BDBM141165 US11547697, Compound 525::US9682141, 525

SMILES COc1ncc(cc1NS(C)(=O)=O)-c1ccc2ncn(C3CCN(C)CC3)c(=O)c2c1

InChI Key InChIKey=VDIDUPVPJHCFHE-UHFFFAOYSA-N

Data  7 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 141165   

LigandPNGBDBM141165(US9682141, 525 | US11547697, Compound 525)
Affinity DataIC50: 100nMAssay Description:An exemplary system is PI 3-Kinase (human) HTRF Assay from Upstate. The assay can be carried out according to the procedures suggested by the manufac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
US Patent

LigandPNGBDBM141165(US9682141, 525 | US11547697, Compound 525)
Affinity DataIC50: 100nMAssay Description:An exemplary system is PI 3-Kinase (human) HTRF Assay from Upstate. The assay can be carried out according to the procedures suggested by the manufac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
US Patent

LigandPNGBDBM141165(US9682141, 525 | US11547697, Compound 525)
Affinity DataIC50: 100nMT: 2°CAssay Description:Briefly, the assay is a time resolved FRET assay that indirectly measures PIP3 product formed by the activity of a PI3-K. The kinase reaction is perf...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2018
Entry Details
US Patent

LigandPNGBDBM141165(US9682141, 525 | US11547697, Compound 525)
Affinity DataIC50: 1.00E+3nMAssay Description:An exemplary system is PI 3-Kinase (human) HTRF Assay from Upstate. The assay can be carried out according to the procedures suggested by the manufac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
US Patent

LigandPNGBDBM141165(US9682141, 525 | US11547697, Compound 525)
Affinity DataIC50: 1.00E+3nMT: 2°CAssay Description:Briefly, the assay is a time resolved FRET assay that indirectly measures PIP3 product formed by the activity of a PI3-K. The kinase reaction is perf...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2018
Entry Details
US Patent

LigandPNGBDBM141165(US9682141, 525 | US11547697, Compound 525)
Affinity DataIC50: 1.00E+4nMAssay Description:An exemplary system is PI 3-Kinase (human) HTRF Assay from Upstate. The assay can be carried out according to the procedures suggested by the manufac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
US Patent

LigandPNGBDBM141165(US9682141, 525 | US11547697, Compound 525)
Affinity DataIC50: 1.00E+4nMT: 2°CAssay Description:Briefly, the assay is a time resolved FRET assay that indirectly measures PIP3 product formed by the activity of a PI3-K. The kinase reaction is perf...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2018
Entry Details
US Patent