Compile Data Set for Download or QSAR
Report error Found 204 of affinity data for UniProtKB/TrEMBL: P49430
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024903(6-Chloro-3-(4-imidazol-1-yl-butyl)-1H-quinazoline-...)
Affinity DataIC50: 2nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024948(6-Chloro-3-(7-imidazol-1-yl-heptyl)-1H-quinazoline...)
Affinity DataIC50: 2nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037039(2-Amino-5,7-dimethyl-4-pyridin-3-ylmethyl-benzothi...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against the production of thromboxane B2 (TXB2) in glycogen-induced peritoneal cells of ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024906(3-(3-Imidazol-1-yl-2-methyl-propyl)-6-methyl-1H-qu...)
Affinity DataIC50: 3nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024934(CHEMBL544065 | CHEMBL76234 | 7-Chloro-3-(3-imidazo...)
Affinity DataIC50: 3nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024914(6-Chloro-3-(6-imidazol-1-yl-hexyl)-1H-quinazoline-...)
Affinity DataIC50: 4nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024415(5-Chloro-1H-indole-2-carboxylic acid (5-imidazol-1...)
Affinity DataIC50: 7nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024913(6-Chloro-3-(10-imidazol-1-yl-decyl)-1H-quinazoline...)
Affinity DataIC50: 7nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024903(6-Chloro-3-(4-imidazol-1-yl-butyl)-1H-quinazoline-...)
Affinity DataIC50: 7nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024908(CHEMBL74733 | CHEMBL554990 | 6-Chloro-3-(3-imidazo...)
Affinity DataIC50: 8nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024925(7-Chloro-3-(4-imidazol-1-yl-butyl)-1H-quinazoline-...)
Affinity DataIC50: 9nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024942(8-Chloro-3-(3-imidazol-1-yl-2-methyl-propyl)-1H-qu...)
Affinity DataIC50: 10nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024950(3-(5-Imidazol-1-yl-pentyl)-8-trifluoromethyl-1H-qu...)
Affinity DataIC50: 10nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024908(CHEMBL74733 | CHEMBL554990 | 6-Chloro-3-(3-imidazo...)
Affinity DataIC50: 10nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024936(6-Chloro-3-(5-imidazol-1-yl-pentyl)-1H-quinazoline...)
Affinity DataIC50: 12nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50018179(2-Imidazol-1-ylmethyl-4,5-dihydro-benzo[b]thiophen...)
Affinity DataIC50: 13nMAssay Description:Inhibition of platelet microsomal thromboxane A2 synthetase in rabbitsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037746(5-[2-Imidazol-1-yl-1,3-diphenyl-prop-(Z)-ylideneam...)
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024940(3-(3-Imidazol-1-yl-propyl)-6-methyl-1H-quinazoline...)
Affinity DataIC50: 20nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50018181(CHEMBL23942 | 2-Imidazol-1-ylmethyl-4,5,6,7-tetrah...)
Affinity DataIC50: 26nMAssay Description:Inhibition of thromboxane A2 synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024424(5-Chloro-1H-indole-2-carboxylic acid (8-imidazol-1...)
Affinity DataIC50: 27nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50003795(5-[Pyridin-3-yl-(3-trifluoromethyl-phenyl)-methyle...)
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024931(8-Chloro-3-(4-imidazol-1-yl-butyl)-1H-quinazoline-...)
Affinity DataIC50: 30nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024938(3-(3-Imidazol-1-yl-2-methyl-propyl)-1H-quinazoline...)
Affinity DataIC50: 30nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024946(3-(5-Imidazol-1-yl-pentyl)-6-methyl-1H-quinazoline...)
Affinity DataIC50: 30nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024414(1H-Indole-2-carboxylic acid (4-imidazol-1-yl-butyl...)
Affinity DataIC50: 40nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037725(5-[1-Imidazol-1-ylmethyl-hept-(Z)-ylideneaminooxy]...)
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037743(5-[1-Cyclohexyl-2-imidazol-1-yl-eth-(Z)-ylideneami...)
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024912(6-Chloro-3-(8-imidazol-1-yl-octyl)-3H-quinazolin-4...)
Affinity DataIC50: 40nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024922(3-(6-Imidazol-1-yl-hexyl)-1H-quinazoline-2,4-dione...)
Affinity DataIC50: 40nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024926(8-Chloro-3-(5-imidazol-1-yl-pentyl)-1H-quinazoline...)
Affinity DataIC50: 40nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024408(5-Chloro-1H-indole-2-carboxylic acid (3-imidazol-1...)
Affinity DataIC50: 50nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037757(5-[1-(1-Imidazol-1-yl-2-phenyl-ethyl)-hept-(E)-yli...)
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037750(5-[2-Imidazol-1-yl-1,3-diphenyl-prop-(E)-ylideneam...)
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024910(3-(4-Imidazol-1-yl-butyl)-6-methyl-1H-quinazoline-...)
Affinity DataIC50: 50nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50367468(CHEMBL1743616)
Affinity DataIC50: 50nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024951(3-(4-Imidazol-1-yl-butyl)-8-trifluoromethyl-1H-qui...)
Affinity DataIC50: 50nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037751(5-[3-(4-Fluoro-phenyl)-2-imidazol-1-yl-1-phenyl-pr...)
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037740(5-[1-Cyclohexyl-2-imidazol-1-yl-3-phenyl-prop-(E)-...)
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50367469(CHEMBL1743613)
Affinity DataIC50: 60nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024413(5-Chloro-thiophene-2-carboxylic acid (8-imidazol-1...)
Affinity DataIC50: 70nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037731(5-[1-Cyclohexyl-2-imidazol-1-yl-3-pyrazin-2-yl-pro...)
Affinity DataIC50: 70nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024929(3-(3-Imidazol-1-yl-butyl)-6-methyl-1H-quinazoline-...)
Affinity DataIC50: 70nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024923(2-Amino-5-chloro-N-(3-imidazol-1-yl-2-methyl-propy...)
Affinity DataIC50: 90nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024943(6-Chloro-3-(3-imidazol-1-yl-2-methyl-propyl)-3H-qu...)
Affinity DataIC50: 90nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037037(5,7-Dimethyl-2-methylamino-4-pyridin-3-ylmethyl-be...)
Affinity DataIC50: 90nMAssay Description:Inhibitory activity against the production of thromboxane B2 (TXB2) in glycogen-induced peritoneal cells of ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037051(5,7-Dimethyl-2-propylamino-4-pyridin-3-ylmethyl-be...)
Affinity DataIC50: 90nMAssay Description:Inhibitory activity against the production of thromboxane B2 (TXB2) in glycogen-induced peritoneal cells of ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50026226(4-Chloro-N-(8-imidazol-1-yl-octyl)-benzamide | CHE...)
Affinity DataIC50: 100nMAssay Description:compound was tested for inhibitory activity against thromboxane synthetase,More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50024412(5-Chloro-benzo[b]thiophene-2-carboxylic acid (3-im...)
Affinity DataIC50: 100nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037761(5-[1-Cyclohexyl-2-imidazol-1-yl-3-phenyl-prop-(Z)-...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
Medical Research Division of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50037745(5-[1-Cyclohexyl-3-furan-2-yl-2-imidazol-1-yl-prop-...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees CentigradeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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