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Report error Found 11 of affinity data for UniProtKB/TrEMBL: Q8DP79
TargetPeptide deformylase(Streptococcus pneumoniae)
Glaxosmithkline

LigandPNGBDBM92766(PDF inhibitor, compound 8)
Affinity DataKi:  53.7nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/5/2013
Entry Details Article
PubMed
TargetPeptide deformylase(Streptococcus pneumoniae)
Glaxosmithkline

LigandPNGBDBM92761(PDF inhibitor, compound 3)
Affinity DataKi:  117nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/5/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeptide deformylase(Streptococcus pneumoniae)
Glaxosmithkline

LigandPNGBDBM92764(PDF inhibitor, compound 6)
Affinity DataKi:  213nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/5/2013
Entry Details Article
PubMed
TargetPeptide deformylase(Streptococcus pneumoniae)
Glaxosmithkline

LigandPNGBDBM92760(PDF inhibitor, compound 2)
Affinity DataKi:  334nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/5/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeptide deformylase(Streptococcus pneumoniae)
Glaxosmithkline

LigandPNGBDBM21683(N-hydroxy-N-(3-phenylpropyl)formamide | SB-485345)
Affinity DataIC50: 400nMpH: 7.6 T: 2°CAssay Description:Enzyme assay was carried out in 96-well microtiter plates with a SpectraMax plate reader (Molecular Devices Corp.). PDF activity was measured using a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetPeptide deformylase(Streptococcus pneumoniae)
Glaxosmithkline

LigandPNGBDBM92765(PDF inhibitor, compound 7)
Affinity DataKi:  650nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/5/2013
Entry Details Article
PubMed
TargetPeptide deformylase(Streptococcus pneumoniae)
Glaxosmithkline

LigandPNGBDBM21685(N-hydroxy-N-[3-(6-methylpyridin-2-yl)propyl]formam...)
Affinity DataIC50: 2.20E+3nMpH: 7.6 T: 2°CAssay Description:Enzyme assay was carried out in 96-well microtiter plates with a SpectraMax plate reader (Molecular Devices Corp.). PDF activity was measured using a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeptide deformylase(Streptococcus pneumoniae)
Glaxosmithkline

LigandPNGBDBM21684(N-[2-(3-benzoylphenoxy)ethyl]-N-hydroxyformamide |...)
Affinity DataIC50: 3.90E+3nMpH: 7.6 T: 2°CAssay Description:Enzyme assay was carried out in 96-well microtiter plates with a SpectraMax plate reader (Molecular Devices Corp.). PDF activity was measured using a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeptide deformylase(Streptococcus pneumoniae)
Glaxosmithkline

LigandPNGBDBM92759(PDF inhibitor, compound 1)
Affinity DataKi:  6.31E+3nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/5/2013
Entry Details Article
PubMed
TargetPeptide deformylase(Streptococcus pneumoniae)
Glaxosmithkline

LigandPNGBDBM92762(PDF inhibitor, compound 4)
Affinity DataKi:  2.59E+4nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/5/2013
Entry Details Article
PubMed
TargetPeptide deformylase(Streptococcus pneumoniae)
Glaxosmithkline

LigandPNGBDBM92763(PDF inhibitor, compound 5)
Affinity DataKi:  3.17E+4nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/5/2013
Entry Details Article
PubMed