BDBM196911 US9212196, Derivative 7

SMILES COc1cc(cc(Cl)c1OCC(O)=O)C(O)P(O)(=O)CC[C@@H](N)C(O)=O

InChI Key InChIKey=CITKLHPQBXWCKK-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 196911   

TargetMetabotropic glutamate receptor 4(Rat)
Universite Paris Descartes

US Patent
LigandPNGBDBM196911(US9212196, Derivative 7)
Affinity DataEC50:  130nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
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TargetMetabotropic glutamate receptor 8(Rat)
Universite Paris Descartes

US Patent
LigandPNGBDBM196911(US9212196, Derivative 7)
Affinity DataEC50:  4.40E+4nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
Go to US Patent

TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Descartes

US Patent
LigandPNGBDBM196911(US9212196, Derivative 7)
Affinity DataEC50:  1.14E+4nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
Go to US Patent