BDBM23755 3-({4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}methyl)-4,5-dihydro-1,2,4-oxadiazol-5-one::PMS 1062 piperazine deriv., 24b

SMILES CCCCCCCCCCCCCCCCN1CCN(Cc2ccc(Cc3nc(=O)o[nH]3)cc2)CC1

InChI Key InChIKey=OHGIUXCURGDCJA-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 23755   

TargetPhospholipase A2, membrane associated(Human)
Universite Paris 7-Denis Diderot

LigandPNGBDBM23755(3-({4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}me...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2008
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Universite Paris 7-Denis Diderot

LigandPNGBDBM23755(3-({4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}me...)
Affinity DataIC50: 1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2008
Entry Details Article
PubMed