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35 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Strategy for designing selectivea-l-rhamnosidase inhibitors: Synthesis and biological evaluation of l-DMDP cyclic isothioureas.EBI
University of Toyama
Structural Insight into the Interactions between Death-Associated Protein Kinase 1 and Natural Flavonoids.EBI
University of Toyama
In silico and pharmacological screenings identify novel serine racemase inhibitors.EBI
University of Toyama
Inhibitory activities of propolis and its promising component, caffeic acid phenethyl ester, against amyloidogenesis of human transthyretin.EBI
University of Toyama
Docking and SAR studies of calystegines: binding orientation and influence on pharmacological chaperone effects for Gaucher's disease.EBI
University of Toyama
Synthesis and biological evaluation of N-(2-fluorophenyl)-2ß-deoxyfuconojirimycin acetamide as a potent inhibitor fora-l-fucosidases.EBI
University of Toyama
Rational design and synthesis of 4-substituted 2-pyridin-2-ylamides with inhibitory effects on SH2 domain-containing inositol 5'-phosphatase 2 (SHIP2).EBI
University of Toyama
Sesquiterpenes from the rhizomes of Curcuma heyneana.EBI
University of Toyama
Synthesis and evaluation of novel photoreactive alpha-amino acid analog carrying acidic and cleavable functions.EBI
University of Toyama
a-1-C-butyl-1,4-dideoxy-1,4-imino-l-arabinitol as a second-generation iminosugar-based orala-glucosidase inhibitor for improving postprandial hyperglycemia.EBI
University of Toyama
Cytochrome P450 3A4 inhibitory constituents of the wood of Taxus yunnanensis.EBI
University of Toyama
Isolation of glycosidase-inhibiting hyacinthacines and related alkaloids from Scilla socialis.EBI
University of Toyama
Design, synthesis, and biological evaluation of novel (1-thioxo-1,2,3,4-tetrahydro-ß-carbolin-9-yl)acetic acids as selective inhibitors for AKR1B1.EBI
University of Toyama
Docking and SAR studies of D- and L-isofagomine isomers as humanß-glucocerebrosidase inhibitors.EBI
University of Toyama
6,7-Dihydroxy-4-phenylcoumarin as inhibitor of aldose reductase 2.EBI
University of Toyama
2,5-Dideoxy-2,5-imino-d-altritol as a new class of pharmacological chaperone for Fabry disease.EBI
University of Toyama
Synthesis and evaluation of A-seco type triterpenoids for anti-HIV-1protease activity.EBI
University of Toyama
Possible involvement of radical intermediates in the inhibition of cysteine proteases by allenyl esters and amides.EBI
University of Toyama
Synthesis of poison-frog alkaloids 233A, 235U, and 251AA and their inhibitory effects on neuronal nicotinic acetylcholine receptors.EBI
University of Toyama
Resveratrol Derivatives Inhibit Transthyretin Fibrillization: Structural Insights into the Interactions between Resveratrol Derivatives and Transthyretin.EBI
University of Toyama
Design and Pharmacological Chaperone Effects of EBI
University of Toyama
Benziodarone and 6-hydroxybenziodarone are potent and selective inhibitors of transthyretin amyloidogenesis.EBI
University of Toyama
Chlorinated Naringenin Analogues as Potential Inhibitors of Transthyretin Amyloidogenesis.EBI
University of Toyama
Design and synthesis of pyrido[2,3-d]pyrimidine derivatives for a novel PAC1 receptor antagonist.EBI
University of Toyama
5-EBI
University of Toyama
Repositioning of the Anthelmintic Drugs Bithionol and Triclabendazole as Transthyretin Amyloidogenesis Inhibitors.EBI
University of Toyama
Inhibitory activities of anthraquinone and xanthone derivatives against transthyretin amyloidogenesis.EBI
University of Toyama
Transthyretin Amyloidogenesis Inhibitors: From Discovery to Current Developments.EBI
University of Toyama
Synthesis of a novel and potent small-molecule antagonist of PAC1 receptor for the treatment of neuropathic pain.EBI
University of Toyama
Crown Ethers as Transthyretin Amyloidogenesis Inhibitors.EBI
University of Toyama
Discovery of a new class of MTH1 inhibitor by X-ray crystallographic screening.EBI
University of Toyama
Inhibition of the dimerization and active site of HIV-1 protease by secondary metabolites from the Vietnamese mushroom Ganoderma colossum.EBI
University of Toyama
Synthesis of dammarane-type triterpene derivatives and their ability to inhibit HIV and HCV proteases.EBI
University of Toyama
Anti-HIV-1 protease activity of lanostane triterpenes from the vietnamese mushroom Ganoderma colossum.EBI
University of Toyama
Design and synthesis of novel anti-hyperalgesic agents based on 6-prenylnaringenin as the T-type calcium channel blockers.EBI
University of Toyama