BDBM270923 7-(benzenesulfonyl)-4-cyclohexyl-2-methyl-5H-pyrrolo[3,2-d]pyrimidin-6-amine::US10059713, Example 40
SMILES Cc1nc(C2CCCCC2)c2[nH]c(N)c(c2n1)S(=O)(=O)c1ccccc1
InChI Key InChIKey=FTSXZSDAYGPPCY-UHFFFAOYSA-N
Data 1 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 270923
Affinity DataEC50: 37nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair
