BDBM270895 6-amino-4-(cyclohex-1-en-1-yl)-N-(4-methoxyphenyl)-N-methyl-5H-pyrrolo[3,2-d]pyrimidine-7-sulfonamide::US10059713, Example 14

SMILES COc1ccc(cc1)N(C)S(=O)(=O)c1c(N)[nH]c2c(ncnc12)C1=CCCCC1

InChI Key InChIKey=ATQGBTGRQWFIPY-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 270895   

TargetFree fatty acid receptor 2(Human)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM270895(6-amino-4-(cyclohex-1-en-1-yl)-N-(4-methoxyphenyl)...)
Affinity DataEC50:  267nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent