BDBM310287 US10150760, Example 83.0::US10150760, Example 84.0

SMILES CO[C@@H]([C@H](C)S(=O)(=O)Nc1nnc([C@H]2CCCCO2)n1-c1c(OC)cccc1OC)c1ncc(Cl)cn1

InChI Key InChIKey=PTNMUXPIZNNNNU-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 310287   

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310287(US10150760, Example 83.0 | US10150760, Example 84....)
Affinity DataEC50:  0.800nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310287(US10150760, Example 83.0 | US10150760, Example 84....)
Affinity DataEC50:  10nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
US Patent