BDBM270888 7-(benzenesulfonyl)-4-(morpholin-4-yl)-5H-pyrrolo[3,2-d]pyrimidin-6-amine::US10059713, Example 6

SMILES Nc1[nH]c2c(ncnc2c1S(=O)(=O)c1ccccc1)N1CCOCC1

InChI Key InChIKey=YTDBHTZELLWIGP-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 270888   

TargetFree fatty acid receptor 2(Human)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM270888(7-(benzenesulfonyl)-4-(morpholin-4-yl)-5H-pyrrolo[...)
Affinity DataEC50:  273nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent