BDBM310902 6-methyl-4-[4-(1-methyl-4-piperidyl)phenyl]-1H-pyrrolo[2,3-c]pyridin-7-one::US10150767, Example 42

SMILES CN1CCC(CC1)c1ccc(cc1)-c1cn(C)c(=O)c2[nH]ccc12

InChI Key InChIKey=VAGZNNSTEOVTJS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 310902   

TargetBromodomain-containing protein 9 [134-239](Human)
Genentech

US Patent
LigandPNGBDBM310902(US10150767, Example 42 | 6-methyl-4-[4-(1-methyl-4...)
Affinity DataIC50: 53nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
US Patent