BDBM310417 US10150760, Example 240.0

SMILES CO[C@@H]([C@H](C)S(=O)(=O)Nc1nnc([C@@H]2CCCO2)n1-c1ccccc1OC)c1ncc(Cl)cn1

InChI Key InChIKey=OIHYWUQDIRVTRY-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 310417   

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM310417(US10150760, Example 240.0)
Affinity DataEC50:  1.30nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
US Patent