BDBM161991 US9682991, 40

SMILES CC1CN(C)c2c(NCC3CCN(C)CC3)nn3c(nnc3c2O1)-c1cccc(OC(F)(F)F)c1

InChI Key InChIKey=YJHZIINCQHGQNE-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 161991   

TargetSerine/threonine-protein kinase pim-1(Human)
FundaciÓN Centro Nacional De Investigaciones Oncologicas Carlos Iii

US Patent
LigandPNGBDBM161991(US9682991, 40)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure PIM-1 activity relies on the ADP Hunter assay kit (DiscoveRx Corp., Cat. #90-0077), that determines the amount of AD...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-3(Human)
FundaciÓN Centro Nacional De Investigaciones Oncologicas Carlos Iii

US Patent
LigandPNGBDBM161991(US9682991, 40)
Affinity DataIC50: 100nMAssay Description:The biochemical assay to measure PIM-3 activity relies on the ADP Hunter assay kit (DiscoveRx Corp., Cat. #90-0077), that determines the amount of AD...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-2(Human)
FundaciÓN Centro Nacional De Investigaciones Oncologicas Carlos Iii

US Patent
LigandPNGBDBM161991(US9682991, 40)
Affinity DataIC50: 550nMAssay Description:The biochemical assay to measure PIM-2 activity relies on the ADP Hunter assay kit (DiscoveRx Corp., Cat. #90-0077), that determines the amount of AD...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent