BDBM20479 1-(2-bromophenyl)-3-{2-[methyl(3-methylphenyl)amino]ethyl}urea::urea TRPV1 antagonist, 12

SMILES CN(CCNC(=O)Nc1ccccc1Br)c1cccc(C)c1

InChI Key InChIKey=GECSVPIMSOPKGK-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20479   

LigandPNGBDBM20479(1-(2-bromophenyl)-3-{2-[methyl(3-methylphenyl)amin...)
Affinity DataEC50:  40nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2008
Entry Details Article
PubMed