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Report error Found 2271 for UniProtKB: P30874
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065450(2-Amino-3-phenyl-N-{4-[(2S,5S,8S,14S,17R)-8,10,14-...)
Affinity DataKd:  3nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst2) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065453(CHEMBL421362 | L-361,301 | L-363,301 | L-363301 | ...)
Affinity DataKd:  0.760nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst2) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataEC50:  0.100nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50169468(4-{3-[2-(6-Fluoro-1H-indol-3-yl)-ethylsulfanyl]-5-...)
Affinity DataEC50:  14nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50169462(4-{3-[2-(7-Methyl-1H-indol-3-yl)-ethylsulfanyl]-5-...)
Affinity DataEC50:  22nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50169465(3-[4-(4-Amino-butyl)-5-quinolin-2-yl-4H-[1,2,4]tri...)
Affinity DataEC50:  4nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50169467(4-{3-[2-(5-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-...)
Affinity DataEC50:  6.30nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065452(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  6.20nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst2) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065451(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  407nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst2) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098603(10-(4-Amino-butyl)-19-[(2-amino-3-phenyl-propionyl...)
Affinity DataKd:  1.04nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098610(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  56.2nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098611(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  120nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098613(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd:  9.74nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098616(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  1.84nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098608(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  13.2nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098607(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  14.3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098619(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  0.150nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098606(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  40.1nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098602(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098605(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  61.4nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098618(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  10.3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098609(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  14.8nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098604(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  8.96nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098614(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  56.2nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098612(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd:  1.03nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098617(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  26.2nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098615(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  23.5nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50165159(4-[(4R,7S,10S,13R,16S)-4-{[(1S)-1-carboxy-2-hydrox...)
Affinity DataEC50:  2.13nMAssay Description:Relative effective concentration against human somatostatin receptor type 2 expressed in CHO cells; (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50165173(4-[(4R,7S,10S,13R,16S)-4-{[(2R)-1,3-dihydroxybutan...)
Affinity DataEC50:  2.96nMAssay Description:Relative effective concentration against human somatostatin receptor type 2 expressed in CHO cells; (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50165174(Radiolabeled octreotide derivative | 4-[(4R,7S,10S...)
Affinity DataEC50:  1.01nMAssay Description:Relative effective concentration against human somatostatin receptor type 2 expressed in CHO cells; (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50165168(4-[(4R,7S,10S,13R,16S)-4-{[(1S)-1-carboxy-2-hydrox...)
Affinity DataEC50:  2.51nMAssay Description:Relative effective concentration against human somatostatin receptor type 2 expressed in CHO cells; (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50165177(4-[(4R,7S,10S,13R,16S)-4-{[(2R)-1,3-dihydroxybutan...)
Affinity DataEC50:  1.43nMAssay Description:Relative effective concentration against human somatostatin receptor type 2 expressed in CHO cells; (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50165180(4-[(4R,7S,10S,13R,16S)-4-{[(1S)-1-carboxy-2-hydrox...)
Affinity DataEC50:  1.81nMAssay Description:Relative effective concentration against human somatostatin receptor type 2 expressed in CHO cells; (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50165167(4-[(4R,7S,10S,13R,16S)-19-(2-azaniumyl-3-phenylpro...)
Affinity DataEC50:  1.70nMAssay Description:Relative effective concentration against human somatostatin receptor type 2 expressed in CHO cells; (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50165160(Radiolabeled octreotide derivative | 4-[(4R,7S,10S...)
Affinity DataEC50:  1.12nMAssay Description:Relative effective concentration against human somatostatin receptor type 2 expressed in CHO cells; (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50165185(4-[(4R,7S,10S,13R,16S)-4-{[(2R)-1,3-dihydroxybutan...)
Affinity DataEC50:  2.62nMAssay Description:Relative effective concentration against human somatostatin receptor type 2 expressed in CHO cells; (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50165172(4-[(4R,7S,10S,13R,16S)-19-(2-azaniumyl-3-phenylpro...)
Affinity DataEC50:  1nMAssay Description:Relative effective concentration against human somatostatin receptor type 2 expressed in CHO cells; (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50192018(CHEMBL3350037)
Affinity DataKd:  0.610nMAssay Description:Binding affinity to human SST2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2018
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50192019(CHEMBL3966064)
Affinity DataKd:  16nMAssay Description:Binding affinity to human SST2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2018
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423297(Obelin | CHEMBL251541)
Affinity DataKd:  3.63E+4nMAssay Description:Binding affinity to human recombinant sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423465(ERGOLINE)
Affinity DataKd:  1.23E+4nMAssay Description:Binding affinity to human recombinant sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423464(CHEMBL252231)
Affinity DataKd:  9.33E+3nMAssay Description:Binding affinity to human recombinant sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  6.76E+3nMAssay Description:Binding affinity to human recombinant sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423458(CHEMBL252232)
Affinity DataKd:  3.89E+3nMAssay Description:Binding affinity to human recombinant sst2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM405554(US10351547, Compound 1-2 | US10597377, Compound 1-...)
Affinity DataEC50: <10nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC #CCL-61) stably expressing the human SSTR2 are plated in each well of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2020
Entry Details
Go to US Patent

TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM405555(US10351547, Compound 1-3 | US10597377, Compound 1-...)
Affinity DataEC50:  550nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC #CCL-61) stably expressing the human SSTR2 are plated in each well of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2020
Entry Details
Go to US Patent

TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM405553(US10351547, Compound 1-1 | US10597377, Compound 1-...)
Affinity DataEC50: <10nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC #CCL-61) stably expressing the human SSTR2 are plated in each well of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2020
Entry Details
Go to US Patent

TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM405556(US10351547, Compound 1-4 | US10597377, Compound 1-...)
Affinity DataEC50: <10nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC #CCL-61) stably expressing the human SSTR2 are plated in each well of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2020
Entry Details
Go to US Patent

TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM405557(US10351547, Compound 1-5 | US10597377, Compound 1-...)
Affinity DataEC50: <10nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC #CCL-61) stably expressing the human SSTR2 are plated in each well of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2020
Entry Details
Go to US Patent

TargetSomatostatin receptor type 2(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM405558(US10351547, Compound 1-6 | US10597377, Compound 1-...)
Affinity DataEC50: <10nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC #CCL-61) stably expressing the human SSTR2 are plated in each well of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2020
Entry Details
Go to US Patent

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