24 articles for thisTarget
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Amino derivatives of platanic acid act as selective and potent inhibitors of butyrylcholinesterase.
Martin-Luther-University Halle-Wittenberg
Repurposing N,N'-bis-(arylamidino)-1,4-piperazinedicarboxamidines: An unexpected class of potent inhibitors of cholinesterases.
Martin-Luther-University Halle-Wittenberg
Discovery of substituted 1,4-dihydroquinolines as novel promising class of P-glycoprotein inhibitors: First structure-activity relationships and bioanalytical studies.
Martin-Luther-University Halle-Wittenberg
Discovery of 4-anilinoa-carbolines as novel Brk inhibitors.
Martin-Luther-University Halle-Wittenberg
Evaluation of potential Myt1 kinase inhibitors by TR-FRET based binding assay.
Martin-Luther-University Halle-Wittenberg
Multitargeted drug development: Discovery and profiling of dihydroxy substituted 1-aza-9-oxafluorenes as lead compounds targeting Alzheimer disease relevant kinases.
Martin-Luther-University Halle-Wittenberg
Three-dimensional quantitative structure-activity relationship analyses of beta-lactam antibiotics and tripeptides as substrates of the mammalian H+/peptide cotransporter PEPT1.
Martin-Luther-University Halle-Wittenberg
Evaluation of the first cytostatically active 1-aza-9-oxafluorenes as novel selective CDK1 inhibitors with P-glycoprotein modulating properties.
Martin-Luther-University Halle-Wittenberg
Three-dimensional quantitative structure-activity relationship analyses of peptide substrates of the mammalian H+/peptide cotransporter PEPT1.
Martin-Luther-University Halle-Wittenberg
In vitro and in silico studies on substrate recognition and acceptance of human PKMYT1, a Cdk1 inhibitory kinase.
Martin-Luther-University Halle-Wittenberg
Three-dimensional quantitative structure-activity relationship analyses of substrates of the human proton-coupled amino acid transporter 1 (hPAT1).
Martin-Luther-University Halle-Wittenberg
Discovery and selectivity-profiling of 4-benzylamino 1-aza-9-oxafluorene derivatives as lead structures for IGF-1R inhibitors.
Martin-Luther-University Halle-Wittenberg
Structural requirements for the substrates of the H+/peptide cotransporter PEPT2 determined by three-dimensional quantitative structure-activity relationship analysis.
Martin-Luther-University Halle-Wittenberg
Biological evaluation of bishydroxymethyl-substituted cage dimeric 1,4-dihydropyridines as a novel class of p-glycoprotein modulating agents in cancer cells.
Martin-Luther-University Halle-Wittenberg
Synthesis and biological evaluation of the first N-alkyl cage dimeric 4-aryl-1,4-dihydropyridines as novel nonpeptidic HIV-1 protease inhibitors.
Martin-Luther-University Halle-Wittenberg
Caffeic acid phenethyl ester (CAPE)-derivatives act as selective inhibitors of acetylcholinesterase.
Martin-Luther-University Halle-Wittenberg
Computer-aided design, synthesis and biological characterization of novel inhibitors for PKMYT1.
Martin-Luther-University Halle-Wittenberg
Evidence for the absolute conformational specificity of the intestinal H+/peptide symporter, PEPT1.
Martin-Luther-University Halle-Wittenberg
A novel inhibitor of the mammalian peptide transporter PEPT1.
Martin-Luther-University Halle-Wittenberg
Unexpected AChE inhibitory activity of (2E)α,β-unsaturated fatty acids.
Martin-Luther-University Halle-Wittenberg
Identification of PKMYT1 inhibitors by screening the GSK published protein kinase inhibitor set I and II.
Martin-Luther-University Halle-Wittenberg
Potent and Selective Inhibitors of Human Sirtuin 5.
Martin-Luther-University Halle-Wittenberg
Discovery of novel substituted benzo-anellated 4-benzylamino pyrrolopyrimidines as dual EGFR and VEGFR2 inhibitors.
Martin-Luther-University Halle-Wittenberg
