BDBM310379 US10150760, Example 199.0::US10150760, Example 200.0

SMILES CO[C@@H]([C@H](C)S(=O)(=O)Nc1nnc([C@H]2CC[C@@H](C)O2)n1C1(C)CC1)c1ncc(Cl)cn1

InChI Key InChIKey=ARNRZJBJDGPFBC-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 310379   

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310379(US10150760, Example 199.0 | US10150760, Example 20...)
Affinity DataEC50:  2.70nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310379(US10150760, Example 199.0 | US10150760, Example 20...)
Affinity DataEC50:  290nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
US Patent