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BindingDB contains 3.1M data for 1.3M Compounds and 9.6K Targets. Of those, 1.5M data for 708K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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9 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Small molecules that target phosphorylation dependent protein-protein interaction.EBI
Riken
Identification of Cyproheptadine as an Inhibitor of SET Domain Containing Lysine Methyltransferase 7/9 (Set7/9) That Regulates Estrogen-Dependent Transcription.EBI
Riken
Identification of new SUMO activating enzyme 1 inhibitors using virtual screening and scaffold hopping.EBI
Riken
Structural revision of kynapcin-12 by total synthesis, and inhibitory activities against prolyl oligopeptidase and cancer cells.EBI
Riken
Identification of quinazolinyloxy biaryl urea as a new class of SUMO activating enzyme 1 inhibitors.EBI
Riken
Contribution of Cage-Shaped Structure of Physalins to Their Mode of Action in Inhibition of NF-kB ActivationEBI
Riken
Design and synthesis of lignostilbene-alpha,beta-dioxygenase inhibitors.EBI
Riken
Discovery of Novel Spiroindoline Derivatives as Selective Tankyrase Inhibitors.EBI
Riken
Aminopyridine derivatives and their use as selective ALK-2 inhibitorsBDB
Novartis