BDBM18601 6-[bis(2,2,2-trifluoroethyl)amino]-4-methyl-1,2-dihydroquinolin-2-one::6-bisalkylamino-2-quinolinone, 7b

SMILES Cc1cc(=O)[nH]c2ccc(cc12)N(CC(F)(F)F)CC(F)(F)F

InChI Key InChIKey=VGAKCOHWSSQOBR-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 18601   

TargetAndrogen receptor(Human)
Ligand Pharmaceuticals

LigandPNGBDBM18601(6-[bis(2,2,2-trifluoroethyl)amino]-4-methyl-1,2-di...)
Affinity DataKi:  1.40nM EC50:  0.800nMAssay Description:The compounds were evaluated in a transcriptional activation assay with hAR in a mammalian cell background (CV-1) as the primary in vitro assay. Rece...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2007
Entry Details Article
PubMed