Compile Data Set for Download or QSAR
Report error Found 152 of affinity data for UniProtKB/TrEMBL: Q5PPG3
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22911(2-(3H-imidazol-4-yl)ethylsulfanylmethanimidamide |...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22911(2-(3H-imidazol-4-yl)ethylsulfanylmethanimidamide |...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50074629(CHEMBL278462 | 4-[(1R,2R)-2-(5,5-Dimethyl-hex-1-yn...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22911(2-(3H-imidazol-4-yl)ethylsulfanylmethanimidamide |...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM85023(GR-168320 | GR 168320)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM85023(GR-168320 | GR 168320)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22916(5-{3-[(4-iodophenyl)methoxy]propyl}-1H-imidazole |...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22911(2-(3H-imidazol-4-yl)ethylsulfanylmethanimidamide |...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50074629(CHEMBL278462 | 4-[(1R,2R)-2-(5,5-Dimethyl-hex-1-yn...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22530(N(alpha)-Methylhistamine | [2-(1H-imidazol-5-yl)et...)
Affinity DataKi:  0.390nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM27213(CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...)
Affinity DataKi:  0.427nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22530(N(alpha)-Methylhistamine | [2-(1H-imidazol-5-yl)et...)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22904(CHEMBL268229 | Alpha-Methylhistane-R | (2R)-1-(1H-...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22904(CHEMBL268229 | Alpha-Methylhistane-R | (2R)-1-(1H-...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22542(4-(1H-imidazol-4-ylmethyl)piperidine | 4-(1H-imida...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM27213(CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...)
Affinity DataKi:  0.510nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM27213(CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...)
Affinity DataKi:  0.510nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM27213(CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...)
Affinity DataKi:  0.630nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM27213(CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...)
Affinity DataKi:  0.630nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM27213(CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...)
Affinity DataKi:  0.654nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22530(N(alpha)-Methylhistamine | [2-(1H-imidazol-5-yl)et...)
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50158601(CHEMBL361355 | A-317920 | Furan-2-carboxylic acid ...)
Affinity DataKi:  0.710nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50158601(CHEMBL361355 | A-317920 | Furan-2-carboxylic acid ...)
Affinity DataKi:  0.720nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22530(N(alpha)-Methylhistamine | [2-(1H-imidazol-5-yl)et...)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50070214(CHEMBL280076 | GT 2293 | 4-(7,7-Dimethyl-oct-3-yny...)
Affinity DataKi:  0.830nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22541(VUF 9153 | N''-[(4-chlorophenyl)methyl]{[3-(1H-imi...)
Affinity DataKi:  0.870nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22916(5-{3-[(4-iodophenyl)methoxy]propyl}-1H-imidazole |...)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50070220(GT 2286 | CHEMBL274977 | 4-(6-Cyclopentyl-hex-3-yn...)
Affinity DataKi:  0.950nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22913(CHEMBL1237146 | CHEMBL498770 | {[3-(1H-imidazol-5-...)
Affinity DataKi:  0.970nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22911(2-(3H-imidazol-4-yl)ethylsulfanylmethanimidamide |...)
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM85407(GT 2231)
In Depth
Date in BDB:
4/8/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22904(CHEMBL268229 | Alpha-Methylhistane-R | (2R)-1-(1H-...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22530(N(alpha)-Methylhistamine | [2-(1H-imidazol-5-yl)et...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50139391((R)-4-(2-(2-(2-methylpyrrolidin-1-yl)ethyl)benzofu...)
Affinity DataKi:  1.23nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22904(CHEMBL268229 | Alpha-Methylhistane-R | (2R)-1-(1H-...)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM86061(A-304121)
Affinity DataKi:  1.26nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50159110(1-(3-(4-(piperidin-1-ylmethyl)phenoxy)propyl)piper...)
Affinity DataKi:  1.26nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22542(4-(1H-imidazol-4-ylmethyl)piperidine | 4-(1H-imida...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)
Affinity DataKi:  1.45nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2012
Entry Details Article
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22913(CHEMBL1237146 | CHEMBL498770 | {[3-(1H-imidazol-5-...)
Affinity DataKi:  1.48nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22530(N(alpha)-Methylhistamine | [2-(1H-imidazol-5-yl)et...)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details
PubMed
TargetHrh3 protein(Rat)
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM22904(CHEMBL268229 | Alpha-Methylhistane-R | (2R)-1-(1H-...)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details
PubMed
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