BDBM148072 US8962609, DMX-6

SMILES COc1ccc(Nc2nccc(n2)-c2ccc(N3CCCC3)c(c2)C#N)cc1

InChI Key InChIKey=PEDJYEKGYANTDW-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 148072   

TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Human)
Domainex

US Patent

LigandBDBM148072(US8962609, DMX-6)Copy SMILESCopy InChI

Affinity DataIC50: 30nMpH: 7.5Assay Description:Inhibitions studies were performed using a time-resolved fluorescence-based Lanthascreen assay. Phosphorylation of a fluorescein-labelled substrate p...More data for this Ligand-Target Pair

Target InfoKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
7/15/2015
Entry Details
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