BDBM115261 US8637500, 68

SMILES OCC1CCN(CC1)c1cccnc1Oc1ccc(Nc2ccccn2)cc1

InChI Key InChIKey=CEOWZGDETRETFE-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 115261   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Rat)
Amgen

US Patent

LigandBDBM115261(US8637500, 68)Copy SMILESCopy InChI

Affinity DataIC50: 1.66nMT: 2°CAssay Description:An IMAP TR-FRET assay was used to analyze the enzyme activity (Molecular Devices Corp., Sunnyvale Calif.). 5 μL of serial diluted PDE10A (BPS Bi...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/22/2014
Entry Details
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