BDBM183026 US9150544, 60

SMILES CN(C)c1ccc(cn1)S(=O)(=O)N[C@H]1CCN([C@H](Cc2cc3ccnc(N)c3cc2OC(F)(F)F)C(O)=O)C1=O

InChI Key InChIKey=ZZCAKOUFQSCCCF-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 183026   

TargetCoagulation factor IX(Human)
Sanofi

US Patent
LigandPNGBDBM183026(US9150544, 60)
Affinity DataIC50: 130nMAssay Description:The compounds according to the invention are tested in a range of concentrations (4.9 nM to 5 µM final) and deposited in a proportion of 25 µl per we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
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TargetCoagulation factor X(Human)
Sanofi

US Patent
LigandPNGBDBM183026(US9150544, 60)
Affinity DataIC50: 34nMpH: 7.0Assay Description:The compounds according to the invention are tested in a range of concentrations (10pM to 10 µM final) in assay buffer (50 mM TRIS, 100 mM NaCl, 0.1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2016
Entry Details
Go to US Patent