Compile Data Set for Download or QSAR
Report error Found 31 of affinity data for UniProtKB/TrEMBL: Q16798
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405810(CHEMBL5284610)
Affinity DataIC50: 60nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405814(CHEMBL5285899)
Affinity DataIC50: 70nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405806(CHEMBL5275653)
Affinity DataIC50: 80nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405807(CHEMBL5287773)
Affinity DataIC50: 90nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405803(CHEMBL5284469)
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405805(CHEMBL5289840)
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405801(CHEMBL5289950)
Affinity DataIC50: 110nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405802(CHEMBL5278951)
Affinity DataIC50: 110nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405811(CHEMBL5277536)
Affinity DataIC50: 120nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405813(CHEMBL5288731)
Affinity DataIC50: 130nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405804(CHEMBL5279230)
Affinity DataIC50: 130nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405808(CHEMBL5279096)
Affinity DataIC50: 130nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405818(CHEMBL5273550)
Affinity DataIC50: 140nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50177180(3-(4-(4-hydroxyphenyl)piperazin-1-yl)-1-phenylpyrr...)
Affinity DataIC50: 150nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405817(CHEMBL5267542)
Affinity DataIC50: 150nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405824(CHEMBL5279589)
Affinity DataIC50: 160nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405815(CHEMBL5278596)
Affinity DataIC50: 200nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405812(CHEMBL5281297)
Affinity DataIC50: 230nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405825(CHEMBL5286488)
Affinity DataIC50: 240nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405826(CHEMBL5290463)
Affinity DataIC50: 250nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405822(CHEMBL5274945)
Affinity DataIC50: 310nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405809(CHEMBL5283020)
Affinity DataIC50: 330nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405823(CHEMBL5286064)
Affinity DataIC50: 360nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405816(CHEMBL5291081)
Affinity DataIC50: 390nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405819(CHEMBL5282439)
Affinity DataIC50: 410nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405820(CHEMBL5270965)
Affinity DataIC50: 470nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405821(CHEMBL5281258)
Affinity DataIC50: 580nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405798(CHEMBL5218866)
Affinity DataIC50: 900nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405799(CHEMBL5283717)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405797(CHEMBL5277143)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetNADP-dependent malic enzyme, mitochondrial(Human)
Sun Pharma Advanced Research Company

Curated by ChEMBL
LigandPNGBDBM50405800(CHEMBL5267207)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of His-tagged human recombinant ME3 (26 to 604 residues) using L-malate and beta-NADP+ as substrate preincubated with enzyme for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed