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17 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Functional 1,3a,6a-triazapentalene scaffold: Design of fluorescent probes for kinesin spindle protein (KSP).EBI
University of Shizuoka
Structure-Guided Design of Novel l-Cysteine Derivatives as Potent KSP Inhibitors.EBI
University of Shizuoka
Structure-Activity Relationship Study on Isothiocyanates: Comparison of TRPA1-Activating Ability between Allyl Isothiocyanate and Specific Flavor Components of Wasabi, Horseradish, and White Mustard.EBI
University of Shizuoka
Identification of Indole Alkaloid Structural Units Important for Stimulus-Selective TRPM8 Inhibition: SAR Study of Naturally Occurring Iboga Derivatives.EBI
University of Shizuoka
Activation and inhibition of thermosensitive TRP channels by voacangine, an alkaloid present in Voacanga africana, an African tree.EBI
University of Shizuoka
S-benzylisothiourea derivatives as small-molecule inhibitors of indoleamine-2,3-dioxygenase.EBI
University of Shizuoka
Ellagitannins and hexahydroxydiphenoyl esters as inhibitors of vertebrate squalene epoxidase.EBI
University of Shizuoka
Inhibition of vertebrate squalene epoxidase by isoprenyl gallates and phenylalkyl gallates.EBI
University of Shizuoka
Syntheses of 2-deoxy-2,3-didehydro-N-acetylneuraminic acid analogues modified by N-sulfonylamidino groups at the C-4 position and biological evaluation as inhibitors of human parainfluenza virus type 1.EBI
University of Shizuoka
Selective inhibition of methoxyflavonoids on human CYP1B1 activity.EBI
University of Shizuoka
Phenolic constituents of the aerial parts of Cimicifuga simplex and Cimicifuga japonica.EBI
University of Shizuoka
Bis(hetero)aryl derivatives as unique kinesin spindle protein inhibitors.EBI
University of Shizuoka
Synthesis and biological evaluation of L-cysteine derivatives as mitotic kinesin Eg5 inhibitors.EBI
University of Shizuoka
Ligand Screening System for the RXRα Heterodimer Using the Fluorescence RXR Agonist CU-6PMN.EBI
University of Shizuoka
Design, synthesis, and evaluation of a novel prodrug, a S-trityl-EBI
University of Shizuoka
Propolis Components from Stingless Bees Collected on South Sulawesi, Indonesia, and Their Xanthine Oxidase Inhibitory Activity.EBI
University of Shizuoka
Ligand-Phospholipid Conjugation: A Versatile Strategy for Developing Long-Acting Ligands That Bind to Membrane Proteins by Restricting the Subcellular Localization of the Ligand.EBI
University of Shizuoka