Compile Data Set for Download or QSAR
Report error Found 10 of affinity data for UniProtKB/TrEMBL: Q28524
TargetBeta-3 adrenergic receptor(Rhesus macaque)
Merck And

Curated by ChEMBL
LigandPNGBDBM50448786(CHEMBL3128194)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at rhesus monkey beta-3 adrenergic receptor expressed in CHO cells assessed as increase in intracellular cAMP accumulation after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rhesus macaque)
Merck And

Curated by ChEMBL
LigandPNGBDBM50092645(N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-...)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at rhesus monkey beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rhesus macaque)
Merck And

Curated by ChEMBL
LigandPNGBDBM50146154(KRP-114V | MK-4618 | Vibegron)
Affinity DataEC50:  0.570nMAssay Description:Agonist activity at rhesus monkey beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rhesus macaque)
Merck And

Curated by ChEMBL
LigandPNGBDBM50448787(CHEMBL3128178)
Affinity DataEC50:  2nMAssay Description:Agonist activity at rhesus monkey beta-3 adrenergic receptor expressed in CHO cells assessed as increase in intracellular cAMP accumulation after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rhesus macaque)
Merck And

Curated by ChEMBL
LigandPNGBDBM50146160(CHEMBL3765335)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at rhesus monkey beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rhesus macaque)
Merck And

Curated by ChEMBL
LigandPNGBDBM50146156(CHEMBL3764088)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at rhesus monkey beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rhesus macaque)
Merck And

Curated by ChEMBL
LigandPNGBDBM50448789(CHEMBL3128188)
Affinity DataEC50:  4.70nMAssay Description:Agonist activity at rhesus monkey beta-3 adrenergic receptor expressed in CHO cells assessed as increase in intracellular cAMP accumulation after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rhesus macaque)
Merck And

Curated by ChEMBL
LigandPNGBDBM50146154(KRP-114V | MK-4618 | Vibegron)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at rhesus monkey beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assay in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rhesus macaque)
Merck And

Curated by ChEMBL
LigandPNGBDBM50146160(CHEMBL3765335)
Affinity DataEC50:  12nMAssay Description:Agonist activity at rhesus monkey beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assay in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Rhesus macaque)
Merck And

Curated by ChEMBL
LigandPNGBDBM50092645(N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-...)
Affinity DataEC50:  17nMAssay Description:Agonist activity at rhesus monkey beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cAMP after 30 mins by TR-FRET assay in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed