Compile Data Set for Download or QSAR
Report error Found 894 of affinity data for UniProtKB/TrEMBL: P09467
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50293594(5-(2-amino-5-isobutylthiazol-4-yl)furan-2-ylphosph...)
Affinity DataEC50:  16nMAssay Description:Inhibition of human liver FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50504454(CHEMBL4593275)
Affinity DataKd:  5.40E+4nMAssay Description:Binding affinity to human FBPase expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant at 100 uM by UV-visible spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50310094({[(7-carbamoyl-8H-indeno[1,2-d][1,3]thiazol-4-yl)o...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50322036(Ethyl(2S,6S)-4-{[(7-carbamoyl-8H-indeno[1,2-d][1,3...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50273103(3-[(3-methylbenzene)sulfonyl]-1-({4-[({[(3-methylb...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50310095((7-(methylcarbamoyl)-8H-indeno[1,2-d]thiazol-4-ylo...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50322037(Ethyl(2S,6S)-2,6-dimethyl-4-({[7-(methylcarbamoyl)...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50273103(3-[(3-methylbenzene)sulfonyl]-1-({4-[({[(3-methylb...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50310093((7-(pyrimidin-5-yl)-8H-indeno[1,2-d]thiazol-4-ylox...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50273102(3-[(3-chlorobenzene)sulfonyl]-1-({4-[({[(3-chlorob...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50272993(N,N'-(heptane-1,7-diyldicarbamoyl)bis(3-chlorobenz...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50272994(1-[(3-methylbenzene)sulfonyl]-3-[7-({[(3-methylben...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50273104(3-[(3-methylbenzene)sulfonyl]-1-({3-[({[(3-methylb...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50273102(3-[(3-chlorobenzene)sulfonyl]-1-({4-[({[(3-chlorob...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50272991(1-[(3-chlorobenzene)sulfonyl]-3-[6-({[(3-chloroben...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50273035(3-[(3-methylbenzene)sulfonyl]-1-[8-({[(3-methylben...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50310086((7-chloro-8H-indeno[1,2-d]thiazol-4-yloxy)methylph...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50310083((7-methyl-8H-indeno[1,2-d]thiazol-4-yloxy)methylph...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50322039(Ethyl(2S,6S)-2,6-dimethyl-4-{[(7-methyl-8H-indeno[...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50272993(N,N'-(heptane-1,7-diyldicarbamoyl)bis(3-chlorobenz...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50310091((7-(pyridin-3-yl)-8H-indeno[1,2-d]thiazol-4-yloxy)...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50310092((7-(pyridin-4-yl)-8H-indeno[1,2-d]thiazol-4-yloxy)...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50310088((6,7-difluoro-8H-indeno[1,2-d]thiazol-4-yloxy)meth...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50273193(1-[(3-chlorobenzene)sulfonyl]-3-(2-{[2-({[(3-chlor...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50293594(5-(2-amino-5-isobutylthiazol-4-yl)furan-2-ylphosph...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human liver FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50310087((6,7-dimethyl-8H-indeno[1,2-d]thiazol-4-yloxy)meth...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50293594(5-(2-amino-5-isobutylthiazol-4-yl)furan-2-ylphosph...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50335039(2-Amino-5-cyclopropylmethyl-4-[2-(5-phosphono)fura...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human liver FBPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50317151((2S,2'S)-diethyl 2,2'-(((6,7-dimethyl-8H-indeno[1,...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50322041(Isopropyl(2S,6S)-4-{[(6,7-dimethyl-8H-indeno[1,2-d...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50322042(Ethyl4-{[(6,7-dimethyl-8H-indeno[1,2-d][1,3]thiazo...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50322043(MB06322 | (2S,2'S)-diethyl 2,2'-((5-(2-amino-5-iso...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50310084((7-ethyl-8H-indeno[1,2-d]thiazol-4-yloxy)methylpho...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50322038(Ethyl(2S,6S)-4-[({7-[(2,2-dimethylpropyl)carbamoyl...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50322040(Ethyl(2S,6S)-4-{[(7-ethyl-8H-indeno[1,2-d][1,3]thi...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50615534(CHEMBL5271686)
Affinity DataIC50: 11nMAssay Description:Inhibition of human liver FBPase by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50273194(1-[(3-methylbenzene)sulfonyl]-3-(2-{[2-({[(3-methy...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50272992(1-[(3-methylbenzene)sulfonyl]-3-[6-({[(3-methylben...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50273104(3-[(3-methylbenzene)sulfonyl]-1-({3-[({[(3-methylb...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50272994(1-[(3-methylbenzene)sulfonyl]-3-[7-({[(3-methylben...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphataseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50273070(3-[(3-methylbenzene)sulfonyl]-1-[6-({[(3-methylben...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50310082((8H-indeno[1,2-d]thiazol-4-yloxy)methylphosphonic ...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human liver recombinant FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50335036(2-Amino-5-cyclobutyl-4-[2-(5-phosphono)furanyl]thi...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human liver FBPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50335069(2-Amino-5-(2-naphthyl)-4-[2-(5-phosphono)furanyl]t...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human liver FBPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50302495(2-amino-4,5-dihydronaphtho[1,2-d][1,3]thiazol-8-yl...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human liver FBPaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50335065(2-Amino-5-(4-chlorophenyl)-4-[2-(5-phosphono)furan...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human liver FBPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50273036(1-[(3-chlorobenzene)sulfonyl]-3-[(3E)-6-({[(3-chlo...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human liver fructose-1,6-bisphosphatase in presence of fructose-2,6-bisphosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50335054(2-Amino-4-[2-(5-phosphono)furanyl]-5-ethoxycarbony...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human liver FBPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50335057(5-(2-amino-5-phenylthiazol-4-yl)furan-2-ylphosphon...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human liver FBPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
Boston College

Curated by ChEMBL
LigandPNGBDBM50335063(2-Amino-5-(4-methoxycarbonylphenyl)-4-[2-(5-phosph...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human liver FBPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
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