Compile Data Set for Download or QSAR
Report error Found 4 for UniProtKB: Q6PAJ1
TargetBreakpoint cluster region protein(Mouse)
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM13530(cid_5291 | STI571 | N-(4-methyl-3-{[4-(pyridin-3-y...)
Affinity DataIC50: 38nMAssay Description:Inhibition of Bcr-Abl phosphorylation in BALB/c mouse 3T3 by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetBreakpoint cluster region protein(Mouse)
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50290422(4-(4-Methyl-piperazin-1-ylmethyl)-N-[3-(4-pyridin-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Bcr-Abl phosphorylation in BALB/c mouse 3T3 by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetBCR/ABL1(Mouse)
Hangzhou Medical College

Curated by ChEMBL
LigandPNGBDBM50590370(Vodobatinib | K-0706 | K0706 | Sco-088 | VODOBATIN...)
Affinity DataIC50: 165nMAssay Description:Inhibition of BCR-ABL E255V mutant phosphorylation in mouse BaF3 cells incubated for 4 hrs by immunoblotting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetBreakpoint cluster region protein(Mouse)
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50590370(Vodobatinib | K-0706 | K0706 | Sco-088 | VODOBATIN...)
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of BCR-ABL T315I mutant phosphorylation in mouse BaF3 cells incubated for 4 hrs by immunoblotting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed