BDBM2655 (Phenylindolyl)maleimide deriv. 77::3-(2,5-dimethylphenyl)-4-(1-methyl-1H-indol-3-yl)-2,5-dihydro-1H-pyrrole-2,5-dione

SMILES Cc1ccc(C)c(c1)C1=C(C(=O)NC1=O)c1cn(C)c2ccccc12

InChI Key InChIKey=AJAGWKXGNBDGDQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 2655   

TargetProtein kinase C beta type(Rat)
Roche Products

LigandPNGBDBM2655(3-(2,5-dimethylphenyl)-4-(1-methyl-1H-indol-3-yl)-...)
Affinity DataIC50: 1.20E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2004
Entry Details Article
PubMed
LigandPNGBDBM2655(3-(2,5-dimethylphenyl)-4-(1-methyl-1H-indol-3-yl)-...)
Affinity DataIC50: 8.20E+4nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2004
Entry Details Article
PubMed