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Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50371998(CHEMBL404372)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to rat 5HT5A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50051944(3-((1R,2S)-2-Dipropylamino-cyclopropyl)-phenol | C...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50371996(CHEMBL541993)
Affinity DataKi:  2.90nMAssay Description:Binding affinity to rat 5HT5A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50051956(2-((1R,2S)-2-Dipropylamino-cyclopropyl)-phenol | C...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50027065(12'-hydroxy-2'-methyl-5'alpha-(phenylmethyl)ergota...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM21392([3H]-5-carboxamidotryptamine | CHEMBL18840 | 5-car...)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50027065(12'-hydroxy-2'-methyl-5'alpha-(phenylmethyl)ergota...)
Affinity DataKi:  15.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50051950([(1S,2R)-2-(2-Methoxy-phenyl)-cyclopropyl]-dipropy...)
Affinity DataKi:  17nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM78940(methanesulfonic acid;1-methyl-4-(3-methylsulfanyl-...)
Affinity DataKi:  28.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50288778(3-((1S,2R)-2-Dipropylaminomethyl-cyclopropyl)-phen...)
Affinity DataKi:  58nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM78940(methanesulfonic acid;1-methyl-4-(3-methylsulfanyl-...)
Affinity DataKi:  146nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50288773(3-((1S,2S)-2-Dipropylaminomethyl-cyclopropyl)-phen...)
Affinity DataKi:  186nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50031942(CHEMBL1065 | Sansert | (6aR,9R)-4-Methyl-4,6,6a,7,...)
Affinity DataKi:  195nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2011
Entry Details Article
PubMed
LigandPNGBDBM50025223(CHEMBL343529)
Affinity DataIC50: 220nMAssay Description:Evaluated for inhibition of specific [3H]5-HT receptor binding in rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50288781([(1S,2S)-2-(2-Methoxy-phenyl)-cyclopropylmethyl]-d...)
Affinity DataKi:  239nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50288780([(1S,2S)-2-(3-Methoxy-phenyl)-cyclopropylmethyl]-d...)
Affinity DataKi:  310nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50288782(2-((1S,2R)-2-Dipropylaminomethyl-cyclopropyl)-phen...)
Affinity DataKi:  379nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50288775([(1R,2S)-2-(3-Methoxy-phenyl)-cyclopropylmethyl]-d...)
Affinity DataKi:  388nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50288783(Diethyl-[(1S,2S)-2-(2-methoxy-phenyl)-cyclopropylm...)
Affinity DataKi:  431nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50288776(2-((1S,2S)-2-Diethylaminomethyl-cyclopropyl)-pheno...)
Affinity DataKi:  506nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50028124(CHEMBL337825 | 6-MeOT | 2-(6-methoxy-1H-indol-3-yl...)
Affinity DataIC50: 630nMAssay Description:Evaluated for inhibition of specific [3H]5-HT receptor binding in rat cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50288774([(1R,2R)-2-(3-Methoxy-phenyl)-cyclopropyl]-dipropy...)
Affinity DataKi:  736nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50288779(2-((1S,2S)-2-Dipropylaminomethyl-cyclopropyl)-phen...)
Affinity DataKi:  752nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50288777([(1R,2S)-2-(2-Methoxy-phenyl)-cyclopropylmethyl]-d...)
Affinity DataKi:  998nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity at serotonin 5-HT1-type site receptor in rat cortex by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM28582([125I]2,5-dimethoxy-4-iodoamphetamine | DOI,(-) | ...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50024204(MESULERGINE | CHEMBL12314 | 4,7-dimethyl-(6aR,9S,1...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50031942(CHEMBL1065 | Sansert | (6aR,9R)-4-Methyl-4,6,6a,7,...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM35234(Noradrenaline,(+) | NOREPINEPHRINE | DL-[7-3H]nore...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM30704(METERGOLINE | (phenylmethyl) N-[[(6aR,9S,10aR)-4,7...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50010301(SKF 83566 | CHEMBL324017 | 8-Bromo-3-methyl-5-phen...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50106251(2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethylamine | C...)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]LSD as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  1.33E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50106246([1-Benzenesulfonyl-4-(2-dimethylamino-ethyl)-1H-in...)
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]LSD as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50106249([2-(1-Benzenesulfonyl-1H-indol-4-yl)-ethyl]-dimeth...)
Affinity DataKi:  3.40E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]LSD as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50106250([2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethyl]-dimeth...)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]LSD as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50106252([3-(2-Dimethylamino-ethyl)-5-hydroxy-indol-1-yl]-p...)
Affinity DataKi:  4.50E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]LSD as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM34141(CHEMBL76237 | MS-245)
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]LSD as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50106248(4-Dimethylamino-1-(toluene-4-sulfonyl)-1,3,4,5-tet...)
Affinity DataKi: >6.40E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 5A receptor in HEK 293 cells was determined using [3H]LSD as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM85330(NSC_68647 | CAS_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity was measured on 5-hydroxytryptamine receptor uptake receptor using [3H]- paroxetine as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50231569(Cilansetron | KC-9946)
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity was measured on 5-hydroxytryptamine receptor uptake receptor using [3H]- paroxetine as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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