Compile Data Set for Download or QSAR
Report error Found 113 of affinity data for UniProtKB/TrEMBL: Q12830
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50098250(CHEMBL3590389)
Affinity DataKd: <1.00E+5nMAssay Description:Binding affinity to BPTF in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2016
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50098305(CHEMBL3590405)
Affinity DataKd: <1.00E+5nMAssay Description:Binding affinity to BPTF in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2016
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50098311(CHEMBL3590408)
Affinity DataKd: <1.00E+5nMAssay Description:Binding affinity to BPTF in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2016
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50157526(TCMDC-133606 | CHEMBL586426 | D3RKN_107)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to BPTF (unknown origin) by isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50239563(CHEMBL4095390)
Affinity DataKd:  6.80E+6nMAssay Description:Binding affinity to 5FW-labeled BPTF (unknown origin) by PrOF NMR spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50366670(CHEMBL4173488)
Affinity DataKd: >5.00E+3nMAssay Description:Binding affinity to human FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOScan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50455480(CHEMBL4218735)
Affinity DataKd: <3.02E+4nMAssay Description:Binding affinity to human partial length DNA-tagged FALZ isoform1 expressed in bacteria by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM179481(US9675697, Cpd. No. 73)
Affinity DataKd: >4.00E+3nMAssay Description:Binding affinity to human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50453949(CHEMBL4208820 | US11247989, Example 87)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM249277(US9458145, 1020-18 | US10017501, Compound 1020-18)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system after 1 hr by bromoscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50512964(CHEMBL4574669)
Affinity DataKd:  917nMAssay Description:Binding affinity to human N-terminal His-tagged FALZ by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50539801(CHEMBL4648912 | US11840533, Compound 70)
Affinity DataKd: <1nMAssay Description:Binding affinity to human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  1.89E+3nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: S2791-H2911More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50157526(TCMDC-133606 | CHEMBL586426 | D3RKN_107)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to BPTF (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50571297(CHEMBL4846718)
Affinity DataKd:  428nMAssay Description:Binding affinity to BPTF (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50571296(CHEMBL4873093)
Affinity DataKd:  71nMAssay Description:Binding affinity to BPTF (unknown origin) by BLI assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50571299(CHEMBL4858897)
Affinity DataKd:  3.55E+4nMAssay Description:Binding affinity to BPTF (unknown origin) by BLI assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM25121(4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,...)
Affinity DataKd:  3.70E+4nMAssay Description:Binding affinity to 5FW-labelled BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by 19F-NMR spectraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50157526(TCMDC-133606 | CHEMBL586426 | D3RKN_107)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to 5FW-labelled BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by 19F-NMR spectraMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573836(CHEMBL4861375)
Affinity DataKd:  2.81E+3nMAssay Description:Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573840(CHEMBL4860578)
Affinity DataKd:  4.96E+4nMAssay Description:Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573844(CHEMBL4873042)
Affinity DataKd:  2.07E+4nMAssay Description:Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573844(CHEMBL4873042)
Affinity DataEC50:  120nMAssay Description:Displacement of Halo-tagged histone H4 from NanoLuc-tagged BPTF (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573851(CHEMBL4872422)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to human BPTF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataKd:  120nMAssay Description:Binding affinity to BPTF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573852(CHEMBL4780673)
Affinity DataKd:  71nMAssay Description:Binding affinity to BPTF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50571298(CHEMBL4846726)
Affinity DataKd:  1.79E+4nMAssay Description:Binding affinity to BPTF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataKd:  200nMAssay Description:Binding affinity to BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50234923(CHEMBL4069412)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573183(CHEMBL4867912)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50157526(TCMDC-133606 | CHEMBL586426 | D3RKN_107)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to 5FW-labeled BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by BODIPY-BI2536 tracer ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataKd:  1.20E+5nMAssay Description:Binding affinity to 5FW-labeled BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by BODIPY-BI2536 tracer ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataKd:  6.30nMAssay Description:Binding affinity to BPTF (unknown origin) by by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573200(CHEMBL4861491)
Affinity DataKd:  9.30nMAssay Description:Binding affinity to BPTF (unknown origin) by by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573201(CHEMBL4848701)
Affinity DataKd:  70nMAssay Description:Binding affinity to BPTF (unknown origin) by by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573203(CHEMBL4863631)
Affinity DataKd:  200nMAssay Description:Binding affinity to BPTF (unknown origin) by by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50584925(CHEMBL5079885)
Affinity DataKd: <316nMAssay Description:Binding affinity to human FALZ bromodomain by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50615275(CHEMBL5282240)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM321437((E)-6-(but-2-en-1-yl)-4-(4-(2-hydroxypropan-2-yl)-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50615276(CHEMBL5270178)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM321424(6-[(E)-but-2-enyl]-4-[2,5-dimethoxy-4-(morpholine-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50571296(CHEMBL4873093)
Affinity DataIC50: 16nMAssay Description:Inhibition of BPTF in human HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573840(CHEMBL4860578)
Affinity DataIC50: 16nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573844(CHEMBL4873042)
Affinity DataIC50: 27nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573839(CHEMBL4870170)
Affinity DataIC50: 29nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50571296(CHEMBL4873093)
Affinity DataIC50: 30nMAssay Description:Inhibition of BPTF (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573837(CHEMBL4867072)
Affinity DataIC50: 33nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573200(CHEMBL4861491)
Affinity DataIC50: 36nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573838(CHEMBL4868713)
Affinity DataIC50: 37nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50573201(CHEMBL4848701)
Affinity DataIC50: 56nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
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