Compile Data Set for Download or QSAR
Report error Found 16 of affinity data for UniProtKB/TrEMBL: Q8RT60
TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50021959(antibiotic MM 14151 | CHEMBL777 | MM 14151 | clavu...)
Affinity DataIC50: 30.1nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212638(CHEMBL302512)
Affinity DataIC50: 72nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212634(CHEMBL309009)
Affinity DataIC50: 83.7nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 106nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212640(CHEMBL423309)
Affinity DataIC50: 230nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212641(Brobactam)
Affinity DataIC50: 285nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212637(CHEMBL72046)
Affinity DataIC50: 370nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212639(CHEMBL302241)
Affinity DataIC50: 376nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212646(CHEMBL72972)
Affinity DataIC50: 524nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212635(CHEMBL415266)
Affinity DataIC50: 634nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212642(CHEMBL70269)
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212645(CHEMBL305908)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212643(CHEMBL308516)
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212644(CHEMBL73450)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50021954(UNASYN | 3,3-Dimethyl-4,4,7-trioxo-4lambda*6*-thia...)
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212636(CHEMBL310221)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details