BDBM24371 2-{3-[(5-chloro-1H-indole-2-)amido]-2-oxo-1,2,3,4-tetrahydroquinolin-1-yl}acetic acid::3,4-dihydro-2-quinolone (DHQ) derivative, 10

SMILES OC(=O)CN1C(=O)C(Cc2ccccc12)NC(=O)c1cc2cc(Cl)ccc2[nH]1

InChI Key InChIKey=CCGBIWYBXDWOOH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 24371   

TargetGlycogen phosphorylase, liver form(Human)
Astrazeneca

LigandPNGBDBM24371(2-{3-[(5-chloro-1H-indole-2-)amido]-2-oxo-1,2,3,4-...)
Affinity DataIC50: 237nMpH: 7.2 T: 2°CAssay Description:The inhibitory activity of the test compounds against human recombinant glycogen phosphorylase a (GPa) was monitored using 96-well microplate format....More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2008
Entry Details Article
PubMed