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15 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis, pharmacology and pharmacokinetics of 3-(4-aryl-piperazin-1-ylalkyl)-uracils as uroselective alpha1A-antagonists.EBI
Roche Bioscience
N-arylpiperazinyl-N'-propylamino derivatives of heteroaryl amides as functional uroselective alpha 1-adrenoceptor antagonists.EBI
Roche Bioscience
Amino acid derived sulfonamide hydroxamates as inhibitors of procollagen C-proteinase: solid-phase synthesis of ornithine analogues.EBI
Roche Bioscience
Amino acid derived sulfonamide hydroxamates as inhibitors of procollagen C-proteinase. Part 2: Solid-phase optimization of side chains.EBI
Roche Bioscience
Solid-phase synthesis of di- and tripeptidic hydroxamic acids as inhibitors of procollagen C-proteinase.EBI
Roche Bioscience
Structure-based design of six novel classes of nonpeptide antagonists of the bradykinin B2 receptor.EBI
Roche Bioscience
1-sulfonyl piperidine derivatives as modulators of prokineticin receptorsBDB
Takeda Pharmaceutical
Radiolabeled compoundsBDB
Takeda Pharmaceutical
Dipeptidyl nitrile inhibitors of Cathepsin L.BDB
Astrazeneca
2-Cyclohexylcarbonylbenzimidazoles as potent, orally available and brain-penetrable opioid receptor-like 1 (ORL1) antagonists.BDB
Banyu Pharmaceutical
Second generation of BACE-1 inhibitors part 3: Towards non hydroxyethylamine transition state mimetics.BDB
Gsk
Identification and characterization of small molecule inhibitors of a class I histone deacetylase from Plasmodium falciparum.BDB
Harvard Medical School
Molecular cloning, characterization, and inhibition studies of the Rv1284 beta-carbonic anhydrase from Mycobacterium tuberculosis with sulfonamides and a sulfamate.BDB
Kochi Medical School