Compile Data Set for Download or QSAR
Report error Found 542 of affinity data for UniProtKB/TrEMBL: Q9JKC1
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50235800(CHEBI:553827 | Bambuterol)
Affinity DataIC50: 3nMAssay Description:Inhibition of rat BChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50014107(CHEMBL74950 | 1,3alpha,8-trimethyl-1,2,3,3alpha,8,...)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of rat plasma BChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50004000(CHEMBL94 | physostigmine | Antilirium | Eserine | ...)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of rat plasma BChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50100592(CHEMBL3321889)
Affinity DataIC50: 8nMAssay Description:Inhibition of BChE in rat serum using butyrylthiocholine iodide substrate incubated for 15 mins by UV spectroscopy based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2016
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50004000(CHEMBL94 | physostigmine | Antilirium | Eserine | ...)
Affinity DataIC50: 8.10nMAssay Description:In vitro inhibitory concentration against butyrylcholinesterase (BuChE) obtained from rat plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50004000(CHEMBL94 | physostigmine | Antilirium | Eserine | ...)
Affinity DataIC50: 8.10nMAssay Description:Inhibitory concentration was determined in in vitro for Butyrylcholinesterase in rat plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50004000(CHEMBL94 | physostigmine | Antilirium | Eserine | ...)
Affinity DataIC50: 8.10nMAssay Description:ButyrylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50313191(1,3alpha,8-trimethyl-1,2,3,3alpha,8,8alpha-hexahyd...)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of rat plasma BChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 9nMAssay Description:Inhibition of rat plasma butyrylcholine esterase in presence of butyrylcholine substrate by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50100597(CHEMBL3321877)
Affinity DataIC50: 10nMAssay Description:Inhibition of BChE in rat serum using butyrylthiocholine iodide substrate incubated for 15 mins by UV spectroscopy based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2016
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50100578(CHEMBL3321887)
Affinity DataIC50: 12nMAssay Description:Inhibition of BChE in rat serum using butyrylthiocholine iodide substrate incubated for 15 mins by UV spectroscopy based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2016
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8980(N-[(1-benzylpiperidin-4-yl)methyl]-2-(1,2,3,4-tetr...)
Affinity DataIC50: 12.4nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The appearance of product was monitored at 412 nm for 5 min us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2006
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50313194(1,3alpha,8-trimethyl-1,2,3,3alpha,8,8alpha-hexahyd...)
Affinity DataIC50: 14.1nMAssay Description:Inhibition of rat plasma BChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50313184(1,3alpha,8-trimethyl-1,2,3,3alpha,8,8alpha-hexahyd...)
Affinity DataIC50: 14.9nMAssay Description:Inhibition of rat plasma BChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50100594(CHEMBL3321874)
Affinity DataIC50: 18nMAssay Description:Inhibition of BChE in rat serum using butyrylthiocholine iodide substrate incubated for 15 mins by UV spectroscopy based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2016
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50100576(CHEMBL3321885)
Affinity DataIC50: 24nMAssay Description:Inhibition of BChE in rat serum using butyrylthiocholine iodide substrate incubated for 15 mins by UV spectroscopy based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2016
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50100570(CHEMBL3321879)
Affinity DataIC50: 29nMAssay Description:Inhibition of BChE in rat serum using butyrylthiocholine iodide substrate incubated for 15 mins by UV spectroscopy based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2016
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50100572(CHEMBL3321881)
Affinity DataIC50: 34nMAssay Description:Inhibition of BChE in rat serum using butyrylthiocholine iodide substrate incubated for 15 mins by UV spectroscopy based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2016
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50100579(CHEMBL3321888)
Affinity DataIC50: 35nMAssay Description:Inhibition of BChE in rat serum using butyrylthiocholine iodide substrate incubated for 15 mins by UV spectroscopy based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2016
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50313188(1,3alpha,8-trimethyl-1,2,3,3alpha,8,8alpha-hexahyd...)
Affinity DataIC50: 39.6nMAssay Description:Inhibition of rat plasma BChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 44nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2006
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 44nMAssay Description:Inhibition of rat serum butyrylcholinesterase using butyrylthiocholine as substrate in presence of AChE inhibitor BW284C51 by spectrophotometric meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 55nMAssay Description:Compound was tested in vitro for inhibitory activity against ButyrylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50004000(CHEMBL94 | physostigmine | Antilirium | Eserine | ...)
Affinity DataIC50: 58.4nMAssay Description:Inhibition of BuChE in Wistar rat plasma using acetylthiocholine iodide as substrate after 0.5 hrs by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50313183(1,3alpha,8-trimethyl-1,2,3,3alpha,8,8alpha-hexahyd...)
Affinity DataIC50: 61.3nMAssay Description:Inhibition of rat plasma BChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50100595(CHEMBL3321875)
Affinity DataIC50: 63nMAssay Description:Inhibition of BChE in rat serum using butyrylthiocholine iodide substrate incubated for 15 mins by UV spectroscopy based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2016
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 73nMAssay Description:In vitro inhibitory concentration against Butyrylcholinesterase obtained from rat plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 73nMAssay Description:Inhibitory concentration was determined in in vitro for Butyrylcholinesterase in rat plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 73nMAssay Description:ButyrylcholinesteraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 74nMAssay Description:Inhibition of rat cortex homogenate BuChE by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8979(CHEMBL486901 | N-[2-(1-benzylpiperidin-4-yl)ethyl]...)
Affinity DataIC50: 76nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The appearance of product was monitored at 412 nm for 5 min us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2006
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8979(CHEMBL486901 | N-[2-(1-benzylpiperidin-4-yl)ethyl]...)
Affinity DataIC50: 76nMAssay Description:Inhibition of rat serum BChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8979(CHEMBL486901 | N-[2-(1-benzylpiperidin-4-yl)ethyl]...)
Affinity DataIC50: 76nMAssay Description:Inhibition of rat serum butyrylcholinesterase by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50100571(CHEMBL3321880)
Affinity DataIC50: 79nMAssay Description:Inhibition of BChE in rat serum using butyrylthiocholine iodide substrate incubated for 15 mins by UV spectroscopy based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2016
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 80nMAssay Description:Inhibition of rat serum BChE using butyrylthiocholine iodide as substrate after 20 mins by by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2020
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50100574(CHEMBL3321883)
Affinity DataIC50: 82nMAssay Description:Inhibition of BChE in rat serum using butyrylthiocholine iodide substrate incubated for 15 mins by UV spectroscopy based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2016
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50080157((RS)-tacrine(10)-hupyridone | 5-[10-(1,2,3,4-Tetra...)
Affinity DataIC50: 82nMAssay Description:Inhibitory potency against rat serum Butyrylcholinesterase with BW284c51 as AChE inhibitorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50080157((RS)-tacrine(10)-hupyridone | 5-[10-(1,2,3,4-Tetra...)
Affinity DataIC50: 82nMAssay Description:Inhibition of rat BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50313187(1,3alpha,8-trimethyl-1,2,3,3alpha,8,8alpha-hexahyd...)
Affinity DataIC50: 88.7nMAssay Description:Inhibition of rat plasma BChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 92nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The appearance of product was monitored at 412 nm for 5 min us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2006
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 92nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2006
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 92nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2006
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 92nMAssay Description:Inhibition of rat serum BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 92nMAssay Description:Inhibitory potency against rat serum Butyrylcholinesterase with BW284c51 as AChE inhibitorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 92nMAssay Description:Inhibition of rat serum BChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50272632(CHEMBL4128689)
Affinity DataIC50: 100nMAssay Description:Inhibition of rat serum BChE using butyrylthiocholine iodide as substrate after 20 mins by by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2020
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM10478(A2A.2HCl | CHEMBL213377 | N-[2-(1,2,3,4-tetrahydro...)
Affinity DataIC50: 102nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2006
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM10478(A2A.2HCl | CHEMBL213377 | N-[2-(1,2,3,4-tetrahydro...)
Affinity DataIC50: 102nMAssay Description:Inhibition of rat serum BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM10958((3aS,8aR)-1,3a,8-trimethyl-1H,2H,3H,3aH,8H,8aH-pyr...)
Affinity DataIC50: 104nMAssay Description:Inhibition of rat plasma BChE by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM8964(CHEMBL75274 | N-[8-(1,2,3,4-tetrahydroacridin-9-yl...)
Affinity DataIC50: 105nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2006
Entry Details Article
PubMed
Displayed 1 to 50 (of 542 total ) | Next | Last >>
Jump to: