Compile Data Set for Download or QSAR
Report error Found 62 of affinity data for UniProtKB/TrEMBL: P15208
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50459972(CHEMBL4226003)
Affinity DataEC50:  4nMAssay Description:Agonist activity at B6D2F1 mouse insulin receptor assessed as increase in glucose incorporation into lipid phase after 2 hrs in presence of D-[3-3H]g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50296348(NVP-AEW541 | 7-(3-(azetidin-1-yl)cyclobutyl)-5-(3-...)
Affinity DataIC50: 140nMAssay Description:Inhibition of insulin receptor-mediated proliferation of mouse NIH/3T3 cells after 48 hrs by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 200nMAssay Description:Inhibition of Insulin receptor kinase in P19 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50384721(CHEMBL2037224)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of Tel-fused INSR in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50377967(CHEMBL1627107)
Affinity DataEC50:  5.00E+3nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50384734(CHEMBL2037211)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of Tel-fused INSR in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50384725(CHEMBL2037209)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of Tel-fused INSR in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50384726(CHEMBL2037208)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of Tel-fused INSR in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253185(2-Chloro-5-{[(7-{[(7-{[(4-chloro-3-sulfophenyl)ami...)
Affinity DataEC50:  6.00E+3nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50066982(5-[1,4-Bis-(4-methoxy-benzyl)-1H-imidazol-2-ylamin...)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of insulin receptor mediated mitogenesis of NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50384727(CHEMBL2037226)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of Tel-fused INSR in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253181(2-Hydroxy-5-{[(7-{[(7-sulfo(2-naphthyl))amino]carb...)
Affinity DataEC50:  9.00E+3nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50066983(5-[1-(4-Hydroxy-benzyl)-4-(4-methoxy-benzyl)-1H-im...)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of insulin receptor mediated mitogenesis of NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50162998(3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-(...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Insulin receptor kinase in P19 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50162991(3-(1-Benzo[b]thiophen-2-yl-1H-indol-3-yl)-4-[1-(3-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Insulin receptor kinase in P19 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50162994(3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-[...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Insulin receptor kinase in P19 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50162996(3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-[...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Insulin receptor kinase in P19 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50162990(3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-(...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Insulin receptor kinase in P19 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50162993(3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-(...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Insulin receptor kinase in P19 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50384720(CHEMBL2037220)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Tel-fused INSR in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253179(5-{[(7-{[(7-{[(3-Carboxy-4-chlorophenyl)amino]sulf...)
Affinity DataEC50:  1.60E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253178(5-{[(7-{[(7-{[(3-Carboxy-4-chlorophenyl)amino]sulf...)
Affinity DataEC50:  1.80E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50271906(6-benzyl-N4-(3-bromophenyl)-7H-pyrrolo[2,3-d]pyrim...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of insulin receptor-mediated proliferation of mouse NIH/3T3 cells after 48 hrs by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50271907(2-(2-chlorobenzyl)-N4-(3-bromophenyl)-1H-indole-4,...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of insulin receptor-mediated proliferation of mouse NIH/3T3 cells after 48 hrs by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50377968(CHEMBL1627106)
Affinity DataEC50:  2.20E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253166(3-{7-[({7-[(3-carboxyphenyl)sulfamoyl]naphthalen-2...)
Affinity DataEC50:  2.40E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253159(3-{[(4-Hydroxy-7-{[(5-hydroxy-7-{[(3-sulfophenyl)a...)
Affinity DataEC50:  2.60E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253182(5-{7-[({7-[(3-carboxy-4-nitrophenyl)sulfamoyl]naph...)
Affinity DataEC50:  4.00E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253177(2-{7-[({7-[(2-carboxyphenyl)sulfamoyl]naphthalen-2...)
Affinity DataEC50:  4.10E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253180(5-{[(7-{[(7-{[(3-Carboxy-4-hydroxyphenyl)amino]sul...)
Affinity DataEC50:  4.30E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253165(3-{7-[({7-[(3-carboxyphenyl)sulfamoyl]-5-hydroxyna...)
Affinity DataEC50:  4.30E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253168(1,3-bis(7-{[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]sul...)
Affinity DataEC50:  5.40E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253189(5-[({7-[3-(7-{[(3-Carboxy-4-chlorophenyl)amino]sul...)
Affinity DataEC50:  5.60E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253167(1,3-bis(5-hydroxy-7-{[3-(1H-1,2,3,4-tetrazol-1-yl)...)
Affinity DataEC50:  7.30E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50377965(CHEMBL436679)
Affinity DataEC50:  9.00E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253192(disodium 3-{N-methyl7-[({7-[methyl(3-sulfonatophen...)
Affinity DataEC50:  9.10E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253175(2-{7-[({7-[(2-carboxyphenyl)sulfamoyl]-5-hydroxyna...)
Affinity DataEC50:  9.30E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253173(disodium 4-{7-[({7-[(4-sulfonatophenyl)sulfamoyl]n...)
Affinity DataEC50:  9.40E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253174(4-{7-[({7-[(4-carboxyphenyl)sulfamoyl]-5-hydroxyna...)
Affinity DataEC50:  1.03E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253184(3-{7-[({7-[(3-carboxy-2-chlorophenyl)sulfamoyl]-5-...)
Affinity DataEC50:  1.21E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253183(3-{7-[({7-[(3-carboxy-2-hydroxyphenyl)sulfamoyl]na...)
Affinity DataEC50:  1.50E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253195(5-({[7-({[(7-{[(3-Carboxy-4-chlorophenyl)amino]sul...)
Affinity DataEC50:  1.62E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253196(5-{[(7-{2-Amino-1-aza-2-[(7-{[(3-carboxy-4-chlorop...)
Affinity DataEC50:  1.79E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253176(4-{7-[({7-[(4-carboxyphenyl)sulfamoyl]naphthalen-2...)
Affinity DataEC50:  1.83E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253194(5-({[7-({2-[(7-{[(3-Carboxy-4-chlorophenyl)amino]s...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50377966(CHEMBL1627108)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253172(2-[3-(7-{[(7-{[3-(carboxymethyl)phenyl]sulfamoyl}-...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253197(5-[7-(1-{7-[(3-carboxy-4-chlorophenyl)sulfamoyl]na...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253163(1,3-bis({7-[(3-cyanophenyl)sulfamoyl]naphthalen-2-...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetInsulin receptor(Mouse)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253199(5-{[(7-{[N-(7-{[(3-Carboxy-4-chlorophenyl)amino]su...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
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