Compile Data Set for Download or QSAR
Report error Found 114 of affinity data for UniProtKB/TrEMBL: Q28044
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50405521(ALO 1401-02 | ALO-1401-02 | Betaxolol | BETAXOLOL ...)
Affinity DataKd:  1.86E+5nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421717(Tulobuterol Hydrochloride | TULOBUTEROL)
Affinity DataKd:  130nMAssay Description:Apparent binding affinity constant to beta-2 adrenergic receptor determined using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421727(CHEMBL349845)
Affinity DataKd:  1.03E+3nMAssay Description:Apparent binding affinity constant to beta-2 adrenergic receptor determined using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421721(SKF-56301 | CHEMBL1159712)
Affinity DataKd:  560nMAssay Description:Apparent binding affinity constant to beta-2 adrenergic receptor determined using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM27958(Planipart | 1-(4-amino-3,5-dichlorophenyl)-2-(tert...)
Affinity DataKd:  37nMAssay Description:Apparent binding affinity constant to beta-2 adrenergic receptor determined using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421732(VUF8303 | CHEMBL1159711)
Affinity DataKd:  6.47E+3nMAssay Description:Apparent binding affinity constant to beta-2 adrenergic receptor determined using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM92678(2-(tert-butylamino)-1-phenylethan-1-ol, 4)
Affinity DataKd:  2.94E+3nMAssay Description:Apparent binding affinity constant to beta-2 adrenergic receptor determined using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421733(CHEMBL1159887)
Affinity DataKd:  1.35E+3nMAssay Description:Apparent binding affinity constant to beta-2 adrenergic receptor determined using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421728(COLTEROL)
Affinity DataKd:  670nMAssay Description:Apparent binding affinity constant to beta-2 adrenergic receptor determined using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421715(Du-28663 | CHEMBL1159710)
Affinity DataKd:  2.17E+3nMAssay Description:Apparent binding affinity constant to beta-2 adrenergic receptor determined using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM25770(Terbutaline,(+/-) | Brethine | 5-[2-(tert-butylami...)
Affinity DataKd:  4.48E+3nMAssay Description:Apparent binding affinity constant to beta-2 adrenergic receptor determined using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM25769(Levalbuterol | Salbutamol,(+/-) | albuterol | Prov...)
Affinity DataKd:  570nMAssay Description:Apparent binding affinity constant to beta-2 adrenergic receptor determined using [3H]DHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM60973(MLS001333595 | (2R)-1-(1-naphthalenyloxy)-3-(propa...)
Affinity DataKd:  0.891nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM27958(Planipart | 1-(4-amino-3,5-dichlorophenyl)-2-(tert...)
Affinity DataKd:  36nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421715(Du-28663 | CHEMBL1159710)
Affinity DataKd:  2.04E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM25769(Levalbuterol | Salbutamol,(+/-) | albuterol | Prov...)
Affinity DataKd:  520nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM25760(1-(naphthalen-2-yl)-2-(propan-2-ylamino)ethan-1-ol...)
Affinity DataKd:  160nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421716(Phenol metabolite | PRENALTEROL)
Affinity DataKd:  1.07E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421717(Tulobuterol Hydrochloride | TULOBUTEROL)
Affinity DataKd:  130nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM92679(3-{1-hydroxy-2-[(propan-2-yl)amino]ethyl}phenol, 7)
Affinity DataKd:  910nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50295572(5-(1-Hydroxy-2-isopropylamino-ethyl)-benzene-1,3-d...)
Affinity DataKd:  9.12E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM25770(Terbutaline,(+/-) | Brethine | 5-[2-(tert-butylami...)
Affinity DataKd:  3.98E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421718(Du-21117 | CHEMBL1159719)
Affinity DataKd:  5.13E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421719(Ko 707 | CHEMBL1159714)
Affinity DataKd:  10nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421720(Isophenethanol | NIFENALOL)
Affinity DataKd:  1.32E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM92680(4-{1-hydroxy-2-[(propan-2-yl)amino]ethyl}phenol, 8)
Affinity DataKd:  4.27E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataKd:  330nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421721(SKF-56301 | CHEMBL1159712)
Affinity DataKd:  520nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421722(CHEMBL1159890)
Affinity DataKd:  2.14E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421723(CHEMBL321468)
Affinity DataKd:  3.16E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421724(SD-2124-01 | PROCINOLOL)
Affinity DataKd:  0.389nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421725(CHEMBL1159889)
Affinity DataKd:  18nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421726(CHEMBL1159891)
Affinity DataKd:  50.1nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421727(CHEMBL349845)
Affinity DataKd:  470nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421728(COLTEROL)
Affinity DataKd:  600nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM25762(Sotalol,(-) | CHEMBL471 | cid_66245 | Sotalol,(+) ...)
Affinity DataKd:  580nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50241366((S)-1-(isopropylamino)-3-(m-tolyloxy)propan-2-ol (...)
Affinity DataKd:  43.7nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421729(CHEMBL6920)
Affinity DataKd:  10nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50169785(1-Isopropylamino-3-phenoxy-propan-2-ol | (2-Hydrox...)
Affinity DataKd:  5.37E+4nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM25749(Practolol,(-) | Practolol,(+) | N-{4-[2-hydroxy-3-...)
Affinity DataKd:  2.04E+4nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM81447(CAS_43216 | NSC_43216 | Dihydroalprenolol,(+/-))
Affinity DataKd:  0.630nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421730(CHEMBL1159888)
Affinity DataKd:  22nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421731(CHEMBL1159713)
Affinity DataKd:  58nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421732(VUF8303 | CHEMBL1159711)
Affinity DataKd:  1.95E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421733(CHEMBL1159887)
Affinity DataKd:  1.26E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM92679(3-{1-hydroxy-2-[(propan-2-yl)amino]ethyl}phenol, 7)
Affinity DataKd:  910nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421727(CHEMBL349845)
Affinity DataKd:  93nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM81447(CAS_43216 | NSC_43216 | Dihydroalprenolol,(+/-))
Affinity DataKd:  0.631nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50421720(Isophenethanol | NIFENALOL)
Affinity DataKd:  1.32E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50405521(ALO 1401-02 | ALO-1401-02 | Betaxolol | BETAXOLOL ...)
Affinity DataKd:  93nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
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