Affinity DataEC50: >1.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 64nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 330nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 280nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 91nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 240nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 350nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
Affinity DataEC50: 920nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
Affinity DataEC50: 370nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Agonist activity at human NK3R expressed in CHO cells assessed as potentiation of senktide-induced effectMore data for this Ligand-Target Pair
Affinity DataEC50: 6.60nMAssay Description:Activity at human NK3 receptor expressed in CHO cells assessed as increase in inositol phosphate generationMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Activity at human NK3 receptor expressed in CHO cells assessed as increase in inositol phosphate generationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at human NK3 receptor expressed in cells assessed as accumulation of [3H]inositol phosphateMore data for this Ligand-Target Pair
Affinity DataKd: 0.220nMAssay Description:Apparent binding affinity to human NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.200nMAssay Description:Equilibrium binding affinity to human NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 36nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.90nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.90nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.30nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 81nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 48nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.12E+3nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 690nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.50E+3nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.90nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.20nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.70nMAssay Description:Antagonist activity at human NK3 receptor expressed in CHO cells assessed as inhibition of senktide-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
