Compile Data Set for Download or QSAR
Report error Found 262 of affinity data for UniProtKB/TrEMBL: O70526
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074994(5-[({[4-Methoxy-3-(2-methyl-quinolin-8-yloxymethyl...)
Affinity DataEC50:  480nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074982((E)-N-({[2,4-Dichloro-3-(2-methyl-benzothiazol-4-y...)
Affinity DataEC50:  54nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074998((E)-N-({[4-Methoxy-3-(2-methyl-quinolin-8-yloxymet...)
Affinity DataEC50:  220nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074984((E)-N-({[2,4-Dichloro-3-(2-methyl-benzothiazol-4-y...)
Affinity DataEC50:  23nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074989((E)-N-({[2,4-Dichloro-3-(2-phenyl-benzothiazol-4-y...)
Affinity DataEC50:  2.00E+4nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074987(N-[2-Cyano-4-methoxy-3-(2-methyl-quinolin-8-yloxym...)
Affinity DataEC50:  450nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074988((E)-N-({[3-(Benzothiazol-4-yloxymethyl)-2,4-dichlo...)
Affinity DataEC50:  1.30E+3nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074991((E)-Penta-2,4-dienoic acid ({[2,4-dichloro-3-(2-me...)
Affinity DataEC50:  260nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074992((E)-N-({[4-Chloro-2-methoxy-3-(2-methyl-quinolin-8...)
Affinity DataEC50:  55nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074997((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[4-methoxy-...)
Affinity DataEC50:  59nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074983((E)-N-({[2-Chloro-4-methoxy-3-(2-methyl-quinolin-8...)
Affinity DataEC50:  130nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074990(4-[3-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-yl...)
Affinity DataEC50:  400nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074995((E)-N-({[2-Methoxy-3-(2-methyl-quinolin-8-yloxymet...)
Affinity DataEC50:  1.10E+3nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074979((E)-3-(4-Methoxy-phenyl)-N-({methyl-[3-(2-methyl-q...)
Affinity DataEC50:  660nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50075000((E)-N-({[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-y...)
Affinity DataEC50:  4.10nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074978(2-[3-(4-Amino-butyl)-ureido]-N-[4-chloro-2-cyano-3...)
Affinity DataEC50:  350nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074986(N-(2-((4-chloro-2-cyano-3-((2-methylquinolin-8-ylo...)
Affinity DataEC50:  56nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074980((E)-N-({[2,4-Dichloro-3-(2-methyl-benzothiazol-4-y...)
Affinity DataEC50:  100nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074999(N-[4-Chloro-2-cyano-3-(2-methyl-quinolin-8-yloxyme...)
Affinity DataEC50:  290nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50419902(CHEMBL1956722)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at guinea pig bradykinin B2 receptor in longitudinal smooth muscle assessed as inhibition of bradykinin-induced contractile respo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50408815(B-9430 | CHEMBL384857)
Affinity DataKd:  6.31nMAssay Description:Antagonistic activity against Bradykinin receptor B2 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50408806(B-9858 | CHEMBL410358)
Affinity DataKd:  3.16E+3nMAssay Description:Antagonistic activity against Bradykinin receptor B2 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataIC50: 0.0900nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataIC50: 0.0900nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067317(N-({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxymeth...)
Affinity DataIC50: 0.130nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067929(4-(2-{[(E)-3-(4-Dimethylcarbamoyl-phenyl)-acryloyl...)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50074986(N-(2-((4-chloro-2-cyano-3-((2-methylquinolin-8-ylo...)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]bradykinin from guinea pig B2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067263(5-{2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...)
Affinity DataIC50: 0.360nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067242(3-(6-Acetylamino-pyridin-3-yl)-N-({[3-(3-bromo-2-m...)
Affinity DataIC50: 0.380nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067248(5-{2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...)
Affinity DataIC50: 0.440nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067301(FK-3657 | (E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[...)
Affinity DataIC50: 0.460nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067301(FK-3657 | (E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[...)
Affinity DataIC50: 0.460nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067290(5-{2-[({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxy...)
Affinity DataIC50: 0.460nMAssay Description:Displacement of [3H]BK from Bradykinin B2 Receptor in guinea pig ileum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067305((E)-N-({[2,4-Dimethyl-3-(2-methyl-quinolin-8-yloxy...)
Affinity DataIC50: 0.470nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067247(4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyr...)
Affinity DataIC50: 0.5nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067247(4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyr...)
Affinity DataIC50: 0.5nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067283((E)-3-(4-Acetylamino-phenyl)-N-({[2,4-dichloro-3-(...)
Affinity DataIC50: 0.5nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067281(CHEMBL439737 | CHEMBL542096 | 4-{(E)-2-[({[2,4-Dic...)
Affinity DataIC50: 0.510nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067281(CHEMBL439737 | CHEMBL542096 | 4-{(E)-2-[({[2,4-Dic...)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067253((E)-3-(4-Acetylamino-phenyl)-N-({[3-(3-bromo-2-met...)
Affinity DataIC50: 0.550nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067274((E)-N-({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxy...)
Affinity DataIC50: 0.550nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067932((E)-N-({Methyl-[3-(2-methyl-quinolin-8-yloxymethyl...)
Affinity DataIC50: 0.550nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067923(3-(6-Acetylamino-pyridin-3-yl)-N-{1-[2,4-bis-acety...)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067917((E)-N-{1-[3-(2-Methyl-quinolin-8-yloxymethyl)-2,4-...)
Affinity DataIC50: 0.580nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067240((E)-N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...)
Affinity DataIC50: 0.590nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067294(4-{2-[({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxy...)
Affinity DataIC50: 0.620nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067930(4-[(E)-2-({1-[2,4-Dichloro-3-(2-methyl-quinolin-8-...)
Affinity DataIC50: 0.640nMAssay Description:Inhibition of the specific binding of [3H]BK to Bradykinin receptor B2 in guinea pig ileum membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067289((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[2,4-dichlo...)
Affinity DataIC50: 0.650nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067251(4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyr...)
Affinity DataIC50: 0.660nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Guinea pig)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50067251(4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyr...)
Affinity DataIC50: 0.660nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
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