-3,8,11,26H2,(H,28,30)(H,29,31)	HDYYBVOXXIVGQL-UHFFFAOYSA-N	794814	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[[(2S)-oxolan-2-yl]methoxy]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C37	Myelin transcription factor 1	Homo sapiens		 3.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794814	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794814&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293784	528826277							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126431	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCC3(F)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H17F2N5O2/c24-15-4-3-11(14-9-28-30-20(14)15)17-13-8-16(32-10-23(25)5-6-23)21-12(2-1-7-27-21)19(13)29-22(31)18(17)26/h1-4,7-9H,5-6,10,26H2,(H,28,30)(H,29,31)	NQGCRTKJMIASGM-UHFFFAOYSA-N	794815	3-Amino-6-[(1-fluorocyclopropyl)methoxy]-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C38	Myelin transcription factor 1	Homo sapiens		 5.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794815	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794815&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293895	528826278							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126432	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCC3CC(F)(F)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H18F3N5O2/c25-16-4-3-12(15-9-30-32-21(15)16)18-14-6-17(34-10-11-7-24(26,27)8-11)22-13(2-1-5-29-22)20(14)31-23(33)19(18)28/h1-6,9,11H,7-8,10,28H2,(H,30,32)(H,31,33)	RJZUECQZQYPIKP-UHFFFAOYSA-N	794816	3-Amino-6-[(3,3-difluorocyclobutyl)methoxy]-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C39	Myelin transcription factor 1	Homo sapiens		 6.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794816	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794816&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293832	528826279							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126433	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCC3(F)COC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H17F2N5O3/c24-15-4-3-11(14-7-28-30-20(14)15)17-13-6-16(33-10-23(25)8-32-9-23)21-12(2-1-5-27-21)19(13)29-22(31)18(17)26/h1-7H,8-10,26H2,(H,28,30)(H,29,31)	GWECDIDNKYCVCJ-UHFFFAOYSA-N	794817	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[(3-fluorooxetan-3-yl)methoxy]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C40	Myelin transcription factor 1	Homo sapiens		 4.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794817	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794817&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293283	528826280							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126434	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC3CC4(COC4)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C25H20FN5O3/c26-17-4-3-13(16-9-29-31-22(16)17)19-15-6-18(34-12-7-25(8-12)10-33-11-25)23-14(2-1-5-28-23)21(15)30-24(32)20(19)27/h1-6,9,12H,7-8,10-11,27H2,(H,29,31)(H,30,32)	FZFFWGFJBFLXFR-UHFFFAOYSA-N	794818	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(2-oxaspiro[3,3]heptan-6-yloxy)-1H-1,7-one::US20260062412, Compound C41	Myelin transcription factor 1	Homo sapiens		 6.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794818	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794818&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293610	528826281							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126435	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(O[C@H]3C[C@H](F)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H17F2N5O2/c24-10-6-11(7-10)32-17-8-14-18(12-3-4-16(25)21-15(12)9-28-30-21)19(26)23(31)29-20(14)13-2-1-5-27-22(13)17/h1-5,8-11H,6-7,26H2,(H,28,30)(H,29,31)	SXVHVHDRZDKHET-UHFFFAOYSA-N	794819	3-Amino-6-((1r,3r)-3-fluorocyclobutyl)oxy-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C42	Myelin transcription factor 1	Homo sapiens		 2.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794819	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794819&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293666	528826282							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126436	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCCOC(F)(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C22H15F4N5O3/c23-14-4-3-10(13-9-29-31-19(13)14)16-12-8-15(33-6-7-34-22(24,25)26)20-11(2-1-5-28-20)18(12)30-21(32)17(16)27/h1-5,8-9H,6-7,27H2,(H,29,31)(H,30,32)	KKKSEOBFAKVVMG-UHFFFAOYSA-N	794820	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[2-(trifluoromethoxy)ethoxy]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C43	Myelin transcription factor 1	Homo sapiens		 19.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794820	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794820&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293412	528826283							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126437	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCC3(C(F)(F)F)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H17F4N5O2/c25-15-4-3-11(14-9-31-33-20(14)15)17-13-8-16(35-10-23(5-6-23)24(26,27)28)21-12(2-1-7-30-21)19(13)32-22(34)18(17)29/h1-4,7-9H,5-6,10,29H2,(H,31,33)(H,32,34)	JHIAKUZHRVUFNZ-UHFFFAOYSA-N	794821	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[[1-(trifluoromethyl)cyclopropyl]methoxy]-1H-1,7-one::US20260062412, Compound C44	Myelin transcription factor 1	Homo sapiens		 5.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794821	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794821&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293274	528826284							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126438	CO[C@@H](C)COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C23H20FN5O3/c1-11(31-2)10-32-17-8-14-18(12-5-6-16(24)21-15(12)9-27-29-21)19(25)23(30)28-20(14)13-4-3-7-26-22(13)17/h3-9,11H,10,25H2,1-2H3,(H,27,29)(H,28,30)	YLLSAWYFGFOHGN-UHFFFAOYSA-N	794822	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[(2S)-2-methoxypropoxy]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C45	Myelin transcription factor 1	Homo sapiens		 3.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794822	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794822&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293138	528826285							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126439	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(O[C@@H]3CCCOC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20FN5O3/c25-17-6-5-13(16-10-28-30-22(16)17)19-15-9-18(33-12-3-2-8-32-11-12)23-14(4-1-7-27-23)21(15)29-24(31)20(19)26/h1,4-7,9-10,12H,2-3,8,11,26H2,(H,28,30)(H,29,31)	ZHEMYMMLWAGGFK-UHFFFAOYSA-N	794823	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[(3R)-oxan-3-yl]oxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C46	Myelin transcription factor 1	Homo sapiens		 2.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794823	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794823&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293693	528826286							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126440	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC3CCS(=O)(=O)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20FN5O4S/c25-17-4-3-13(16-11-28-30-22(16)17)19-15-10-18(34-12-5-8-35(32,33)9-6-12)23-14(2-1-7-27-23)21(15)29-24(31)20(19)26/h1-4,7,10-12H,5-6,8-9,26H2,(H,28,30)(H,29,31)	ZTSKBVOICGKHEV-UHFFFAOYSA-N	794824	3-Amino-6-(1,1-dioxothian-4-yl)oxy-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C47	Myelin transcription factor 1	Homo sapiens		 4.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794824	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794824&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293584	528826287							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126441	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC3CCC(F)(F)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C25H20F3N5O2/c26-17-4-3-13(16-11-31-33-22(16)17)19-15-10-18(35-12-5-7-25(27,28)8-6-12)23-14(2-1-9-30-23)21(15)32-24(34)20(19)29/h1-4,9-12H,5-8,29H2,(H,31,33)(H,32,34)	GOUSRXWJZDLUGX-UHFFFAOYSA-N	794825	3-Amino-6-(4,4-difluorocyclohexyl)oxy-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C48	Myelin transcription factor 1	Homo sapiens		 10.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794825	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794825&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293793	528826288							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126442	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCC34CC(C3)C4)c3ncccc3c2[nH]c1=O	InChI=1S/C25H20FN5O2/c26-17-4-3-13(16-10-29-31-22(16)17)19-15-6-18(33-11-25-7-12(8-25)9-25)23-14(2-1-5-28-23)21(15)30-24(32)20(19)27/h1-6,10,12H,7-9,11,27H2,(H,29,31)(H,30,32)	FXNSSVVWNOJVRK-UHFFFAOYSA-N	794826	3-Amino-6-(1-bicyclo[1.1.1]pentanylmethoxy)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C49	Myelin transcription factor 1	Homo sapiens		 1.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794826	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794826&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293593	528826289							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126443	CO[C@H](C)COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C23H20FN5O3/c1-11(31-2)10-32-17-8-14-18(12-5-6-16(24)21-15(12)9-27-29-21)19(25)23(30)28-20(14)13-4-3-7-26-22(13)17/h3-9,11H,10,25H2,1-2H3,(H,27,29)(H,28,30)	YLLSAWYFGFOHGN-UHFFFAOYSA-N	794827	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[(2R)-2-methoxypropoxy]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C50	Myelin transcription factor 1	Homo sapiens		 4.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794827	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794827&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293195	528826290							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126444	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(O[C@H]3CCCOC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20FN5O3/c25-17-6-5-13(16-10-28-30-22(16)17)19-15-9-18(33-12-3-2-8-32-11-12)23-14(4-1-7-27-23)21(15)29-24(31)20(19)26/h1,4-7,9-10,12H,2-3,8,11,26H2,(H,28,30)(H,29,31)	ZHEMYMMLWAGGFK-UHFFFAOYSA-N	794828	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[(3S)-oxan-3-yl]oxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C51	Myelin transcription factor 1	Homo sapiens		 1.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794828	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794828&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293538	528826291							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126445	CC1(COc2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC(F)(F)C1	InChI=1S/C25H20F3N5O2/c1-24(9-25(27,28)10-24)11-35-17-7-14-18(12-4-5-16(26)21-15(12)8-31-33-21)19(29)23(34)32-20(14)13-3-2-6-30-22(13)17/h2-8H,9-11,29H2,1H3,(H,31,33)(H,32,34)	BXLKAOUJZIVIAL-UHFFFAOYSA-N	794829	3-Amino-6-[(3,3-difluoro-1-methylcyclobutyl)methoxy]-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-one::US20260062412, Compound C52	Myelin transcription factor 1	Homo sapiens		 2.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794829	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794829&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293828	528826292							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126446	COC1(COc2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC1	InChI=1S/C24H20FN5O3/c1-32-24(6-7-24)11-33-17-9-14-18(12-4-5-16(25)21-15(12)10-28-30-21)19(26)23(31)29-20(14)13-3-2-8-27-22(13)17/h2-5,8-10H,6-7,11,26H2,1H3,(H,28,30)(H,29,31)	HHPBBHTUBCMNGF-UHFFFAOYSA-N	794830	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[(1-methoxycyclopropyl)methoxy]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C53	Myelin transcription factor 1	Homo sapiens		 4.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794830	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794830&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293653	528826293							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126447	N#CC1(COc2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC1	InChI=1S/C24H17FN6O2/c25-16-4-3-12(15-9-29-31-21(15)16)18-14-8-17(33-11-24(10-26)5-6-24)22-13(2-1-7-28-22)20(14)30-23(32)19(18)27/h1-4,7-9H,5-6,11,27H2,(H,29,31)(H,30,32)	IAXAJNZKTOLLBJ-UHFFFAOYSA-N	794831	1-[[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]oxymethyl]cyclopropane-1-carbonitrile::US20260062412, Compound C54	Myelin transcription factor 1	Homo sapiens		 1.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794831	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794831&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293785	528826294							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126448	N#CC1(COc2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CCC1	InChI=1S/C25H19FN6O2/c26-17-5-4-13(16-10-30-32-22(16)17)19-15-9-18(34-12-25(11-27)6-2-7-25)23-14(3-1-8-29-23)21(15)31-24(33)20(19)28/h1,3-5,8-10H,2,6-7,12,28H2,(H,30,32)(H,31,33)	INKRRSTXHMWJBC-UHFFFAOYSA-N	794832	1-[[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]oxymethyl]cyclobutane-1-carbonitrile::US20260062412, Compound C55	Myelin transcription factor 1	Homo sapiens		 0.920							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794832	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794832&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293730	528826295							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126449	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCC3(F)CCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H19F2N5O2/c25-16-5-4-12(15-10-29-31-21(15)16)18-14-9-17(33-11-24(26)6-2-7-24)22-13(3-1-8-28-22)20(14)30-23(32)19(18)27/h1,3-5,8-10H,2,6-7,11,27H2,(H,29,31)(H,30,32)	NMOHAQSRVJPKPP-UHFFFAOYSA-N	794833	3-Amino-6-[(1-fluorocyclobutyl)methoxy]-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C56	Myelin transcription factor 1	Homo sapiens		 1.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794833	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794833&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293751	528826296							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126450	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC3CC(C(F)(F)F)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H17F4N5O2/c25-16-4-3-12(15-9-31-33-21(15)16)18-14-8-17(35-11-6-10(7-11)24(26,27)28)22-13(2-1-5-30-22)20(14)32-23(34)19(18)29/h1-5,8-11H,6-7,29H2,(H,31,33)(H,32,34)	MAXREWTYCNOKLF-UHFFFAOYSA-N	794834	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[3-(trifluoromethyl)cyclobutyl]oxy-1H-1,7-one::US20260062412, Compound C57	Myelin transcription factor 1	Homo sapiens		 2.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794834	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794834&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293719	528826297							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126451	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC3CC(C(F)F)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H18F3N5O2/c25-16-4-3-12(15-9-30-32-21(15)16)18-14-8-17(34-11-6-10(7-11)23(26)27)22-13(2-1-5-29-22)20(14)31-24(33)19(18)28/h1-5,8-11,23H,6-7,28H2,(H,30,32)(H,31,33)	KIPYZLRZNXKCFM-UHFFFAOYSA-N	794835	3-Amino-6-[3-(difluoromethyl)cyclobutyl]oxy-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C58	Myelin transcription factor 1	Homo sapiens		 1.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794835	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794835&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293941	528826298							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126452	CC(C)(COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12)C(F)(F)F	InChI=1S/C24H19F4N5O2/c1-23(2,24(26,27)28)10-35-16-8-13-17(11-5-6-15(25)20-14(11)9-31-33-20)18(29)22(34)32-19(13)12-4-3-7-30-21(12)16/h3-9H,10,29H2,1-2H3,(H,31,33)(H,32,34)	ALJVKNDIFKSQPN-UHFFFAOYSA-N	794836	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(3,3,3-trifluoro-2,2-dimethylpropoxy)-1H-1,7-one::US20260062412, Compound C59	Myelin transcription factor 1	Homo sapiens		 5.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794836	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794836&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293403	528826299							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126453	CCCOc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H18FN5O2/c1-2-8-30-16-9-13-17(11-5-6-15(23)20-14(11)10-26-28-20)18(24)22(29)27-19(13)12-4-3-7-25-21(12)16/h3-7,9-10H,2,8,24H2,1H3,(H,26,28)(H,27,29)	FQAZWBJIECDGJM-UHFFFAOYSA-N	794837	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-propoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C60	Myelin transcription factor 1	Homo sapiens		 0.850							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794837	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794837&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293282	528826300							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126454	C[C@@H](F)COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H17F2N5O2/c1-10(23)9-31-16-7-13-17(11-4-5-15(24)20-14(11)8-27-29-20)18(25)22(30)28-19(13)12-3-2-6-26-21(12)16/h2-8,10H,9,25H2,1H3,(H,27,29)(H,28,30)	VNYGQUDVMXLQAN-UHFFFAOYSA-N	794838	(R)-3-amino-4-(7-fluoro-1H-indazol-4-yl)-6-(2-fluoropropoxy)-1,7-phenanthrolin-2(1H)-one::US20260062412, Compound C61	Myelin transcription factor 1	Homo sapiens		 1.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794838	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794838&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293323	528826301							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126455	N#CCOc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H13FN6O2/c22-14-4-3-10(13-9-26-28-19(13)14)16-12-8-15(30-7-5-23)20-11(2-1-6-25-20)18(12)27-21(29)17(16)24/h1-4,6,8-9H,7,24H2,(H,26,28)(H,27,29)	WAQFSPBXIHPQIE-UHFFFAOYSA-N	794839	2-[[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]oxy]acetonitrile::US20260062412, Compound C62	Myelin transcription factor 1	Homo sapiens		 1.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794839	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794839&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293454	528826302							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126456	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(SC(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C20H12F3N5OS/c21-12-4-3-8(11-7-26-28-17(11)12)14-10-6-13(30-20(22)23)18-9(2-1-5-25-18)16(10)27-19(29)15(14)24/h1-7,20H,24H2,(H,26,28)(H,27,29)	RXSYFKTUQSMKNE-UHFFFAOYSA-N	794840	3-Amino-6-(difluoromethylsulfanyl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C63	Myelin transcription factor 1	Homo sapiens		 1.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794840	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794840&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293847	528826303							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126457	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(F)c3ncccc3c2[nH]c1=O	InChI=1S/C19H11F2N5O/c20-12-4-3-8(11-7-24-26-18(11)12)14-10-6-13(21)17-9(2-1-5-23-17)16(10)25-19(27)15(14)22/h1-7H,22H2,(H,24,26)(H,25,27)	DZGCMIUGLPUCIS-UHFFFAOYSA-N	794841	3-Amino-6-fluoro-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C64	Myelin transcription factor 1	Homo sapiens		 7.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794841	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794841&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293174	528826304							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126458	COc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H13F2N5O2/c1-29-13-6-10-14(9-5-12(21)15(22)19-11(9)7-25-27-19)16(23)20(28)26-17(10)8-3-2-4-24-18(8)13/h2-7H,23H2,1H3,(H,25,27)(H,26,28)	XFZXIJLXMACSSN-UHFFFAOYSA-N	794842	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-methoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C65	Myelin transcription factor 1	Homo sapiens		 3.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794842	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794842&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293543	528826305							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126459	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(Br)c3ncccc3c2[nH]c1=O	InChI=1S/C19H10BrF2N5O/c20-11-4-9-13(8-5-12(21)14(22)18-10(8)6-25-27-18)15(23)19(28)26-16(9)7-2-1-3-24-17(7)11/h1-6H,23H2,(H,25,27)(H,26,28)	SERHMTCBVBXPEB-UHFFFAOYSA-N	794843	3-Amino-6-bromo-4-(6,7-difluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C66	Myelin transcription factor 1	Homo sapiens		 4.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794843	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794843&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293943	528826306							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126460	CCOc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H15F2N5O2/c1-2-30-14-7-11-15(10-6-13(22)16(23)20-12(10)8-26-28-20)17(24)21(29)27-18(11)9-4-3-5-25-19(9)14/h3-8H,2,24H2,1H3,(H,26,28)(H,27,29)	ZDYACGZBLWVWLA-UHFFFAOYSA-N	794844	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-ethoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C67	Myelin transcription factor 1	Homo sapiens		 2.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794844	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794844&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293625	528826307							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126461	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(OCC(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C21H13F4N5O2/c22-12-4-9(11-6-28-30-20(11)16(12)25)15-10-5-13(32-7-14(23)24)19-8(2-1-3-27-19)18(10)29-21(31)17(15)26/h1-6,14H,7,26H2,(H,28,30)(H,29,31)	JWLNDIFXGALLQK-UHFFFAOYSA-N	794845	3-Amino-6-(2,2-difluoroethoxy)-4-(6,7-difluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C68	Myelin transcription factor 1	Homo sapiens		 1.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794845	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794845&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293328	528826308							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126462	CC(C)Oc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H17F2N5O2/c1-9(2)31-15-7-12-16(11-6-14(23)17(24)21-13(11)8-27-29-21)18(25)22(30)28-19(12)10-4-3-5-26-20(10)15/h3-9H,25H2,1-2H3,(H,27,29)(H,28,30)	GTSCSJYLNSFNGR-UHFFFAOYSA-N	794846	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-propan-2-yloxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C69	Myelin transcription factor 1	Homo sapiens		 2.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794846	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794846&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293576	528826309							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126463	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(OCC3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H17F2N5O2/c24-15-6-12(14-8-28-30-22(14)18(15)25)17-13-7-16(32-9-10-3-4-10)21-11(2-1-5-27-21)20(13)29-23(31)19(17)26/h1-2,5-8,10H,3-4,9,26H2,(H,28,30)(H,29,31)	ZAIOEEQXKUPDPX-UHFFFAOYSA-N	794847	3-Amino-6-(cyclopropylmethoxy)-4-(6,7-difluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C70	Myelin transcription factor 1	Homo sapiens		 1.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794847	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794847&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293267	528826310							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126464	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(OCC3(F)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H16F3N5O2/c24-14-6-11(13-8-29-31-21(13)17(14)25)16-12-7-15(33-9-23(26)3-4-23)20-10(2-1-5-28-20)19(12)30-22(32)18(16)27/h1-2,5-8H,3-4,9,27H2,(H,29,31)(H,30,32)	GGJTZJWWISAYEJ-UHFFFAOYSA-N	794848	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-[(1-fluorocyclopropyl)methoxy]-1H-1,7-one::US20260062412, Compound C71	Myelin transcription factor 1	Homo sapiens		 1.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794848	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794848&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293169	528826311							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126465	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(OC(F)(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C20H10F5N5O2/c21-11-4-8(10-6-28-30-18(10)14(11)22)13-9-5-12(32-20(23,24)25)17-7(2-1-3-27-17)16(9)29-19(31)15(13)26/h1-6H,26H2,(H,28,30)(H,29,31)	MNLBBZJSJRXHJI-UHFFFAOYSA-N	794849	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-(trifluoromethoxy)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C72	Myelin transcription factor 1	Homo sapiens		 6.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794849	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794849&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293208	528826312							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126466	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Br)c3ncccc3c2[nH]c1=O	InChI=1S/C19H11BrClN5O/c20-12-6-10-14(8-3-4-13(21)18-11(8)7-24-26-18)15(22)19(27)25-16(10)9-2-1-5-23-17(9)12/h1-7H,22H2,(H,24,26)(H,25,27)	HRLAXGHROUXRRK-UHFFFAOYSA-N	794850	3-Amino-6-bromo-4-(7-chloro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C73	Myelin transcription factor 1	Homo sapiens		<14.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794850	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794850&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293539	528826313							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126467	COc1cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H14ClN5O2/c1-28-14-7-11-15(9-4-5-13(21)18-12(9)8-24-26-18)16(22)20(27)25-17(11)10-3-2-6-23-19(10)14/h2-8H,22H2,1H3,(H,24,26)(H,25,27)	IPOHKFXAYVMCSO-UHFFFAOYSA-N	794851	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-methoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C74	Myelin transcription factor 1	Homo sapiens		 0.830							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794851	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794851&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293748	528826314							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126468	Nc1c(-c2cc(F)c(Cl)c3[nH]ncc23)c2cc(Br)c3ncccc3c2[nH]c1=O	InChI=1S/C19H10BrClFN5O/c20-11-4-9-13(8-5-12(22)14(21)18-10(8)6-25-27-18)15(23)19(28)26-16(9)7-2-1-3-24-17(7)11/h1-6H,23H2,(H,25,27)(H,26,28)	RRNRYLCRXNXUMG-UHFFFAOYSA-N	794852	3-Amino-6-bromo-4-(7-chloro-6-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C75	Myelin transcription factor 1	Homo sapiens		 1.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794852	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794852&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293380	528826315							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126469	COc1cc2c(-c3cc(F)c(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H13ClFN5O2/c1-29-13-6-10-14(9-5-12(22)15(21)19-11(9)7-25-27-19)16(23)20(28)26-17(10)8-3-2-4-24-18(8)13/h2-7H,23H2,1H3,(H,25,27)(H,26,28)	AKGZZODTYNYXCP-UHFFFAOYSA-N	794853	3-Amino-4-(7-chloro-6-fluoro-1H-indazol-4-yl)-6-methoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C76	Myelin transcription factor 1	Homo sapiens		 1.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794853	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794853&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293729	528826316							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126470	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Cl)c3ncccc3c2[nH]c1=O	InChI=1S/C19H11Cl2N5O/c20-12-4-3-8(11-7-24-26-18(11)12)14-10-6-13(21)17-9(2-1-5-23-17)16(10)25-19(27)15(14)22/h1-7H,22H2,(H,24,26)(H,25,27)	BRJQEZUPISCKTB-UHFFFAOYSA-N	794854	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C77	Myelin transcription factor 1	Homo sapiens		 8.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794854	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794854&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293878	528826317							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126471	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Cl)c3ncccc3c2[nH]c1=O	InChI=1S/C19H11ClFN5O/c20-12-6-10-14(8-3-4-13(21)18-11(8)7-24-26-18)15(22)19(27)25-16(10)9-2-1-5-23-17(9)12/h1-7H,22H2,(H,24,26)(H,25,27)	CWHCCNDDZMAHAF-UHFFFAOYSA-N	794855	3-Amino-6-chloro-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C78	Myelin transcription factor 1	Homo sapiens		 3.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794855	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794855&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293671	528826318							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126472	Nc1c(-c2cccc3[nH]ncc23)c2cc(Cl)c3ncccc3c2[nH]c1=O	InChI=1S/C19H12ClN5O/c20-13-7-11-15(9-3-1-5-14-12(9)8-23-25-14)16(21)19(26)24-17(11)10-4-2-6-22-18(10)13/h1-8H,21H2,(H,23,25)(H,24,26)	WLXVQQBMMOFSOX-UHFFFAOYSA-N	794856	3-Amino-6-chloro-4-(1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C79	Myelin transcription factor 1	Homo sapiens		 11.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794856	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794856&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293190	528826319							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126473	Nc1c(-c2cncc3[nH]ncc23)c2cc(Br)c3ncccc3c2[nH]c1=O	InChI=1S/C18H11BrN6O/c19-12-4-9-14(11-5-21-7-13-10(11)6-23-25-13)15(20)18(26)24-16(9)8-2-1-3-22-17(8)12/h1-7H,20H2,(H,23,25)(H,24,26)	UENKAQLMHWJBAO-UHFFFAOYSA-N	794857	3-Amino-6-bromo-4-(1H-pyrazolo[3,4-c]pyridin-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C80	Myelin transcription factor 1	Homo sapiens		 100.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794857	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794857&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293343	528826320							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126474	Nc1c(-c2ccnc3[nH]ncc23)c2cc(Br)c3ncccc3c2[nH]c1=O	InChI=1S/C18H11BrN6O/c19-12-6-10-13(8-3-5-22-17-11(8)7-23-25-17)14(20)18(26)24-15(10)9-2-1-4-21-16(9)12/h1-7H,20H2,(H,24,26)(H,22,23,25)	XJDMKFPFDMXXPR-UHFFFAOYSA-N	794858	3-Amino-6-bromo-4-(1H-pyrazolo[3,4-b]pyridin-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C81	Myelin transcription factor 1	Homo sapiens		 49.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794858	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794858&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293237	528826321							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126475	Nc1c(-c2ccnc3[nH]ncc23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C21H16N6O/c22-17-16(11-5-7-24-20-15(11)9-25-27-20)14-8-13(10-3-4-10)18-12(2-1-6-23-18)19(14)26-21(17)28/h1-2,5-10H,3-4,22H2,(H,26,28)(H,24,25,27)	QTZJOLXANCOGEX-UHFFFAOYSA-N	794859	3-Amino-6-cyclopropyl-4-(1H-pyrazolo[3,4-b]pyridin-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C82	Myelin transcription factor 1	Homo sapiens		 11.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794859	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794859&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293164	528826322							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126476	Nc1c(-c2ccc(F)c3[nH]ncc23)c2ccc3ncccc3c2[nH]c1=O	InChI=1S/C19H12FN5O/c20-13-5-3-9(12-8-23-25-18(12)13)15-11-4-6-14-10(2-1-7-22-14)17(11)24-19(26)16(15)21/h1-8H,21H2,(H,23,25)(H,24,26)	CVGSWRGEMHJVNE-UHFFFAOYSA-N	794860	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C83	Myelin transcription factor 1	Homo sapiens		 2.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794860	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794860&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293470	528826323							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126477	Nc1c(C2=CC=C(F)C3NN=CC23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H18FN5O/c23-16-6-5-11(15-9-26-28-21(15)16)17-14-8-13(10-3-4-10)19-12(2-1-7-25-19)20(14)27-22(29)18(17)24/h1-2,5-10,15,21,28H,3-4,24H2,(H,27,29)	BTIVOCRMOOPVQU-UHFFFAOYSA-N	794861	3-Amino-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one solvate::US20260062412, Compound C84	Myelin transcription factor 1	Homo sapiens		 2.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794861	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794861&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			178423166	528826324							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126478	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H14FN5O/c1-9-7-12-15(10-4-5-14(21)19-13(10)8-24-26-19)16(22)20(27)25-18(12)11-3-2-6-23-17(9)11/h2-8H,22H2,1H3,(H,24,26)(H,25,27)	JLHGHMDSERVGHA-UHFFFAOYSA-N	794862	3-Amino-4-(7-fluoro-1H-inadazol-4-yl)-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C85	Myelin transcription factor 1	Homo sapiens		 2.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794862	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794862&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293256	528826325							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126479	CCc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H16FN5O/c1-2-10-8-13-16(11-5-6-15(22)20-14(11)9-25-27-20)17(23)21(28)26-19(13)12-4-3-7-24-18(10)12/h3-9H,2,23H2,1H3,(H,25,27)(H,26,28)	QYLIZLBBMCBRMJ-UHFFFAOYSA-N	794863	3-Amino-6-ethyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C86	Myelin transcription factor 1	Homo sapiens		 4.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794863	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794863&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293665	528826326							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126480	N#Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H11FN6O/c21-14-4-3-10(13-8-25-27-19(13)14)15-12-6-9(7-22)17-11(2-1-5-24-17)18(12)26-20(28)16(15)23/h1-6,8H,23H2,(H,25,27)(H,26,28)	OYLMIDNPBXSSAE-UHFFFAOYSA-N	794864	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthroline-6-carbonitrile::US20260062412, Compound C87	Myelin transcription factor 1	Homo sapiens		 18.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794864	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794864&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293457	528826327							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126481	Cn1cc(-c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)cn1	InChI=1S/C23H16FN7O/c1-31-10-11(8-28-31)14-7-15-18(12-4-5-17(24)22-16(12)9-27-30-22)19(25)23(32)29-21(15)13-3-2-6-26-20(13)14/h2-10H,25H2,1H3,(H,27,30)(H,29,32)	ZJTGYVFOQIBZDZ-UHFFFAOYSA-N	794865	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-methylpyrazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C88	Myelin transcription factor 1	Homo sapiens		 4.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794865	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794865&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293932	528826328							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126482	C=Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H14FN5O/c1-2-10-8-13-16(11-5-6-15(22)20-14(11)9-25-27-20)17(23)21(28)26-19(13)12-4-3-7-24-18(10)12/h2-9H,1,23H2,(H,25,27)(H,26,28)	XSEPYVQLBUZJIO-UHFFFAOYSA-N	794866	3-Amino-6-ethenyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C89	Myelin transcription factor 1	Homo sapiens		 3.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794866	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794866&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293712	528826329							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126483	CC#Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H14FN5O/c1-2-4-11-9-14-17(12-6-7-16(23)21-15(12)10-26-28-21)18(24)22(29)27-20(14)13-5-3-8-25-19(11)13/h3,5-10H,24H2,1H3,(H,26,28)(H,27,29)	KEPIYZUVCGDMQA-UHFFFAOYSA-N	794867	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-prop-1-inyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C90	Myelin transcription factor 1	Homo sapiens		 14.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794867	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794867&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293405	528826330							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126484	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H18FN5O/c24-17-7-6-12(16-10-27-29-22(16)17)18-15-9-14(11-3-1-4-11)20-13(5-2-8-26-20)21(15)28-23(30)19(18)25/h2,5-11H,1,3-4,25H2,(H,27,29)(H,28,30)	IYIBINXWVNMQSD-UHFFFAOYSA-N	794868	3-Amino-6-cyclobutyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C91	Myelin transcription factor 1	Homo sapiens		 10.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794868	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794868&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293184	528826331							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126485	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20FN5O/c25-18-8-7-13(17-11-28-30-23(17)18)19-16-10-15(12-4-1-2-5-12)21-14(6-3-9-27-21)22(16)29-24(31)20(19)26/h3,6-12H,1-2,4-5,26H2,(H,28,30)(H,29,31)	MWAVRFFPFNYBKQ-UHFFFAOYSA-N	794869	3-Amino-6-cyclopentyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C92	Myelin transcription factor 1	Homo sapiens		 19.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794869	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794869&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293709	528826332							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126486	CN(C)C(=O)Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C23H19FN6O2/c1-30(2)17(31)9-11-8-14-18(12-5-6-16(24)22-15(12)10-27-29-22)19(25)23(32)28-21(14)13-4-3-7-26-20(11)13/h3-8,10H,9,25H2,1-2H3,(H,27,29)(H,28,32)	IZHLTROUVRDWHN-UHFFFAOYSA-N	794870	2-[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]-N,N-dimethylacetamide::US20260062412, Compound C93	Myelin transcription factor 1	Homo sapiens		 32.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794870	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794870&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293465	528826333							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126487	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3=COCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H16FN5O2/c24-17-4-3-12(16-9-27-29-22(16)17)18-15-8-14(11-5-7-31-10-11)20-13(2-1-6-26-20)21(15)28-23(30)19(18)25/h1-4,6,8-10H,5,7,25H2,(H,27,29)(H,28,30)	HALFHOGQTFBODD-UHFFFAOYSA-N	794871	3-Amino-6-(2,3-dihydrofuran-4-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C94	Myelin transcription factor 1	Homo sapiens		 8.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794871	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794871&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293166	528826334							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126488	N#CC1(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC1	InChI=1S/C23H15FN6O/c24-16-4-3-11(14-9-28-30-21(14)16)17-13-8-15(23(10-25)5-6-23)20-12(2-1-7-27-20)19(13)29-22(31)18(17)26/h1-4,7-9H,5-6,26H2,(H,28,30)(H,29,31)	JBMYLTRNBIBUFS-UHFFFAOYSA-N	794872	1-[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]cyclopropane-1-carbonitrile::US20260062412, Compound C95	Myelin transcription factor 1	Homo sapiens		 8.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794872	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794872&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293733	528826335							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126489	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCCO3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H18FN5O2/c24-16-6-5-11(15-10-27-29-22(15)16)18-14-9-13(17-4-2-8-31-17)20-12(3-1-7-26-20)21(14)28-23(30)19(18)25/h1,3,5-7,9-10,17H,2,4,8,25H2,(H,27,29)(H,28,30)	RRMAUIBKWPVUET-UHFFFAOYSA-N	794873	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(oxolan-2-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C96	Myelin transcription factor 1	Homo sapiens		 5.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794873	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794873&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293421	528826336							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126490	CC(C)(C)OC(=O)N1CC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)C1	InChI=1S/C27H25FN6O3/c1-27(2,3)37-26(36)34-11-13(12-34)16-9-17-20(14-6-7-19(28)24-18(14)10-31-33-24)21(29)25(35)32-23(17)15-5-4-8-30-22(15)16/h4-10,13H,11-12,29H2,1-3H3,(H,31,33)(H,32,35)	YERSSFQYAAYGQU-UHFFFAOYSA-N	794874	tert-Butyl 3-[3-amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]azetidine-1-carboxylate::US20260062412, Compound C97	Myelin transcription factor 1	Homo sapiens		 22.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794874	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794874&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293424	528826337							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126491	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCOCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20FN5O2/c25-18-4-3-13(17-11-28-30-23(17)18)19-16-10-15(12-5-8-32-9-6-12)21-14(2-1-7-27-21)22(16)29-24(31)20(19)26/h1-4,7,10-12H,5-6,8-9,26H2,(H,28,30)(H,29,31)	UEVYVEVCJPPKMX-UHFFFAOYSA-N	794875	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(oxan-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C98	Myelin transcription factor 1	Homo sapiens		 2.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794875	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794875&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293552	528826338							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126492	CC(C)(C)OC(=O)N1CCC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC1	InChI=1S/C29H29FN6O3/c1-29(2,3)39-28(38)36-11-8-15(9-12-36)18-13-19-22(16-6-7-21(30)26-20(16)14-33-35-26)23(31)27(37)34-25(19)17-5-4-10-32-24(17)18/h4-7,10,13-15H,8-9,11-12,31H2,1-3H3,(H,33,35)(H,34,37)	DBODRHQKYMAAFP-UHFFFAOYSA-N	794876	tert-Butyl 4-[3-amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]piperidine-1-carboxylate::US20260062412, Compound C99	Myelin transcription factor 1	Homo sapiens		 21.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794876	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794876&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293351	528826339							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126493	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(/C=C/CCO)c3ncccc3c2[nH]c1=O	InChI=1S/C23H18FN5O2/c24-17-7-6-13(16-11-27-29-22(16)17)18-15-10-12(4-1-2-9-30)20-14(5-3-8-26-20)21(15)28-23(31)19(18)25/h1,3-8,10-11,30H,2,9,25H2,(H,27,29)(H,28,31)	SBLFOWRRUBVDBB-UHFFFAOYSA-N	794877	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[(E)-4-hydroxybut-1-enyl]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C100	Myelin transcription factor 1	Homo sapiens		 1.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794877	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794877&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293275	528826340							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126494	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCC4(CC3)OCCO4)c3ncccc3c2[nH]c1=O	InChI=1S/C27H24FN5O3/c28-20-4-3-15(19-13-31-33-25(19)20)21-18-12-17(14-5-7-27(8-6-14)35-10-11-36-27)23-16(2-1-9-30-23)24(18)32-26(34)22(21)29/h1-4,9,12-14H,5-8,10-11,29H2,(H,31,33)(H,32,34)	XLQZDMCJBNNSKA-UHFFFAOYSA-N	794878	3-Amino-6-(1,4-dioxaspiro[4.5]decan-8-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one 2,2,2-trifluoroacetate::US20260062412, Compound C101	Myelin transcription factor 1	Homo sapiens		 6.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794878	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794878&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293685	528826341							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126495	CC(C)(O)C#Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C24H18FN5O2/c1-24(2,32)8-7-12-10-15-18(13-5-6-17(25)22-16(13)11-28-30-22)19(26)23(31)29-21(15)14-4-3-9-27-20(12)14/h3-6,9-11,32H,26H2,1-2H3,(H,28,30)(H,29,31)	JXGCFCCRLPERLA-UHFFFAOYSA-N	794879	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(3-hydroxy-3-methylbut-1-inyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C102	Myelin transcription factor 1	Homo sapiens		 3.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794879	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794879&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293718	528826342							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126496	C=C(C)c1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H16FN5O/c1-10(2)13-8-14-17(11-5-6-16(23)21-15(11)9-26-28-21)18(24)22(29)27-20(14)12-4-3-7-25-19(12)13/h3-9H,1,24H2,2H3,(H,26,28)(H,27,29)	IKQFQEXCLZUMSY-UHFFFAOYSA-N	794880	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-prop-1-en-2-yl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C103	Myelin transcription factor 1	Homo sapiens		 4.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794880	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794880&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293598	528826343							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126497	CC(C)c1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H18FN5O/c1-10(2)13-8-14-17(11-5-6-16(23)21-15(11)9-26-28-21)18(24)22(29)27-20(14)12-4-3-7-25-19(12)13/h3-10H,24H2,1-2H3,(H,26,28)(H,27,29)	CCOXGUWPHRPDMI-UHFFFAOYSA-N	794881	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-propan-2-yl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C104	Myelin transcription factor 1	Homo sapiens		 3.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794881	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794881&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293559	528826344							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126498	CC(C)Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C23H20FN5O/c1-11(2)8-12-9-15-18(13-5-6-17(24)22-16(13)10-27-29-22)19(25)23(30)28-21(15)14-4-3-7-26-20(12)14/h3-7,9-11H,8,25H2,1-2H3,(H,27,29)(H,28,30)	SWJSDOTZVNMVNO-UHFFFAOYSA-N	794882	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(2-methylpropyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C105	Myelin transcription factor 1	Homo sapiens		 5.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794882	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794882&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293580	528826345							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126499	CCCc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H18FN5O/c1-2-4-11-9-14-17(12-6-7-16(23)21-15(12)10-26-28-21)18(24)22(29)27-20(14)13-5-3-8-25-19(11)13/h3,5-10H,2,4,24H2,1H3,(H,26,28)(H,27,29)	HBJPIMIGQBXMQG-UHFFFAOYSA-N	794883	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-propyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C106	Myelin transcription factor 1	Homo sapiens		 2.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794883	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794883&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293529	528826346							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126500	CC(C)CCc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C24H22FN5O/c1-12(2)5-6-13-10-16-19(14-7-8-18(25)23-17(14)11-28-30-23)20(26)24(31)29-22(16)15-4-3-9-27-21(13)15/h3-4,7-12H,5-6,26H2,1-2H3,(H,28,30)(H,29,31)	FESIRFXMGSUNST-UHFFFAOYSA-N	794884	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(3-methylbutyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C107	Myelin transcription factor 1	Homo sapiens		 8.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794884	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794884&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293888	528826347							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126501	CCC(CC)c1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C24H22FN5O/c1-3-12(4-2)15-10-16-19(13-7-8-18(25)23-17(13)11-28-30-23)20(26)24(31)29-22(16)14-6-5-9-27-21(14)15/h5-12H,3-4,26H2,1-2H3,(H,28,30)(H,29,31)	CQJVQDWFIACMQC-UHFFFAOYSA-N	794885	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-pentan-3-yl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C108	Myelin transcription factor 1	Homo sapiens		 37.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794885	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794885&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293700	528826348							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126502	CCC(C)c1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C23H20FN5O/c1-3-11(2)14-9-15-18(12-6-7-17(24)22-16(12)10-27-29-22)19(25)23(30)28-21(15)13-5-4-8-26-20(13)14/h4-11H,3,25H2,1-2H3,(H,27,29)(H,28,30)	YAXVWRGRDWRVFG-UHFFFAOYSA-N	794886	3-Amino-6-butan-2-yl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C109	Myelin transcription factor 1	Homo sapiens		 4.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794886	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794886&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293707	528826349							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126503	CP(C)(=O)c1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H17FN5O2P/c1-30(2,29)15-8-12-16(10-5-6-14(22)19-13(10)9-25-27-19)17(23)21(28)26-18(12)11-4-3-7-24-20(11)15/h3-9H,23H2,1-2H3,(H,25,27)(H,26,28)	LKSGPHZHMJHMEI-UHFFFAOYSA-N	794887	3-Amino-6-dimethylphosphoryl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C110	Myelin transcription factor 1	Homo sapiens		 14.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794887	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794887&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293601	528826350							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126504	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(I)c3ncccc3c2[nH]c1=O	InChI=1S/C19H11FIN5O/c20-12-4-3-8(11-7-24-26-17(11)12)14-10-6-13(21)18-9(2-1-5-23-18)16(10)25-19(27)15(14)22/h1-7H,22H2,(H,24,26)(H,25,27)	NHERPMQKEFJMGI-UHFFFAOYSA-N	794888	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-iodo-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C111	Myelin transcription factor 1	Homo sapiens		 4.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794888	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794888&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293201	528826351							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126505	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCCC3=O)c3ncccc3c2[nH]c1=O	InChI=1S/C23H17FN6O2/c24-15-6-5-11(14-10-27-29-21(14)15)18-13-9-16(30-8-2-4-17(30)31)22-12(3-1-7-26-22)20(13)28-23(32)19(18)25/h1,3,5-7,9-10H,2,4,8,25H2,(H,27,29)(H,28,32)	UUVFHXRZUFMDSL-UHFFFAOYSA-N	794889	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(2-oxopyrrolidin-1-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C112	Myelin transcription factor 1	Homo sapiens		 78.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794889	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794889&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293258	528826352							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126506	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H19FN6O/c24-16-6-5-12(15-11-27-29-21(15)16)18-14-10-17(30-8-1-2-9-30)22-13(4-3-7-26-22)20(14)28-23(31)19(18)25/h3-7,10-11H,1-2,8-9,25H2,(H,27,29)(H,28,31)	PKLLYYHGBDELCN-UHFFFAOYSA-N	794890	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-pyrrolidin-1-yl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C113	Myelin transcription factor 1	Homo sapiens		 4.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794890	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794890&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293717	528826353							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126507	CN1CCN(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC1	InChI=1S/C24H22FN7O/c1-31-7-9-32(10-8-31)18-11-15-19(13-4-5-17(25)22-16(13)12-28-30-22)20(26)24(33)29-21(15)14-3-2-6-27-23(14)18/h2-6,11-12H,7-10,26H2,1H3,(H,28,30)(H,29,33)	NMCJOGBRUXNSCK-UHFFFAOYSA-N	794891	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(4-methylpiperazin-1-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C114	Myelin transcription factor 1	Homo sapiens		 2.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794891	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794891&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293306	528826354							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126508	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCC(F)(F)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H17F3N6O/c24-15-4-3-11(14-9-29-31-20(14)15)17-13-8-16(32-7-5-23(25,26)10-32)21-12(2-1-6-28-21)19(13)30-22(33)18(17)27/h1-4,6,8-9H,5,7,10,27H2,(H,29,31)(H,30,33)	PATQVGVLEUHJDF-UHFFFAOYSA-N	794892	3-Amino-6-(3,3-difluoropyrrolidin-1-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C115	Myelin transcription factor 1	Homo sapiens		 3.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794892	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794892&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293298	528826355							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126509	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCC(O)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H19FN6O2/c24-16-4-3-12(15-9-27-29-21(15)16)18-14-8-17(30-7-5-11(31)10-30)22-13(2-1-6-26-22)20(14)28-23(32)19(18)25/h1-4,6,8-9,11,31H,5,7,10,25H2,(H,27,29)(H,28,32)	MSWYRCAKZJAEPK-UHFFFAOYSA-N	794893	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(3-hydroxypyrrolidin-1-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C116	Myelin transcription factor 1	Homo sapiens		 2.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794893	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794893&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293563	528826356							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126510	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCC(N4CCOCC4)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C28H28FN7O2/c29-21-4-3-17(20-15-32-34-26(20)21)23-19-14-22(36-8-5-16(6-9-36)35-10-12-38-13-11-35)27-18(2-1-7-31-27)25(19)33-28(37)24(23)30/h1-4,7,14-16H,5-6,8-13,30H2,(H,32,34)(H,33,37)	JYBOTYRDCBQIOG-UHFFFAOYSA-N	794894	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(4-morpholin-4-ylpiperidin-1-yl)-1H-1,7-one::US20260062412, Compound C117	Myelin transcription factor 1	Homo sapiens		 3.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794894	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794894&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293739	528826357							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126511	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CC4(COC4)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H19FN6O2/c25-16-4-3-12(15-7-28-30-21(15)16)18-14-6-17(31-8-24(9-31)10-33-11-24)22-13(2-1-5-27-22)20(14)29-23(32)19(18)26/h1-7H,8-11,26H2,(H,28,30)(H,29,32)	ZVKYKKQDXLQUQH-UHFFFAOYSA-N	794895	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(2-oxa-6-azaspiro[3,3]heptan-6-yl)-1H-1,7-one::US20260062412, Compound C118	Myelin transcription factor 1	Homo sapiens		 2.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794895	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794895&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293532	528826358							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126512	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCC(N4CCCC4)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C28H28FN7O/c29-21-6-5-17(20-15-32-34-26(20)21)23-19-14-22(36-12-7-16(8-13-36)35-10-1-2-11-35)27-18(4-3-9-31-27)25(19)33-28(37)24(23)30/h3-6,9,14-16H,1-2,7-8,10-13,30H2,(H,32,34)(H,33,37)	ATMVINRFAAGOQY-UHFFFAOYSA-N	794896	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(4-pyrrolidin-1-ylpiperidin-1-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C119	Myelin transcription factor 1	Homo sapiens		 2.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794896	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794896&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293803	528826359							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126513	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCC4(COC4)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C25H21FN6O2/c26-17-4-3-13(16-9-29-31-22(16)17)19-15-8-18(32-7-5-25(10-32)11-34-12-25)23-14(2-1-6-28-23)21(15)30-24(33)20(19)27/h1-4,6,8-9H,5,7,10-12,27H2,(H,29,31)(H,30,33)	RPKNXURRIUFQNE-UHFFFAOYSA-N	794897	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(2-oxa-7-azaspiro[3.4]octan-7-yl)-1H-1,7-one::US20260062412, Compound C120	Myelin transcription factor 1	Homo sapiens		 2.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794897	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794897&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293714	528826360							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126514	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H17FN6O/c23-15-5-4-11(14-10-26-28-20(14)15)17-13-9-16(29-7-2-8-29)21-12(3-1-6-25-21)19(13)27-22(30)18(17)24/h1,3-6,9-10H,2,7-8,24H2,(H,26,28)(H,27,30)	FNYUNBPHLSMYDX-UHFFFAOYSA-N	794898	3-Amino-6-(azetidin-1-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C121	Myelin transcription factor 1	Homo sapiens		 3.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794898	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794898&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293175	528826361							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126515	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCOCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H19FN6O2/c24-16-4-3-12(15-11-27-29-21(15)16)18-14-10-17(30-6-8-32-9-7-30)22-13(2-1-5-26-22)20(14)28-23(31)19(18)25/h1-5,10-11H,6-9,25H2,(H,27,29)(H,28,31)	DRECSFOVGPRWKE-UHFFFAOYSA-N	794899	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-morpholin-4-yl-1H-1,7-phenanthrolin-2-one 2,2,2-trifluoroacetate::US20260062412, Compound C122	Myelin transcription factor 1	Homo sapiens		 4.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794899	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794899&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293147	528826362							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126516	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CC(F)(F)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H15F3N6O/c23-14-4-3-10(13-7-28-30-19(13)14)16-12-6-15(31-8-22(24,25)9-31)20-11(2-1-5-27-20)18(12)29-21(32)17(16)26/h1-7H,8-9,26H2,(H,28,30)(H,29,32)	FRBDIZWRANOAQW-UHFFFAOYSA-N	794900	3-Amino-6-(3,3-difluoroazetidin-1-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C123	Myelin transcription factor 1	Homo sapiens		 3.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794900	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794900&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293696	528826363							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126517	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCS(=O)(=O)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H19FN6O3S/c24-16-4-3-12(15-11-27-29-21(15)16)18-14-10-17(30-6-8-34(32,33)9-7-30)22-13(2-1-5-26-22)20(14)28-23(31)19(18)25/h1-5,10-11H,6-9,25H2,(H,27,29)(H,28,31)	TZQCYVINVQUEQQ-UHFFFAOYSA-N	794901	3-Amino-6-(1,1-dioxo-1,4-thiazinan-4-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C124	Myelin transcription factor 1	Homo sapiens		 3.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794901	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794901&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293157	528826364							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126518	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCCCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H21FN6O/c25-17-7-6-13(16-12-28-30-22(16)17)19-15-11-18(31-9-2-1-3-10-31)23-14(5-4-8-27-23)21(15)29-24(32)20(19)26/h4-8,11-12H,1-3,9-10,26H2,(H,28,30)(H,29,32)	ACYAGUYRLMZUSJ-UHFFFAOYSA-N	794902	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-piperidin-1-yl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C125	Myelin transcription factor 1	Homo sapiens		 5.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794902	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794902&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293204	528826365							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126519	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCC(F)(F)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H19F3N6O/c25-16-4-3-12(15-11-30-32-21(15)16)18-14-10-17(33-8-5-24(26,27)6-9-33)22-13(2-1-7-29-22)20(14)31-23(34)19(18)28/h1-4,7,10-11H,5-6,8-9,28H2,(H,30,32)(H,31,34)	SCMOJPFBUSMOFR-UHFFFAOYSA-N	794903	3-Amino-6-(4,4-difluoropiperidin-1-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C126	Myelin transcription factor 1	Homo sapiens		 4.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794903	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794903&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293211	528826366							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126520	CS(=O)(=O)Nc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H15FN6O3S/c1-31(29,30)27-14-7-11-15(9-4-5-13(21)18-12(9)8-24-26-18)16(22)20(28)25-17(11)10-3-2-6-23-19(10)14/h2-8,27H,22H2,1H3,(H,24,26)(H,25,28)	SUJCARYUCNJZFO-UHFFFAOYSA-N	794904	N-[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]methanesulfonamide::US20260062412, Compound C127	Myelin transcription factor 1	Homo sapiens		 1.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794904	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794904&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293747	528826367							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126521	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CC4CC(C3)O4)c3ncccc3c2[nH]c1=O	InChI=1S/C24H19FN6O2/c25-17-4-3-13(16-8-28-30-22(16)17)19-15-7-18(31-9-11-6-12(10-31)33-11)23-14(2-1-5-27-23)21(15)29-24(32)20(19)26/h1-5,7-8,11-12H,6,9-10,26H2,(H,28,30)(H,29,32)	QKBINLQNRSARRQ-UHFFFAOYSA-N	794905	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(6-oxa-3-azabicyclo[3.1.1]heptan-3-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C128	Myelin transcription factor 1	Homo sapiens		 5.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794905	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794905&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293462	528826368							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126522	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3C4COCC3C4)c3ncccc3c2[nH]c1=O	InChI=1S/C24H19FN6O2/c25-17-4-3-13(16-8-28-30-22(16)17)19-15-7-18(31-11-6-12(31)10-33-9-11)23-14(2-1-5-27-23)21(15)29-24(32)20(19)26/h1-5,7-8,11-12H,6,9-10,26H2,(H,28,30)(H,29,32)	ANJVZCWNWSXOMR-UHFFFAOYSA-N	794906	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(3-oxa-6-azabicyclo[3.1.1]heptan-6-yl)-1H-1,7-one::US20260062412, Compound C129	Myelin transcription factor 1	Homo sapiens		 3.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794906	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794906&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293518	528826369							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126523	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(NS(=O)(=O)C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H17FN6O3S/c23-15-6-5-11(14-9-26-28-20(14)15)17-13-8-16(29-33(31,32)10-3-4-10)21-12(2-1-7-25-21)19(13)27-22(30)18(17)24/h1-2,5-10,29H,3-4,24H2,(H,26,28)(H,27,30)	MSDFPABFKQDBOL-UHFFFAOYSA-N	794907	N-[3-amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]cyclopropanesulfonamide::US20260062412, Compound C130	Myelin transcription factor 1	Homo sapiens		 3.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794907	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794907&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293670	528826370							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126524	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCN(C(F)(F)F)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H19F4N7O/c25-16-4-3-12(15-11-31-33-21(15)16)18-14-10-17(34-6-8-35(9-7-34)24(26,27)28)22-13(2-1-5-30-22)20(14)32-23(36)19(18)29/h1-5,10-11H,6-9,29H2,(H,31,33)(H,32,36)	LOIFXYSKIOAGPG-UHFFFAOYSA-N	794908	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[4-(trifluoromethyl) piperidin-1-yl]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C131	Myelin transcription factor 1	Homo sapiens		 33.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794908	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794908&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			178423167	528826371							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126525	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CNC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H17FN6O/c23-16-4-3-11(15-9-27-29-21(15)16)17-14-6-13(10-7-25-8-10)19-12(2-1-5-26-19)20(14)28-22(30)18(17)24/h1-6,9-10,25H,7-8,24H2,(H,27,29)(H,28,30)	IPHKDALKECPAKS-UHFFFAOYSA-N	794909	3-Amino-6-(azetidin-3-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one; formate::US20260062412, Compound C132	Myelin transcription factor 1	Homo sapiens		 11.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794909	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794909&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293692	528826372							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126526	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCNCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H21FN6O/c25-18-4-3-13(17-11-29-31-23(17)18)19-16-10-15(12-5-8-27-9-6-12)21-14(2-1-7-28-21)22(16)30-24(32)20(19)26/h1-4,7,10-12,27H,5-6,8-9,26H2,(H,29,31)(H,30,32)	JXDKWQCCEWQQKU-UHFFFAOYSA-N	794910	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-piperidin-4-yl-1H-1,7-phenanthrolin-2-one; hydrochloride::US20260062412, Compound C133	Myelin transcription factor 1	Homo sapiens		 1.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794910	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794910&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293618	528826373							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126527	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCN(C4CCC4)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C28H27FN6O/c29-22-7-6-17(21-14-32-34-27(21)22)23-20-13-19(15-8-11-35(12-9-15)16-3-1-4-16)25-18(5-2-10-31-25)26(20)33-28(36)24(23)30/h2,5-7,10,13-16H,1,3-4,8-9,11-12,30H2,(H,32,34)(H,33,36)	VWTRXZWWARKGDY-UHFFFAOYSA-N	794911	3-Amino-6-(1-cyclobutylpiperidin-4-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C134	Myelin transcription factor 1	Homo sapiens		 3.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794911	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794911&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293261	528826374							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126528	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCN(C4COC4)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C27H25FN6O2/c28-21-4-3-16(20-11-31-33-26(20)21)22-19-10-18(14-5-8-34(9-6-14)15-12-36-13-15)24-17(2-1-7-30-24)25(19)32-27(35)23(22)29/h1-4,7,10-11,14-15H,5-6,8-9,12-13,29H2,(H,31,33)(H,32,35)	PHEOLMVLSIREMF-UHFFFAOYSA-N	794912	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[1-(oxetan-3-yl) piperidin-4-yl]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C135	Myelin transcription factor 1	Homo sapiens		 2.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794912	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794912&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293369	528826375							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126529	CC(C)N1CCC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC1	InChI=1S/C27H27FN6O/c1-14(2)34-10-7-15(8-11-34)18-12-19-22(16-5-6-21(28)26-20(16)13-31-33-26)23(29)27(35)32-25(19)17-4-3-9-30-24(17)18/h3-6,9,12-15H,7-8,10-11,29H2,1-2H3,(H,31,33)(H,32,35)	MTFMIKRWXSZUTI-UHFFFAOYSA-N	794913	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-propan-2-ylpiperidin-4-yl)-1H-1,7-phenanthrolin-2-one; formate::US20260062412, Compound C136	Myelin transcription factor 1	Homo sapiens		 3.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794913	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794913&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293435	528826376							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126530	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCN(C4CCOCC4)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C29H29FN6O2/c30-23-4-3-18(22-15-33-35-28(22)23)24-21-14-20(16-5-10-36(11-6-16)17-7-12-38-13-8-17)26-19(2-1-9-32-26)27(21)34-29(37)25(24)31/h1-4,9,14-17H,5-8,10-13,31H2,(H,33,35)(H,34,37)	KPWJXXMETFKFFG-UHFFFAOYSA-N	794914	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[1-(oxan-4-yl) piperidin-4-yl]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C137	Myelin transcription factor 1	Homo sapiens		 4.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794914	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794914&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293507	528826377							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126531	CN1CCC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC1	InChI=1S/C25H23FN6O/c1-32-9-6-13(7-10-32)16-11-17-20(14-4-5-19(26)24-18(14)12-29-31-24)21(27)25(33)30-23(17)15-3-2-8-28-22(15)16/h2-5,8,11-13H,6-7,9-10,27H2,1H3,(H,29,31)(H,30,33)	JHZHSGNLORZFDL-UHFFFAOYSA-N	794915	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-methylpiperidin-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C138	Myelin transcription factor 1	Homo sapiens		 2.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794915	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794915&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293171	528826378							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126532	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCC(=O)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C25H20FN5O2/c26-19-8-7-14(18-11-29-31-24(18)19)20-17-10-16(12-3-5-13(32)6-4-12)22-15(2-1-9-28-22)23(17)30-25(33)21(20)27/h1-2,7-12H,3-6,27H2,(H,29,31)(H,30,33)	BFOJFEOOVMACAM-UHFFFAOYSA-N	794916	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(4-oxocyclohexyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C139	Myelin transcription factor 1	Homo sapiens		 3.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794916	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794916&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293880	528826379							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126533	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc([C@H]3CC[C@H](O)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C25H22FN5O2/c26-19-8-7-14(18-11-29-31-24(18)19)20-17-10-16(12-3-5-13(32)6-4-12)22-15(2-1-9-28-22)23(17)30-25(33)21(20)27/h1-2,7-13,32H,3-6,27H2,(H,29,31)(H,30,33)	ZTDZYEUDHPMYPI-UHFFFAOYSA-N	794917	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-((1r, 4r)-4-hydroxycyclohexyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C140	Myelin transcription factor 1	Homo sapiens		 1.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794917	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794917&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			176112735	528826380							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126534	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc([C@H]3CC[C@@H](O)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C25H22FN5O2/c26-19-8-7-14(18-11-29-31-24(18)19)20-17-10-16(12-3-5-13(32)6-4-12)22-15(2-1-9-28-22)23(17)30-25(33)21(20)27/h1-2,7-13,32H,3-6,27H2,(H,29,31)(H,30,33)	ZTDZYEUDHPMYPI-UHFFFAOYSA-N	794918	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-((1s, 4s)-4-hydroxycyclohexyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C141	Myelin transcription factor 1	Homo sapiens		 4.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794918	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794918&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			176112735	528826381							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126535	CC1(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC1	InChI=1S/C23H18FN5O/c1-23(6-7-23)15-9-13-17(11-4-5-16(24)21-14(11)10-27-29-21)18(25)22(30)28-19(13)12-3-2-8-26-20(12)15/h2-5,8-10H,6-7,25H2,1H3,(H,27,29)(H,28,30)	QALJEILAITWSSD-UHFFFAOYSA-N	794919	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-methylcyclopropyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C142	Myelin transcription factor 1	Homo sapiens		 18.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794919	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794919&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293484	528826382							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126536	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H16ClN5O/c23-16-6-5-11(15-9-26-28-21(15)16)17-14-8-13(10-3-4-10)19-12(2-1-7-25-19)20(14)27-22(29)18(17)24/h1-2,5-10H,3-4,24H2,(H,26,28)(H,27,29)	CULBTRFDPALKTG-UHFFFAOYSA-N	794920	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-cyclopropyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C143	Myelin transcription factor 1	Homo sapiens		 2.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794920	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794920&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293414	528826383							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126537	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2ccc3ncccc3c2[nH]c1=O	InChI=1S/C19H12ClN5O/c20-13-5-3-9(12-8-23-25-18(12)13)15-11-4-6-14-10(2-1-7-22-14)17(11)24-19(26)16(15)21/h1-8H,21H2,(H,23,25)(H,24,26)	VICZQFFWCKFLGI-UHFFFAOYSA-N	794921	3-Amino-4-(7-chloro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C144	Myelin transcription factor 1	Homo sapiens		 7.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794921	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794921&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293864	528826384							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126538	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C22H14F3N5O/c23-15-4-3-9(13-8-28-30-20(13)15)16-12-6-11(14-7-22(14,24)25)18-10(2-1-5-27-18)19(12)29-21(31)17(16)26/h1-6,8,14H,7,26H2,(H,28,30)(H,29,31)	WYOKELCARWSKQM-UHFFFAOYSA-N	794922	3-Amino-6-(2,2-difluorocyclopropyl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C145	Myelin transcription factor 1	Homo sapiens		 3.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794922	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794922&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293321	528826385							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126539	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCNC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H19FN6O/c24-17-4-3-12(16-10-28-30-22(16)17)18-15-8-14(11-5-7-26-9-11)20-13(2-1-6-27-20)21(15)29-23(31)19(18)25/h1-4,6,8,10-11,26H,5,7,9,25H2,(H,28,30)(H,29,31)	ASKXOJLWFWUBQH-UHFFFAOYSA-N	794923	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-pyrrolidin-3-yl-1H-1,7-phenanthrolin-2-one; formate::US20260062412, Compound C146	Myelin transcription factor 1	Homo sapiens		 3.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794923	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794923&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293340	528826386							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126540	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C3CCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H18ClN5O/c24-17-7-6-12(16-10-27-29-22(16)17)18-15-9-14(11-3-1-4-11)20-13(5-2-8-26-20)21(15)28-23(30)19(18)25/h2,5-11H,1,3-4,25H2,(H,27,29)(H,28,30)	RDSFUWNQKSEQKM-UHFFFAOYSA-N	794924	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-cyclobutyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C147	Myelin transcription factor 1	Homo sapiens		 5.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794924	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794924&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293483	528826387							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126541	N#Cc1cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H11ClN6O/c21-14-4-3-10(13-8-25-27-19(13)14)15-12-6-9(7-22)17-11(2-1-5-24-17)18(12)26-20(28)16(15)23/h1-6,8H,23H2,(H,25,27)(H,26,28)	AJHMLDBTXHCZBE-UHFFFAOYSA-N	794925	3-Amino-4-(7-chloro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthroline-6-carbonitrile::US20260062412, Compound C148	Myelin transcription factor 1	Homo sapiens		 4.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794925	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794925&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293342	528826388							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126542	N#Cc1cc2c(-c3ccc(C#N)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H11N7O/c22-7-10-3-4-12(15-9-26-28-19(10)15)16-14-6-11(8-23)18-13(2-1-5-25-18)20(14)27-21(29)17(16)24/h1-6,9H,24H2,(H,26,28)(H,27,29)	JHHALFDXAUAVHT-UHFFFAOYSA-N	794926	3-Amino-4-(7-cyano-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthroline-6-carbonitrile::US20260062412, Compound C149	Myelin transcription factor 1	Homo sapiens		 380							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794926	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794926&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293773	528826389							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126543	CCc1cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H16ClN5O/c1-2-10-8-13-16(11-5-6-15(22)20-14(11)9-25-27-20)17(23)21(28)26-19(13)12-4-3-7-24-18(10)12/h3-9H,2,23H2,1H3,(H,25,27)(H,26,28)	MAQGUZXVPSPIDB-UHFFFAOYSA-N	794927	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-ethyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C150	Myelin transcription factor 1	Homo sapiens		 1.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794927	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794927&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293315	528826390							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126544	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C3CCCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20ClN5O/c25-18-8-7-13(17-11-28-30-23(17)18)19-16-10-15(12-4-1-2-5-12)21-14(6-3-9-27-21)22(16)29-24(31)20(19)26/h3,6-12H,1-2,4-5,26H2,(H,28,30)(H,29,31)	WIGGCHWDROKEBZ-UHFFFAOYSA-N	794928	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-cyclopentyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C151	Myelin transcription factor 1	Homo sapiens		 10.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794928	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794928&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293142	528826391							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126545	Cc1cc2c(-c3ccc(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H14ClN5O/c1-9-7-12-15(10-4-5-14(21)19-13(10)8-24-26-19)16(22)20(27)25-18(12)11-3-2-6-23-17(9)11/h2-8H,22H2,1H3,(H,24,26)(H,25,27)	VYALUQWZZAXGTE-UHFFFAOYSA-N	794929	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C152	Myelin transcription factor 1	Homo sapiens		 4.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794929	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794929&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293562	528826392							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126546	Cc1cc2c(-c3ccc(C)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H17N5O/c1-10-5-6-12(15-9-24-26-19(10)15)16-14-8-11(2)18-13(4-3-7-23-18)20(14)25-21(27)17(16)22/h3-9H,22H2,1-2H3,(H,24,26)(H,25,27)	HXMKSJWILDFESP-UHFFFAOYSA-N	794930	3-Amino-6-methyl-4-(7-methyl-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C153	Myelin transcription factor 1	Homo sapiens		 4.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794930	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794930&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293180	528826393							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126547	Nc1c(-c2c(F)ccc3[nH]ncc23)c2cc(Br)c3ncccc3c2[nH]c1=O	InChI=1S/C19H11BrFN5O/c20-11-6-9-15(14-10-7-24-26-13(10)4-3-12(14)21)16(22)19(27)25-17(9)8-2-1-5-23-18(8)11/h1-7H,22H2,(H,24,26)(H,25,27)	HPWJCKCKCWKLMN-UHFFFAOYSA-N	794931	3-Amino-6-bromo-4-(5-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C154	Myelin transcription factor 1	Homo sapiens		 3.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794931	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794931&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293603	528826394							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126548	Cc1cc2c(-c3c(F)ccc4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H14FN5O/c1-9-7-11-16(15-12-8-24-26-14(12)5-4-13(15)21)17(22)20(27)25-19(11)10-3-2-6-23-18(9)10/h2-8H,22H2,1H3,(H,24,26)(H,25,27)	CEJSSNRTXYXSRE-UHFFFAOYSA-N	794932	3-Amino-4-(5-fluoro-1H-indazol-4-yl)-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C155	Myelin transcription factor 1	Homo sapiens		 2.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794932	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794932&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293247	528826395							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126549	Nc1c(-c2c(F)ccc3[nH]ncc23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H16FN5O/c23-15-5-6-16-14(9-26-28-16)17(15)18-13-8-12(10-3-4-10)20-11(2-1-7-25-20)21(13)27-22(29)19(18)24/h1-2,5-10H,3-4,24H2,(H,26,28)(H,27,29)	PEYWJOJLYYNZDL-UHFFFAOYSA-N	794933	3-Amino-6-cyclopropyl-4-(5-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one (racemate)::US20260062412, Compound C156	Myelin transcription factor 1	Homo sapiens		 2.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794933	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794933&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293776	528826396							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
126550	Nc1c(-c2c(F)ccc3[nH]ncc23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H16FN5O/c23-15-5-6-16-14(9-26-28-16)17(15)18-13-8-12(10-3-4-10)20-11(2-1-7-25-20)21(13)27-22(29)19(18)24/h1-2,5-10H,3-4,24H2,(H,26,28)(H,27,29)	PEYWJOJLYYNZDL-UHFFFAOYSA-N	794934	(R)-3-amino-6-cyclopropyl-4-(5-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C157	Myelin transcription factor 1	Homo sapiens		 310							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794934	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794934&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293776	528826397							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237483	Nc1c(-c2c(F)ccc3[nH]ncc23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H16FN5O/c23-15-5-6-16-14(9-26-28-16)17(15)18-13-8-12(10-3-4-10)20-11(2-1-7-25-20)21(13)27-22(29)19(18)24/h1-2,5-10H,3-4,24H2,(H,26,28)(H,27,29)	PEYWJOJLYYNZDL-UHFFFAOYSA-N	794935	(S)-3-amino-6-cyclopropyl-4-(5-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C158	Myelin transcription factor 1	Homo sapiens		 1.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794935	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794935&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293776	528826398							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237484	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCOC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H18FN5O2/c24-17-4-3-12(16-9-27-29-22(16)17)18-15-8-14(11-5-7-31-10-11)20-13(2-1-6-26-20)21(15)28-23(30)19(18)25/h1-4,6,8-9,11H,5,7,10,25H2,(H,27,29)(H,28,30)	QIJWPVRHTUPDLM-UHFFFAOYSA-N	794936	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(oxolan-3-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C159	Myelin transcription factor 1	Homo sapiens		 2.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794936	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794936&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293762	528826399							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237485	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(CCCF)c3ncccc3c2[nH]c1=O	InChI=1S/C22H17F2N5O/c23-7-1-3-11-9-14-17(12-5-6-16(24)21-15(12)10-27-29-21)18(25)22(30)28-20(14)13-4-2-8-26-19(11)13/h2,4-6,8-10H,1,3,7,25H2,(H,27,29)(H,28,30)	SVFSGXMKXKKQII-UHFFFAOYSA-N	794937	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(3-fluoropropyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C160	Myelin transcription factor 1	Homo sapiens		 2.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794937	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794937&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293645	528826400							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237486	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(CCC(F)(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C22H15F4N5O/c23-15-4-3-11(14-9-29-31-20(14)15)16-13-8-10(5-6-22(24,25)26)18-12(2-1-7-28-18)19(13)30-21(32)17(16)27/h1-4,7-9H,5-6,27H2,(H,29,31)(H,30,32)	FTMBARDTVTVMOU-UHFFFAOYSA-N	794938	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(3,3,3-trifluoropropyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C161	Myelin transcription factor 1	Homo sapiens		 8.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794938	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794938&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293631	528826401							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237487	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCC(F)(F)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H18F3N5O/c25-17-4-3-12(16-10-30-32-22(16)17)18-15-8-14(11-5-6-24(26,27)9-11)20-13(2-1-7-29-20)21(15)31-23(33)19(18)28/h1-4,7-8,10-11H,5-6,9,28H2,(H,30,32)(H,31,33)	WNGHOOHHBDAQOQ-UHFFFAOYSA-N	794939	3-Amino-6-(3,3-difluorocyclopentyl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C162	Myelin transcription factor 1	Homo sapiens		 12.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794939	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794939&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293446	528826402							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237488	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCC(F)(F)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C25H20F3N5O/c26-18-4-3-13(17-11-31-33-23(17)18)19-16-10-15(12-5-7-25(27,28)8-6-12)21-14(2-1-9-30-21)22(16)32-24(34)20(19)29/h1-4,9-12H,5-8,29H2,(H,31,33)(H,32,34)	AJYQKUPPMNVCPZ-UHFFFAOYSA-N	794940	3-Amino-6-(4,4-difluorocyclohexyl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C163	Myelin transcription factor 1	Homo sapiens		 24.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794940	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794940&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293860	528826403							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237489	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC(F)(F)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H16F3N5O/c24-16-4-3-11(15-9-29-31-21(15)16)17-14-6-13(10-7-23(25,26)8-10)19-12(2-1-5-28-19)20(14)30-22(32)18(17)27/h1-6,9-10H,7-8,27H2,(H,29,31)(H,30,32)	BOTSEWVNGZQLHE-UHFFFAOYSA-N	794941	3-Amino-6-(3,3-difluorocyclobutyl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C164	Myelin transcription factor 1	Homo sapiens		 8.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794941	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794941&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293531	528826404							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237490	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(CC(F)(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C21H13F4N5O/c22-14-4-3-10(13-8-28-30-19(13)14)15-12-6-9(7-21(23,24)25)17-11(2-1-5-27-17)18(12)29-20(31)16(15)26/h1-6,8H,7,26H2,(H,28,30)(H,29,31)	SFSVMXXBJRGNJF-UHFFFAOYSA-N	794942	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(2,2,2-trifluoroethyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C165	Myelin transcription factor 1	Homo sapiens		 7.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794942	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794942&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293131	528826405							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237491	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC4(C3)CC(F)(F)C4)c3ncccc3c2[nH]c1=O	InChI=1S/C26H20F3N5O/c27-18-4-3-13(17-9-32-34-23(17)18)19-16-6-15(12-7-25(8-12)10-26(28,29)11-25)21-14(2-1-5-31-21)22(16)33-24(35)20(19)30/h1-6,9,12H,7-8,10-11,30H2,(H,32,34)(H,33,35)	WCFLAHRVWNXLDS-UHFFFAOYSA-N	794943	3-Amino-6-(2,2-difluorospiro[3,3]heptan-6-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C166	Myelin transcription factor 1	Homo sapiens		 2.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794943	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794943&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293417	528826406							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237492	CC1(C)CC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)C1	InChI=1S/C25H22FN5O/c1-25(2)9-12(10-25)15-8-16-19(13-5-6-18(26)23-17(13)11-29-31-23)20(27)24(32)30-22(16)14-4-3-7-28-21(14)15/h3-8,11-12H,9-10,27H2,1-2H3,(H,29,31)(H,30,32)	UNQQRQAAKAJPEP-UHFFFAOYSA-N	794944	3-Amino-6-(3,3-dimethylcyclobutyl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C167	Myelin transcription factor 1	Homo sapiens		 46.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794944	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794944&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293753	528826407							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237493	CC(c1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12)C(F)(F)F	InChI=1S/C22H15F4N5O/c1-9(22(24,25)26)12-7-13-16(10-4-5-15(23)20-14(10)8-29-31-20)17(27)21(32)30-19(13)11-3-2-6-28-18(11)12/h2-9H,27H2,1H3,(H,29,31)(H,30,32)	LYKOGNYBXYXDGI-UHFFFAOYSA-N	794945	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1,1,1-trifluoropropan-2-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C168	Myelin transcription factor 1	Homo sapiens		 54.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794945	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794945&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293481	528826408							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237494	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC4(CCC4)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C26H22FN5O/c27-19-5-4-14(18-12-30-32-24(18)19)20-17-9-16(13-10-26(11-13)6-2-7-26)22-15(3-1-8-29-22)23(17)31-25(33)21(20)28/h1,3-5,8-9,12-13H,2,6-7,10-11,28H2,(H,30,32)(H,31,33)	XMDNUDHKYNTRJS-UHFFFAOYSA-N	794946	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-spiro[3,3]heptan-2-yl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C169	Myelin transcription factor 1	Homo sapiens		 86.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794946	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794946&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293820	528826409							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237495	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(CC(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C21H14F3N5O/c22-14-4-3-10(13-8-27-29-20(13)14)16-12-6-9(7-15(23)24)18-11(2-1-5-26-18)19(12)28-21(30)17(16)25/h1-6,8,15H,7,25H2,(H,27,29)(H,28,30)	XKWOJPMEKNCZIV-UHFFFAOYSA-N	794947	3-Amino-6-(2,2-difluoroethyl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C170	Myelin transcription factor 1	Homo sapiens		 3.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794947	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794947&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293246	528826410							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237496	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(CCC(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C22H16F3N5O/c23-15-5-4-11(14-9-28-30-21(14)15)17-13-8-10(3-6-16(24)25)19-12(2-1-7-27-19)20(13)29-22(31)18(17)26/h1-2,4-5,7-9,16H,3,6,26H2,(H,28,30)(H,29,31)	KAELLXMNVIFLOS-UHFFFAOYSA-N	794948	3-Amino-6-(3,3-difluoropropyl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C171	Myelin transcription factor 1	Homo sapiens		 2.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794948	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794948&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293344	528826411							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237497	CC(C)(C)C1CC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)C1	InChI=1S/C27H26FN5O/c1-27(2,3)14-9-13(10-14)17-11-18-21(15-6-7-20(28)25-19(15)12-31-33-25)22(29)26(34)32-24(18)16-5-4-8-30-23(16)17/h4-8,11-14H,9-10,29H2,1-3H3,(H,31,33)(H,32,34)	ABJIRAVXQFMLON-UHFFFAOYSA-N	794949	3-Amino-6-(3-tert-butylcyclobutyl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C173	Myelin transcription factor 1	Homo sapiens		 95.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794949	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794949&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293294	528826412							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237498	CC1(C)CC2(CC(c3cc4c(-c5ccc(F)c6[nH]ncc56)c(N)c(=O)[nH]c4c4cccnc34)C2)C1	InChI=1S/C28H26FN5O/c1-27(2)12-28(13-27)9-14(10-28)17-8-18-21(15-5-6-20(29)25-19(15)11-32-34-25)22(30)26(35)33-24(18)16-4-3-7-31-23(16)17/h3-8,11,14H,9-10,12-13,30H2,1-2H3,(H,32,34)(H,33,35)	RBIOQYXBSFIRJR-UHFFFAOYSA-N	794950	3-Amino-6-(2,2-dimethylspiro[3,3]heptan-6-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-one::US20260062412, Compound C174	Myelin transcription factor 1	Homo sapiens		 140							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794950	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794950&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293516	528826413							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237499	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC4(CC4)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C25H20FN5O/c26-18-4-3-13(17-11-29-31-23(17)18)19-16-8-15(12-9-25(10-12)5-6-25)21-14(2-1-7-28-21)22(16)30-24(32)20(19)27/h1-4,7-8,11-12H,5-6,9-10,27H2,(H,29,31)(H,30,32)	ALDNMJYHCZGTTC-UHFFFAOYSA-N	794951	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-spiro[2.3]hexan-5-yl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C175	Myelin transcription factor 1	Homo sapiens		 16.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794951	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794951&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293651	528826414							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237500	N#CC1CC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)C1	InChI=1S/C24H17FN6O/c25-18-4-3-13(17-10-29-31-23(17)18)19-16-8-15(12-6-11(7-12)9-26)21-14(2-1-5-28-21)22(16)30-24(32)20(19)27/h1-5,8,10-12H,6-7,27H2,(H,29,31)(H,30,32)	HXYUUPCAXWZXNT-UHFFFAOYSA-N	794952	3-[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]cyclobutane-1-carbonitrile::US20260062412, Compound C176	Myelin transcription factor 1	Homo sapiens		 2.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794952	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794952&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293265	528826415							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237501	N#CC1(Cc2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC1	InChI=1S/C24H17FN6O/c25-17-4-3-13(16-10-29-31-22(16)17)18-15-8-12(9-24(11-26)5-6-24)20-14(2-1-7-28-20)21(15)30-23(32)19(18)27/h1-4,7-8,10H,5-6,9,27H2,(H,29,31)(H,30,32)	VUKQCKOYOHEGFC-UHFFFAOYSA-N	794953	1-[[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]methyl]cyclopropane-1-carbonitrile::US20260062412, Compound C177	Myelin transcription factor 1	Homo sapiens		 2.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794953	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794953&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293939	528826416							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237502	N#C[C@H]1C[C@@H](c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc32)C1	InChI=1S/C24H17FN6O/c25-18-4-3-13(17-10-29-31-23(17)18)19-16-8-15(12-6-11(7-12)9-26)21-14(2-1-5-28-21)22(16)30-24(32)20(19)27/h1-5,8,10-12H,6-7,27H2,(H,29,31)(H,30,32)	HXYUUPCAXWZXNT-UHFFFAOYSA-N	794954	(1s,3s)-3-[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]cyclobutane-1-carbonitrile::US20260062412, Compound C178	Myelin transcription factor 1	Homo sapiens		 2.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794954	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794954&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293265	528826417							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237503	N#C[C@H]1C[C@H](c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc32)C1	InChI=1S/C24H17FN6O/c25-18-4-3-13(17-10-29-31-23(17)18)19-16-8-15(12-6-11(7-12)9-26)21-14(2-1-5-28-21)22(16)30-24(32)20(19)27/h1-5,8,10-12H,6-7,27H2,(H,29,31)(H,30,32)	HXYUUPCAXWZXNT-UHFFFAOYSA-N	794955	(1r,3r)-3-[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]cyclobutane-1-carbonitrile::US20260062412, Compound C179	Myelin transcription factor 1	Homo sapiens		 0.840							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794955	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794955&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293265	528826418							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237504	CC(C)(C)c1ccc2c(ccc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c32)n1	InChI=1S/C23H20FN5O/c1-23(2,3)17-9-6-12-16(27-17)8-5-13-18(19(25)22(30)28-20(12)13)11-4-7-15(24)21-14(11)10-26-29-21/h4-10H,25H2,1-3H3,(H,26,29)(H,28,30)	GEJMKJLZGZNVBA-UHFFFAOYSA-N	794956	3-Amino-8-tert-butyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C180	Myelin transcription factor 1	Homo sapiens		 41.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794956	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794956&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293920	528826419							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237505	Cc1ccc2c(n1)c(I)cc1c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C20H13FIN5O/c1-8-2-3-10-17-11(6-14(22)19(10)25-8)15(16(23)20(28)26-17)9-4-5-13(21)18-12(9)7-24-27-18/h2-7H,23H2,1H3,(H,24,27)(H,26,28)	HFMMMHZOYDLUDM-UHFFFAOYSA-N	794957	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-iodo-8-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C181	Myelin transcription factor 1	Homo sapiens		 23.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794957	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794957&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293573	528826420							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237506	Cc1ccc2c(n1)c(C1CC1)cc1c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C23H18FN5O/c1-10-2-5-13-20(27-10)14(11-3-4-11)8-15-18(19(25)23(30)28-21(13)15)12-6-7-17(24)22-16(12)9-26-29-22/h2,5-9,11H,3-4,25H2,1H3,(H,26,29)(H,28,30)	CRGKVLURGDNFDE-UHFFFAOYSA-N	794958	3-Amino-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-8-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C182	Myelin transcription factor 1	Homo sapiens		 5.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794958	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794958&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293737	528826421							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237507	Cc1ccc2c(ccc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c32)n1	InChI=1S/C20H14FN5O/c1-9-2-3-11-15(24-9)7-5-12-16(17(22)20(27)25-18(11)12)10-4-6-14(21)19-13(10)8-23-26-19/h2-8H,22H2,1H3,(H,23,26)(H,25,27)	WVXWXTPINJPFSP-UHFFFAOYSA-N	794959	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-8-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C183	Myelin transcription factor 1	Homo sapiens		 110							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794959	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794959&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293839	528826422							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237508	Nc1c(-c2cccc(O)c2)c2ccc3ncccc3c2[nH]c1=O	InChI=1S/C18H13N3O2/c19-16-15(10-3-1-4-11(22)9-10)13-6-7-14-12(5-2-8-20-14)17(13)21-18(16)23/h1-9,22H,19H2,(H,21,23)	XBBICBUIAYBGGZ-UHFFFAOYSA-N	794960	3-Amino-4-(3-hydroxyphenyl)-1H-1,7-phenanthrolin-2-one; hydrobromide::US20260062412, Compound C184	Myelin transcription factor 1	Homo sapiens		 10.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794960	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794960&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293575	528826423							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237509	Nc1c(-c2cccc3[nH]ncc23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H17N5O/c23-19-18(12-3-1-5-17-16(12)10-25-27-17)15-9-14(11-6-7-11)20-13(4-2-8-24-20)21(15)26-22(19)28/h1-5,8-11H,6-7,23H2,(H,25,27)(H,26,28)	SESIRVHTVJUFCA-UHFFFAOYSA-N	794961	3-Amino-6-cyclopropyl-4-(1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C185	Myelin transcription factor 1	Homo sapiens		 2.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794961	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794961&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293679	528826424							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237510	Nc1c(-c2cccc3[nH]ncc23)c2ccc3ncccc3c2[nH]c1=O	InChI=1S/C19H13N5O/c20-17-16(10-3-1-5-15-13(10)9-22-24-15)12-6-7-14-11(4-2-8-21-14)18(12)23-19(17)25/h1-9H,20H2,(H,22,24)(H,23,25)	DNTCJROXICERMW-UHFFFAOYSA-N	794962	3-Amino-4-(1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C186	Myelin transcription factor 1	Homo sapiens		 6.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794962	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794962&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293189	528826425							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237511	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C(F)(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C20H11F4N5O/c21-13-4-3-8(11-7-27-29-18(11)13)14-10-6-12(20(22,23)24)17-9(2-1-5-26-17)16(10)28-19(30)15(14)25/h1-7H,25H2,(H,27,29)(H,28,30)	GPWRSKGDHQSKNZ-UHFFFAOYSA-N	794963	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(trifluoromethyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C187	Myelin transcription factor 1	Homo sapiens		 20.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794963	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794963&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293319	528826426							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237512	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OC(F)(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C20H11F4N5O2/c21-12-4-3-8(11-7-27-29-17(11)12)14-10-6-13(31-20(22,23)24)18-9(2-1-5-26-18)16(10)28-19(30)15(14)25/h1-7H,25H2,(H,27,29)(H,28,30)	HMRKCTCFCXWNRQ-UHFFFAOYSA-N	794964	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(trifluoromethoxy)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C188	Myelin transcription factor 1	Homo sapiens		 4.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794964	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794964&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293774	528826427							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237513	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cc(B(O)O)cnc12	InChI=1S/C20H15BFN5O3/c1-8-4-11-15(10-2-3-14(22)19-13(10)7-25-27-19)16(23)20(28)26-18(11)12-5-9(21(29)30)6-24-17(8)12/h2-7,29-30H,23H2,1H3,(H,25,27)(H,26,28)	QPKNAEGSVFKZPT-UHFFFAOYSA-N	794965	[3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-methyl-2-oxo-1H-1,7-phenanthrolin-9-yl]boronic acid::US20260062412, Compound C189	Myelin transcription factor 1	Homo sapiens		 18.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794965	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794965&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293311	528826428							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237514	Cc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H13F2N5O/c1-8-5-11-14(10-6-13(21)15(22)19-12(10)7-25-27-19)16(23)20(28)26-18(11)9-3-2-4-24-17(8)9/h2-7H,23H2,1H3,(H,25,27)(H,26,28)	SMHSNABIWLRGHW-UHFFFAOYSA-N	794966	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C190	Myelin transcription factor 1	Homo sapiens		 2.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794966	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794966&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293229	528826429							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237515	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H15F2N5O/c23-15-7-12(14-8-27-29-21(14)17(15)24)16-13-6-11(9-3-4-9)19-10(2-1-5-26-19)20(13)28-22(30)18(16)25/h1-2,5-9H,3-4,25H2,(H,27,29)(H,28,30)	IUCLREGYFCIISK-UHFFFAOYSA-N	794967	3-Amino-6-cyclopropyl-4-(6,7-difluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C191	Myelin transcription factor 1	Homo sapiens		 6.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794967	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794967&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293534	528826430							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237516	CCc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H15F2N5O/c1-2-9-6-12-15(11-7-14(22)16(23)20-13(11)8-26-28-20)17(24)21(29)27-19(12)10-4-3-5-25-18(9)10/h3-8H,2,24H2,1H3,(H,26,28)(H,27,29)	KJCJSYJJDZGPHB-UHFFFAOYSA-N	794968	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-ethyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C192	Myelin transcription factor 1	Homo sapiens		 3.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794968	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794968&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293385	528826431							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237517	CCOc1cc2c(-c3cc(F)c(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H15ClFN5O2/c1-2-30-14-7-11-15(10-6-13(23)16(22)20-12(10)8-26-28-20)17(24)21(29)27-18(11)9-4-3-5-25-19(9)14/h3-8H,2,24H2,1H3,(H,26,28)(H,27,29)	CXDCHRKKMXWASR-UHFFFAOYSA-N	794969	3-Amino-4-(7-chloro-6-fluoro-1H-indazol-4-yl)-6-ethoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C193	Myelin transcription factor 1	Homo sapiens		 1.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794969	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794969&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293325	528826432							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237518	CC(C)Oc1cc2c(-c3cc(F)c(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H17ClFN5O2/c1-9(2)31-15-7-12-16(11-6-14(24)17(23)21-13(11)8-27-29-21)18(25)22(30)28-19(12)10-4-3-5-26-20(10)15/h3-9H,25H2,1-2H3,(H,27,29)(H,28,30)	VYWLZGNCUQBVCX-UHFFFAOYSA-N	794970	3-Amino-4-(7-chloro-6-fluoro-1H-indazol-4-yl)-6-propan-2-yloxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C194	Myelin transcription factor 1	Homo sapiens		 1.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794970	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794970&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293273	528826433							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237519	Nc1c(-c2cc(F)c(Cl)c3[nH]ncc23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H15ClFN5O/c23-17-15(24)7-12(14-8-27-29-21(14)17)16-13-6-11(9-3-4-9)19-10(2-1-5-26-19)20(13)28-22(30)18(16)25/h1-2,5-9H,3-4,25H2,(H,27,29)(H,28,30)	XPQKJTUGNBBJRG-UHFFFAOYSA-N	794971	3-Amino-4-(7-chloro-6-fluoro-1H-indazol-4-yl)-6-cyclopropyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C195	Myelin transcription factor 1	Homo sapiens		 2.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794971	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794971&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293301	528826434							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237520	Cc1cc2c(-c3cc(F)c(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H13ClFN5O/c1-8-5-11-14(10-6-13(22)15(21)19-12(10)7-25-27-19)16(23)20(28)26-18(11)9-3-2-4-24-17(8)9/h2-7H,23H2,1H3,(H,25,27)(H,26,28)	WCSWMOOWXOIMAU-UHFFFAOYSA-N	794972	3-Amino-4-(7-chloro-6-fluoro-1H-indazol-4-yl)-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C196	Myelin transcription factor 1	Homo sapiens		 3.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794972	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794972&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293648	528826435							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237521	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2ccc3ncccc3c2[nH]c1=O	InChI=1S/C19H11F2N5O/c20-12-6-10(11-7-24-26-18(11)15(12)21)14-9-3-4-13-8(2-1-5-23-13)17(9)25-19(27)16(14)22/h1-7H,22H2,(H,24,26)(H,25,27)	UTIISVAYMGAUML-UHFFFAOYSA-N	794973	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C197	Myelin transcription factor 1	Homo sapiens		 20.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794973	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794973&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293312	528826436							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237522	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(Cl)c3ncccc3c2[nH]c1=O	InChI=1S/C19H10ClF2N5O/c20-11-4-9-13(8-5-12(21)14(22)18-10(8)6-25-27-18)15(23)19(28)26-16(9)7-2-1-3-24-17(7)11/h1-6H,23H2,(H,25,27)(H,26,28)	VVMFPXPOZYMITF-UHFFFAOYSA-N	794974	3-Amino-6-chloro-4-(6,7-difluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C198	Myelin transcription factor 1	Homo sapiens		 3.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794974	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794974&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293639	528826437							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237523	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(O)c3ncccc3c2[nH]c1=O	InChI=1S/C19H11F2N5O2/c20-11-4-8(10-6-24-26-18(10)14(11)21)13-9-5-12(27)17-7(2-1-3-23-17)16(9)25-19(28)15(13)22/h1-6,27H,22H2,(H,24,26)(H,25,28)	DHIAFMSKRXLZFC-UHFFFAOYSA-N	794975	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-hydroxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C199	Myelin transcription factor 1	Homo sapiens		 3.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794975	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794975&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293938	528826438							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237524	CC(=O)c1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H14FN5O2/c1-9(28)12-7-13-16(10-4-5-15(22)20-14(10)8-25-27-20)17(23)21(29)26-19(13)11-3-2-6-24-18(11)12/h2-8H,23H2,1H3,(H,25,27)(H,26,29)	YSXBNYZSSJMQOR-UHFFFAOYSA-N	794976	6-Acetyl-3-amino-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C200	Myelin transcription factor 1	Homo sapiens		 2.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794976	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794976&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293548	528826439							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237525	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(C3CCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H17F2N5O/c24-16-8-13(15-9-28-30-22(15)18(16)25)17-14-7-12(10-3-1-4-10)20-11(5-2-6-27-20)21(14)29-23(31)19(17)26/h2,5-10H,1,3-4,26H2,(H,28,30)(H,29,31)	MRVAHKOCBDBWOK-UHFFFAOYSA-N	794977	3-Amino-6-cyclobutyl-4-(6,7-difluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C201	Myelin transcription factor 1	Homo sapiens		 5.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794977	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794977&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293468	528826440							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237526	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(C3CCCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H19F2N5O/c25-17-9-14(16-10-29-31-23(16)19(17)26)18-15-8-13(11-4-1-2-5-11)21-12(6-3-7-28-21)22(15)30-24(32)20(18)27/h3,6-11H,1-2,4-5,27H2,(H,29,31)(H,30,32)	FNWKSPRVTXDMBY-UHFFFAOYSA-N	794978	3-Amino-6-cyclopentyl-4-(6,7-difluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C202	Myelin transcription factor 1	Homo sapiens		 7.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794978	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794978&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293361	528826441							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237527	CC(C)Cc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C23H19F2N5O/c1-10(2)6-11-7-14-17(13-8-16(24)18(25)22-15(13)9-28-30-22)19(26)23(31)29-21(14)12-4-3-5-27-20(11)12/h3-5,7-10H,6,26H2,1-2H3,(H,28,30)(H,29,31)	XCUVMRPNQMBYSO-UHFFFAOYSA-N	794979	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-(2-methylpropyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C203	Myelin transcription factor 1	Homo sapiens		 17.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794979	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794979&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293837	528826442							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237528	C=Cc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H13F2N5O/c1-2-9-6-12-15(11-7-14(22)16(23)20-13(11)8-26-28-20)17(24)21(29)27-19(12)10-4-3-5-25-18(9)10/h2-8H,1,24H2,(H,26,28)(H,27,29)	CAFBZNSOVMGALM-UHFFFAOYSA-N	794980	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-ethenyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C204	Myelin transcription factor 1	Homo sapiens		 10.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794980	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794980&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293449	528826443							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237529	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(OC(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C20H11F4N5O2/c21-11-4-8(10-6-27-29-18(10)14(11)22)13-9-5-12(31-20(23)24)17-7(2-1-3-26-17)16(9)28-19(30)15(13)25/h1-6,20H,25H2,(H,27,29)(H,28,30)	XTLYPJYCMNUNEO-UHFFFAOYSA-N	794981	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-(difluoromethoxy)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C205	Myelin transcription factor 1	Homo sapiens		 3.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794981	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794981&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293749	528826444							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237530	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(OC3CCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H17F2N5O2/c24-15-7-12(14-9-28-30-22(14)18(15)25)17-13-8-16(32-10-3-1-4-10)21-11(5-2-6-27-21)20(13)29-23(31)19(17)26/h2,5-10H,1,3-4,26H2,(H,28,30)(H,29,31)	RCCUJHIIJIZLLQ-UHFFFAOYSA-N	794982	3-Amino-6-cyclobutyloxy-4-(6,7-difluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C206	Myelin transcription factor 1	Homo sapiens		 4.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794982	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794982&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293478	528826445							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237531	Cn1cc(-c2cc3c(-c4cc(F)c(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)cn1	InChI=1S/C23H15F2N7O/c1-32-9-10(7-29-32)12-5-14-17(13-6-16(24)18(25)22-15(13)8-28-31-22)19(26)23(33)30-21(14)11-3-2-4-27-20(11)12/h2-9H,26H2,1H3,(H,28,31)(H,30,33)	AJWAYAHMOQOCEK-UHFFFAOYSA-N	794983	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-(1-methylpyrazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C207	Myelin transcription factor 1	Homo sapiens		 1.000							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794983	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794983&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293186	528826446							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237532	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(N3CCOCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H18F2N6O2/c24-15-8-12(14-10-28-30-22(14)18(15)25)17-13-9-16(31-4-6-33-7-5-31)21-11(2-1-3-27-21)20(13)29-23(32)19(17)26/h1-3,8-10H,4-7,26H2,(H,28,30)(H,29,32)	NBVHZMHAFMKXIX-UHFFFAOYSA-N	794984	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-morpholin-4-yl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C208	Myelin transcription factor 1	Homo sapiens		 2.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794984	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794984&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293230	528826447							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237533	CN1CCN(c2cc3c(-c4cc(F)c(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC1	InChI=1S/C24H21F2N7O/c1-32-5-7-33(8-6-32)17-10-14-18(13-9-16(25)19(26)23-15(13)11-29-31-23)20(27)24(34)30-21(14)12-3-2-4-28-22(12)17/h2-4,9-11H,5-8,27H2,1H3,(H,29,31)(H,30,34)	BZCJXVDNQIHGIE-UHFFFAOYSA-N	794985	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-(4-methylpiperazin-1-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C209	Myelin transcription factor 1	Homo sapiens		 1.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794985	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794985&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293287	528826448							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237534	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(O[C@H]3C[C@H](F)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H16F3N5O2/c24-9-4-10(5-9)33-16-7-13-17(12-6-15(25)18(26)22-14(12)8-29-31-22)19(27)23(32)30-20(13)11-2-1-3-28-21(11)16/h1-3,6-10H,4-5,27H2,(H,29,31)(H,30,32)	ZGUHEJAWHIZKPK-UHFFFAOYSA-N	794986	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-((1r,3r)-3-fluorocyclobutyl)oxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C210	Myelin transcription factor 1	Homo sapiens		 1.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794986	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794986&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293668	528826449							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237535	N#C[C@H]1C[C@H](Oc2cc3c(-c4cc(F)c(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)C1	InChI=1S/C24H16F2N6O2/c25-16-6-13(15-9-30-32-23(15)19(16)26)18-14-7-17(34-11-4-10(5-11)8-27)22-12(2-1-3-29-22)21(14)31-24(33)20(18)28/h1-3,6-7,9-11H,4-5,28H2,(H,30,32)(H,31,33)	VGYRLHJDSYXRAE-UHFFFAOYSA-N	794987	(1r,3r)-3-[[3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]oxy]cyclobutane-1-carbonitrile::US20260062412, Compound C211	Myelin transcription factor 1	Homo sapiens		 0.870							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794987	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794987&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293389	528826450							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237536	N#C[C@H]1C[C@@H](Oc2cc3c(-c4cc(F)c(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)C1	InChI=1S/C24H16F2N6O2/c25-16-6-13(15-9-30-32-23(15)19(16)26)18-14-7-17(34-11-4-10(5-11)8-27)22-12(2-1-3-29-22)21(14)31-24(33)20(18)28/h1-3,6-7,9-11H,4-5,28H2,(H,30,32)(H,31,33)	VGYRLHJDSYXRAE-UHFFFAOYSA-N	794988	(1s,3s)-3-[[3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-2-oxo-1H-1,7-phenanthrolin-6-yl]oxy]cyclobutane-1-carbonitrile::US20260062412, Compound C212	Myelin transcription factor 1	Homo sapiens		 1.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794988	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794988&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293389	528826451							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237537	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(O[C@H]3C[C@@H](F)C3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H16F3N5O2/c24-9-4-10(5-9)33-16-7-13-17(12-6-15(25)18(26)22-14(12)8-29-31-22)19(27)23(32)30-20(13)11-2-1-3-28-21(11)16/h1-3,6-10H,4-5,27H2,(H,29,31)(H,30,32)	ZGUHEJAWHIZKPK-UHFFFAOYSA-N	794989	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-((1s,3s)-3-fluorocyclobutyl)oxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C213	Myelin transcription factor 1	Homo sapiens		 0.830							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794989	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794989&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293668	528826452							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237538	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(OCCC(F)F)c3ncccc3c2[nH]c1=O	InChI=1S/C22H15F4N5O2/c23-13-6-10(12-8-29-31-21(12)17(13)26)16-11-7-14(33-5-3-15(24)25)20-9(2-1-4-28-20)19(11)30-22(32)18(16)27/h1-2,4,6-8,15H,3,5,27H2,(H,29,31)(H,30,32)	NIUZEKNZFFHIRY-UHFFFAOYSA-N	794990	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-(3,3-difluoropropoxy)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C214	Myelin transcription factor 1	Homo sapiens		 1.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794990	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794990&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293333	528826453							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237539	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(-c3cccnc3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H14F2N6O/c25-17-8-14(16-10-30-32-23(16)19(17)26)18-15-7-13(11-3-1-5-28-9-11)21-12(4-2-6-29-21)22(15)31-24(33)20(18)27/h1-10H,27H2,(H,30,32)(H,31,33)	KXVDNINCCKVUQQ-UHFFFAOYSA-N	794991	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-pyridin-3-yl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C215	Myelin transcription factor 1	Homo sapiens		 2.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794991	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794991&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293904	528826454							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237540	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3ccncc3c2[nH]c1=O	InChI=1S/C19H11BrFN5O/c20-13-5-10-15(9-1-2-14(21)18-12(9)7-24-26-18)16(22)19(27)25-17(10)11-6-23-4-3-8(11)13/h1-7H,22H2,(H,24,26)(H,25,27)	QOKQASVIJODQTG-UHFFFAOYSA-N	794992	3-Amino-6-bromo-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D1	Myelin transcription factor 1	Homo sapiens		 9.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794992	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794992&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			178423168	528826455							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237541	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3cccnc3c2[nH]c1=O	InChI=1S/C22H16FN5O/c23-16-6-5-11(15-9-26-28-19(15)16)17-14-8-13(10-3-4-10)12-2-1-7-25-20(12)21(14)27-22(29)18(17)24/h1-2,5-10H,3-4,24H2,(H,26,28)(H,27,29)	WTUSPBCHWZGEOK-UHFFFAOYSA-N	794993	3-Amino-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D2	Myelin transcription factor 1	Homo sapiens		 4.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794993	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794993&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293600	528826456							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237542	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ncccc12	InChI=1S/C20H14FN5O/c1-9-7-12-15(11-4-5-14(21)17-13(11)8-24-26-17)16(22)20(27)25-19(12)18-10(9)3-2-6-23-18/h2-8H,22H2,1H3,(H,24,26)(H,25,27)	YICOBQSGJQQLKB-UHFFFAOYSA-N	794994	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-methyl-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D3	Myelin transcription factor 1	Homo sapiens		 4.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794994	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794994&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293877	528826457							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237543	Nc1c(-c2ccc(F)c3[nH]ncc23)c2ccc3cccnc3c2[nH]c1=O	InChI=1S/C19H12FN5O/c20-13-6-5-10(12-8-23-25-17(12)13)14-11-4-3-9-2-1-7-22-16(9)18(11)24-19(26)15(14)21/h1-8H,21H2,(H,23,25)(H,24,26)	LQDXSCISJZMTDU-UHFFFAOYSA-N	794995	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D4	Myelin transcription factor 1	Homo sapiens		 15.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794995	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794995&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293891	528826458							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237544	CCc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ncccc12	InChI=1S/C21H16FN5O/c1-2-10-8-13-16(12-5-6-15(22)18-14(12)9-25-27-18)17(23)21(28)26-20(13)19-11(10)4-3-7-24-19/h3-9H,2,23H2,1H3,(H,25,27)(H,26,28)	LJORVTJROORRTH-UHFFFAOYSA-N	794996	3-Amino-6-ethyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D5	Myelin transcription factor 1	Homo sapiens		 6.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794996	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794996&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293735	528826459							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237545	CN1CCN(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3ncccc23)CC1	InChI=1S/C24H22FN7O/c1-31-7-9-32(10-8-31)18-11-15-19(13-4-5-17(25)21-16(13)12-28-30-21)20(26)24(33)29-23(15)22-14(18)3-2-6-27-22/h2-6,11-12H,7-10,26H2,1H3,(H,28,30)(H,29,33)	QGLZSHYEUMHMPO-UHFFFAOYSA-N	794997	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(4-methylpiperazin-1-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D6	Myelin transcription factor 1	Homo sapiens		 2.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794997	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794997&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293192	528826460							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237546	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCC(N4CCOCC4)CC3)c3cccnc3c2[nH]c1=O	InChI=1S/C28H28FN7O2/c29-21-4-3-17(20-15-32-34-25(20)21)23-19-14-22(36-8-5-16(6-9-36)35-10-12-38-13-11-35)18-2-1-7-31-26(18)27(19)33-28(37)24(23)30/h1-4,7,14-16H,5-6,8-13,30H2,(H,32,34)(H,33,37)	RUTJGGPVWCEHQR-UHFFFAOYSA-N	794998	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(4-morpholin-4-ylpiperidin-1-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D7	Myelin transcription factor 1	Homo sapiens		 15.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794998	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794998&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293276	528826461							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237547	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCC(F)(F)C3)c3cccnc3c2[nH]c1=O	InChI=1S/C23H17F3N6O/c24-15-4-3-11(14-9-29-31-19(14)15)17-13-8-16(32-7-5-23(25,26)10-32)12-2-1-6-28-20(12)21(13)30-22(33)18(17)27/h1-4,6,8-9H,5,7,10,27H2,(H,29,31)(H,30,33)	CPVYPWWAWTXVIO-UHFFFAOYSA-N	794999	3-Amino-6-(3,3-difluoropyrrolidin-1-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D8	Myelin transcription factor 1	Homo sapiens		 10.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794999	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794999&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293861	528826462							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237548	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCOCC3)c3cccnc3c2[nH]c1=O	InChI=1S/C23H19FN6O2/c24-16-4-3-12(15-11-27-29-20(15)16)18-14-10-17(30-6-8-32-9-7-30)13-2-1-5-26-21(13)22(14)28-23(31)19(18)25/h1-5,10-11H,6-9,25H2,(H,27,29)(H,28,31)	LIWHMJPJSXTSNB-UHFFFAOYSA-N	795000	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-morpholin-4-yl-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D9	Myelin transcription factor 1	Homo sapiens		 22.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795000	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795000&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293617	528826463							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237549	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CC4(COC4)C3)c3cccnc3c2[nH]c1=O	InChI=1S/C24H19FN6O2/c25-16-4-3-12(15-7-28-30-20(15)16)18-14-6-17(31-8-24(9-31)10-33-11-24)13-2-1-5-27-21(13)22(14)29-23(32)19(18)26/h1-7H,8-11,26H2,(H,28,30)(H,29,32)	HWZNJMGABAVSPB-UHFFFAOYSA-N	795001	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(2-oxa-6-azaspiro[3,3]heptan-6-yl)-1H-1,10-one::US20260062412, Compound D10	Myelin transcription factor 1	Homo sapiens		 3.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795001	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795001&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293546	528826464							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237550	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CC(N4CC(F)(F)C4)C3)c3cccnc3c2[nH]c1=O	InChI=1S/C25H20F3N7O/c26-17-4-3-13(16-7-31-33-21(16)17)19-15-6-18(34-8-12(9-34)35-10-25(27,28)11-35)14-2-1-5-30-22(14)23(15)32-24(36)20(19)29/h1-7,12H,8-11,29H2,(H,31,33)(H,32,36)	KBIHCNDWVZKGHC-UHFFFAOYSA-N	795002	3-Amino-6-[3-(3,3-difluoroazetidin-1-yl) azetidin-1-yl]-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D11	Myelin transcription factor 1	Homo sapiens		 20.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795002	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795002&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293165	528826465							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237551	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCN4CCOC[C@H]4C3)c3cccnc3c2[nH]c1=O	InChI=1S/C26H24FN7O2/c27-19-4-3-15(18-11-30-32-23(18)19)21-17-10-20(34-7-6-33-8-9-36-13-14(33)12-34)16-2-1-5-29-24(16)25(17)31-26(35)22(21)28/h1-5,10-11,14H,6-9,12-13,28H2,(H,30,32)(H,31,35)	QGCHHDKAEMEOQG-UHFFFAOYSA-N	795003	6-[(9aR)-3,4,6,7,9,9a-hexahydro-1H-pyrazino[2,1-c][1,4]oxazin-8-yl]-3-amino-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D12	Myelin transcription factor 1	Homo sapiens		 49.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795003	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795003&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293794	528826466							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237552	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCN4CCOC[C@@H]4C3)c3cccnc3c2[nH]c1=O	InChI=1S/C26H24FN7O2/c27-19-4-3-15(18-11-30-32-23(18)19)21-17-10-20(34-7-6-33-8-9-36-13-14(33)12-34)16-2-1-5-29-24(16)25(17)31-26(35)22(21)28/h1-5,10-11,14H,6-9,12-13,28H2,(H,30,32)(H,31,35)	QGCHHDKAEMEOQG-UHFFFAOYSA-N	795004	6-[(9aS)-3,4,6,7,9,9a-hexahydro-1H-pyrazino[2,1-c][1,4]oxazin-8-yl]-3-amino-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D13	Myelin transcription factor 1	Homo sapiens		 25.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795004	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795004&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293586	528826467							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237553	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCN(CC(F)F)CC3)c3cccnc3c2[nH]c1=O	InChI=1S/C25H22F3N7O/c26-17-4-3-13(16-11-31-33-22(16)17)20-15-10-18(35-8-6-34(7-9-35)12-19(27)28)14-2-1-5-30-23(14)24(15)32-25(36)21(20)29/h1-5,10-11,19H,6-9,12,29H2,(H,31,33)(H,32,36)	HCMULOKJVFDUKG-UHFFFAOYSA-N	795005	3-Amino-6-[4-(2,2-difluoroethyl) piperazin-1-yl]-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D14	Myelin transcription factor 1	Homo sapiens		 33.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795005	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795005&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293393	528826468							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237554	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(N3CCN(CC(F)(F)F)CC3)c3cccnc3c2[nH]c1=O	InChI=1S/C25H21F4N7O/c26-17-4-3-13(16-11-32-34-21(16)17)19-15-10-18(36-8-6-35(7-9-36)12-25(27,28)29)14-2-1-5-31-22(14)23(15)33-24(37)20(19)30/h1-5,10-11H,6-9,12,30H2,(H,32,34)(H,33,37)	OYVJHXOKKDDDBL-UHFFFAOYSA-N	795006	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[4-(2,2,2-trifluoroethyl) piperazin-1-yl]-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D15	Myelin transcription factor 1	Homo sapiens		 69.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795006	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795006&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293501	528826469							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237555	CS(=O)(=O)Nc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ncccc12	InChI=1S/C20H15FN6O3S/c1-31(29,30)27-14-7-11-15(9-4-5-13(21)17-12(9)8-24-26-17)16(22)20(28)25-19(11)18-10(14)3-2-6-23-18/h2-8,27H,22H2,1H3,(H,24,26)(H,25,28)	JNUZFBSOPBEQNE-UHFFFAOYSA-N	795007	N-[8-Amino-7-(7-fluoro-1H-indazol-4-yl)-9-oxo-10H-1,10-phenanthroline-5-yl]methanesulfonamide::US20260062412, Compound D16	Myelin transcription factor 1	Homo sapiens		 2.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795007	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795007&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293933	528826470							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237556	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(NS(=O)(=O)C3CC3)c3cccnc3c2[nH]c1=O	InChI=1S/C22H17FN6O3S/c23-15-6-5-11(14-9-26-28-19(14)15)17-13-8-16(29-33(31,32)10-3-4-10)12-2-1-7-25-20(12)21(13)27-22(30)18(17)24/h1-2,5-10,29H,3-4,24H2,(H,26,28)(H,27,30)	JGWCQPXRLGBOHJ-UHFFFAOYSA-N	795008	N-[8-amino-7-(7-fluoro-1H-indazol-4-yl)-9-oxo-10H-1,10-phenanthrolin-5-yl]cyclopropanesulfonamide::US20260062412, Compound D17	Myelin transcription factor 1	Homo sapiens		 3.10							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795008	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795008&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293698	528826471							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237557	COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ncccc12	InChI=1S/C20H14FN5O2/c1-28-14-7-11-15(9-4-5-13(21)17-12(9)8-24-26-17)16(22)20(27)25-19(11)18-10(14)3-2-6-23-18/h2-8H,22H2,1H3,(H,24,26)(H,25,27)	GFQLJFVSONUSMB-UHFFFAOYSA-N	795009	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-methoxy-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D18	Myelin transcription factor 1	Homo sapiens		 0.250							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795009	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795009&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293652	528826472							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237558	CC(=O)Nc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ncccc12	InChI=1S/C21H15FN6O2/c1-9(29)26-15-7-12-16(10-4-5-14(22)18-13(10)8-25-28-18)17(23)21(30)27-20(12)19-11(15)3-2-6-24-19/h2-8H,23H2,1H3,(H,25,28)(H,26,29)(H,27,30)	LLJKWXCPRRVFAG-UHFFFAOYSA-N	795010	N-[8-amino-7-(7-fluoro-1H-indazol-4-yl)-9-oxo-10H-1,10-phenanthrolin-5-yl]acetamide::US20260062412, Compound D19	Myelin transcription factor 1	Homo sapiens		 22.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795010	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795010&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293410	528826473							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237559	CC(C)Nc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ncccc12	InChI=1S/C22H19FN6O/c1-10(2)27-16-8-13-17(11-5-6-15(23)19-14(11)9-26-29-19)18(24)22(30)28-21(13)20-12(16)4-3-7-25-20/h3-10,27H,24H2,1-2H3,(H,26,29)(H,28,30)	OUCIEXYMLIAHHN-UHFFFAOYSA-N	795011	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(propan-2-ylamino)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D20	Myelin transcription factor 1	Homo sapiens		 7.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795011	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795011&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293875	528826474							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237560	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCNCC3)c3cccnc3c2[nH]c1=O	InChI=1S/C24H21FN6O/c25-18-4-3-13(17-11-29-31-21(17)18)19-16-10-15(12-5-8-27-9-6-12)14-2-1-7-28-22(14)23(16)30-24(32)20(19)26/h1-4,7,10-12,27H,5-6,8-9,26H2,(H,29,31)(H,30,32)	JKWOWOGYQHGBSF-UHFFFAOYSA-N	795012	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-piperidin-4-yl-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D21	Myelin transcription factor 1	Homo sapiens		 3.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795012	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795012&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293646	528826475							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237561	CN1CCC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3ncccc23)CC1	InChI=1S/C25H23FN6O/c1-32-9-6-13(7-10-32)16-11-17-20(14-4-5-19(26)22-18(14)12-29-31-22)21(27)25(33)30-24(17)23-15(16)3-2-8-28-23/h2-5,8,11-13H,6-7,9-10,27H2,1H3,(H,29,31)(H,30,33)	VTVODBOCCDLWTD-UHFFFAOYSA-N	795013	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-methylpiperidin-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D22	Myelin transcription factor 1	Homo sapiens		 2.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795013	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795013&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293240	528826476							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237562	CC(C)N1CCC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3ncccc23)CC1	InChI=1S/C27H27FN6O/c1-14(2)34-10-7-15(8-11-34)18-12-19-22(16-5-6-21(28)24-20(16)13-31-33-24)23(29)27(35)32-26(19)25-17(18)4-3-9-30-25/h3-6,9,12-15H,7-8,10-11,29H2,1-2H3,(H,31,33)(H,32,35)	YNCJYDBMGLTNQS-UHFFFAOYSA-N	795014	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-propan-2-ylpiperidin-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D23	Myelin transcription factor 1	Homo sapiens		 6.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795014	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795014&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293148	528826477							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237563	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCN(C4CCC4)CC3)c3cccnc3c2[nH]c1=O	InChI=1S/C28H27FN6O/c29-22-7-6-17(21-14-32-34-25(21)22)23-20-13-19(15-8-11-35(12-9-15)16-3-1-4-16)18-5-2-10-31-26(18)27(20)33-28(36)24(23)30/h2,5-7,10,13-16H,1,3-4,8-9,11-12,30H2,(H,32,34)(H,33,36)	BEEVGBUHCURGOR-UHFFFAOYSA-N	795015	3-Amino-6-(1-cyclobutylpiperidin-4-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D24	Myelin transcription factor 1	Homo sapiens		 6.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795015	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795015&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293764	528826478							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237564	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCN(C4CCOCC4)CC3)c3cccnc3c2[nH]c1=O	InChI=1S/C29H29FN6O2/c30-23-4-3-18(22-15-33-35-26(22)23)24-21-14-20(16-5-10-36(11-6-16)17-7-12-38-13-8-17)19-2-1-9-32-27(19)28(21)34-29(37)25(24)31/h1-4,9,14-17H,5-8,10-13,31H2,(H,33,35)(H,34,37)	BLNLSMSLDYZUNH-UHFFFAOYSA-N	795016	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[1-(oxan-4-yl) piperidin-4-yl]-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D25	Myelin transcription factor 1	Homo sapiens		 7.80							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795016	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795016&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293172	528826479							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237565	CCN1CCC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3ncccc23)CC1	InChI=1S/C26H25FN6O/c1-2-33-10-7-14(8-11-33)17-12-18-21(15-5-6-20(27)23-19(15)13-30-32-23)22(28)26(34)31-25(18)24-16(17)4-3-9-29-24/h3-6,9,12-14H,2,7-8,10-11,28H2,1H3,(H,30,32)(H,31,34)	TUBXLOWWKSERIR-UHFFFAOYSA-N	795017	3-Amino-6-(1-ethylpiperidin-4-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D26	Myelin transcription factor 1	Homo sapiens		 3.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795017	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795017&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293526	528826480							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237566	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCN(C4COC4)CC3)c3cccnc3c2[nH]c1=O	InChI=1S/C27H25FN6O2/c28-21-4-3-16(20-11-31-33-24(20)21)22-19-10-18(14-5-8-34(9-6-14)15-12-36-13-15)17-2-1-7-30-25(17)26(19)32-27(35)23(22)29/h1-4,7,10-11,14-15H,5-6,8-9,12-13,29H2,(H,31,33)(H,32,35)	GFKZOYZBCLUCLL-UHFFFAOYSA-N	795018	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[1-(oxetan-3-yl) piperidin-4-yl]-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D27	Myelin transcription factor 1	Homo sapiens		 0.530							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795018	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795018&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293596	528826481							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237567	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CNC3)c3cccnc3c2[nH]c1=O	InChI=1S/C22H17FN6O/c23-16-4-3-11(15-9-27-29-19(15)16)17-14-6-13(10-7-25-8-10)12-2-1-5-26-20(12)21(14)28-22(30)18(17)24/h1-6,9-10,25H,7-8,24H2,(H,27,29)(H,28,30)	YUGLZTGWGMTMPB-UHFFFAOYSA-N	795019	3-Amino-6-(azetidin-3-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D28	Myelin transcription factor 1	Homo sapiens		 1.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795019	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795019&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293514	528826482							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237568	CC(C)N1CC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3ncccc23)C1	InChI=1S/C25H23FN6O/c1-12(2)32-10-13(11-32)16-8-17-20(14-5-6-19(26)22-18(14)9-29-31-22)21(27)25(33)30-24(17)23-15(16)4-3-7-28-23/h3-9,12-13H,10-11,27H2,1-2H3,(H,29,31)(H,30,33)	WABWDRSUOFVIHZ-UHFFFAOYSA-N	795020	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-propan-2-ylazetidin-3-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D29	Myelin transcription factor 1	Homo sapiens		 5.70							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795020	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795020&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293493	528826483							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237569	CN1CC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3ncccc23)C1	InChI=1S/C23H19FN6O/c1-30-9-11(10-30)14-7-15-18(12-4-5-17(24)20-16(12)8-27-29-20)19(25)23(31)28-22(15)21-13(14)3-2-6-26-21/h2-8,11H,9-10,25H2,1H3,(H,27,29)(H,28,31)	QPFCVEVEHVCXCH-UHFFFAOYSA-N	795021	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-methylazetidin-3-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D30	Myelin transcription factor 1	Homo sapiens		 2.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795021	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795021&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293913	528826484							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237570	Nc1c(-c2cccc3[nH]ncc23)c2ccccc2oc1=O	InChI=1S/C16H11N3O2/c17-15-14(9-5-3-6-12-11(9)8-18-19-12)10-4-1-2-7-13(10)21-16(15)20/h1-8H,17H2,(H,18,19)	OEDPKRRRGGVHKB-UHFFFAOYSA-N	795022	3-Amino-4-(1H-indazol-4-yl) chromen-2-one::US20260062412, Compound E1	Myelin transcription factor 1	Homo sapiens		 1100							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795022	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795022&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293780	528826485							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237571	O=c1[nH]c2ccccc2c(-c2cccc3[nH]ncc23)c1O	InChI=1S/C16H11N3O2/c20-15-14(9-5-3-7-13-11(9)8-17-19-13)10-4-1-2-6-12(10)18-16(15)21/h1-8,20H,(H,17,19)(H,18,21)	YZJFIEVIWCLAGA-UHFFFAOYSA-N	795023	3-Hydroxy-4-(1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound E2	Myelin transcription factor 1	Homo sapiens		 840							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795023	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795023&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293447	528826486							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237572	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3ncc(F)cc3c2[nH]c1=O	InChI=1S/C19H10BrF2N5O/c20-12-4-9-14(8-1-2-13(22)18-11(8)6-25-27-18)15(23)19(28)26-16(9)10-3-7(21)5-24-17(10)12/h1-6H,23H2,(H,25,27)(H,26,28)	WUMPWTRZDNBASN-UHFFFAOYSA-N	795024	3-Amino-6-bromo-9-fluoro-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound F1	Myelin transcription factor 1	Homo sapiens		 12.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795024	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795024&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293811	528826487							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237573	COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cc(F)cnc12	InChI=1S/C20H13F2N5O2/c1-29-14-5-10-15(9-2-3-13(22)18-12(9)7-25-27-18)16(23)20(28)26-17(10)11-4-8(21)6-24-19(11)14/h2-7H,23H2,1H3,(H,25,27)(H,26,28)	WDBQVRVVKUTHCJ-UHFFFAOYSA-N	795025	3-Amino-9-fluoro-4-(7-fluoro-1H-indazol-4-yl)-6-methoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound F2	Myelin transcription factor 1	Homo sapiens		 1.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795025	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795025&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293286	528826488							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237574	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cc(F)cnc12	InChI=1S/C20H13F2N5O/c1-8-4-11-15(10-2-3-14(22)19-13(10)7-25-27-19)16(23)20(28)26-18(11)12-5-9(21)6-24-17(8)12/h2-7H,23H2,1H3,(H,25,27)(H,26,28)	FSWAJLAGQAAPPN-UHFFFAOYSA-N	795026	3-Amino-9-fluoro-4-(7-fluoro-1H-indazol-4-yl)-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound F3	Myelin transcription factor 1	Homo sapiens		 4.00							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795026	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795026&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293606	528826489							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237575	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2cc(Br)c3ncc(F)cc3c2[nH]c1=O	InChI=1S/C19H9BrF3N5O/c20-11-2-8-13(7-3-12(22)14(23)18-10(7)5-26-28-18)15(24)19(29)27-16(8)9-1-6(21)4-25-17(9)11/h1-5H,24H2,(H,26,28)(H,27,29)	ZXIYCZQBJAUAGZ-UHFFFAOYSA-N	795027	3-Amino-6-bromo-4-(6,7-difluoro-1H-indazol-4-yl)-9-fluoro-1H-1,7-phenanthrolin-2-one::US20260062412, Compound F4	Myelin transcription factor 1	Homo sapiens		 22.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795027	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795027&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293687	528826490							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237576	COc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cc(F)cnc12	InChI=1S/C20H12F3N5O2/c1-30-13-4-9-14(8-3-12(22)15(23)19-11(8)6-26-28-19)16(24)20(29)27-17(9)10-2-7(21)5-25-18(10)13/h2-6H,24H2,1H3,(H,26,28)(H,27,29)	XQQKKFCEBKDKMR-UHFFFAOYSA-N	795028	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-9-fluoro-6-methoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound F5	Myelin transcription factor 1	Homo sapiens		 3.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795028	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795028&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293688	528826491							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237577	Cc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cc(F)cnc12	InChI=1S/C20H12F3N5O/c1-7-2-10-14(9-4-13(22)15(23)19-12(9)6-26-28-19)16(24)20(29)27-18(10)11-3-8(21)5-25-17(7)11/h2-6H,24H2,1H3,(H,26,28)(H,27,29)	KHEHSZOWNGWIDW-UHFFFAOYSA-N	795029	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-9-fluoro-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound F6	Myelin transcription factor 1	Homo sapiens		 9.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795029	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795029&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293308	528826492							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237578	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3nccnc3c2[nH]c1=O	InChI=1S/C18H10BrFN6O/c19-10-5-8-12(7-1-2-11(20)14-9(7)6-24-26-14)13(21)18(27)25-15(8)17-16(10)22-3-4-23-17/h1-6H,21H2,(H,24,26)(H,25,27)	LSVFSCOPXGCFLR-UHFFFAOYSA-N	795030	8-Amino-5-bromo-7-(7-fluoro-1H-indazol-4-yl)-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G1	Myelin transcription factor 1	Homo sapiens		 16.0							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795030	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795030&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293427	528826493							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237579	O=c1[nH]c2c(cc(Br)c3nccnc32)c(-c2ccc(F)c3[nH]ncc23)c1Cl	InChI=1S/C18H8BrClFN5O/c19-10-5-8-12(7-1-2-11(21)14-9(7)6-24-26-14)13(20)18(27)25-15(8)17-16(10)22-3-4-23-17/h1-6H,(H,24,26)(H,25,27)	JXXUGOBNEIZFDM-UHFFFAOYSA-N	795031	5-Bromo-8-chloro-7-(7-fluoro-1H-indazol-4-yl)-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G2	Myelin transcription factor 1	Homo sapiens		 270							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795031	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795031&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293713	528826494							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237580	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2nccnc12	InChI=1S/C19H13FN6O/c1-8-6-10-13(9-2-3-12(20)16-11(9)7-24-26-16)14(21)19(27)25-17(10)18-15(8)22-4-5-23-18/h2-7H,21H2,1H3,(H,24,26)(H,25,27)	AHKWAJCZYQYITA-UHFFFAOYSA-N	795032	8-Amino-7-(7-fluoro-1H-indazol-4-yl)-5-methyl-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G3	Myelin transcription factor 1	Homo sapiens		 7.90							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795032	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795032&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293817	528826495							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237581	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3nccnc3c2[nH]c1=O	InChI=1S/C21H15FN6O/c22-14-4-3-10(13-8-26-28-17(13)14)15-12-7-11(9-1-2-9)18-20(25-6-5-24-18)19(12)27-21(29)16(15)23/h3-9H,1-2,23H2,(H,26,28)(H,27,29)	LZRBNGIQGVYYEQ-UHFFFAOYSA-N	795033	8-Amino-5-cyclopropyl-7-(7-fluoro-1H-indazol-4-yl)-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G4	Myelin transcription factor 1	Homo sapiens		 3.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795033	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795033&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293855	528826496							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237582	CS(=O)(=O)Nc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2nccnc12	InChI=1S/C19H14FN7O3S/c1-31(29,30)27-12-6-9-13(8-2-3-11(20)15-10(8)7-24-26-15)14(21)19(28)25-16(9)18-17(12)22-4-5-23-18/h2-7,27H,21H2,1H3,(H,24,26)(H,25,28)	RUUPSXDACZVRMG-UHFFFAOYSA-N	795034	N-[8-amino-7-(7-fluoro-1H-indazol-4-yl)-9-oxo-10H-pyrido[2,3-f]quinoxalin-5-yl]methanesulfonamide::US20260062412, Compound G5	Myelin transcription factor 1	Homo sapiens		 9.30							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795034	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795034&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293212	528826497							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237583	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(NS(=O)(=O)C3CC3)c3nccnc3c2[nH]c1=O	InChI=1S/C21H16FN7O3S/c22-13-4-3-10(12-8-26-28-17(12)13)15-11-7-14(29-33(31,32)9-1-2-9)19-20(25-6-5-24-19)18(11)27-21(30)16(15)23/h3-9,29H,1-2,23H2,(H,26,28)(H,27,30)	UFUZJFSQCMAYAT-UHFFFAOYSA-N	795035	N-[8-amino-7-(7-fluoro-1H-indazol-4-yl)-9-oxo-10H-pyrido[2,3-f]quinoxalin-5-yl]cyclopropanesulfonamide::US20260062412, Compound G6	Myelin transcription factor 1	Homo sapiens		 7.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795035	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795035&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293703	528826498							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237584	CN1CCN(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3nccnc23)CC1	InChI=1S/C23H21FN8O/c1-31-6-8-32(9-7-31)16-10-13-17(12-2-3-15(24)19-14(12)11-28-30-19)18(25)23(33)29-20(13)22-21(16)26-4-5-27-22/h2-5,10-11H,6-9,25H2,1H3,(H,28,30)(H,29,33)	JYUNJIZMPQUNFH-UHFFFAOYSA-N	795036	8-Amino-7-(7-fluoro-1H-indazol-4-yl)-5-(4-methylpiperazin-1-yl)-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G7	Myelin transcription factor 1	Homo sapiens		 2.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795036	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795036&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293633	528826499							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237585	CC(=O)Nc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2nccnc12	InChI=1S/C20H14FN7O2/c1-8(29)26-13-6-10-14(9-2-3-12(21)16-11(9)7-25-28-16)15(22)20(30)27-17(10)19-18(13)23-4-5-24-19/h2-7H,22H2,1H3,(H,25,28)(H,26,29)(H,27,30)	MXZVEGRTPGYIEP-UHFFFAOYSA-N	795037	N-[8-amino-7-(7-fluoro-1H-indazol-4-yl)-9-oxo-10H-pyrido[2,3-f]quinoxalin-5-yl]acetamide::US20260062412, Compound G8	Myelin transcription factor 1	Homo sapiens		 1.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795037	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795037&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293193	528826500							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237586	CC(C)Nc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2nccnc12	InChI=1S/C21H18FN7O/c1-9(2)27-14-7-11-15(10-3-4-13(22)17-12(10)8-26-29-17)16(23)21(30)28-18(11)20-19(14)24-5-6-25-20/h3-9,27H,23H2,1-2H3,(H,26,29)(H,28,30)	UPVIYKXHJNSUPR-UHFFFAOYSA-N	795038	8-Amino-7-(7-fluoro-1H-indazol-4-yl)-5-(propan-2-ylamino)-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G9	Myelin transcription factor 1	Homo sapiens		 4.40							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795038	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795038&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293143	528826501							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237587	COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2nccnc12	InChI=1S/C19H13FN6O2/c1-28-12-6-9-13(8-2-3-11(20)15-10(8)7-24-26-15)14(21)19(27)25-16(9)18-17(12)22-4-5-23-18/h2-7H,21H2,1H3,(H,24,26)(H,25,27)	IUKYKLQQWBRINI-UHFFFAOYSA-N	795039	8-Amino-7-(7-fluoro-1H-indazol-4-yl)-5-methoxy-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G10	Myelin transcription factor 1	Homo sapiens		 2.20							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795039	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795039&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293480	528826502							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237588	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCC3CC3)c3nccnc3c2[nH]c1=O	InChI=1S/C22H17FN6O2/c23-14-4-3-11(13-8-27-29-18(13)14)16-12-7-15(31-9-10-1-2-10)20-21(26-6-5-25-20)19(12)28-22(30)17(16)24/h3-8,10H,1-2,9,24H2,(H,27,29)(H,28,30)	JJKLLAVFXDITBW-UHFFFAOYSA-N	795040	8-Amino-5-(cyclopropylmethoxy)-7-(7-fluoro-1H-indazol-4-yl)-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G11	Myelin transcription factor 1	Homo sapiens		 2.50							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795040	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795040&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293587	528826503							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237589	N#C[C@H]1C[C@H](Oc2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3nccnc23)C1	InChI=1S/C23H16FN7O2/c24-15-2-1-12(14-9-29-31-19(14)15)17-13-7-16(33-11-5-10(6-11)8-25)21-22(28-4-3-27-21)20(13)30-23(32)18(17)26/h1-4,7,9-11H,5-6,26H2,(H,29,31)(H,30,32)	PLRLYHKXQPODAK-UHFFFAOYSA-N	795041	(1r,3r)-3-[[8-Amino-7-(7-fluoro-1H-indazol-4-yl)-9-oxo-10H-pyrido[2,3-f]quinoxalin-5-yl]oxy]cyclobutane-1-carbonitrile::US20260062412, Compound G12	Myelin transcription factor 1	Homo sapiens		 0.950							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795041	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795041&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293542	528826504							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237590	CC[C@H](C)Oc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2nccnc12	InChI=1S/C22H19FN6O2/c1-3-10(2)31-15-8-12-16(11-4-5-14(23)18-13(11)9-27-29-18)17(24)22(30)28-19(12)21-20(15)25-6-7-26-21/h4-10H,3,24H2,1-2H3,(H,27,29)(H,28,30)	SGAOXFXXQXBAGB-UHFFFAOYSA-N	795042	8-Amino-5-[(2S)-butan-2-yl]oxy-7-(7-fluoro-1H-indazol-4-yl)-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G13	Myelin transcription factor 1	Homo sapiens		 0.490							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795042	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795042&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293469	528826505							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237591	CC[C@@H](C)Oc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2nccnc12	InChI=1S/C22H19FN6O2/c1-3-10(2)31-15-8-12-16(11-4-5-14(23)18-13(11)9-27-29-18)17(24)22(30)28-19(12)21-20(15)25-6-7-26-21/h4-10H,3,24H2,1-2H3,(H,27,29)(H,28,30)	SGAOXFXXQXBAGB-UHFFFAOYSA-N	795043	8-Amino-5-[(2R)-butan-2-yl]oxy-7-(7-fluoro-1H-indazol-4-yl)-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G14	Myelin transcription factor 1	Homo sapiens		 0.690							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795043	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795043&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293272	528826506							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237592	CC(C)Oc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2nccnc12	InChI=1S/C21H17FN6O2/c1-9(2)30-14-7-11-15(10-3-4-13(22)17-12(10)8-26-28-17)16(23)21(29)27-18(11)20-19(14)24-5-6-25-20/h3-9H,23H2,1-2H3,(H,26,28)(H,27,29)	DIHCBEWYOWWSSM-UHFFFAOYSA-N	795044	8-Amino-7-(7-fluoro-1H-indazol-4-yl)-5-propan-2-yloxy-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G15	Myelin transcription factor 1	Homo sapiens		 1.60							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795044	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795044&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293901	528826507							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237593	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(O[C@H]3C[C@H](F)C3)c3nccnc3c2[nH]c1=O	InChI=1S/C22H16F2N6O2/c23-9-5-10(6-9)32-15-7-12-16(11-1-2-14(24)18-13(11)8-28-30-18)17(25)22(31)29-19(12)21-20(15)26-3-4-27-21/h1-4,7-10H,5-6,25H2,(H,28,30)(H,29,31)	RUEFIPXCJVWKRU-UHFFFAOYSA-N	795045	8-Amino-5-((1,3r)-3-fluorocyclobutyl)oxy-7-(7-fluoro-1H-indazol-4-yl)-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G16	Myelin transcription factor 1	Homo sapiens		 0.910							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795045	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795045&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293778	528826508							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
237594	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(O[C@H]3C[C@@H](F)C3)c3nccnc3c2[nH]c1=O	InChI=1S/C22H16F2N6O2/c23-9-5-10(6-9)32-15-7-12-16(11-1-2-14(24)18-13(11)8-28-30-18)17(25)22(31)29-19(12)21-20(15)26-3-4-27-21/h1-4,7-10H,5-6,25H2,(H,28,30)(H,29,31)	RUEFIPXCJVWKRU-UHFFFAOYSA-N	795046	8-Amino-5-((1s,3s)-3-fluorocyclobutyl)oxy-7-(7-fluoro-1H-indazol-4-yl)-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G17	Myelin transcription factor 1	Homo sapiens		 0.850							US Patent		10.7270/Q2S75N9Z			US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795046	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795046&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293778	528826509							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741140	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(OCCC(F)F)c3nccnc3c2[nH]c1=O	InChI=1S/C21H15F3N6O2/c22-12-2-1-9(11-8-28-30-17(11)12)15-10-7-13(32-6-3-14(23)24)19-20(27-5-4-26-19)18(10)29-21(31)16(15)25/h1-2,4-5,7-8,14H,3,6,25H2,(H,28,30)(H,29,31)	WQXNCSFGABHUPG-UHFFFAOYSA-N	795047	8-Amino-5-(3,3-difluoropropoxy)-7-(7-fluoro-1H-indazol-4-yl)-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G18	Myelin transcription factor 1	Homo sapiens		 0.790							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795047	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795047&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293264	528826510							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741141	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3cnsc3c2[nH]c1=O	InChI=1S/C17H9BrFN5OS/c18-10-3-7-12(6-1-2-11(19)14-8(6)4-21-24-14)13(20)17(25)23-15(7)16-9(10)5-22-26-16/h1-5H,20H2,(H,21,24)(H,23,25)	SHPWWFBPBWAWAI-UHFFFAOYSA-N	795048	7-Amino-4-bromo-6-(7-fluoro-1H-indazol-4-yl)-9H-[1,2]thiazolo[4,5-h]quinolin-8-one::US20260062412, Compound H1	Myelin transcription factor 1	Homo sapiens		 6.20							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795048	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795048&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293219	528826511							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741142	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2sncc12	InChI=1S/C18H12FN5OS/c1-7-4-9-13(8-2-3-12(19)15-11(8)5-21-24-15)14(20)18(25)23-16(9)17-10(7)6-22-26-17/h2-6H,20H2,1H3,(H,21,24)(H,23,25)	NTCYIEKXQXYXGU-UHFFFAOYSA-N	795049	7-Amino-6-(7-fluoro-1H-indazol-4-yl)-4-methyl-9H-[1.2]thiazolo[4,5-h]quinolin-8-one::US20260062412, Compound H2	Myelin transcription factor 1	Homo sapiens		 1.80							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795049	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795049&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293928	528826512							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741143	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3cnsc3c2[nH]c1=O	InChI=1S/C20H14FN5OS/c21-14-4-3-9(12-6-23-26-17(12)14)15-11-5-10(8-1-2-8)13-7-24-28-19(13)18(11)25-20(27)16(15)22/h3-8H,1-2,22H2,(H,23,26)(H,25,27)	YQGCROOYJXQTLY-UHFFFAOYSA-N	795050	7-Amino-4-cyclopropyl-6-(7-fluoro-1H-indazol-4-yl)-9H-[1,2]thiazolo[4,5-h]quinolin-8-one::US20260062412, Compound H3	Myelin transcription factor 1	Homo sapiens		 2.70							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795050	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795050&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293170	528826513							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741144	Cn1ncc2c(Br)cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c21	InChI=1S/C18H12BrFN6O/c1-26-17-10(6-23-26)11(19)4-8-13(14(21)18(27)24-16(8)17)7-2-3-12(20)15-9(7)5-22-25-15/h2-6H,21H2,1H3,(H,22,25)(H,24,27)	YUKVGTKTAKBBPR-UHFFFAOYSA-N	795051	7-Amino-4-bromo-6-(7-fluoro-1H-indazol-4-yl)-1-methyl-9H-pyrazolo[4,3-h]quinolin-8-one::US20260062412, Compound I1	Myelin transcription factor 1	Homo sapiens		 33.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795051	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795051&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293801	528826514							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741145	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2c1cnn2C	InChI=1S/C19H15FN6O/c1-8-5-10-14(9-3-4-13(20)16-12(9)6-22-25-16)15(21)19(27)24-17(10)18-11(8)7-23-26(18)2/h3-7H,21H2,1-2H3,(H,22,25)(H,24,27)	ISXTWOQAUQKUAO-UHFFFAOYSA-N	795052	7-Amino-6-(7-fluoro-1H-indazol-4-yl)-1,4-dimethyl-9H-pyrazolo[4,3-h]quinolin-8-one::US20260062412, Compound I2	Myelin transcription factor 1	Homo sapiens		 16.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795052	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795052&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293822	528826515							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741146	Cn1ncc2c(C3CC3)cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c21	InChI=1S/C21H17FN6O/c1-28-20-14(8-25-28)11(9-2-3-9)6-12-16(17(23)21(29)26-19(12)20)10-4-5-15(22)18-13(10)7-24-27-18/h4-9H,2-3,23H2,1H3,(H,24,27)(H,26,29)	PNDCYYMHOIYGNV-UHFFFAOYSA-N	795053	7-Amino-4-cyclopropyl-6-(7-fluoro-1H-indazol-4-yl)-1-methyl-9H-pyrazolo[4,3-h]quinolin-8-one::US20260062412, Compound I3	Myelin transcription factor 1	Homo sapiens		 8.00							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795053	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795053&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293818	528826516							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741147	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3cncnc3c2[nH]c1=O	InChI=1S/C18H10BrFN6O/c19-11-3-8-13(7-1-2-12(20)15-9(7)5-24-26-15)14(21)18(27)25-17(8)16-10(11)4-22-6-23-16/h1-6H,21H2,(H,24,26)(H,25,27)	QAEILQZDGZYSAV-UHFFFAOYSA-N	795054	8-Amino-5-bromo-7-(7-fluoro-1H-indazol-4-yl)-10H-pyrido[3,2-h]quinazolin-9-one::US20260062412, Compound J1	Myelin transcription factor 1	Homo sapiens		 7.30							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795054	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795054&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293544	528826517							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741148	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ncncc12	InChI=1S/C19H13FN6O/c1-8-4-10-14(9-2-3-13(20)16-12(9)6-24-26-16)15(21)19(27)25-18(10)17-11(8)5-22-7-23-17/h2-7H,21H2,1H3,(H,24,26)(H,25,27)	IJPICBDRPQANDE-UHFFFAOYSA-N	795055	8-Amino-7-(7-fluoro-1H-indazol-4-yl)-5-methyl-10H-pyrido[3,2-h]quinazolin-9-one::US20260062412, Compound J2	Myelin transcription factor 1	Homo sapiens		 3.10							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795055	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795055&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293669	528826518							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741149	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3cncnc3c2[nH]c1=O	InChI=1S/C21H15FN6O/c22-15-4-3-10(14-7-26-28-18(14)15)16-12-5-11(9-1-2-9)13-6-24-8-25-19(13)20(12)27-21(29)17(16)23/h3-9H,1-2,23H2,(H,26,28)(H,27,29)	UURQTSAKXONDQY-UHFFFAOYSA-N	795056	8-Amino-5-cyclopropyl-7-(7-fluoro-1H-indazol-4-yl)-10H-pyrido[3,2-h]quinazolin-9-one::US20260062412, Compound J3	Myelin transcription factor 1	Homo sapiens		 3.50							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795056	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795056&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293295	528826519							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741150	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3ncsc3c2[nH]c1=O	InChI=1S/C17H9BrFN5OS/c18-9-3-7-11(6-1-2-10(19)13-8(6)4-22-24-13)12(20)17(25)23-14(7)16-15(9)21-5-26-16/h1-5H,20H2,(H,22,24)(H,23,25)	BQUKVEWGKPTVTF-UHFFFAOYSA-N	795057	7-Amino-4-bromo-6-(7-fluoro-1H-indazol-4-yl)-9H-[1,3]thiazolo[4,5-h]quinolin-8-one::US20260062412, Compound K1	Myelin transcription factor 1	Homo sapiens		 1.70							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795057	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795057&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293456	528826520							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741151	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2scnc12	InChI=1S/C18H12FN5OS/c1-7-4-9-12(8-2-3-11(19)15-10(8)5-22-24-15)13(20)18(25)23-16(9)17-14(7)21-6-26-17/h2-6H,20H2,1H3,(H,22,24)(H,23,25)	AIHUPSYXHAVAEG-UHFFFAOYSA-N	795058	7-Amino-6-(7-fluoro-1H-indazol-4-yl)-4-methyl-9H-[1,3]thiazolo[4,5-h]quinolin-8-one::US20260062412, Compound K2	Myelin transcription factor 1	Homo sapiens		 1.20							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795058	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795058&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293279	528826521							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741152	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3ncsc3c2[nH]c1=O	InChI=1S/C20H14FN5OS/c21-13-4-3-9(12-6-24-26-16(12)13)14-11-5-10(8-1-2-8)17-19(28-7-23-17)18(11)25-20(27)15(14)22/h3-8H,1-2,22H2,(H,24,26)(H,25,27)	LBLGVAWQALSOLT-UHFFFAOYSA-N	795059	7-Amino-4-cyclopropyl-6-(7-fluoro-1H-indazol-4-yl)-9H-[1,3]thiazolo[4,5-h]quinolin-8-one::US20260062412, Compound K3	Myelin transcription factor 1	Homo sapiens		 50.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795059	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795059&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293929	528826522							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741153	Cc1nc2c(C)cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c2s1	InChI=1S/C19H14FN5OS/c1-7-5-10-13(9-3-4-12(20)16-11(9)6-22-25-16)14(21)19(26)24-17(10)18-15(7)23-8(2)27-18/h3-6H,21H2,1-2H3,(H,22,25)(H,24,26)	YFGJKPUTQXNLMI-UHFFFAOYSA-N	795060	7-Amino-6-(7-fluoro-1H-indazol-4-yl)-2,4-dimethyl-9H-[1,3]thiazolo[4,5-h]quinolin-8-one::US20260062412, Compound K4	Myelin transcription factor 1	Homo sapiens		 2.70							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795060	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795060&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293876	528826523							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741154	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3ccsc3c2[nH]c1=O	InChI=1S/C18H10BrFN4OS/c19-11-5-9-13(7-1-2-12(20)15-10(7)6-22-24-15)14(21)18(25)23-16(9)17-8(11)3-4-26-17/h1-6H,21H2,(H,22,24)(H,23,25)	HVMBYAPIXYMPBE-UHFFFAOYSA-N	795061	7-Amino-4-bromo-6-(7-fluoro-1H-indazol-4-yl)-9H-thieno[3,2-h]quinolin-8-one::US20260062412, Compound L1	Myelin transcription factor 1	Homo sapiens		 3.00							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795061	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795061&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293224	528826524							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741155	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2sccc12	InChI=1S/C19H13FN4OS/c1-8-6-11-14(10-2-3-13(20)16-12(10)7-22-24-16)15(21)19(25)23-17(11)18-9(8)4-5-26-18/h2-7H,21H2,1H3,(H,22,24)(H,23,25)	SUGPOOQINLZYNO-UHFFFAOYSA-N	795062	7-Amino-6-(7-fluoro-1H-indazol-4-yl)-4-methyl-9H-thieno[3,2-h]quinolin-8-one::US20260062412, Compound L2	Myelin transcription factor 1	Homo sapiens		 1.80							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795062	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795062&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293509	528826525							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741156	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3ccsc3c2[nH]c1=O	InChI=1S/C21H15FN4OS/c22-15-4-3-10(14-8-24-26-18(14)15)16-13-7-12(9-1-2-9)11-5-6-28-20(11)19(13)25-21(27)17(16)23/h3-9H,1-2,23H2,(H,24,26)(H,25,27)	SRWCLKJWOZKHJN-UHFFFAOYSA-N	795063	7-Amino-4-cyclopropyl-6-(7-fluoro-1H-indazol-4-yl)-9H-thieno[3,2-h]quinolin-8-one::US20260062412, Compound L3	Myelin transcription factor 1	Homo sapiens		 2.30							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795063	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795063&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293850	528826526							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741157	Cn1cnc2c3[nH]c(=O)c(N)c(-c4ccc(F)c5[nH]ncc45)c3cc(Br)c21	InChI=1S/C18H12BrFN6O/c1-26-6-22-16-15-8(4-10(19)17(16)26)12(13(21)18(27)24-15)7-2-3-11(20)14-9(7)5-23-25-14/h2-6H,21H2,1H3,(H,23,25)(H,24,27)	BUYNGWLQFOPSPG-UHFFFAOYSA-N	795064	7-Amino-4-bromo-6-(7-fluoro-1H-indazol-4-yl)-3-methyl-9H-imidazo[4,5-h]quinolin-8-one::US20260062412, Compound M1	Myelin transcription factor 1	Homo sapiens		 10.00							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795064	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795064&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293681	528826527							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741158	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ncn(C)c12	InChI=1S/C19H15FN6O/c1-8-5-10-13(9-3-4-12(20)15-11(9)6-23-25-15)14(21)19(27)24-16(10)17-18(8)26(2)7-22-17/h3-7H,21H2,1-2H3,(H,23,25)(H,24,27)	YYWLXWQKOXMCBQ-UHFFFAOYSA-N	795065	7-Amino-6-(7-fluoro-1H-indazol-4-yl)-3,4-dimethyl-9H-imidazo[4,5-h]quinolin-8-one::US20260062412, Compound M2	Myelin transcription factor 1	Homo sapiens		 14.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795065	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795065&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293558	528826528							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741159	Cn1cnc2c3[nH]c(=O)c(N)c(-c4ccc(F)c5[nH]ncc45)c3ccc21	InChI=1S/C18H13FN6O/c1-25-7-21-17-12(25)5-3-9-13(14(20)18(26)23-16(9)17)8-2-4-11(19)15-10(8)6-22-24-15/h2-7H,20H2,1H3,(H,22,24)(H,23,26)	HQSIFBZXOCFIJE-UHFFFAOYSA-N	795066	7-Amino-6-(7-fluoro-1H-indazol-4-yl)-3-methyl-9H-imidazo[4,5-h]quinolin-8-one::US20260062412, Compound M3	Myelin transcription factor 1	Homo sapiens		 99.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795066	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795066&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293132	528826529							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741160	Cn1cnc2c3[nH]c(=O)c(N)c(-c4ccc(F)c5[nH]ncc45)c3cc(C3CC3)c21	InChI=1S/C21H17FN6O/c1-28-8-24-19-18-12(6-11(20(19)28)9-2-3-9)15(16(23)21(29)26-18)10-4-5-14(22)17-13(10)7-25-27-17/h4-9H,2-3,23H2,1H3,(H,25,27)(H,26,29)	PTBBGWGLAVEBMH-UHFFFAOYSA-N	795067	7-Amino-4-cyclopropyl-6-(7-fluoro-1H-indazol-4-yl)-3-methyl-9H-imidazo[4,5-h]quinolin-8-one::US20260062412, Compound M4	Myelin transcription factor 1	Homo sapiens		 19.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795067	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795067&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293524	528826530							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741161	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3scnc3c2[nH]c1=O	InChI=1S/C17H9BrFN5OS/c18-9-3-7-11(6-1-2-10(19)13-8(6)4-22-24-13)12(20)17(25)23-14(7)15-16(9)26-5-21-15/h1-5H,20H2,(H,22,24)(H,23,25)	AYOLKKDRIBAHOZ-UHFFFAOYSA-N	795068	7-Amino-4-bromo-6-(7-fluoro-1H-indazol-4-yl)-9H-[1,3]thiazolo[5,4-h]quinolin-8-one::US20260062412, Compound N1	Myelin transcription factor 1	Homo sapiens		 5.30							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795068	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795068&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293280	528826531							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741162	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3scnc3c2[nH]c1=O	InChI=1S/C20H14FN5OS/c21-13-4-3-9(12-6-24-26-16(12)13)14-11-5-10(8-1-2-8)19-18(23-7-28-19)17(11)25-20(27)15(14)22/h3-8H,1-2,22H2,(H,24,26)(H,25,27)	FUJNVWAUENNRPF-UHFFFAOYSA-N	795069	7-Amino-4-cyclopropyl-6-(7-fluoro-1H-indazol-4-yl)-9H-[1,3]thiazolo[5,4-h]quinolin-8-one::US20260062412, Compound N2	Myelin transcription factor 1	Homo sapiens		 3.30							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795069	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795069&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293253	528826532							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741163	Cc1nc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C19H13FN6O/c1-8-15-10(3-2-6-22-15)17-18(24-8)13(14(21)19(27)25-17)9-4-5-12(20)16-11(9)7-23-26-16/h2-7H,21H2,1H3,(H,23,26)(H,25,27)	NHPNZAYUPBUIQJ-UHFFFAOYSA-N	795070	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-methyl-1H-pyrido[2,3-h][1,5]naphthyridin-2-one::US20260062412, Compound O1	Myelin transcription factor 1	Homo sapiens		 1.10							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795070	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795070&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293459	528826533							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741164	Nc1c(-c2cccc3[nH]ncc23)c2cc(C3CC3)c3cnccc3c2[nH]c1=O	InChI=1S/C22H17N5O/c23-20-19(12-2-1-3-18-17(12)10-25-27-18)15-8-14(11-4-5-11)16-9-24-7-6-13(16)21(15)26-22(20)28/h1-3,6-11H,4-5,23H2,(H,25,27)(H,26,28)	XVHRRRWCVFHSER-UHFFFAOYSA-N	795071	3-Amino-6-cyclopropyl-4-(1H-indazol-4-yl)-1H-1,8-phenanthrolin-2-one::US20260062412, Compound P1	Myelin transcription factor 1	Homo sapiens		 1.80							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795071	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795071&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293330	528826534							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741165	Cc1nccc2c1c(Br)cc1c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C20H13BrFN5O/c1-8-15-10(4-5-24-8)18-11(6-13(15)21)16(17(23)20(28)26-18)9-2-3-14(22)19-12(9)7-25-27-19/h2-7H,23H2,1H3,(H,25,27)(H,26,28)	KMZCSKFMXAWGIF-UHFFFAOYSA-N	795072	3-Amino-6-bromo-4-(7-fluoro-1H-indazol-4-yl)-7-methyl-1H-1,8-phenanthrolin-2-one::US20260062412, Compound P2	Myelin transcription factor 1	Homo sapiens		 13.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795072	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795072&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293746	528826535							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741166	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3cnccc3c2[nH]c1=O	InChI=1S/C19H11BrFN5O/c20-13-5-10-15(8-1-2-14(21)18-12(8)7-24-26-18)16(22)19(27)25-17(10)9-3-4-23-6-11(9)13/h1-7H,22H2,(H,24,26)(H,25,27)	ZHUHQMMVPXISEX-UHFFFAOYSA-N	795073	3-Amino-6-bromo-4-(7-fluoro-1H-indazol-4-yl)-1H-1,8-phenanthrolin-2-one::US20260062412, Compound P3	Myelin transcription factor 1	Homo sapiens		 12.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795073	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795073&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293154	528826536							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741167	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3cnccc3c2[nH]c1=O	InChI=1S/C22H16FN5O/c23-17-4-3-11(16-9-26-28-21(16)17)18-14-7-13(10-1-2-10)15-8-25-6-5-12(15)20(14)27-22(29)19(18)24/h3-10H,1-2,24H2,(H,26,28)(H,27,29)	XJHHNXUOQBEFJY-UHFFFAOYSA-N	795074	3-Amino-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,8-phenanthrolin-2-one 2,2,2-trifluoroacetate::US20260062412, Compound P4	Myelin transcription factor 1	Homo sapiens		 6.10							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795074	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795074&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293259	528826537							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741168	Nc1c(-c2cccc(O)c2)c2ccc3cnccc3c2[nH]c1=O	InChI=1S/C18H13N3O2/c19-16-15(10-2-1-3-12(22)8-10)14-5-4-11-9-20-7-6-13(11)17(14)21-18(16)23/h1-9,22H,19H2,(H,21,23)	DLNHEKJTVHYITM-UHFFFAOYSA-N	795075	3-Amino-4-(3-hydroxyphenyl)-1H-1,8-phenanthrolin-2-one; hydrobromide::US20260062412, Compound P5	Myelin transcription factor 1	Homo sapiens		 3.90							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795075	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795075&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293263	528826538							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741169	Nc1c(-c2cccc3[nH]ncc23)c2cc(C3CC3)c3ccncc3c2[nH]c1=O	InChI=1S/C22H17N5O/c23-20-19(13-2-1-3-18-16(13)10-25-27-18)15-8-14(11-4-5-11)12-6-7-24-9-17(12)21(15)26-22(20)28/h1-3,6-11H,4-5,23H2,(H,25,27)(H,26,28)	BKEXKGVSTVZXJB-UHFFFAOYSA-N	795076	3-Amino-6-cyclopropyl-4-(1H-indazol-4-yl)-1H-1,9-phenanthrolin-2-one::US20260062412, Compound Q1	Myelin transcription factor 1	Homo sapiens		 9.30							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795076	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795076&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293150	528826539							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741170	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cnc3ccccc3c2[nH]c1=O	InChI=1S/C19H12FN5O/c20-13-6-5-9(11-8-23-25-18(11)13)15-12-7-22-14-4-2-1-3-10(14)17(12)24-19(26)16(15)21/h1-8H,21H2,(H,23,25)(H,24,26)	NMIGXJHOMYINIX-UHFFFAOYSA-N	795077	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h][1,6]naphthyridin-2-one::US20260062412, Compound R1	Myelin transcription factor 1	Homo sapiens		 3.40							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795077	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795077&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293436	528826540							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741171	Cc1cc2c(nn1)c(Br)cc1c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C19H12BrFN6O/c1-7-4-10-16-9(5-12(20)17(10)27-25-7)14(15(22)19(28)24-16)8-2-3-13(21)18-11(8)6-23-26-18/h2-6H,22H2,1H3,(H,23,26)(H,24,28)	XZCJGYSNSIOLPM-UHFFFAOYSA-N	795078	3-Amino-6-bromo-4-(7-fluoro-1H-indazol-4-yl)-9-methyl-1H-pyrido[2,3-f]cinnolin-2-one::US20260062412, Compound S1	Myelin transcription factor 1	Homo sapiens		 370							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795078	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795078&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			176112739	528826541							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741172	COc1ccc2c(n1)c(OC)cc1c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C21H16FN5O3/c1-29-14-7-11-16(9-3-5-13(22)19-12(9)8-24-27-19)17(23)21(28)26-18(11)10-4-6-15(30-2)25-20(10)14/h3-8H,23H2,1-2H3,(H,24,27)(H,26,28)	KLDAJPXNMSTVJS-UHFFFAOYSA-N	795079	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6,8-dimethoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound T1	Myelin transcription factor 1	Homo sapiens		 4.90							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795079	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795079&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293477	528826542							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741173	COc1ccc2c(n1)c(OC(C)C)cc1c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c12	InChI=1S/C23H20FN5O3/c1-10(2)32-16-8-13-18(11-4-6-15(24)21-14(11)9-26-29-21)19(25)23(30)28-20(13)12-5-7-17(31-3)27-22(12)16/h4-10H,25H2,1-3H3,(H,26,29)(H,28,30)	WISKCXAXZJLREL-UHFFFAOYSA-N	795080	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-8-methoxy-6-propan-2-yloxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound T2	Myelin transcription factor 1	Homo sapiens		 7.60							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795080	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795080&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293218	528826543							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741174	CCOc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccc(OC)nc12	InChI=1S/C22H18FN5O3/c1-3-31-15-8-12-17(10-4-6-14(23)20-13(10)9-25-28-20)18(24)22(29)27-19(12)11-5-7-16(30-2)26-21(11)15/h4-9H,3,24H2,1-2H3,(H,25,28)(H,27,29)	QYZCZENBKDUCPD-UHFFFAOYSA-N	795081	3-Amino-6-ethoxy-4-(7-fluoro-1H-indazol-4-yl)-8-methoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound T3	Myelin transcription factor 1	Homo sapiens		 6.10							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795081	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795081&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293783	528826544							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741175	COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccc(=O)[nH]c12	InChI=1S/C20H14FN5O3/c1-29-13-6-10-15(8-2-4-12(21)18-11(8)7-23-26-18)16(22)20(28)25-17(10)9-3-5-14(27)24-19(9)13/h2-7H,22H2,1H3,(H,23,26)(H,24,27)(H,25,28)	DNKACRFGXVKQJE-UHFFFAOYSA-N	795082	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-methoxy-1,7-dihydro-1,7-phenanthroline-2,8-dione::US20260062412, Compound T4	Myelin transcription factor 1	Homo sapiens		 3.20							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795082	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795082&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293554	528826545							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741176	CC(C)Oc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccc(=O)[nH]c12	InChI=1S/C22H18FN5O3/c1-9(2)31-15-7-12-17(10-3-5-14(23)20-13(10)8-25-28-20)18(24)22(30)27-19(12)11-4-6-16(29)26-21(11)15/h3-9H,24H2,1-2H3,(H,25,28)(H,26,29)(H,27,30)	GTBRKARIFCGGBQ-UHFFFAOYSA-N	795083	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-propan-2-yloxy-1,7-dihydro-1,7-phenanthroline-2,8-dione::US20260062412, Compound T5	Myelin transcription factor 1	Homo sapiens		 3.50							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795083	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795083&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293438	528826546							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741177	CCOc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccc(=O)[nH]c12	InChI=1S/C21H16FN5O3/c1-2-30-14-7-11-16(9-3-5-13(22)19-12(9)8-24-27-19)17(23)21(29)26-18(11)10-4-6-15(28)25-20(10)14/h3-8H,2,23H2,1H3,(H,24,27)(H,25,28)(H,26,29)	DRJFOVZSQCWMIX-UHFFFAOYSA-N	795084	3-Amino-6-ethoxy-4-(7-fluoro-1H-indazol-4-yl)-1,7-dihydro-1,7-phenanthroline-2,8-dione::US20260062412, Compound T6	Myelin transcription factor 1	Homo sapiens		 2.20							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795084	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795084&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293498	528826547							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741178	Cc1c(C)c2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H15F2N5O/c1-8-9(2)18-10(4-3-5-25-18)19-14(8)15(17(24)21(29)27-19)11-6-13(22)16(23)20-12(11)7-26-28-20/h3-7H,24H2,1-2H3,(H,26,28)(H,27,29)	BEYQRIMLWKTWKP-UHFFFAOYSA-N	795085	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-5,6-dimethyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C216	Myelin transcription factor 1	Homo sapiens		 3.40							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795085	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795085&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293382	528826548							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741179	Cc1c(C2CC2)c2ncccc2c2[nH]c(=O)c(N)c(-c3cc(F)c(F)c4[nH]ncc34)c12	InChI=1S/C23H17F2N5O/c1-9-15(10-4-5-10)20-11(3-2-6-27-20)21-16(9)17(19(26)23(31)29-21)12-7-14(24)18(25)22-13(12)8-28-30-22/h2-3,6-8,10H,4-5,26H2,1H3,(H,28,30)(H,29,31)	PPJQGFBQSSHWTA-UHFFFAOYSA-N	795086	3-Amino-6-cyclopropyl-4-(6,7-difluoro-1H-indazol-4-yl)-5-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C217	Myelin transcription factor 1	Homo sapiens		 1.80							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795086	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795086&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293396	528826549							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741180	Cc1cc2ncccc2c2[nH]c(=O)c(N)c(-c3cc(F)c(F)c4[nH]ncc34)c12	InChI=1S/C20H13F2N5O/c1-8-5-13-9(3-2-4-24-13)18-14(8)15(17(23)20(28)26-18)10-6-12(21)16(22)19-11(10)7-25-27-19/h2-7H,23H2,1H3,(H,25,27)(H,26,28)	SYFRZWVJYQEMKP-UHFFFAOYSA-N	795087	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-5-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C218	Myelin transcription factor 1	Homo sapiens		 0.430							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795087	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795087&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293602	528826550							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741181	Cc1c(F)c2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H12F3N5O/c1-7-14(22)13-12(9-5-11(21)15(23)19-10(9)6-26-28-19)16(24)20(29)27-18(13)8-3-2-4-25-17(7)8/h2-6H,24H2,1H3,(H,26,28)(H,27,29)	ZDEHZYMJFMCCDC-UHFFFAOYSA-N	795088	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-5-fluoro-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C219	Myelin transcription factor 1	Homo sapiens		 2.10							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795088	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795088&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293191	528826551							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741182	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2c(F)c(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H14F3N5O/c23-12-6-10(11-7-28-30-21(11)16(12)24)14-15-17(25)13(8-3-4-8)19-9(2-1-5-27-19)20(15)29-22(31)18(14)26/h1-2,5-8H,3-4,26H2,(H,28,30)(H,29,31)	YRQKGNHGFVLDBB-UHFFFAOYSA-N	795089	3-Amino-6-cyclopropyl-4-(6,7-difluoro-1H-indazol-4-yl)-5-fluoro-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C220	Myelin transcription factor 1	Homo sapiens		 4.10							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795089	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795089&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293327	528826552							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741183	Nc1c(-c2cc(F)c(F)c3[nH]ncc23)c2c(F)cc3ncccc3c2[nH]c1=O	InChI=1S/C19H10F3N5O/c20-10-5-12-7(2-1-3-24-12)17-14(10)13(16(23)19(28)26-17)8-4-11(21)15(22)18-9(8)6-25-27-18/h1-6H,23H2,(H,25,27)(H,26,28)	IFCZSZNGNVZPSC-UHFFFAOYSA-N	795090	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-5-fluoro-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C221	Myelin transcription factor 1	Homo sapiens		 0.720							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795090	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795090&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293160	528826553							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741184	Cc1cc2c(-c3c(F)cc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H13F2N5O/c1-8-5-10-15(14-11-7-25-27-19(11)13(22)6-12(14)21)16(23)20(28)26-18(10)9-3-2-4-24-17(8)9/h2-7H,23H2,1H3,(H,25,27)(H,26,28)	ZQAFAOBMLWIYKH-UHFFFAOYSA-N	795091	3-Amino-4-(5,7-difluoro-1H-indazol-4-yl)-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C222	Myelin transcription factor 1	Homo sapiens		 1.40							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795091	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795091&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293133	528826554							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741185	Cc1cc2c(-c3nccc4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C19H14N6O/c1-9-7-11-14(18-12-8-23-25-13(12)4-6-22-18)15(20)19(26)24-17(11)10-3-2-5-21-16(9)10/h2-8H,20H2,1H3,(H,23,25)(H,24,26)	XUEUTQWEWQEFLO-UHFFFAOYSA-N	795092	3-Amino-6-methyl-4-(1H-pyrazolo[4,3-c]pyridin-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C223	Myelin transcription factor 1	Homo sapiens		 750							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795092	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795092&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293655	528826555							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741186	Cc1cc2c(-c3cccc4[nH]nnc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C19H14N6O/c1-9-8-12-14(10-4-2-6-13-18(10)24-25-23-13)15(20)19(26)22-17(12)11-5-3-7-21-16(9)11/h2-8H,20H2,1H3,(H,22,26)(H,23,24,25)	GNAWLUVJSKWDSB-UHFFFAOYSA-N	795093	3-Amino-4-(1H-benzotriazol-4-yl)-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C224	Myelin transcription factor 1	Homo sapiens		 3000							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795093	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795093&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293940	528826556							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741187	CC(C)(C)c1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C23H20FN5O/c1-23(2,3)15-9-13-17(11-6-7-16(24)21-14(11)10-27-29-21)18(25)22(30)28-19(13)12-5-4-8-26-20(12)15/h4-10H,25H2,1-3H3,(H,27,29)(H,28,30)	XTHJCBZZASKXPQ-UHFFFAOYSA-N	795094	3-Amino-6-(tert-butyl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C225	Myelin transcription factor 1	Homo sapiens		 1000							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795094	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795094&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293461	528826557							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741188	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Cl)c(Br)cc2[nH]c1=O	InChI=1S/C16H9BrCl2N4O/c17-9-4-12-7(3-11(9)19)13(14(20)16(24)22-12)6-1-2-10(18)15-8(6)5-21-23-15/h1-5H,20H2,(H,21,23)(H,22,24)	KTSKQHONYLQJGZ-UHFFFAOYSA-N	794684	3-Amino-7-bromo-6-chloro-4-(7-chloro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A27	Myelin transcription factor 1	Homo sapiens		 0.520							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794684	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794684&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293616	528826147							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741189	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Cl)c(OC(F)F)cc2[nH]c1=O	InChI=1S/C17H10Cl2F2N4O2/c18-9-2-1-6(8-5-23-25-15(8)9)13-7-3-10(19)12(27-17(20)21)4-11(7)24-16(26)14(13)22/h1-5,17H,22H2,(H,23,25)(H,24,26)	YNIHNDYYBMUDRX-UHFFFAOYSA-N	794687	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-7-(difluoromethoxy)-1H-quinolin-2-one::US20260062412, Compound A30	Myelin transcription factor 1	Homo sapiens		 0.710							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794687	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794687&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293316	528826150							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741190	Nc1c(-c2cc(F)cc3[nH]ncc23)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H10ClFN4O/c17-7-1-2-12-10(3-7)14(15(19)16(23)21-12)9-4-8(18)5-13-11(9)6-20-22-13/h1-6H,19H2,(H,20,22)(H,21,23)	CTYWKJSVQRBRSV-UHFFFAOYSA-N	794712	3-Amino-6-chloro-4-(6-fluoro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A56	Myelin transcription factor 1	Homo sapiens		 1.10							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794712	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794712&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293140	528826175							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741191	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H10ClFN4O/c17-7-1-4-12-9(5-7)13(14(19)16(23)21-12)8-2-3-11(18)15-10(8)6-20-22-15/h1-6H,19H2,(H,20,22)(H,21,23)	USGRRVXARARGEO-UHFFFAOYSA-N	794713	3-Amino-6-chloro-4-(7-fluoro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A57	Myelin transcription factor 1	Homo sapiens		 0.610							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794713	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794713&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293831	528826176							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741192	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C16H10Cl2N4O/c17-7-1-4-12-9(5-7)13(14(19)16(23)21-12)8-2-3-11(18)15-10(8)6-20-22-15/h1-6H,19H2,(H,20,22)(H,21,23)	YXKVRHAAENFPKJ-UHFFFAOYSA-N	794715	3-Amino-6-chloro-4-(7-chloro-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A59	Myelin transcription factor 1	Homo sapiens		 0.600							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794715	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794715&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293613	528826178							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741193	Cc1ccc(-c2c(N)c(=O)[nH]c3ccc(Cl)cc23)c2cn[nH]c12	InChI=1S/C17H13ClN4O/c1-8-2-4-10(12-7-20-22-16(8)12)14-11-6-9(18)3-5-13(11)21-17(23)15(14)19/h2-7H,19H2,1H3,(H,20,22)(H,21,23)	RQHRSWSSLBGBBW-UHFFFAOYSA-N	794716	3-Amino-6-chloro-4-(7-methyl-1H-indazol-4-yl)-1H-quinolin-2-one::US20260062412, Compound A60	Myelin transcription factor 1	Homo sapiens		 0.550							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794716	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794716&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293475	528826179							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741194	Nc1c(-c2ccc(C(F)(F)F)c3[nH]ncc23)c2cc(Cl)ccc2[nH]c1=O	InChI=1S/C17H10ClF3N4O/c18-7-1-4-12-9(5-7)13(14(22)16(26)24-12)8-2-3-11(17(19,20)21)15-10(8)6-23-25-15/h1-6H,22H2,(H,23,25)(H,24,26)	NMVHRSCBOHNZMV-UHFFFAOYSA-N	794717	3-Amino-6-chloro-4-[7-(trifluoromethyl)-1H-indazol-4-yl]-1H-quinolin-2-one::US20260062412, Compound A61	Myelin transcription factor 1	Homo sapiens		 5.00							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794717	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794717&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293441	528826180							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741195	Nc1c(-c2cccc(O)c2)c2ccc3ccccc3c2[nH]c1=O	InChI=1S/C19H14N2O2/c20-17-16(12-5-3-6-13(22)10-12)15-9-8-11-4-1-2-7-14(11)18(15)21-19(17)23/h1-10,22H,20H2,(H,21,23)	MBPNONCSDWAHCA-UHFFFAOYSA-N	794729	3-Amino-4-(3-hydroxyphenyl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B2	Myelin transcription factor 1	Homo sapiens		 4.00							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794729	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794729&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293937	528826192							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741196	Nc1c(-c2cccc(O)c2)c2cc(C3CC3)c3ccccc3c2[nH]c1=O	InChI=1S/C22H18N2O2/c23-20-19(13-4-3-5-14(25)10-13)18-11-17(12-8-9-12)15-6-1-2-7-16(15)21(18)24-22(20)26/h1-7,10-12,25H,8-9,23H2,(H,24,26)	BPJSTDLWYAENHZ-UHFFFAOYSA-N	794730	3-Amino-6-cyclopropyl-4-(3-hydroxyphenyl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B3	Myelin transcription factor 1	Homo sapiens		 0.520							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794730	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794730&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293234	528826193							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741197	N#Cc1cc2c(-c3cccc(O)c3)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C20H13N3O2/c21-10-12-9-16-17(11-4-3-5-13(24)8-11)18(22)20(25)23-19(16)15-7-2-1-6-14(12)15/h1-9,24H,22H2,(H,23,25)	YHYNXXIZLMHJKC-UHFFFAOYSA-N	794734	3-Amino-4-(3-hydroxyphenyl)-2-oxo-1H-benzo[h]quinoline-6-carbonitrile::US20260062412, Compound B7	Myelin transcription factor 1	Homo sapiens		 5.70							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794734	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794734&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293881	528826197							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741198	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3ccccc3c2[nH]c1=O	InChI=1S/C23H17FN4O/c24-18-8-7-13(17-10-26-28-22(17)18)19-16-9-15(11-5-6-11)12-3-1-2-4-14(12)21(16)27-23(29)20(19)25/h1-4,7-11H,5-6,25H2,(H,26,28)(H,27,29)	ZMVUHEXIDZMTQF-UHFFFAOYSA-N	794749	3-Amino-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B22	Myelin transcription factor 1	Homo sapiens		 0.250							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794749	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794749&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293622	528826212							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741199	CCc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C22H17FN4O/c1-2-11-9-15-18(13-7-8-17(23)21-16(13)10-25-27-21)19(24)22(28)26-20(15)14-6-4-3-5-12(11)14/h3-10H,2,24H2,1H3,(H,25,27)(H,26,28)	WXFGCKNRGPCFQC-UHFFFAOYSA-N	794750	3-Amino-6-ethyl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B23	Myelin transcription factor 1	Homo sapiens		 0.260							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794750	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794750&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293398	528826213							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741200	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCC3)c3ccccc3c2[nH]c1=O	InChI=1S/C24H19FN4O/c25-19-9-8-14(18-11-27-29-23(18)19)20-17-10-16(12-4-3-5-12)13-6-1-2-7-15(13)22(17)28-24(30)21(20)26/h1-2,6-12H,3-5,26H2,(H,27,29)(H,28,30)	WSIHCUQKGHWPIW-UHFFFAOYSA-N	794751	3-Amino-6-cyclobutyl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B24	Myelin transcription factor 1	Homo sapiens		 0.620							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794751	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794751&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293214	528826214							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741201	N#Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C21H12FN5O/c22-16-6-5-12(15-9-25-27-20(15)16)17-14-7-10(8-23)11-3-1-2-4-13(11)19(14)26-21(28)18(17)24/h1-7,9H,24H2,(H,25,27)(H,26,28)	YUBIURDSEFTDEV-UHFFFAOYSA-N	794753	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-2-oxo-1H-benzo[h]quinoline-6-carbonitrile::US20260062412, Compound B26	Myelin transcription factor 1	Homo sapiens		 0.370							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794753	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794753&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293500	528826216							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741202	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C21H15FN4O/c1-10-8-14-17(12-6-7-16(22)20-15(12)9-24-26-20)18(23)21(27)25-19(14)13-5-3-2-4-11(10)13/h2-9H,23H2,1H3,(H,24,26)(H,25,27)	QMANJWPRNPRPCY-UHFFFAOYSA-N	794754	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-methyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B27	Myelin transcription factor 1	Homo sapiens		 0.210							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794754	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794754&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293854	528826217							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741203	CP(C)(=O)c1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2ccccc12	InChI=1S/C22H18FN4O2P/c1-30(2,29)17-9-14-18(12-7-8-16(23)21-15(12)10-25-27-21)19(24)22(28)26-20(14)13-6-4-3-5-11(13)17/h3-10H,24H2,1-2H3,(H,25,27)(H,26,28)	KATJVJFDXQPFPI-UHFFFAOYSA-N	794758	3-Amino-6-dimethylphosphoryl-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B31	Myelin transcription factor 1	Homo sapiens		 0.320							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794758	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794758&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293657	528826221							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741204	Nc1c(-c2ccc(F)c3[nH]ncc23)c2ccc3ccccc3c2[nH]c1=O	InChI=1S/C20H13FN4O/c21-15-8-7-12(14-9-23-25-19(14)15)16-13-6-5-10-3-1-2-4-11(10)18(13)24-20(26)17(16)22/h1-9H,22H2,(H,23,25)(H,24,26)	AFCDRYCMAJNTBS-UHFFFAOYSA-N	794759	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B32	Myelin transcription factor 1	Homo sapiens		 0.260							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794759	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794759&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293220	528826222							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741205	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Cl)c3ccccc3c2[nH]c1=O	InChI=1S/C20H12ClFN4O/c21-14-7-12-16(10-5-6-15(22)19-13(10)8-24-26-19)17(23)20(27)25-18(12)11-4-2-1-3-9(11)14/h1-8H,23H2,(H,24,26)(H,25,27)	LZYBABQGXSNVHJ-UHFFFAOYSA-N	794761	3-Amino-6-chloro-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B34	Myelin transcription factor 1	Homo sapiens		 0.860							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794761	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794761&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293813	528826224							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741206	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(F)c3ccccc3c2[nH]c1=O	InChI=1S/C20H12F2N4O/c21-14-6-5-10(13-8-24-26-19(13)14)16-12-7-15(22)9-3-1-2-4-11(9)18(12)25-20(27)17(16)23/h1-8H,23H2,(H,24,26)(H,25,27)	JNZVVFYRJTWAJV-UHFFFAOYSA-N	794762	3-Amino-6-fluoro-4-(7-fluoro-1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B35	Myelin transcription factor 1	Homo sapiens		 0.440							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794762	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794762&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293568	528826225							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741207	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C3CC3)c3ccccc3c2[nH]c1=O	InChI=1S/C23H17ClN4O/c24-18-8-7-13(17-10-26-28-22(17)18)19-16-9-15(11-5-6-11)12-3-1-2-4-14(12)21(16)27-23(29)20(19)25/h1-4,7-11H,5-6,25H2,(H,26,28)(H,27,29)	NKEOCOBPKVNCLZ-UHFFFAOYSA-N	794764	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-cyclopropyl-1H-benzo[h]quinolin-2-one::US20260062412, Compound B37	Myelin transcription factor 1	Homo sapiens		 0.750							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794764	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794764&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293443	528826227							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741208	Nc1c(-c2cccc3[nH]ncc23)c2ccc3ccccc3c2[nH]c1=O	InChI=1S/C20H14N4O/c21-18-17(13-6-3-7-16-15(13)10-22-24-16)14-9-8-11-4-1-2-5-12(11)19(14)23-20(18)25/h1-10H,21H2,(H,22,24)(H,23,25)	QMDOHABESUHWFL-UHFFFAOYSA-N	794773	3-Amino-4-(1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B46	Myelin transcription factor 1	Homo sapiens		 6.40							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794773	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794773&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293254	528826236							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741209	Nc1c(-c2cccc3[nH]ncc23)c2cc(C3CC3)c3ccc(F)cc3c2[nH]c1=O	InChI=1S/C23H17FN4O/c24-12-6-7-13-15(11-4-5-11)9-17-20(14-2-1-3-19-18(14)10-26-28-19)21(25)23(29)27-22(17)16(13)8-12/h1-3,6-11H,4-5,25H2,(H,26,28)(H,27,29)	MJDLGQBGEZVCMO-UHFFFAOYSA-N	794774	3-Amino-6-cyclopropyl-9-fluoro-4-(1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one::US20260062412, Compound B47	Myelin transcription factor 1	Homo sapiens		 1.10							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794774	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794774&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293334	528826237							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741210	Nc1c(-c2cccc3[nH]ncc23)c2cc(C3CC3)c3cc(F)ccc3c2[nH]c1=O	InChI=1S/C23H17FN4O/c24-12-6-7-14-16(8-12)15(11-4-5-11)9-17-20(21(25)23(29)27-22(14)17)13-2-1-3-19-18(13)10-26-28-19/h1-3,6-11H,4-5,25H2,(H,26,28)(H,27,29)	MPSOQTIARBCFIO-UHFFFAOYSA-N	794775	3-Amino-6-cyclopropyl-8-fluoro-4-(1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one; hydrochloride::US20260062412, Compound B48	Myelin transcription factor 1	Homo sapiens		 2.50							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794775	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794775&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293249	528826238							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741211	Nc1c(-c2cccc3[nH]ncc23)c2cc(C3CC3)c3ccccc3c2[nH]c1=O	InChI=1S/C23H18N4O/c24-21-20(14-6-3-7-19-18(14)11-25-27-19)17-10-16(12-8-9-12)13-4-1-2-5-15(13)22(17)26-23(21)28/h1-7,10-12H,8-9,24H2,(H,25,27)(H,26,28)	QHZKNLUIVZGKCR-UHFFFAOYSA-N	794776	3-Amino-6-cyclopropyl-4-(1H-indazol-4-yl)-1H-benzo[h]quinolin-2-one 2-propanol solvate::US20260062412, Compound B49	Myelin transcription factor 1	Homo sapiens		 6.40							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794776	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794776&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293863	528826239							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741212	Nc1c(-c2cccc(F)c2)c2ccc3ccccc3c2[nH]c1=O	InChI=1S/C19H13FN2O/c20-13-6-3-5-12(10-13)16-15-9-8-11-4-1-2-7-14(11)18(15)22-19(23)17(16)21/h1-10H,21H2,(H,22,23)	NSOFAMMWRKVIDV-UHFFFAOYSA-N	794777	3-Amino-4-(3-fluorophenyl)-1H-benzo[h]quinolin-2-one; hydrochloride::US20260062412, Compound B50	Myelin transcription factor 1	Homo sapiens		 210							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794777	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794777&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293371	528826240							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741213	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3ncccc3c2[nH]c1=O	InChI=1S/C19H11BrFN5O/c20-12-6-10-14(8-3-4-13(21)18-11(8)7-24-26-18)15(22)19(27)25-16(10)9-2-1-5-23-17(9)12/h1-7H,22H2,(H,24,26)(H,25,27)	DQRRECKYKYCQAW-UHFFFAOYSA-N	794778	3-Amino-6-bromo-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C1	Myelin transcription factor 1	Homo sapiens		<0.170							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794778	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794778&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293706	528826241							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741214	COc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H14FN5O2/c1-28-14-7-11-15(9-4-5-13(21)18-12(9)8-24-26-18)16(22)20(27)25-17(11)10-3-2-6-23-19(10)14/h2-8H,22H2,1H3,(H,24,26)(H,25,27)	UZGVOKWMDFZQCU-UHFFFAOYSA-N	794781	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-methoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C4	Myelin transcription factor 1	Homo sapiens		 0.150							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794781	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794781&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293492	528826244							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741215	CCOc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H16FN5O2/c1-2-29-15-8-12-16(10-5-6-14(22)19-13(10)9-25-27-19)17(23)21(28)26-18(12)11-4-3-7-24-20(11)15/h3-9H,2,23H2,1H3,(H,25,27)(H,26,28)	MRTXNVJHKIGLQK-UHFFFAOYSA-N	794785	3-Amino-6-ethoxy-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C8	Myelin transcription factor 1	Homo sapiens		 0.300							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794785	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794785&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293442	528826248							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741216	CC(C)Oc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H18FN5O2/c1-10(2)30-16-8-13-17(11-5-6-15(23)20-14(11)9-26-28-20)18(24)22(29)27-19(13)12-4-3-7-25-21(12)16/h3-10H,24H2,1-2H3,(H,26,28)(H,27,29)	JHGYBATVADJEKA-UHFFFAOYSA-N	794790	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-propan-2-yloxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C13	Myelin transcription factor 1	Homo sapiens		 0.150							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794790	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794790&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293767	528826253							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741217	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(F)c3ncccc3c2[nH]c1=O	InChI=1S/C19H11F2N5O/c20-12-4-3-8(11-7-24-26-18(11)12)14-10-6-13(21)17-9(2-1-5-23-17)16(10)25-19(27)15(14)22/h1-7H,22H2,(H,24,26)(H,25,27)	DZGCMIUGLPUCIS-UHFFFAOYSA-N	794841	3-Amino-6-fluoro-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C64	Myelin transcription factor 1	Homo sapiens		 0.200							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794841	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794841&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293174	528826304							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741218	COc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H13F2N5O2/c1-29-13-6-10-14(9-5-12(21)15(22)19-11(9)7-25-27-19)16(23)20(28)26-17(10)8-3-2-4-24-18(8)13/h2-7H,23H2,1H3,(H,25,27)(H,26,28)	XFZXIJLXMACSSN-UHFFFAOYSA-N	794842	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-methoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C65	Myelin transcription factor 1	Homo sapiens		 0.083							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794842	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794842&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293543	528826305							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741219	CCOc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H15F2N5O2/c1-2-30-14-7-11-15(10-6-13(22)16(23)20-12(10)8-26-28-20)17(24)21(29)27-18(11)9-4-3-5-25-19(9)14/h3-8H,2,24H2,1H3,(H,26,28)(H,27,29)	ZDYACGZBLWVWLA-UHFFFAOYSA-N	794844	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-ethoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C67	Myelin transcription factor 1	Homo sapiens		 0.100							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794844	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794844&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293625	528826307							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741220	CC(C)Oc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H17F2N5O2/c1-9(2)31-15-7-12-16(11-6-14(23)17(24)21-13(11)8-27-29-21)18(25)22(30)28-19(12)10-4-3-5-26-20(10)15/h3-9H,25H2,1-2H3,(H,27,29)(H,28,30)	GTSCSJYLNSFNGR-UHFFFAOYSA-N	794846	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-propan-2-yloxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C69	Myelin transcription factor 1	Homo sapiens		 0.100							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794846	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794846&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293576	528826309							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741221	COc1cc2c(-c3cc(F)c(Cl)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H13ClFN5O2/c1-29-13-6-10-14(9-5-12(22)15(21)19-11(9)7-25-27-19)16(23)20(28)26-17(10)8-3-2-4-24-18(8)13/h2-7H,23H2,1H3,(H,25,27)(H,26,28)	AKGZZODTYNYXCP-UHFFFAOYSA-N	794853	3-Amino-4-(7-chloro-6-fluoro-1H-indazol-4-yl)-6-methoxy-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C76	Myelin transcription factor 1	Homo sapiens		 0.092							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794853	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794853&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293729	528826316							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741222	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Cl)c3ncccc3c2[nH]c1=O	InChI=1S/C19H11ClFN5O/c20-12-6-10-14(8-3-4-13(21)18-11(8)7-24-26-18)15(22)19(27)25-16(10)9-2-1-5-23-17(9)12/h1-7H,22H2,(H,24,26)(H,25,27)	CWHCCNDDZMAHAF-UHFFFAOYSA-N	794855	3-Amino-6-chloro-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C78	Myelin transcription factor 1	Homo sapiens		<0.170							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794855	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794855&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293671	528826318							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741223	Nc1c(-c2cccc3[nH]ncc23)c2cc(Cl)c3ncccc3c2[nH]c1=O	InChI=1S/C19H12ClN5O/c20-13-7-11-15(9-3-1-5-14-12(9)8-23-25-14)16(21)19(26)24-17(11)10-4-2-6-22-18(10)13/h1-8H,21H2,(H,23,25)(H,24,26)	WLXVQQBMMOFSOX-UHFFFAOYSA-N	794856	3-Amino-6-chloro-4-(1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C79	Myelin transcription factor 1	Homo sapiens		 0.300							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794856	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794856&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293190	528826319							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741224	Nc1c(-c2ccc(F)c3[nH]ncc23)c2ccc3ncccc3c2[nH]c1=O	InChI=1S/C19H12FN5O/c20-13-5-3-9(12-8-23-25-18(12)13)15-11-4-6-14-10(2-1-7-22-14)17(11)24-19(26)16(15)21/h1-8H,21H2,(H,23,25)(H,24,26)	CVGSWRGEMHJVNE-UHFFFAOYSA-N	794860	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C83	Myelin transcription factor 1	Homo sapiens		 0.200							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794860	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794860&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293470	528826323							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741225	Nc1c(C2=CC=C(F)C3NN=CC23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H18FN5O/c23-16-6-5-11(15-9-26-28-21(15)16)17-14-8-13(10-3-4-10)19-12(2-1-7-25-19)20(14)27-22(29)18(17)24/h1-2,5-10,15,21,28H,3-4,24H2,(H,27,29)	BTIVOCRMOOPVQU-UHFFFAOYSA-N	794861	3-Amino-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one solvate::US20260062412, Compound C84	Myelin transcription factor 1	Homo sapiens		 0.250							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794861	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794861&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			178423166	528826324							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741226	Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H14FN5O/c1-9-7-12-15(10-4-5-14(21)19-13(10)8-24-26-19)16(22)20(27)25-18(12)11-3-2-6-23-17(9)11/h2-8H,22H2,1H3,(H,24,26)(H,25,27)	JLHGHMDSERVGHA-UHFFFAOYSA-N	794862	3-Amino-4-(7-fluoro-1H-inadazol-4-yl)-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C85	Myelin transcription factor 1	Homo sapiens		 0.190							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794862	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794862&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293256	528826325							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741227	CCc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H16FN5O/c1-2-10-8-13-16(11-5-6-15(22)20-14(11)9-25-27-20)17(23)21(28)26-19(13)12-4-3-7-24-18(10)12/h3-9H,2,23H2,1H3,(H,25,27)(H,26,28)	QYLIZLBBMCBRMJ-UHFFFAOYSA-N	794863	3-Amino-6-ethyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C86	Myelin transcription factor 1	Homo sapiens		<0.170							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794863	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794863&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293665	528826326							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741228	Cn1cc(-c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)cn1	InChI=1S/C23H16FN7O/c1-31-10-11(8-28-31)14-7-15-18(12-4-5-17(24)22-16(12)9-27-30-22)19(25)23(32)29-21(15)13-3-2-6-26-20(13)14/h2-10H,25H2,1H3,(H,27,30)(H,29,32)	ZJTGYVFOQIBZDZ-UHFFFAOYSA-N	794865	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-methylpyrazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C88	Myelin transcription factor 1	Homo sapiens		<0.170							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794865	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794865&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293932	528826328							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741229	CC#Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C22H14FN5O/c1-2-4-11-9-14-17(12-6-7-16(23)21-15(12)10-26-28-21)18(24)22(29)27-20(14)13-5-3-8-25-19(11)13/h3,5-10H,24H2,1H3,(H,26,28)(H,27,29)	KEPIYZUVCGDMQA-UHFFFAOYSA-N	794867	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-prop-1-inyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C90	Myelin transcription factor 1	Homo sapiens		 0.420							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794867	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794867&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293405	528826330							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741230	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H18FN5O/c24-17-7-6-12(16-10-27-29-22(16)17)18-15-9-14(11-3-1-4-11)20-13(5-2-8-26-20)21(15)28-23(30)19(18)25/h2,5-11H,1,3-4,25H2,(H,27,29)(H,28,30)	IYIBINXWVNMQSD-UHFFFAOYSA-N	794868	3-Amino-6-cyclobutyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C91	Myelin transcription factor 1	Homo sapiens		 1.10							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794868	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794868&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293184	528826331							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741231	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20FN5O/c25-18-8-7-13(17-11-28-30-23(17)18)19-16-10-15(12-4-1-2-5-12)21-14(6-3-9-27-21)22(16)29-24(31)20(19)26/h3,6-12H,1-2,4-5,26H2,(H,28,30)(H,29,31)	MWAVRFFPFNYBKQ-UHFFFAOYSA-N	794869	3-Amino-6-cyclopentyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C92	Myelin transcription factor 1	Homo sapiens		 1.70							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794869	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794869&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293709	528826332							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741232	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCOCC3)c3ncccc3c2[nH]c1=O	InChI=1S/C24H20FN5O2/c25-18-4-3-13(17-11-28-30-23(17)18)19-16-10-15(12-5-8-32-9-6-12)21-14(2-1-7-27-21)22(16)29-24(31)20(19)26/h1-4,7,10-12H,5-6,8-9,26H2,(H,28,30)(H,29,31)	UEVYVEVCJPPKMX-UHFFFAOYSA-N	794875	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(oxan-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C98	Myelin transcription factor 1	Homo sapiens		<4.60							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794875	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794875&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293552	528826338							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741233	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(/C=C/CCO)c3ncccc3c2[nH]c1=O	InChI=1S/C23H18FN5O2/c24-17-7-6-13(16-11-27-29-22(16)17)18-15-10-12(4-1-2-9-30)20-14(5-3-8-26-20)21(15)28-23(31)19(18)25/h1,3-8,10-11,30H,2,9,25H2,(H,27,29)(H,28,31)	SBLFOWRRUBVDBB-UHFFFAOYSA-N	794877	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[(E)-4-hydroxybut-1-enyl]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C100	Myelin transcription factor 1	Homo sapiens		 5.50							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794877	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794877&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293275	528826340							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741234	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCC4(CC3)OCCO4)c3ncccc3c2[nH]c1=O	InChI=1S/C27H24FN5O3/c28-20-4-3-15(19-13-31-33-25(19)20)21-18-12-17(14-5-7-27(8-6-14)35-10-11-36-27)23-16(2-1-9-30-23)24(18)32-26(34)22(21)29/h1-4,9,12-14H,5-8,10-11,29H2,(H,31,33)(H,32,34)	XLQZDMCJBNNSKA-UHFFFAOYSA-N	794878	3-Amino-6-(1,4-dioxaspiro[4.5]decan-8-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one 2,2,2-trifluoroacetate::US20260062412, Compound C101	Myelin transcription factor 1	Homo sapiens		 7.10							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794878	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794878&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293685	528826341							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741235	CC(C)(O)C#Cc1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C24H18FN5O2/c1-24(2,32)8-7-12-10-15-18(13-5-6-17(25)22-16(13)11-28-30-22)19(26)23(31)29-21(15)14-4-3-9-27-20(12)14/h3-6,9-11,32H,26H2,1-2H3,(H,28,30)(H,29,31)	JXGCFCCRLPERLA-UHFFFAOYSA-N	794879	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(3-hydroxy-3-methylbut-1-inyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C102	Myelin transcription factor 1	Homo sapiens		<4.60							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794879	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794879&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293718	528826342							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741236	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCN(C4CCC4)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C28H27FN6O/c29-22-7-6-17(21-14-32-34-27(21)22)23-20-13-19(15-8-11-35(12-9-15)16-3-1-4-16)25-18(5-2-10-31-25)26(20)33-28(36)24(23)30/h2,5-7,10,13-16H,1,3-4,8-9,11-12,30H2,(H,32,34)(H,33,36)	VWTRXZWWARKGDY-UHFFFAOYSA-N	794911	3-Amino-6-(1-cyclobutylpiperidin-4-yl)-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C134	Myelin transcription factor 1	Homo sapiens		 7.60							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794911	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794911&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293261	528826374							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741237	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCN(C4COC4)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C27H25FN6O2/c28-21-4-3-16(20-11-31-33-26(20)21)22-19-10-18(14-5-8-34(9-6-14)15-12-36-13-15)24-17(2-1-7-30-24)25(19)32-27(35)23(22)29/h1-4,7,10-11,14-15H,5-6,8-9,12-13,29H2,(H,31,33)(H,32,35)	PHEOLMVLSIREMF-UHFFFAOYSA-N	794912	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[1-(oxetan-3-yl) piperidin-4-yl]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C135	Myelin transcription factor 1	Homo sapiens		<4.60							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794912	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794912&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293369	528826375							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741238	CC(C)N1CCC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC1	InChI=1S/C27H27FN6O/c1-14(2)34-10-7-15(8-11-34)18-12-19-22(16-5-6-21(28)26-20(16)13-31-33-26)23(29)27(35)32-25(19)17-4-3-9-30-24(17)18/h3-6,9,12-15H,7-8,10-11,29H2,1-2H3,(H,31,33)(H,32,35)	MTFMIKRWXSZUTI-UHFFFAOYSA-N	794913	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-propan-2-ylpiperidin-4-yl)-1H-1,7-phenanthrolin-2-one; formate::US20260062412, Compound C136	Myelin transcription factor 1	Homo sapiens		 8.30							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794913	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794913&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293435	528826376							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741239	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCN(C4CCOCC4)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C29H29FN6O2/c30-23-4-3-18(22-15-33-35-28(22)23)24-21-14-20(16-5-10-36(11-6-16)17-7-12-38-13-8-17)26-19(2-1-9-32-26)27(21)34-29(37)25(24)31/h1-4,9,14-17H,5-8,10-13,31H2,(H,33,35)(H,34,37)	KPWJXXMETFKFFG-UHFFFAOYSA-N	794914	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-[1-(oxan-4-yl) piperidin-4-yl]-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C137	Myelin transcription factor 1	Homo sapiens		 7.70							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794914	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794914&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293507	528826377							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741240	CN1CCC(c2cc3c(-c4ccc(F)c5[nH]ncc45)c(N)c(=O)[nH]c3c3cccnc23)CC1	InChI=1S/C25H23FN6O/c1-32-9-6-13(7-10-32)16-11-17-20(14-4-5-19(26)24-18(14)12-29-31-24)21(27)25(33)30-23(17)15-3-2-8-28-22(15)16/h2-5,8,11-13H,6-7,9-10,27H2,1H3,(H,29,31)(H,30,33)	JHZHSGNLORZFDL-UHFFFAOYSA-N	794915	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(1-methylpiperidin-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C138	Myelin transcription factor 1	Homo sapiens		<4.60							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794915	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794915&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293171	528826378							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741241	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCC(=O)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C25H20FN5O2/c26-19-8-7-14(18-11-29-31-24(18)19)20-17-10-16(12-3-5-13(32)6-4-12)22-15(2-1-9-28-22)23(17)30-25(33)21(20)27/h1-2,7-12H,3-6,27H2,(H,29,31)(H,30,33)	BFOJFEOOVMACAM-UHFFFAOYSA-N	794916	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-(4-oxocyclohexyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C139	Myelin transcription factor 1	Homo sapiens		 19.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794916	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794916&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293880	528826379							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741242	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc([C@H]3CC[C@H](O)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C25H22FN5O2/c26-19-8-7-14(18-11-29-31-24(18)19)20-17-10-16(12-3-5-13(32)6-4-12)22-15(2-1-9-28-22)23(17)30-25(33)21(20)27/h1-2,7-13,32H,3-6,27H2,(H,29,31)(H,30,33)	ZTDZYEUDHPMYPI-UHFFFAOYSA-N	794917	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-((1r, 4r)-4-hydroxycyclohexyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C140	Myelin transcription factor 1	Homo sapiens		<4.60							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794917	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794917&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			176112735	528826380							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741243	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc([C@H]3CC[C@@H](O)CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C25H22FN5O2/c26-19-8-7-14(18-11-29-31-24(18)19)20-17-10-16(12-3-5-13(32)6-4-12)22-15(2-1-9-28-22)23(17)30-25(33)21(20)27/h1-2,7-13,32H,3-6,27H2,(H,29,31)(H,30,33)	ZTDZYEUDHPMYPI-UHFFFAOYSA-N	794918	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-((1s, 4s)-4-hydroxycyclohexyl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C141	Myelin transcription factor 1	Homo sapiens		 11.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794918	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794918&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			176112735	528826381							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741244	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H16ClN5O/c23-16-6-5-11(15-9-26-28-21(15)16)17-14-8-13(10-3-4-10)19-12(2-1-7-25-19)20(14)27-22(29)18(17)24/h1-2,5-10H,3-4,24H2,(H,26,28)(H,27,29)	CULBTRFDPALKTG-UHFFFAOYSA-N	794920	3-Amino-4-(7-chloro-1H-indazol-4-yl)-6-cyclopropyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C143	Myelin transcription factor 1	Homo sapiens		 0.200							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794920	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794920&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293414	528826383							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741245	Nc1c(-c2ccc(Cl)c3[nH]ncc23)c2ccc3ncccc3c2[nH]c1=O	InChI=1S/C19H12ClN5O/c20-13-5-3-9(12-8-23-25-18(12)13)15-11-4-6-14-10(2-1-7-22-14)17(11)24-19(26)16(15)21/h1-8H,21H2,(H,23,25)(H,24,26)	VICZQFFWCKFLGI-UHFFFAOYSA-N	794921	3-Amino-4-(7-chloro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C144	Myelin transcription factor 1	Homo sapiens		 0.320							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794921	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794921&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293864	528826384							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741246	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CCNC3)c3ncccc3c2[nH]c1=O	InChI=1S/C23H19FN6O/c24-17-4-3-12(16-10-28-30-22(16)17)18-15-8-14(11-5-7-26-9-11)20-13(2-1-6-27-20)21(15)29-23(31)19(18)25/h1-4,6,8,10-11,26H,5,7,9,25H2,(H,28,30)(H,29,31)	ASKXOJLWFWUBQH-UHFFFAOYSA-N	794923	3-Amino-4-(7-fluoro-1H-indazol-4-yl)-6-pyrrolidin-3-yl-1H-1,7-phenanthrolin-2-one; formate::US20260062412, Compound C146	Myelin transcription factor 1	Homo sapiens		 16.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794923	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794923&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293340	528826386							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741247	Cc1cc2c(-c3c(F)ccc4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H14FN5O/c1-9-7-11-16(15-12-8-24-26-14(12)5-4-13(15)21)17(22)20(27)25-19(11)10-3-2-6-23-18(9)10/h2-8H,22H2,1H3,(H,24,26)(H,25,27)	CEJSSNRTXYXSRE-UHFFFAOYSA-N	794932	3-Amino-4-(5-fluoro-1H-indazol-4-yl)-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C155	Myelin transcription factor 1	Homo sapiens		<4.60							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794932	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794932&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293247	528826395							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741248	Nc1c(-c2c(F)ccc3[nH]ncc23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H16FN5O/c23-15-5-6-16-14(9-26-28-16)17(15)18-13-8-12(10-3-4-10)20-11(2-1-7-25-20)21(13)27-22(29)19(18)24/h1-2,5-10H,3-4,24H2,(H,26,28)(H,27,29)	PEYWJOJLYYNZDL-UHFFFAOYSA-N	794933	3-Amino-6-cyclopropyl-4-(5-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one (racemate)::US20260062412, Compound C156	Myelin transcription factor 1	Homo sapiens		 6.20							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794933	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794933&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293776	528826396							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741249	Nc1c(-c2cccc(O)c2)c2ccc3ncccc3c2[nH]c1=O	InChI=1S/C18H13N3O2/c19-16-15(10-3-1-4-11(22)9-10)13-6-7-14-12(5-2-8-20-14)17(13)21-18(16)23/h1-9,22H,19H2,(H,21,23)	XBBICBUIAYBGGZ-UHFFFAOYSA-N	794960	3-Amino-4-(3-hydroxyphenyl)-1H-1,7-phenanthrolin-2-one; hydrobromide::US20260062412, Compound C184	Myelin transcription factor 1	Homo sapiens		<4.60							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794960	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794960&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293575	528826423							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741250	Nc1c(-c2cccc3[nH]ncc23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H17N5O/c23-19-18(12-3-1-5-17-16(12)10-25-27-17)15-9-14(11-6-7-11)20-13(4-2-8-24-20)21(15)26-22(19)28/h1-5,8-11H,6-7,23H2,(H,25,27)(H,26,28)	SESIRVHTVJUFCA-UHFFFAOYSA-N	794961	3-Amino-6-cyclopropyl-4-(1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C185	Myelin transcription factor 1	Homo sapiens		 0.310							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794961	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794961&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293679	528826424							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741251	Nc1c(-c2cccc3[nH]ncc23)c2ccc3ncccc3c2[nH]c1=O	InChI=1S/C19H13N5O/c20-17-16(10-3-1-5-15-13(10)9-22-24-15)12-6-7-14-11(4-2-8-21-14)18(12)23-19(17)25/h1-9H,20H2,(H,22,24)(H,23,25)	DNTCJROXICERMW-UHFFFAOYSA-N	794962	3-Amino-4-(1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C186	Myelin transcription factor 1	Homo sapiens		 3.90							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794962	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794962&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293189	528826425							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741252	Cc1cc2c(-c3cc(F)c(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C20H13F2N5O/c1-8-5-11-14(10-6-13(21)15(22)19-12(10)7-25-27-19)16(23)20(28)26-18(11)9-3-2-4-24-17(8)9/h2-7H,23H2,1H3,(H,25,27)(H,26,28)	SMHSNABIWLRGHW-UHFFFAOYSA-N	794966	3-Amino-4-(6,7-difluoro-1H-indazol-4-yl)-6-methyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C190	Myelin transcription factor 1	Homo sapiens		 0.340							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794966	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794966&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293229	528826429							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741253	Nc1c(-c2cc(F)c(Cl)c3[nH]ncc23)c2cc(C3CC3)c3ncccc3c2[nH]c1=O	InChI=1S/C22H15ClFN5O/c23-17-15(24)7-12(14-8-27-29-21(14)17)16-13-6-11(9-3-4-9)19-10(2-1-5-26-19)20(13)28-22(30)18(16)25/h1-2,5-9H,3-4,25H2,(H,27,29)(H,28,30)	XPQKJTUGNBBJRG-UHFFFAOYSA-N	794971	3-Amino-4-(7-chloro-6-fluoro-1H-indazol-4-yl)-6-cyclopropyl-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C195	Myelin transcription factor 1	Homo sapiens		 0.240							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794971	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794971&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293301	528826434							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741254	CC(=O)c1cc2c(-c3ccc(F)c4[nH]ncc34)c(N)c(=O)[nH]c2c2cccnc12	InChI=1S/C21H14FN5O2/c1-9(28)12-7-13-16(10-4-5-15(22)20-14(10)8-25-27-20)17(23)21(29)26-19(13)11-3-2-6-24-18(11)12/h2-8H,23H2,1H3,(H,25,27)(H,26,29)	YSXBNYZSSJMQOR-UHFFFAOYSA-N	794976	6-Acetyl-3-amino-4-(7-fluoro-1H-indazol-4-yl)-1H-1,7-phenanthrolin-2-one::US20260062412, Compound C200	Myelin transcription factor 1	Homo sapiens		 7.00							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794976	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794976&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293548	528826439							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741255	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(Br)c3ccncc3c2[nH]c1=O	InChI=1S/C19H11BrFN5O/c20-13-5-10-15(9-1-2-14(21)18-12(9)7-24-26-18)16(22)19(27)25-17(10)11-6-23-4-3-8(11)13/h1-7H,22H2,(H,24,26)(H,25,27)	QOKQASVIJODQTG-UHFFFAOYSA-N	794992	3-Amino-6-bromo-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D1	Myelin transcription factor 1	Homo sapiens		 17.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794992	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794992&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			178423168	528826455							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741256	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3cccnc3c2[nH]c1=O	InChI=1S/C22H16FN5O/c23-16-6-5-11(15-9-26-28-19(15)16)17-14-8-13(10-3-4-10)12-2-1-7-25-20(12)21(14)27-22(29)18(17)24/h1-2,5-10H,3-4,24H2,(H,26,28)(H,27,29)	WTUSPBCHWZGEOK-UHFFFAOYSA-N	794993	3-Amino-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,10-phenanthrolin-2-one::US20260062412, Compound D2	Myelin transcription factor 1	Homo sapiens		 15.0							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=794993	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=794993&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293600	528826456							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741257	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(O[C@H]3C[C@H](F)C3)c3nccnc3c2[nH]c1=O	InChI=1S/C22H16F2N6O2/c23-9-5-10(6-9)32-15-7-12-16(11-1-2-14(24)18-13(11)8-28-30-18)17(25)22(31)29-19(12)21-20(15)26-3-4-27-21/h1-4,7-10H,5-6,25H2,(H,28,30)(H,29,31)	RUEFIPXCJVWKRU-UHFFFAOYSA-N	795045	8-Amino-5-((1,3r)-3-fluorocyclobutyl)oxy-7-(7-fluoro-1H-indazol-4-yl)-10H-pyrido[2,3-f]quinoxalin-9-one::US20260062412, Compound G16	Myelin transcription factor 1	Homo sapiens		 0.086							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795045	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795045&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293778	528826508							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741258	Nc1c(-c2cccc3[nH]ncc23)c2cc(C3CC3)c3cnccc3c2[nH]c1=O	InChI=1S/C22H17N5O/c23-20-19(12-2-1-3-18-17(12)10-25-27-18)15-8-14(11-4-5-11)16-9-24-7-6-13(16)21(15)26-22(20)28/h1-3,6-11H,4-5,23H2,(H,25,27)(H,26,28)	XVHRRRWCVFHSER-UHFFFAOYSA-N	795071	3-Amino-6-cyclopropyl-4-(1H-indazol-4-yl)-1H-1,8-phenanthrolin-2-one::US20260062412, Compound P1	Myelin transcription factor 1	Homo sapiens		 0.220							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795071	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795071&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293330	528826534							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741259	Nc1c(-c2ccc(F)c3[nH]ncc23)c2cc(C3CC3)c3cnccc3c2[nH]c1=O	InChI=1S/C22H16FN5O/c23-17-4-3-11(16-9-26-28-21(16)17)18-14-7-13(10-1-2-10)15-8-25-6-5-12(15)20(14)27-22(29)19(18)24/h3-10H,1-2,24H2,(H,26,28)(H,27,29)	XJHHNXUOQBEFJY-UHFFFAOYSA-N	795074	3-Amino-6-cyclopropyl-4-(7-fluoro-1H-indazol-4-yl)-1H-1,8-phenanthrolin-2-one 2,2,2-trifluoroacetate::US20260062412, Compound P4	Myelin transcription factor 1	Homo sapiens		 5.90							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795074	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795074&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293259	528826537							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
741260	Nc1c(-c2cccc3[nH]ncc23)c2cc(C3CC3)c3ccncc3c2[nH]c1=O	InChI=1S/C22H17N5O/c23-20-19(13-2-1-3-18-16(13)10-25-27-18)15-8-14(11-4-5-11)12-6-7-24-9-17(12)21(15)26-22(20)28/h1-3,6-11H,4-5,23H2,(H,25,27)(H,26,28)	BKEXKGVSTVZXJB-UHFFFAOYSA-N	795076	3-Amino-6-cyclopropyl-4-(1H-indazol-4-yl)-1H-1,9-phenanthrolin-2-one::US20260062412, Compound Q1	Myelin transcription factor 1	Homo sapiens		 0.830							US Patent		10.7270/Q2S75N9Z		aid1798225	US20260062412	AOKI, T; CHIBA, T; KOCHI, M; TOMIZAWA, M; MURATA, Y; SUYAMA, E	3/5/2026	7/15/2026	Chugai Seiyaku Kabushiki Kaisha	http://www.bindingdb.org/bind/chemsearch/marvin/MolStructure.jsp?monomerid=795076	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=pol&polymerid=50006348&target=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search	http://www.bindingdb.org/rwd/jsp/dbsearch/PrimarySearch_ki.jsp?energyterm=kJ/mole&tag=r21&monomerid=795076&enzyme=Myelin+transcription+factor+1&column=ki&startPg=0&Increment=50&submit=Search			172293150	528826539							1	MSLENEDKRARTRSKALRGPPETTAADLSCPTPGCTGSGHVRGKYSRHRSLQSCPLAKKRKLEGAEAEHLVSKRKSHPLKLALDEGYGVDSDGSEDTEVKDASVSDESEGTLEGAEAETSGQDEIHRPETAEGRSPVKSHFGSNPIGSATASSKGSYSSYQGIIATSLLNLGQIAEETLVEEDLGQAAKPGPGIVHLLQEAAEGAASEEGEKGLFIQPEDAEEVVEVTTERSQDLCPQSLEDAASEESSKQKGILSHEEEDEEEEEEEEEEEEDEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEEAAPDVIFQEDTSHTSAQKAPELRGPESPSPKPEYSVIVEVRSDDDKDEDTHSRKSTVTDESEMQDMMTRGNLGLLEQAIALKAEQVRTVCEPGCPPAEQSQLGLGEPGKAAKPLDTVRKSYYSKDPSRAEKREIKCPTPGCDGTGHVTGLYPHHRSLSGCPHKDRIPPEILAMHENVLKCPTPGCTGQGHVNSNRNTHRSLSGCPIAAAEKLAKSHEKQQPQTGDPSKSSSNSDRILRPMCFVKQLEVPPYGSYRPNVAPATPRANLAKELEKFSKVTFDYASFDAQVFGKRMLAPKIQTSETSPKAFQCFDYSQDAEAAHMAATAILNLSTRCWEMPENLSTKPQDLPSKSVDIEVDENGTLDLSMHKHRKRENAFPSSSSCSSSPGVKSPDASQRHSSTSAPSSSMTSPQSSQASRQDEWDRPLDYTKPSRLREEEPEESEPAAHSFASSEADDQEVSEENFEERKYPGEVTLTNFKLKFLSKDIKKELLTCPTPGCDGSGHITGNYASHRSLSGCPLADKSLRNLMAAHSADLKCPTPGCDGSGHITGNYASHRSLSGCPRAKKSGVKVAPTKDDKEDPELMKCPVPGCVGLGHISGKYASHRSASGCPLAARRQKEGSLNGSSFSWKSLKNEGPTCPTPGCDGSGHANGSFLTHRSLSGCPRATFAGKKGKLSGDEVLSPKFKTSDVLENDEEIKQLNQEIRDLNESNSEMEAAMVQLQSQISSMEKNLKNIEEENKLIEEQNEALFLELSGLSQALIQSLANIRLPHMEPICEQNFDAYVSTLTDMYSNQDPENKDLLESIKQAVRGIQV	2JX1	Myelin transcription factor 1	MYT1_HUMAN	Q01538	E1P5H0 F5H7M8 O94922 Q7Z5W2 Q9UPV2																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																																		
