Compile Data Set for Download or QSAR
Report error Found 45 of affinity data for UniProtKB/TrEMBL: Q8BGY9
LigandPNGBDBM50026216(1-Ethyl-1-(2-hydroxy-ethyl)-aziridinium; chloride ...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro ability to inhibit the transport of [3H]choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50026220(2-hydroxy-N,N,N-trimethylethanaminium | CHEMBL920 ...)
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro ability to inhibit the transport of [3H]choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50026218(1-(2-Hydroxy-ethyl)-1-isopropyl-aziridinium; chlor...)
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro ability to inhibit the transport of [3H]choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50026215(1-Cyclopropyl-1-(2-hydroxy-ethyl)-aziridinium; chl...)
Affinity DataIC50: 3.90E+3nMAssay Description:In vitro ability to inhibit the transport of [3H]choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50026219(1-(2-Hydroxy-ethyl)-1-propyl-aziridinium; chloride...)
Affinity DataIC50: 7.50E+3nMAssay Description:In vitro ability to inhibit the transport of [3H]choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50026217(1-(2-Hydroxy-ethyl)-1-isobutyl-aziridinium; chlori...)
Affinity DataIC50: 3.10E+4nMAssay Description:In vitro ability to inhibit the transport of [3H]choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50026221(1-Butyl-1-(2-hydroxy-ethyl)-aziridinium; chloride ...)
Affinity DataIC50: 1.00E+6nMAssay Description:In vitro ability to inhibit the transport of [3H]choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50416502(CHEMBL1209654)
Affinity DataKi:  20.0nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416489(CHEMBL1209507)
Affinity DataKi:  50nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416490(CHEMBL1209508)
Affinity DataKi:  90.0nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416491(CHEMBL1209577)
Affinity DataKi:  180nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416508(CHEMBL1209578)
Affinity DataKi:  200nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416504(CHEMBL1209579)
Affinity DataKi:  230nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416506(CHEMBL1209581)
Affinity DataKi:  521nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416503(CHEMBL1209713)
Affinity DataKi:  640nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50026220(2-hydroxy-N,N,N-trimethylethanaminium | CHEMBL920 ...)
Affinity DataKi:  681nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50416501(CHEMBL1209653)
Affinity DataKi:  701nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416488(CHEMBL1209506)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50147119(CHEMBL1209422 | CHEMBL317449 | (3-Hydroxy-propyl)-...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50204415(CHEMBL389799 | CHEMBL1209582 | 1-methyl-1-azonia-b...)
Affinity DataKi:  4.70E+3nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50079455(CHEMBL46486 | tetramethylammonium)
Affinity DataKi:  3.01E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM80992(CETYLPYRIDINIUM BROMIDE | cid_8816 | MLS002695907 ...)
Affinity DataKi:  3.21E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416495(CHEMBL1209648)
Affinity DataKi:  4.01E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50060526(2-hydroxy-N,N-dimethylethanaminium | 2-Dimethylami...)
Affinity DataKi:  5.57E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416507(CHEMBL1209649)
Affinity DataKi:  7.21E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM80386(SMR000059200 | MLS000069658 | CHEMBL1209421 | PHEN...)
Affinity DataKi:  7.52E+4nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416505(CHEMBL1209580)
Affinity DataKi:  1.07E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416484(CHEMBL1209503)
Affinity DataKi:  1.90E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50047005(1-Aza-bicyclo[2.2.2]octan-3-ol (3-quinuclidinol) |...)
Affinity DataKi:  2.10E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416496(CHEMBL1209650)
Affinity DataKi:  2.10E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416485(CHEMBL1209504)
Affinity DataKi:  2.70E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416483(CHEMBL1209424)
Affinity DataKi:  2.90E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50147105(CHEMBL102289 | CHEMBL1209423 | (4-Hydroxy-butyl)-t...)
Affinity DataKi:  3.10E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416499(TRIMETHYLAMMONIUM)
Affinity DataKi:  3.40E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416486(CHEMBL1209505)
Affinity DataKi:  3.40E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416500(CHEMBL1209652)
Affinity DataKi:  3.61E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM10458(pyridin-4-amine | CHEMBL284348 | 4-Aminopyridine 1...)
Affinity DataKi:  4.81E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50004108((R,S)-nicotine | (RS)-nicotine | nicotine | (+-)-n...)
Affinity DataKi:  5.20E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416493(CHEMBL354077)
Affinity DataKi:  8.20E+5nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416492(Integrase inhibitor, R3{3} | METHYLAMINE)
Affinity DataKi:  3.51E+7nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM7973(CHEMBL104943 | 2-aminoethan-1-ol | ethanolamine)
Affinity DataKi:  1.50E+8nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416487(CHEMBL1236196 | TETRABUTYLAMMONIUM)
Affinity DataKi:  1.05E+6nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50147120(2-Methylamino-ethanol | 2-hydroxy-N-methylethanami...)
Affinity DataKi:  3.80E+6nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
LigandPNGBDBM50416497(DIMETHYLAMINE)
Affinity DataKi:  9.42E+6nMAssay Description:Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed