Compile Data Set for Download or QSAR
Report error Found 81 of affinity data for UniProtKB/TrEMBL: P20789
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282580((S)-2-{(2S,3S)-2-[(S)-2-{[3-(6-Guanidino-hexyl)-7-...)
Affinity DataKd:  300nMAssay Description:Equilibrium dissociation constant at cloned rat Neurotensin receptor (NT) receptor expressed in CHO-K1 cells; 0.3-0.7 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50548041(CHEMBL4794546)
Affinity DataEC50:  20nMAssay Description:Agonist activity at rat NTR1 expressed in CHO cells assessed as effect on [3H] phosphoinositide accumulation using neurotensin (1 to 13 residues) as ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50322368((S)-5-((S)-1-((S)-2-((S)-1-((S)-1-((S)-1-carboxy-3...)
Affinity DataEC50:  28nMAssay Description:Agonist activity at rat NTR1 expressed in LTK cells assessed as calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2010
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282578((S)-2-{(2S,3S)-2-[(S)-2-{[3-(6-Amino-hexyl)-7-(5-a...)
Affinity DataKd:  300nMAssay Description:Equilibrium dissociation constant at cloned rat Neurotensin receptor (NT) receptor expressed in CHO-K1 cells; 0.3-0.7 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282577((S)-2-{(2S,3S)-2-[(S)-2-{[3-(6-Guanidino-hexyl)-7-...)
Affinity DataKd:  300nMAssay Description:Equilibrium dissociation constant at cloned rat Neurotensin receptor (NT) receptor expressed in CHO-K1 cells; 0.3-0.7 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50124132(CHEMBL3622802)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human NTS1 in Sprague-Dawley rat ileum assessed as inhibition of carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50124146(CHEMBL3622801)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human NTS1 in Sprague-Dawley rat ileum assessed as inhibition of carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50124141(CHEMBL3622805)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human NTS1 in Sprague-Dawley rat ileum assessed as inhibition of carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human NTS1 in Sprague-Dawley rat ileum assessed as inhibition of carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50124138(CHEMBL3622804)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human NTS1 in Sprague-Dawley rat ileum assessed as inhibition of carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50124135(CHEMBL3622803)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human NTS1 in Sprague-Dawley rat ileum assessed as inhibition of carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50130880(pGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-L...)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at rat NTS1 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50240845(2-{(S)-2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guanidin...)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at rat NTS1 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50369070(CHEMBL1793839)
Affinity DataIC50: 5nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50033671((S)-2-{(R)-2-[2-({1-[2-(2-Amino-5-guanidino-pentan...)
Affinity DataIC50: 8nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50240845(2-{(S)-2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guanidin...)
Affinity DataIC50: 10nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50033670((S)-2-[(R)-5-({1-[2-(2-Amino-5-guanidino-pentanoyl...)
Affinity DataIC50: 15nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50248034(CHEMBL506981 | SR 48692 | 2-{[1-(7-Chloro-quinolin...)
Affinity DataIC50: 82nMAssay Description:Displacement of [125I]neurotensin from rat brain NTR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50033677((S,R)5-[1-{1-[2-[1-amino-4-amino(imino)methylamino...)
Affinity DataIC50: 120nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50033667((S,S)2-{1-[2-{1-[2-[1-amino-4-amino(imino)methylam...)
Affinity DataIC50: 180nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT (neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50033668((R,S)5-[1-{1-[2-[1-amino-4-amino(imino)methylamino...)
Affinity DataIC50: 900nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50033678((S,S)5-[1-{1-[2-[1-amino-4-amino(imino)methylamino...)
Affinity DataIC50: 1.20E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50033675((S)-2-[(S)-5-({1-[2-(2-Amino-5-guanidino-pentanoyl...)
Affinity DataIC50: 1.20E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50033679((R,R)5-[1-{1-[2-[1-amino-4-amino(imino)methylamino...)
Affinity DataIC50: 1.50E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50369071(CHEMBL1793838)
Affinity DataIC50: 6.31E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50369072(CHEMBL1793837)
Affinity DataIC50: 8.00E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50033674((S,S)2-{1-[2-{1-[2-[1-amino-4-amino(imino)methylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT (neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280251(UK-73093 | 4-Methyl-N-[2-(3-oxo-1-phenyl-1,3-dihyd...)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibitory concentration required for the displacement of [3H]NT from neurotensin receptor in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50130880(pGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-L...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]neurotensin from rat NTS1 receptor expressed in CHO-K1 cells by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM85050(SR142948A | CAS_184162-64-9 | SR 142948A | SR14294...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]neurotensin from rat NTS1 receptor expressed in CHO-K1 cells by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50130880(pGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-L...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM85050(SR142948A | CAS_184162-64-9 | SR 142948A | SR14294...)
Affinity DataKi:  2nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50248034(CHEMBL506981 | SR 48692 | 2-{[1-(7-Chloro-quinolin...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [125I]NT from rat NTR1 transfected in mouse LTK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50041428(CHEMBL3356855)
Affinity DataKi: >25nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50041429(CHEMBL3356854)
Affinity DataKi: >25nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50041427(CHEMBL3356853)
Affinity DataKi: >25nMAssay Description:Displacement of [125L]NT from rat neurotensin receptor type 1 expressed in CHOK1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50366375(CHEMBL1794002)
Affinity DataKi:  29nMAssay Description:Tested for binding affinity against Neurotensin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281809((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-6-Amino-2-ter...)
Affinity DataKi:  63nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281809((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-6-Amino-2-ter...)
Affinity DataKi:  63nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281812((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-5-Amino-2-ter...)
Affinity DataKi:  82nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281812((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-5-Amino-2-ter...)
Affinity DataKi:  82nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50366303(CHEMBL1790460)
Affinity DataKi:  100nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281811((S)-2-{(2S,3S)-2-[(S)-2-[((S)-1-{(S)-2-[(Adamantan...)
Affinity DataKi:  117nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281811((S)-2-{(2S,3S)-2-[(S)-2-[((S)-1-{(S)-2-[(Adamantan...)
Affinity DataKi:  120nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50019412(CHEMBL3290096)
Affinity DataKi:  177nMAssay Description:Displacement of [I125]neurotensin from rat NTS1 overexpressed in CHO-k1 cells by competitive binding AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50366296(CHEMBL1790463)
Affinity DataKi:  180nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50366308(CHEMBL1790472)
Affinity DataKi:  190nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50366299(CHEMBL1790467)
Affinity DataKi:  220nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50366307(CHEMBL1790457)
Affinity DataKi:  290nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50366298(CHEMBL1790466)
Affinity DataKi:  420nMAssay Description:Binding affinity against rat neurotensin receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

Displayed 1 to 50 (of 81 total ) | Next | Last >>
Jump to: