Compile Data Set for Download or QSAR
Report error Found 3 of affinity data for UniProtKB/TrEMBL: Q8IM71
TargetCholine kinase(Plasmodium falciparum (isolate 3D7))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50166172(Bisquinolinium derivative | CHEMBL192986)
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 choline kinase expressed in Escherichia coli BL21(DE3) assessed as reduction in phosphocholine formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetCholine kinase(Plasmodium falciparum (isolate 3D7))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50342874(1,1'-[4,4'-(Butane-1,4-diyl)bis(1,4-phenylene)]bis...)
Affinity DataIC50: 1.06E+5nMAssay Description:Inhibition of Plasmodium falciparum 3D7 choline kinase expressed in Escherichia coli BL21(DE3) assessed as reduction in phosphocholine formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed
TargetCholine kinase(Plasmodium falciparum (isolate 3D7))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM85206(CAS_312-45-8 | NSC_9399 | Hemicholinium-3)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of Plasmodium falciparum 3D7 choline kinase expressed in Escherichia coli BL21(DE3) assessed as reduction in phosphocholine formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2020
Entry Details Article
PubMed