BDBM270911 7-(benzenesulfonyl)-4-(4-methoxypiperidin-1-yl)-5H-pyrrolo[3,2-d]pyrimidin-6-amine::US10059713, Example 28

SMILES COC1CCN(CC1)c1ncnc2c(c(N)[nH]c12)S(=O)(=O)c1ccccc1

InChI Key InChIKey=QZQXROUEYFPYDJ-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 270911   

TargetFree fatty acid receptor 2(Human)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM270911(7-(benzenesulfonyl)-4-(4-methoxypiperidin-1-yl)-5H...)
Affinity DataEC50:  399nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
US Patent