BDBM17588 bestatin-type inhibitor, 3::ethyl (2S)-2-[(2S,3S)-3-amino-2-hydroxy-4-[(2-methylpropyl)sulfanyl]butanamido]propanoate

SMILES CCOC(=O)[C@H](C)NC(=O)[C@@H](O)[C@H](N)CSCC(C)C

InChI Key InChIKey=MEGZWHWALUAWJD-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 17588   

TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17588(ethyl (2S)-2-[(2S,3S)-3-amino-2-hydroxy-4-[(2-meth...)
Affinity DataIC50: 1.10E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 1(Human)
Abbott Laboratories

LigandPNGBDBM17588(ethyl (2S)-2-[(2S,3S)-3-amino-2-hydroxy-4-[(2-meth...)
Affinity DataIC50: 6.60E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed