Compile Data Set for Download or QSAR
Report error Found 36 of affinity data for UniProtKB/TrEMBL: Q9Y0I0
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105135(N2-(3-((12-((3-((4Amino,6-(methylamino)-1,3,5-tria...)
Affinity DataKi:  135nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089703(N-[4-(3-Nitrooxy-propyl)-phenyl]-[1,3,5]triazine-2...)
Affinity DataKi:  200nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105123(N2-(3-((12-((3-((4Amino,6-(dimethylamino)-1,3,5-tr...)
Affinity DataKi:  240nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105120(N-{3-[12-(3-Amino-propylamino)-dodecylamino]-propy...)
Affinity DataKi:  410nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105124(N2-(3-[12-(3-[(4,6-Diamino-1,3,5-triazin-2-yl)amin...)
Affinity DataKi:  500nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089708(2-(acetylamino)-N-{4-[(4,6-diamino-1,3,5-triazin-2...)
Affinity DataKi:  580nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105137(N-{3-[12-(3-Amino-propylamino)-dodecylamino]-propy...)
Affinity DataKi:  600nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089698(2-(acetylamino)-N-[2-(6-amino-9H-purin-9-yl)ethyl]...)
Affinity DataKi:  620nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105121(N2-(3-((9-((3-((4-Amino-6-(methylamino)-1,3,5-tria...)
Affinity DataKi:  750nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105125(N-{3-[12-(3-Amino-propylamino)-dodecylamino]-propy...)
Affinity DataKi:  1.00E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089705(9-(2-Nitrooxy-ethyl)-9H-purin-6-ylamine | CHEMBL26...)
Affinity DataKi:  1.90E+3nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105139(N1,N9-Di(3-(((4,6-(dimethylamino-1,3,5-triazin-2-y...)
Affinity DataKi:  2.40E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105132(N2-(3-((12-((3-((4,6-Di(dimethylamino)-1,3,5-triaz...)
Affinity DataKi:  2.50E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105141(N2-(3-((12-((3-((4,6-Di(methylamino)-1,3,5-triazin...)
Affinity DataKi:  3.20E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50366636(CHEMBL605462)
Affinity DataKi:  3.47E+3nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105133(N1,N9-Di(3-(((4-amino-6-(dimethylamino-1,3,5-triaz...)
Affinity DataKi:  4.60E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105134(N1,N9-Di(3-(di((4,6-diamino-1,3,5-triazin-2-yl)met...)
Affinity DataKi:  6.70E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105119(N2-(3-((9-((3-((4-Amino-6-(methylamino)-1,3,5-tria...)
Affinity DataKi:  1.00E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM108256(US8609833, 87 | CHEMBL2205239)
Affinity DataKi:  1.23E+4nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105129(N2-(3-((9-((3-((4,6-Di(methylamino)-1,3,5-triazin-...)
Affinity DataKi:  1.40E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105118(N1,N9-Di(3-(((4-amino-6-(dimethylamino-1,3,5-triaz...)
Affinity DataKi:  1.70E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105142(N-{3-[9-(3-Amino-propylamino)-nonylamino]-propyl}-...)
Affinity DataKi:  1.70E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105138(N2-(3-[9-(3-[(4,6-Diamino-1,3,5-triazin-2-yl)amino...)
Affinity DataKi:  1.90E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50421414(Cymelarsan | CYMELARSEN)
Affinity DataKi:  2.29E+4nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105128(N-{3-[12-(3-Amino-propylamino)-dodecylamino]-propy...)
Affinity DataKi:  2.50E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105143(N2-(3-((9-((3-((4,6-Di(dimethylamino)-1,3,5-triazi...)
Affinity DataKi:  2.90E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105131(N1,N9-Di(3-(((4,6-(dimethylamino-1,3,5-triazin-2-y...)
Affinity DataKi:  3.00E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105136(N2-(3-[2-(3-[(4,6-Diamino-1,3,5-triazin-2-yl)amino...)
Affinity DataKi:  5.50E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105130(N2-(3-[4-(3-[(4,6-Diamino-1,3,5-triazin-2-yl)amino...)
Affinity DataKi:  7.20E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105144(N1,N9-Di(3-(di((4,6-diamino-1,3,5-triazin-2-yl)met...)
Affinity DataKi:  8.20E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089701(5,7-Diamino-[1,2,5]oxadiazolo[3,4-d]pyrimidin-1-ol...)
Affinity DataKi:  1.17E+5nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105127(N2-(3-[4-(3-[(4,6-Diamino-1,3,5-triazin-2-yl)amino...)
Affinity DataKi:  1.25E+5nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105122(N2-(3-[2-(3-[(4,6-Diamino-1,3,5-triazin-2-yl)amino...)
Affinity DataKi:  1.63E+5nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089706(2-(acetylamino)-N-(6-aminopyridin-3-yl)-3-methyl-3...)
Affinity DataKi:  4.04E+5nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50089704(nitrooxymethyl-benzene | CHEMBL25961)
Affinity DataKi: >1.00E+6nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50366635(CHEMBL73188)
Affinity DataKi: >1.00E+6nMAssay Description:Compound was tested for inhibition of Adenosine transporter P2 type by using [2-3H]adenosine as radioligand in Trypanosoma equiperdumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed