Compile Data Set for Download or QSAR
Report error Found 259 for UniProtKB: P26255
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50002133((4-{2-[2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-p...)
Affinity DataEC50:  8.40nMAssay Description:In vitro beta adrenergic receptor activity against beta-3 adrenergic receptor in rat epididymal fat pads by stimulation of glycerol release from adip...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  13nMAssay Description:In vitro beta adrenergic receptor activity against beta-3 adrenergic receptor in rat epididymal fat pads by stimulation of glycerol release from adip...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50002134(CL-316243 | CHEMBL32590 | 5-{2-[2-(3-Chloro-phenyl...)
Affinity DataEC50:  3nMAssay Description:In vitro beta adrenergic receptor activity against beta-3 adrenergic receptor in rat epididymal fat pads by stimulation of glycerol release from adip...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50002132(CHEMBL38486 | (BRL 35,135)(4-{2-[2-(3-Chloro-pheny...)
Affinity DataEC50:  16nMAssay Description:In vitro beta adrenergic receptor activity against beta-3 adrenergic receptor in rat epididymal fat pads by stimulation of glycerol release from adip...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50407518(L-ISOPRENALINE | LEVISOPRENALINE | ISOPROTERENOL)
Affinity DataEC50:  6.30E+4nMAssay Description:Activity for beta 3-adrenoceptor was assessed from effect on stimulation of lipolysis in rat adipocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataEC50:  1.58E+3nMAssay Description:Effective dose for contraction of reserpine-pretreated rat vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50193803((S)-6-(4-(2-(2-hydroxy-3-(3-methyl-2-oxo-2,3-dihyd...)
Affinity DataEC50:  25nMAssay Description:Agonist activity at rat beta-3 adrenergic receptor expressed in CHO cells assessed as cAMP levelsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50193805((S)-6-(4-(2-(3-(3-(2-cyclopropylethyl)-2-oxo-2,3-d...)
Affinity DataEC50:  6.80nMAssay Description:Agonist activity at rat beta-3 adrenergic receptor expressed in CHO cells assessed as cAMP levelsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50193804((S)-6-(4-(2-(3-(3-(2-cyclobutylethyl)-2-oxo-2,3-di...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at rat beta-3 adrenergic receptor expressed in CHO cells assessed as cAMP levelsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50108088(CHEMBL3601305)
Affinity DataEC50:  535nMAssay Description:Agonist activity at rat beta3-adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2016
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50218165((R)-1-(pyridin-3-yl)-2-(2-(4-(thiazol-4-yl)phenoxy...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at rat adrenergic beta-3 receptor assessed as cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50218164((R)-2-(2-(4-(2-methylthiazol-4-yl)phenoxy)ethylami...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at rat adrenergic beta-3 receptor assessed as cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50224021((S)-6-(4-(2-(3-(3,3-dimethyl-2-oxoindolin-4-yloxy)...)
Affinity DataEC50:  6.5nMAssay Description:Agonist activity at rat beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50092645(N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-...)
Affinity DataEC50:  3.40E+3nMAssay Description:Agonist activity at rat beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50146156(CHEMBL3764088)
Affinity DataEC50:  615nMAssay Description:Agonist activity at rat beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50146160(CHEMBL3765335)
Affinity DataEC50:  531nMAssay Description:Agonist activity at rat beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50146154(KRP-114V | MK-4618 | Vibegron)
Affinity DataEC50:  86nMAssay Description:Agonist activity at rat beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50146156(CHEMBL3764088)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at rat beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assay in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50146160(CHEMBL3765335)
Affinity DataEC50:  245nMAssay Description:Agonist activity at rat beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assay in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50146154(KRP-114V | MK-4618 | Vibegron)
Affinity DataEC50:  122nMAssay Description:Agonist activity at rat beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assay in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataEC50:  1.00E+5nMAssay Description:Activity for beta 3-adrenoceptor was assessed from effect on stimulation of lipolysis in rat adipocytes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409469(CHEMBL284520)
Affinity DataEC50:  61.7nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409471(CHEMBL32586)
Affinity DataEC50:  5.62nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409472(CHEMBL32391)
Affinity DataEC50:  14.1nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409473(CHEMBL33399)
Affinity DataEC50:  81.3nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409474(CHEMBL417137)
Affinity DataEC50:  158nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409475(CHEMBL32939)
Affinity DataEC50:  575nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  87.1nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. EC50, the mean concentration required to produce 50% relaxation of detrusor before the addition in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50002133((4-{2-[2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-p...)
Affinity DataEC50:  2.19nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM97162(MLS002153782 | RITODRINE | cid_31728 | SMR00123316...)
Affinity DataEC50:  191nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409468(CHEMBL32670)
Affinity DataEC50:  0.933nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409478(CHEMBL285888)
Affinity DataEC50:  457nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50002134(CL-316243 | CHEMBL32590 | 5-{2-[2-(3-Chloro-phenyl...)
Affinity DataEC50:  25.1nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409476(CHEMBL289670)
Affinity DataEC50:  832nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409480(CHEMBL33360)
Affinity DataEC50:  52.5nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409483(CHEMBL32115)
Affinity DataEC50:  11.0nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409484(CHEMBL32470)
Affinity DataEC50:  12.9nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409481(CHEMBL35738)
Affinity DataEC50:  813nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409482(CHEMBL35459)
Affinity DataEC50:  22.9nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409470(CHEMBL32532)
Affinity DataEC50:  24.0nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50409479(CHEMBL32933)
Affinity DataEC50:  7.24nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50379086(CHEMBL2012522 | CHEMBL2012521 | LY-377604)
Affinity DataEC50:  5nMAssay Description:Agonist activity at rat adrenergic beta3 receptor expressed in DHB-11 CHO cells assessed as cAMP accumulation after 20 mins by scintillation proximit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50226716(CHEMBL348176)
Affinity DataKd:  1nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat lung reticulocytes pretreated with alkylating beta-bloc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226717(CHEMBL157881 | (+/-)-Pindobind)
Affinity DataKd:  1.60nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to membrane preparation from rat lung reticulocyte pretreated with alkylating beta-blocker...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226718(CHEMBL156628)
Affinity DataKd:  2nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding sites on beta adrenergic receptor of rat heart reticulocytes pretreated with alkylating be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226719(CHEMBL156754)
Affinity DataKd:  1.60nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytes pretreated with alkylating beta-blo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226719(CHEMBL156754)
Affinity DataKd:  1.20nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat lung reticulocytes pretreated with alkylating beta-bloc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226717(CHEMBL157881 | (+/-)-Pindobind)
Affinity DataKd:  2.40nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226718(CHEMBL156628)
Affinity DataKd:  1.40nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat lung reticulocytes pretreated with alkylating beta-bloc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226716(CHEMBL348176)
Affinity DataKd:  1.60nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytes pretreated with alkylating beta-blo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
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