Affinity DataEC50: 563nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: 1.18E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: >1.80E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: 2.72E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: >4.70E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: >8.22E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: 1.13E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: 857nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: 2.63E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: 870nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: 7.50E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: 1.06E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
Affinity DataKd: 7.94E+3nMAssay Description:Tested for antagonist activity toward NK-3 receptor in rat portal vein against the agonist eledoisin (mean +/-, n=4)More data for this Ligand-Target Pair
Affinity DataKd: 2.51E+3nMAssay Description:Tested antagonist activity toward NK-3 receptor in rat portal vein against the agonist eledoisinMore data for this Ligand-Target Pair
Affinity DataKd: 1.26E+4nMAssay Description:Tested for antagonist activity toward NK-3 receptor in rat portal vein against the agonist eledoisinMore data for this Ligand-Target Pair
Affinity DataKd: 2.00E+3nMAssay Description:Tested for antagonist activity toward NK-3 receptor in rat portal vein against the agonist eledoisinMore data for this Ligand-Target Pair
Affinity DataKd: 3.98E+3nMAssay Description:Tested for antagonist activity toward NK-3 receptor in rat portal vein against the agonist eledoisinMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: 0.5nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein(RPV).More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein(RPV).More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Agonist activity at rat NK3RMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Agonist activity at rat NK3RMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against cloned human Tachykinin receptor 3 in CHO cells labeled with [125I][MePhe7]-NKBMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against cloned human Tachykinin receptor 3 in CHO cells labeled with [125I][MePhe7]-NKBMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Binding affinity to rat NK3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Inhibitory activity against cloned human Tachykinin receptor 3 in CHO cells labeled with [125I][MePhe7]-NKBMore data for this Ligand-Target Pair
Affinity DataIC50: 91nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
