BDBM27488 2-amino-3-(4-{[3-(morpholin-4-yl)propyl]sulfamoyl}phenyl)-5-phenylbenzamide::Amino-substituted diarylbenzamide, 8u

SMILES NC(=O)c1cc(cc(c1N)-c1ccc(cc1)S(=O)(=O)NCCCN1CCOCC1)-c1ccccc1

InChI Key InChIKey=YVHUOVHVRVMPMH-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 27488   

LigandPNGBDBM27488(2-amino-3-(4-{[3-(morpholin-4-yl)propyl]sulfamoyl}...)
Affinity DataIC50: 316nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2009
Entry Details Article
PubMed
LigandPNGBDBM27488(2-amino-3-(4-{[3-(morpholin-4-yl)propyl]sulfamoyl}...)
Affinity DataIC50: 1.00E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2009
Entry Details Article
PubMed
LigandPNGBDBM27488(2-amino-3-(4-{[3-(morpholin-4-yl)propyl]sulfamoyl}...)
Affinity DataIC50: 1.58E+4nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2009
Entry Details Article
PubMed