BDBM27492 2-amino-5-phenyl-3-(4-{[2-(pyrrolidin-1-yl)ethyl]sulfamoyl}phenyl)benzamide::Amino-substituted diarylbenzamide, 8y

SMILES NC(=O)c1cc(cc(c1N)-c1ccc(cc1)S(=O)(=O)NCCN1CCCC1)-c1ccccc1

InChI Key InChIKey=ARAKMVRBBTWPJZ-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 27492   

LigandPNGBDBM27492(2-amino-5-phenyl-3-(4-{[2-(pyrrolidin-1-yl)ethyl]s...)
Affinity DataIC50: 794nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2009
Entry Details Article
PubMed
LigandPNGBDBM27492(2-amino-5-phenyl-3-(4-{[2-(pyrrolidin-1-yl)ethyl]s...)
Affinity DataIC50: 251nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2009
Entry Details Article
PubMed
LigandPNGBDBM27492(2-amino-5-phenyl-3-(4-{[2-(pyrrolidin-1-yl)ethyl]s...)
Affinity DataIC50: 1.58E+4nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2009
Entry Details Article
PubMed